DOI: 10.1055/s-00000083

Synlett

Issue 04 · Volume 2010 · March 2010 DOI: 10.1055/s-002-20806

Editorial

I
Editorial

synform

A22
Zanda, Matteo: SYNFORM ISSUE 2010/03

letter

505
Qian, Zizheng; Baxendale, Ian R.; Ley, Steven V.: A Flow Process Using Microreactors for the Preparation of a Quinolone Derivative as a Potent 5HT1B Antagonist
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509
Silva, Eduarda M. P.; Pye, Richard J.; Cardin, Christine; Harwood, Laurence M.: Probing a Biomimetic Approach to Mycaperoxide B: Hydroperoxidation Studies
https://www.thieme-connect.de/media/synlett/201004/d291_ga.jpg
514
Padwal, Jalindar; Lewis, William; Moody, Christopher J.: Synthesis of the Reported Structure of Crassiflorone, a Pentacyclic Naphthoquinone Isolated from the African Ebony Diospyros crassiflora
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517
Chappell, David; Drew, Michael G. B.; Gibson, Shane; Harwood, Laurence M.; Russell, Andrew T.: Formal Total Synthesis of (±)-Conduramine E Utilising the Bryce-Smith-Gilbert Photoamination Reaction
https://www.thieme-connect.de/media/synlett/201004/d369_ga.jpg
521
Keshipeddy, Santosh; Shi, Yu; Hnatiuk, Nathan; Morton, Martha; Yao, Xudong; Howell, Amy R.: Design and Synthesis of an Activity-Based Probe Template for Protein Kinases
https://www.thieme-connect.de/media/synlett/201004/d238_ga.jpg
Supporting Information
525
Sharma, Pallavi; Moses, John E.: Photochemical Studies of the Tridachiahydropyrones in Seawater
https://www.thieme-connect.de/media/synlett/201004/d269_ga.jpg
529
Macleod, Fraser; Lang, Stuart; Murphy, John A.: The 2-(2-Azidoethyl)cycloalkanone Strategy for Bridged Amides and Medium-Sized Cyclic Amine Derivatives in the Aubé-Schmidt Reaction
https://www.thieme-connect.de/media/synlett/201004/d322_ga.jpg
Supporting Information
535
Hameed, Abdul; Blake, Alexander J.; Hayes, Christopher J.: An Enantioselective Formal Synthesis of (+)-Lactacystin from Hydroxymethyl Glutamic Acid (HMG)
https://www.thieme-connect.de/media/synlett/201004/d324_ga.jpg
539
Crosby, Stuart R.; Sessions, Richard B.; Willis, Christine L.: Intermediates for the Synthesis of 4-Substituted Proline Derivatives
https://www.thieme-connect.de/media/synlett/201004/d011_ga.jpg
543
Clarke, Paul A.; Black, Richard J. G.; Iqbal, Mudassar: Investigation of Transannelation Reactions Across a Cyclononene Ring
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547
Goldring, William P. D.; Mann, John; Brockbank, Paul: A Synthesis of (S)-(-)-Umbelactone and Related α,β-Butenolides
https://www.thieme-connect.de/media/synlett/201004/d293_ga.jpg
Supporting Information
551
Black, Richard J. G; Dungan, Victoria J.; Li, Rebecca Y. T.; Young, Philip G.; Jolliffe, Katrina A.: A Cyclooligomerisation Approach to Backbone-Modified Cyclic Peptides Bearing Guanidinium Arms
https://www.thieme-connect.de/media/synlett/201004/d316_ga.jpg
Supporting Information
555
Chattopadhyay, Shital K.; Singha, Sovan K: Efficient Construction of the Carbon Skeleton of the Novel Polyoxazole-Based Cyclopeptide IB-01211 via a Biomimetic Macrocyclisation
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559
Stockman, Robert A.; McDermott, Paul J.; Newton, Annabella F.; Magnus, Philip: A Versatile Chiral Pyrrolidine Aldehyde Building-Block for Synthesis and Formal Synthesis of ent-Nakadomarin A
https://www.thieme-connect.de/media/synlett/201004/d320_ga.jpg
563
Wang, Lei; Liu, Junyang; Zhang, Hui; Xu, Zhengshuang; Ye, Tao: Progress towards the Total Synthesis of Scytonemin A: Asymmetric Synthesis of (2S,3R,4R)-4-hydroxy-3-methylproline
https://www.thieme-connect.de/media/synlett/201004/d334_ga.jpg
Supporting Information
567
Davies, Stephen G.; Hughes, Deri G.; Price, Paul D.; Roberts, Paul M.; Russell, Angela J.; Smith, Andrew D.; Thomson, James E.; Williams, Oliver M. H.: Asymmetric Synthesis of Piperidines and Octahydroindolizines
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571
Paterson, Ian; Rubenbauer, Philipp: Synthetic Studies towards Iriomoteolide 1a: Stereocontrolled Construction of C1-C9 and C11-C23 Segments Using Lactate Aldol Chemistry
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575
Basar, Norazah; Donnelly, Sam; Liu, Hao; Thomas, Eric J.: 1,5-Stereocontrol in Bismuth-Mediated Reactions between Aldehydes and Allyl Bromides: Stereoselective Synthesis of Open-Chain all-syn- and anti, anti-1,3,5-Disposed Trimethylalkanes
https://www.thieme-connect.de/media/synlett/201004/d34809st-10-1055_s-0029-1219357_ga.jpg
579
Killen, Jonathan C.; Leonard, John; Aggarwal, Varinder K.: A Novel Asymmetric Azaspirocyclisation Using a Morita-Baylis-Hillman-Type Reaction
https://www.thieme-connect.de/media/synlett/201004/d351_ga.jpg
Supporting Information
583
Winzar, Renee; Philips, Jessica; Kiefel, Milton J.: A Simple Synthesis of C-8 Modified 2-Keto-3-deoxy-d-manno-octulosonic Acid (KDO) Derivatives
https://www.thieme-connect.de/media/synlett/201004/d370_ga.jpg
Supporting Information
587
Garrido, Narciso M.; Rubia, Alfonso G.; Nieto, Carlos; Díez, David: Potential of (2E,7E)-Nonadienedioates in Asymmetric Synthesis: Construction of Homopipecolic Acid and an Aminoester Building Block for Peptide Nucleic Acids
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591
Williams, David R.; Fu, Liangfeng: Methodology for the Synthesis of Substituted 1,3-Oxazoles
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595
Chapman, Helen A.; Herbal, Karim; Motherwell, William B.: Studies towards the Taming of the ‘Carbocation’ in the Regioselective Ring Opening of Epoxides to Allylic Alcohols
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599
Bray, Christopher D.; Olasoji, Joy: A Total Synthesis of (+)-Bacillamide B
https://www.thieme-connect.de/media/synlett/201004/d252_ga.jpg
Supporting Information
602
Beltrán-Rodil, Sandra; Edwards, Michael G.; Pugh, David. S.; Reid, Mark; Taylor, Richard J. K.: The Preparation of Substituted Pyrazoles from β,β-Dibromo-enones by a Tandem Condensation/Suzuki-Miyaura Cross-Coupling Process
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607
Roth, Stefanie; Thomas, Neil R.: A Concise Route to l-Azidoamino Acids: l-Azidoalanine, l-Azidohomo­alanine and l-Azidonorvaline
https://www.thieme-connect.de/media/synlett/201004/d280_ga.jpg
610
Clark, Andrew J.; Fullaway, David R.; Murphy, Nicholas P.; Parekh, Hemal: Copper(I) Halide Mediated Tandem 1,4-Aryl Migration-Oxidative Amidyl Radical Cyclisation of Bromosulfonamides
https://www.thieme-connect.de/media/synlett/201004/d287_ga.jpg
615
Brogan, Samantha; Carter, Neil B.; Lam, Hon Wai: Copper-Bisphosphine-Initiated Pentafluorophenylation of Aldehydes and Ketones
https://www.thieme-connect.de/media/synlett/201004/d308_ga.jpg
Supporting Information
618
Lygo, Barry; Beaumont, Douglas J.; Cooke, Jason W. B.; Hirst, David J.: Synthesis of Brombyins II and III, Cyclostachines A and B, and Cyclopiperstachine, Plant-Derived Octahydronaphthalenes
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623
North, Michael; Villuendas, Pedro: Aluminium(salen) and Tetrabutylammonium Bromide Catalysed Synthesis of Cyclic Di- and Trithiocarbonates from Epoxides and Carbon Disulfide
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628
Knight, David W.; Proctor, Anthony J.; Clough, John M.: New Regiospecific Catalytic Approaches to 4,5-Dihydroisoxazoles and 2,5-Dihydroisoxazoles from O-Propargylic Hydroxylamines
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633
Denton, Ross M.; Scragg, James T.: A Concise Synthesis of Dunnianol
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636
Tang, Xiaoping; Rawson, Daniel; Woodward, Simon: Direct Reaction of Aryl Iodides with Activated Aluminium Powder and Reactions of the Derived Aryl Sesquiiodides
https://www.thieme-connect.de/media/synlett/201004/d327_ga.jpg
639
Simpkins, Nigel S.; Taylor, James D.; Weller, Michael D.; Hayes, Christopher J.: Synthesis of Nemorosone via a Difficult Bridgehead Substitution Reaction
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644
Wipf, Peter; George, Kara M.: Regioselective Palladium-Catalyzed Cross-Coupling Reactions of 2,4,7-Trichloroquinazoline
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Supporting Information
649
Kędzia, Jacek L.; Kerr, William J.; McPherson, Allan R.: Regioselective Pauson-Khand Processes with Olefins Possessing Extended Phosphonates
https://www.thieme-connect.de/media/synlett/201004/d386_ga.jpg
654
Jones, Raymond C. F.; Choudhury, Abdul K.; Iley, James N.; Loizou, Georgia; Lumley, Christopher; McKee, Vickie: New Methodologies for the Synthesis of 3-Acylpyridone Metabolites
https://www.thieme-connect.de/media/synlett/201004/d338_ga.jpg
659
Boto, Alicia; Hernández, Rosendo; Saavedra, Carlos J.: One-Pot Conversion of α-Amino Acids into β-Amino Aldehydes or 2-Acetoxyazetidines: Application to the Synthesis of Modified Peptides
https://www.thieme-connect.de/media/synlett/201004/d309_ga.jpg
664
Sançon, Julien; Sweeney, J. B.: Probing the Effect of Allylic Substitution on Cyclic Ammonium Ylid Rearrangements
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667
Zhang, Kai; Gudipati, Venugopal; Curran, Dennis P.: Fluorous Mixture Synthesis of Four Stereoisomers of the C21-C40 Fragment of Tetrafibricin
https://www.thieme-connect.de/media/synlett/201004/d013_ga.jpg
Supporting Information
672
Stevenson, Brett; Lewis, William; Dowden, James: Expedient Route to an Amine Precursor of Halichlorine and Pinnaic Acid from Nitrocyclopent-1-ene
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Supporting Information

addenda and errata

e4
Fluorous Mixture Synthesis of Four Stereoisomers of the C21-C40 Fragment of Tetrafibricin