Synthesis

Issue 05 · March 2025

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table of contents
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review
891
Sajjad, Farrukh; Zhang, Shuyue; Xu, Ming-Hua:
Advances in Transition-Metal Catalysis and Organocatalysis Approaches towards Asymmetric Synthesis of β-Amino Acid Derivatives

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short review
917
Liu, Xigong; Liu, Lei:
Catalytic Asymmetric Syntheses of 3-Monosubstituted Oxindoles

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925
Horwitz, Matthew A.:
Discovery Process Chemistry: An Innovation Hub at the Interface of Academia, the Pharmaceutical Industry, and Contract Research Organizations

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937
Xie, Ke; Li, Ao; Kong, Bao-Rui; Chen, Zhi-Chao; Du, Wei; Chen, Ying-Chun:
Recent Advances in Asymmetric Addition Reactions to Isatins

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Dual Catalysis
953
Atriardi, Shafrizal R.; Anita, Yulia; Woo, Sang Kook:
Harnessing Photoredox and Weak Brønsted Base Dual Catalysis for Selective C(sp³)–H Bond Activation

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feature
965
Mizobuchi, Eduardo F.; Burtoloso, Antonio C. B.:
The Acylation of α-Carbonyl Sulfoxonium Ylides with N-Hydroxyphthalimide Esters

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psp
973
Chaudhury, Subhabrata; Thennakoon, Dulanjali; Wetzel, Edward A.; Donaldson, William A.:
A Scalable, Chromatography-Free Synthesis of the Potent and Highly Selective ERβ Agonist EGX358

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paper
978
Guo, Taijie; Wang, Wei; Xu, Long; Dong, Jiajia:
RNHSO₂F as Reliable Azasulfene Precursors for the Construction of Sulfamates

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SuFEx Chemistry
991
Tao, Guang; Fayad, Eman; Abu Ali, Ola A.; Oyom, Bright; Qin, Hua-Li:
A Convenient One-Pot Process for Converting Thiols into Sulfonyl Fluorides Using H₂O₂ as an Oxidant

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999
Yang, Na; Pei, Guanhua; Li, Hao; Han, Junwei; Wang, Peng; Xie, Lili; Liao, Saihu:
Synthesis of FSO₂-Functionalized Oxindoles via a Radical Fluorosulfonylation/Intramolecular Arylation Cascade

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1007
Dasmahapatra, Upala; Choudhury, Badruzzaman; Ahmad, Md Gulzar; Maiti, Barnali; Chanda, Kaushik:
Direct Access to 5,6-Dihydropyrido[2′,1′:2,3]pyrido-Fused Imidazo [4,5-c]quinolines via Consecutive C–N and C–C Bond Formation in Deep Eutectic Solvent under Microwave Irradiation

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1015
Olu-Igbiloba, Oluwaseun A.; Sitzmann, Helmut; Manolikakes, Georg:
Cobalt-Catalyzed Three-Component Synthesis of α-Substituted N-Sulfonyl Amines via C(sp²)–H Bond Activation

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Dual Catalysis
1025
Wang, Mingze; Zi, Weiwei:
Synergistic Pd/Cu-Catalyzed Asymmetric Csp³–Csp³ Coupling of 1,3-Dienes with 2-Acylimidazoles

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C–S Bond Forming and Cleaving Reactions
1034
Bugaenko, Dmitry I.; Karchava, Alexander V.:
Synthesis of 2-Aminobenzo[b]thiophenes via an Intramolecular Dehydrogenative C–S Bond Formation Effected by Iodine(III) Reagents

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1043
Endo, Koki; Shibahara, Fumitoshi:
Imidazo[1,5-a]pyridin-3-ylidene-Catalyzed Oxidative Esterification of Aldehydes: Remarkable Electronic Effect Regarding π-Accepting Character of Ring-Fused N-Heterocyclic Carbene

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1050
Singroha, Rekha; Onen, Patrick; Yadav, Usha; Kant, Ruchir; Mohanan, Kishor:
Three-Component Synthesis of Cyanopyrazoles Employing Diazoacetonitrile

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1059
Buravov, Oleksandr V.; Tomak, Victor O.; Shishkina, Svitlana V.; Chebanov, Valentyn A.:
First Example of Aryl–Hetaryl Cross-Coupling via [5,5]-Sigmatropic Rearrangement

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1072
Michon, Synthia; Garcia, Maxime; Cavelier, Florine; Salom-Roig, Xavier J.:
Divergent Synthetic Strategy To Access the Polyketide Subunits of Aurilides: Synthesis of the Southern Fragment of Lagunamides D and D′

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