DOI: 10.1055/s-00000131

Synfacts

Issue 02 · Volume 2006 · February 2006 DOI: 10.1055/s-002-4617

Synthesis of Natural Products and Potential Drugs

0095
Magnus, P.; Matthews, K. S.: Synthesis of (±)-Renieramycin G
0096
Itagaki, N.; Sugahara, T.; Iwabuchi, Y.: Synthesis of (-)-CP55,940
0097
Marti, C.; Carreira, E. M.: Synthesis of (-)-Spirotryprostatin B
0098
O’Malley, S. J.; Tan, K. L.; Watzke, A.; Bergman, R. G.; Ellman, J. A.: Synthesis of (+)-Lithospermic Acid
0099
Donohoe, T. J.; Sintim, H. O.; Sisangia, L.; Ace, K. W.; Guyo, P. M.; Cowley, A.; Harling, J. D.: Synthesis of clastro-Lactacystin β-Lactone
0100
Keum, G.; Hwang, C. H.; Kang, S. B.; Kim, Y.; Lee, E.: Synthesis of (+)-Rollimembrin
0101
Muri, D.; Lohse-Fraefel, N.; Carreira, E. M.: Synthesis of Erythronolide
0102
Jiang, X.; Garcia-Fortanet, J.; De Brabander, J. K.: Synthesis of Psymberin/Irciniastatin A
0103
Hamasaki, A.; Zimpleman, J. M.; Hwang, I.; Boger, D. L.: Synthesis of Ningalin D
0104
Suri, J. T.; Steiner, D. D.; Barbas, C. F.: Synthesis of (S)-1-Amino-5-phosphonoindan-1-carboxylic Acid [(S)-APICA]
0105
Zhou, G.; Corey, E. J.: Synthesis of Aflatoxin B2
0106
Fürstner, A.; Domostoj, M. M.; Scheiper, B.: Synthesis of Dictyodendrin B
0107
Kaden, S.; Brockmann, M.; Reissig, H.-U.: Synthesis of Anisomycin
0108
Ding, K.; Lu, Y.; Nikolovska-Coleska, Z.; Qiu, S.; Ding, Y.; Gao, W.; Stuckey, J.; Krajewski, K.; Roller, P. P.; Tomita, Y.; Parrish, D. A.; Deschamps, J. R.; Wang, S.: Synthesis of Spiro-oxindole MDM2 Inhibitors

Synthesis of Heterocycles

0109
Xu, H.-W.; Li, G.-Y.; Wong, M.-K.; Che, C.-M.: Chiral Pyrrolines via Asymmetric 1,3-Dipolar Cycloaddition Reactions
0110
Tsang, W. C. P.; Zheng, N.; Buchwald, S. L.: Synthesis of Carbazoles by Tandem C-H Activation and Buchwald-Hartwig Amination
0111
Feldman, A. K.; Colasson, B.; Sharpless, K. B.; Fokin, V. V.: A Concept for the Regioselective Synthesis of 1,2,3-Triazoles
0112
Konno, T.; Chae, J.; Miyabe, T.; Ishihara, T.: Regioselective Synthesis of 4-Fluoroalkyl Isoquinolines
0113
Duvelleroy, D.; Perrio, C.; Parisel, O.; Lasne, M.-C.: Indium(III)-Mediated Synthesis of Quinoline-4-carboxylic Acid Derivatives
0114
Ohno, H.; Yamamoto, M.; Iuchi, M.; Tanaka, T.: Aromatizing Route to Benzo-, Benzofuranyl-, and N-Tosylindolenyl-isoindolines
0115
Corey, E. J.; Tian, Y.: Synthesis of Azabiaryls by a non-Cross-Coupling Method
0116
Bressy, C.; Alberico, D.; Lautens, M.: A C-H Insertion Route to Fused Indoles
0117
Waldo, J. P.; Larock, R. C.: Convenient Synthesis of Isoxazoles
0118
Kazmaier, U.; Ackermann, S.: Synthesis of Endothiopeptides via Ugi Reaction and their Conversion to Thiazoles
0119
Zhang, L.: Synthesis of Functionalized 2,3-Indoline-Fused Cyclobutanes
0120
Sainz, Y. F.; Raw, S. A.; Taylor, R. J. K.: Multisubstituted Pyridines from 1,2,4-Triazines by Diels-Alder Chemistry
0121
Berkessel, A.; Cleemann, F.; Mukherjee, S.: Oxazinones as Synthetic Intermediates for Enantiomerically Pure β-Amino Acids
0122
Février, F. C.; Smith, E. D.; Comins, D. L.: Regioselective Lithiation of (S)-Nicotine

Synthesis of Materials and Unnatural Products

0123
Toda, M.; Takagaki, A.; Okamira, M.; Kondo, J. N.; Hayashi, S.; Domen, K.; Hara, M.: Biodiesel Made with a Sulfonated Solid Catalyst

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

0125
Moessner, C.; Bolm, C.: Ir-Catalyzed Asymmetric Ketimine Hydrogenation
0126
Hird, A. W.; Hoveyda, A. H.: All-Carbon Quaternary Stereogenic Centers via Cu-Catalyzed Conjugate Additions
0127
Hamze, A.; Provot, O.; Alami, M.; Brion, J.-D.: Regioselective Hydrosilylation of Unsymmetrical Aryl Alkynes
0128
Zhang, D.; Ready, J. M.: Tandem Carbocupration/Oxygenation of Terminal Alkynes
0129
Ma, M.; Peng, L.; Li, C.; Zhang, X.; Wang, J.: [2,3]-Sigmatropic Rearrangement of Sulfur Ylides
0130
Huang, J.; Bunel, E.; Allgeier, A.; Tedrow, J.; Storz, T.; Preston, J.; Correll, T.; Manley, D.; Soukup, T.; Jensen, R.; Syed, R.; Moniz, G.; Larsen, R.; Martinelli, M.; Reider, P. J.: Asymmetric Hydroformylation of [2.2.1]-Bicyclic Olefins
0131
Ma, L.; Du, D.-M.; Xu, J.: Cu-Catalyzed Enantioselective Aziridination of Chalcones
0132
Huang, Y.; Yang, F.; Zhu, C.: Biginelli Reaction Using a New Chiral Ytterbium Catalyst
0133
Aschwanden, P.; Kvaerno, L.; Geisser, R. W.; Kleinbeck, F.; Carreira, E. M.: Synthesis of β-Amino Ketones and β-Amino Alcohols
0134
Schwier, T.; Gevergyan, V.: Trans- and cis-Selective Lewis Acid-Catalyzed Hydrogermylation of Alkynes
0135
Denmark, S. E.; Baiazitov, R. Y.: Intramolecular [4+2] Cycloaddition of Nitroalkenes
0136
Nemoto, T.; Fukuda, T.; Matsumoto, T.; Hitomi, T.; Hamada, Y.: Synthesis of Chiral, All-Carbon Quaternary Centers via Allylic Alkylation
0137
Leitner, A.; Shekar, S.; Pouy, M. J.; Hartwig, J. F.: Ir(I)/Phosphoramidite-Catalyzed Asymmetric Allylic Amination
0138
Cabrera, S.; Arrayás, R. G.; Carretero, J. C.: 1,3-Dipolar Cycloaddition of Azomethine Ylides
0139
Hein, J. E.; Geary, L. M.; Jaworski, A. A.; Hultin, P. G.: Synthesis of Chiral Fluorous Oxazolidinone Auxiliaries
0140
Pohlhaus, P. D.; Johnson, J. S.: Enantiospecific Synthesis of Tetrahydrofurans via Cyclopropane Cycloaddition
0141
Shintani, R.; Yamagami, T.; Kimura, T.; Hayashi, T.: Rhodium-Catalyzed 1,4-Addition of Arylzinc Reagents
0142
Bräse, S.; Höfener, S.: Enantioselective Conjugate Addition of R2Zn to α,β-Unsaturated Aldehydes and Ketones
0143
Bogliotti, N.; Dalko, P. I.; Cossy, J.: One-Pot Conversion of Alkynyl Ketones into Saturated Chiral Alcohols
0144
Wieland, L. C.; Deng, H.; Snapper, M. L.; Hoveyda, A. H.: Al-Catalyzed Enantioselective Dialkylzinc Addition to α-Ketoesters
0145
Mlynarski, J.; Jankowska, J.; Rakiel, B.: Yb(III)-Catalyzed Asymmetric Aldol-Tishchenko Reaction
0146
Hansen, A. L.; Skrydstrup, T.: Regioselective Heck Couplings of α,β-Unsaturated Tosylates and Mesylates

Metal-Mediated Synthesis

0147
Limmert, M. E.; Roy, A. H.; Hartwig, J. F.: Kumada Coupling of Aryl and Vinyl Tosylates under Mild Conditions
0148
Hernandez, E.; Soderquist, J. A.: Asymmetric Propargylation with Trimethylsilyl-9-borabicyclo[3.3.2]decanes
0149
Shimamoto, T.; Chimori, M.; Sogawa, H.; Yamamoto, K.: Pd-Catalyzed Hydrosilylative Coupling of Alkenes with Alkynes
0150
Yamanoi, Y.: Pd-P(t-Bu)3-Catalyzed Cross-Coupling of Silanes with Aryl Halides
0151
Wadamoto, M.; Yamamoto, H.: Silver-Catalyzed Asymmetric Allylation of Ketones with Allyl Silanes
0152
Ison, E.; Trivedi, E. R.; Corbin, R. A.; Abu-Omar, M. M.: Re-Catalyzed Hydrosilylation of Ketones with Et3SiH
0153
Kanno, K.; Liu, Y.; Iesato, A.; Nakajima, K.; Takahashi, T.: Chromium-Mediated Synthesis of Polycyclic Aromatic Compounds
0154
Woodward, A. R.; Burks, H. E.; Chan, L. M.; Morken, J. P.: Catalytic Asymmetric Allene Diboration/Allylation/Functionalization
0155
Lalic, G.; Blum, S.; Bergman, R. G.: Synthesis of Allylic Amines from Allylic Ethers and Zirconocene Imides
0156
Ito, H.; Kawakami, C.; Sawamura, M.: Cu-Catalyzed Stereoselective Reaction of Allylic Carbonates with Diboronate
0157
Jeon, S.-J.; Li, H.; Walsh, P. J.: Solvent-Free Asymmetric Alkylzinc Additions to Ketones
0158
McMahon, J. P.; Ellman, J. A.: Asymmetric Conjugate Addition to α,β-Unsaturated Chiral Sulfinyl Imines
0159
Namba, K.; Wang, J.; Cui, S.; Kishi, Y.: Surprisingly Efficient Catalytic Cr-Mediated Reactions

Organo- and Biocatalysis

0161
Paetzold, J.; Bäckvall, J. E.: Dynamic Kinetic Resolution of Primary Amines
0162
Tozawa, T.; Yamane, Y.; Mukaiyama, T.: Synthesis of 3,4-Dihydropyran-2-ones Catalyzed by Quaternary Ammonium Phenoxide
0163
Pusztai, Z.; Vlád, G.; Bodor, A.; Horváth, I. T.; Laas, H. J.; Halpaap, R.; Richter, F. U.: Mechanism of Phosphine-Catalyzed Cyclo-Oligomerization of Isocyanates
0164
Rowland, G. B.; Zhang, H.; Rowland, E. B.; Chennamadhavuni, S.; Wang, Y.; Antilla, J. C.: Brønsted Acid-Catalyzed Imine Amidation
0165
Svedendahl, M.; Hult, K.; Berglund, P.: Lipase-Catalyzed Michael Addition
0166
Franzén, J.; Marigo, M.; Fielenbach, D.; Wabnitz, T. C.; Kjærsgaard, A.; Jørgensen, K. A.: A General Organocatalyst for the Asymmetric Direct α-Functionalization of Aldehydes
0167
Klein, G.; Humbert, N.; Gradinaru, J.; Ivanova, A.; Gilardoni, F.; Rusbandi, U. E.; Ward, T. R.: Hydrogenation Using Chemogenetically Optimized Chemzymes
0168
Samanta, S.; Liu, J.; Dodda, R.; Zhao, C. G.: A Highly Efficient Catalyst for the Enantioselective Direct Aldol Reaction
0169
Palomo, C.; Oiarbide, M.; Laso, A.; López, R.: Organocatalytic Asymmetric Aza-Henry Reaction
0170
Janey, J. M.; Hsiao, Y.; Armstrong, J. D.: DPP-IV Inhibitor by Proline-Catalyzed Mannich Reaction
0171
Thalji, R. K.; Roush, W. R.: Highly Regioselective Tandem Morita-Baylis-Hillman/Aldol Cyclization

Polymer-Supported Synthesis

0173
Koç, F.; Michalek, F.; Rumi, L.; Bannwarth, W.; Haag, R.: Sintered Polyethylene Chips-Supported Pd, Rh and Ru Catalysts
0174
Blackburn, C.; Achab, A.; Elder, A.; Ghosh, S.; Guo, J.; Harriman, G.; Jones, M.: Synthesis of 3-Amino-1,2,4-benzothiadiazine 1,1-Dioxides
0175
Prousis, K. C.; Detsi, A. D.; Igglessi-Markopoulou, O.: A Traceless Solid-Phase Approach to Functionalized Tetramic Acids
0176
Akagawa, K.; Sakamoto, S.; Kudo, K.: PS-PEG-Supported Proline Catalysis for Aldol Reaction
0177
Papp, A.; Galbàcs, G.; Molnàr, Á: Recycable Ligand-Free Mesoporous Pd Catalysts for Heck Reaction
0178
Aoyama, T.; Takido, T.; Kodomari, M.: Acidic and Basic Supported Reagents for One-Pot Synthesis of Benzo[b]thiophenes
0179
Nefzi, A.; Santos, R. T.: Solid-Phase Synthesis of New Heterocyclic Azoniaspiro Ring Systems
0180
Li, L.; Shi, J.-l: A Highly Active and Reusable Heterogeneous Ruthenium Catalyst
0181
Nielsen, T. E.; Quement, S. L.; Meldal, M.: Solid-Phase Synthesis of Pyrroloisoquinoline
0182
Sabitha, G.; Reddy, K. B.; Yadav, J. S.; Shailaja, D.; Sivudu, K. S.: Ceria/Vinylpyridine Polymer Nanocomposite-Catalyzed Biginelli Reaction
0183
Morelli, C. F.; Saladino, A.; Speranza, G.; Manitto, P.: Solid-Phase Synthesis of Pyrazoledicarboxylic Acid Derivatives
0184
Rudbeck, H. C.; Johannsen, I.; Nielsen, O.; Ruhland, T.; Sommer, M. B.; Tanner, D.; Dancer, R.: Gram-Scale Synthesis of N-Aryl- and N-Aryl-N¢-methylpiperazines on PEG