Synlett

Issue 05 · Volume 2010 · March 2010 DOI: 10.1055/s-002-20856

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675

Shapiro, Nathan D.; Toste, F. Dean: A Reactivity-Driven Approach to the Discovery and Development of Gold-Catalyzed Organic Reactions

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692

Wang, Shaozhong; Zhang, Guozhu; Zhang, Liming: Gold-Catalyzed Reaction of Propargylic Carboxylates via an Initial 3,3-Rearrangement

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letter

707

Wei, Shengwei; Stingl, Kerstin A.; Weiß, Katharina M.; Tsogoeva, Svetlana B.: Thieme Chemistry Journal Awardees - Where Are They Now? Bifunctional Organocatalysis with N-Formyl-l-Proline: A Novel Approach to Epoxide Ring Opening and Sulfide Oxidation

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712

Yadav, Ashok K.; Kumar, Manoj; Yadav, Tripti; Jain, Renuka: (1R,5R)-1-(1′-Dimethylaminoethyl)-2-isopropylidene-5-methylcyclohexanol as a Chiral Ligand in the Enantioselective Addition of Diethylzinc to Aldehydes

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715

Sureshbabu, Vommina V.; Chennakrishnareddy, Gundala; Hemantha, Hosahalli P.: Synthesis of Thioureido-Linked Peptidomimetics, Glycosylated Amino Acids, and Neoglycoconjugates Using Bis(benzotriazolyl)methanethione as Thioacylating Agent

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721

Sreeramamurthy, Kintali; Ashok, Ettam; Mahendar, Velisoju; Santoshkumar, Gourishetti; Das, Parthasarathi: Direct Synthesis of N-Aryl Derivatives of Quinazolin-4(3H)-ones Employing Arylboronic Acids in the Presence of Cu(OAc)₂

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725

Schleiss, Julie; Cerniauskaite, Deimante; Gueyrard, David; Iori, Renato; Rollin, Patrick; Tatibouët, Arnaud: Thioimidate N-Oxides: From Nature to Synthetic Pathways

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729

Frigerio, Fabio; Haseler, Claire A.; Gallagher, Timothy: Synthesis of (+)-Kuraramine

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Supporting Information

731

Ali, Asad; Khera, Rasheed Ahmad; Ibad, Muhammad Farooq; Hussain, Munawar; Langer, Peter: Synthesis of Bis(diaryl)sulfones by Site-Selective Suzuki-Miyaura Reactions of 2,4′-Bis(trifluoromethylsulfonyloxy)diphenylsulfone

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735

Majumdar, K. C.; Taher, Abu; Ponra, Sudipta: Unusual Product from Condensative Cyclization: Pyrano[3,2-f]quinolin-3,10-diones from 6-Amino-5-[(trimethylsilyl)ethynyl]-2H-chromen-2-one and Aryl Aldehydes

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Supporting Information

741

Hajipour, Abdol R.; Ghayeb, Yosof; Sheikhan, Nafisehsadat; Ruoho, Arnold E.: Brønsted Acidic Ionic Liquid as an Efficient and Reusable Catalyst for Synthesis of 14-Aryl- or 14-Alkyl-14H-dibenzo[a,j]xanthenes under Solvent-Free Conditions

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745

Borkin, Dmitry; Carlson, Alena; Török, Béla: K-10-Catalyzed Highly Diastereoselective Synthesis of Aziridines

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749

Baumann, Marcus; Baxendale, Ian R.; Ley, Steven V.: Synthesis of 3-Nitropyrrolidines via Dipolar Cycloaddition Reactions Using a Modular Flow Reactor

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753

Vitoriano, Bruno C.; Carvalho, Luísa C. R.; Estevão, Mónica S.; Sekera, Michael H.; Marques, M. Manuel B.: A Simple Route Toward New Clomiphene Metabolites

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Supporting Information

757

Ramesh, Subburethinam; Gaddam, Vikram; Nagarajan, Rajagopal: A Flexible Approach to the Chromenoquinolines under Copper/Lewis Acid Catalysis

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Supporting Information

761

Hanessian, Stephen; Mi, Xueling: An Organocatalytic Approach to Enantiopure 2,6-Disubstituted Tetrahydropyranols

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765

Niu, Liang-Feng; Xin, Yang-Chun; Wang, Ren-Lin; Jiang, Fan; Xu, Peng-Fei; Hui, Xin-Ping: Asymmetric Aza-Friedel-Crafts Reaction of 2-Naphthol with Tosylimines Catalyzed by a Dinuclear Zinc Complex

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Supporting Information

769

Phillips, David J.; Graham, Andrew E.: Guanidine Bases in Synthesis: Extending the Scope of the Corey-Chaykovsky Epoxidation

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774

Friedmann, Christian; Bräse, Stefan: Synthesis of Paracyclophane Thiols via an Unprecedented Reduction-Deprotection Sequence: Direct Conversion of tert-Butyl Sulfoxides into Thiols with Boron Tribromide

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777

Praveen, C.; Kalyanasundaram, A.; Perumal, P. T.: Gold(III)-Catalyzed Synthesis of Isoxazoles by Cycloisomerization of α,β-Acetylenic Oximes

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782

Körber, Nadine; Rominger, Frank; Müller, Thomas J. J.: Enantioselective One-Pot Rhodium-Catalyzed Cycloisomerization-Wittig Sequence to Chiral Functionalized 4-Alkyl 3-Alkylidene Tetrahydrofuran(on)es

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787

Weisbrod, Samuel H.; Marx, Andreas: Synthesis of Water-Soluble Phosphinophenol for Traceless Staudinger Ligation

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790

Silveira, Claudio C.; Mendes, Samuel R.; Líbero, Francieli M.: Solvent-Free Anti-Markovnikov Addition of Thiols to Alkenes Using Anhydrous Cerium(III) Chloride as Catalyst

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793

Wilding, Emily E.; Gregg, John J.; Mullins, Richard J.: Asymmetric Conjugate Addition of Crotylstannane: Synthesis of (-)-Lasiol

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796

Johnson, Sarah; Drowns, Matt; Tatlock, John; Linton, Angelica; Gonzalez, Javier; Hoffman, Robert; Jewell, Tanya; Patel, Leena; Blazel, Julie; Tang, Mingnam; Li, Hui: Synthetic Route Optimization of PF-00868554, An HCV Polymerase Inhibitor in Clinical Evaluation

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801

Yano, Tomotake; Hoshino, Masakatsu; Kuroboshi, Manabu; Tanaka, Hideo: A Practical One-Pot Transformation of Triphenylphosphine Oxide to Triphenylphosphine by Reduction of in situ Generated Triphenylphosphine Dichloride

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804

Tang, Zhi Yong; Zhang, Yuan; Wang, Tao; Wang, Wei: Rhodium(I)-Catalyzed Synthesis of Aryltriethoxysilanes from Arenediazonium Tosylate Salts with Triethoxysilane

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Supporting Information

809

Cui, Dong-Mei; Zheng, Jin-Zhou; Yang, Liu-Yang; Zhang, Chen: (PPh₃)AuCl/AgOTf-Catalyzed Intermolecular Hydroamination of Alkynes with Sulfonamides To Form N-Sulfonyl Imines

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Supporting Information

812

Barge, Alessandro; Occhiato, Ernesto G.; Prandi, Cristina; Scarpi, Dina; Tabasso, Silvia; Venturello, Paolo: A New, Practical and Efficient Method for Protecting Alcohols as tert-Butyl Ethers

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817

Mukherjee, Sabuj; Sivappa, Rasapalli; Yousufuddin, Muhammed; Lovely, Carl J.: An Approach to the Oxazoline-Containing Fragments of the Oroidin Dimers Nagelamide R and T

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822

Fujitani, Manabu; Tsuchiya, Masami; Okano, Kentaro; Takasu, Kiyosei; Ihara, Masataka; Tokuyama, Hidetoshi: Total Synthesis of (±)-Lepadiformine A via Radical Translocation-Cyclization Reaction

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827

Sakai, Yuki; Ikeuchi, Kazutada; Yamada, Yuji; Wakimoto, Toshiyuki; Kan, Toshiyuki: Modified Julia-Kocienski Reaction Promoted by Means of m-NPT (Nitro­phenyltetrazole) Sulfone

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830

Song, Liping; Li, Xianfu; Xing, Chunhui; Li, Dongmei; Zhu, Shizheng; Deng, Hongmei; Shao, Min: Fluorine-Containing Furan Derivatives from the Michael Addition of Ethyl 4,4,4-Trifluoro-3-oxobutanoate with β-Nitrostyrenes

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Supporting Information

spotlight

835

Yella, Ramesh: Chloroacetylchloride: A Versatile Reagent in Heterocyclic Synthesis

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837

Li, Yanchun: Trimethylsilyl Chloride (TMSCl)

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addenda and errata

839

Chemistry of Lactam-Derived Vinyl Phosphates: Stereoselective Synthesis of (+)-Fagomine

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840

A Practical Synthesis of (S)-Cyclopent-2-enol

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