Synfacts

Issue 01 · January 2007

Issue
Synthesis of Natural Products and Potential Drugs
0001
Wipf, P.; Pierce, J. G.: Synthesis of the α-C-Glycoside Analogue of KRN7000

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0002
Eckelbarger, J. D.; Wilmot, J. T.; Gin, D. Y.: Synthesis of (-)-Deoxyharringtonine

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0003
He, Y.; Funk, R. L.: Synthesis of (±)-β-Erythroidine FREE ACCESS

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0004
Wardrop, D. J.; Fritz, J.: Synthesis of (±)-Magnofargesin

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0005
Wu, Y.; Sun, Y.-P.: Synthesis of Valilactone

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0006
Tang, B.; Bray, C. D.; Pattenden, G.: Synthesis of (+)-Intricarene

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0007
Liu, Z.; Wasmuth, A. S.; Nelson, S. G.: Synthesis of (-)-Rhazinilam

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0008
Xu, F.; Murry, J. A.; Simmons, B.; Corley, E.; Fitch, K.; Karady, S.; Tschaen, D.: Synthesis of DOV21947

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0009
Hoye, T. R.; Eklov, B. M.; Jeon, J.; Khoroosi, M.: Synthesis of (+)-Gigantecin

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0010
Bandur, N. G.; Brückner, D.; Hoffmann, R. W.; Koert, U.: Synthesis of Jimenezin

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0011
Au, C. W. G.; Pyne, S. G.: Synthesis of (-)-Swainsonine

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0012
Göksel, H.; Stark, C. B. W.: Synthesis of cis-Solamin

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0013
Mejia-Oneto, J. M.; Padwa, A.: Synthesis of (±)-Aspidophytine

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0014
Fürstner, A.; Aïssa, C.; Chevrier, C.; Tepl, F.; Nevado, C.; Tremblay, M.; Waser, M.: Synthesis of Iejimalide B

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0015
Boeckman Jr, R. K.; Shao, P.; Wrobleski, S. T.; Boehmler, D. J.; Heintzelman, G. R.; Barbosa, A. J.: Synthesis of (+)-Tetronolide

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Synthesis of Heterocycles
0017
Fayol, A.; Fang, Y.-Q.; Lautens, M.: Pd-Catalyzed Sequential C-N and C-C Coupling Route to 2-Vinylindoles

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0018
Lebeuf, R.; Robert, F.; Schenk, K.; Landais, Y.: Diastereoselective Hydroamination Route to Hexahydroindoles

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0019
Martín, R.; Rivero, M. R.; Buchwald, S. L.: Pyrroles and Pyrazoles by a C-N Coupling-Hydroamination Sequence FREE ACCESS

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0020
Reddy, R. P.; Davies, H. M. L.: Enantioselective Synthesis of Oxazolidinones

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0021
Correa, A.; Tellitu, I.; Domínguez, E.; SanMartin, R.: Synthesis of Benzothiazol-3-ones

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0022
Lamer, A.-C. Le; Gouault, N.; David, M.; Boustie, J.; Uriac, P.: Fluorous-Phase Synthesis of α-Methyleneγ-lactones

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0023
Ichikawa, J.; Nadano, R.; Ito, N.: 4-Difluoromethylene-1-Pyrrolines by Intramolecular Heck Cyclization

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0024
Alajarín, M.; Ortín, M.-M.; Sánchez-Andrada, P.; Vidal, Á: Pericyclic Ring Closure of Ketenimines to Quinolinones

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0025
Guastavino, J. F.; Barolo, S. M.; Rossi, R. A.: An S_RN1 Route to 3-Substituted and Fused Isoquinolin-1-(2H)-ones

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0026
Seregin, I. V.; Gevorgyan, V.: Gold-Catalyzed Synthesis of Pyrrole-Fused Heterocycles

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0027
Rassukana, Y. V.; Khomenko, E. A.; Onys’ko, P. P.; Sinitsa, A. D.: Synthesis of 1,3-Oxathiolan-5-ones and Benzoxathian-4-ones

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0028
Rios, R.; Sundén, H.; Ibrahem, I.; Zhao, G.-L.; Eriksson, L.; CÓrdova, A.: Chiral Benzothiopyrans by Organocatalysis

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0029
Correa, A.; Tellitu, I.; Domínguez, E.; SanMartin, R.: Metal-Free Synthesis of Indolines

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0030
Mross, G.; Holtz, E.; Langer, P.: 2-Alkenylfurans via Feist-Benary and Wittig Reactions

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0031
Li, Y.; Liang, F.; Bi, X.; Liu, Q.: Substituted Thiophenes via Intramolecular Thia-anti-Michael Addition

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Synthesis of Materials and Unnatural Products
0033
Francesconi, O.; Ienco, A.; Moneti, G.; Nativi, C.; Roelens, S.: β-Glucopyranoside Cage Receptor

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0034
He, L.; An, Y.; Yuan, L.; Feng, W.; Li, M.; Zhang, D.; Yamato, K.; Zheng, C.; Zeng, X. C.; Gong, B.: Tetrasulfonamide Macrocycles

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0035
Fokin, A. A.; Schreiner, P. R.; Fokina, N. A.; Tkachenko, B. A.; Hausmann, H.; Serafin, M.; Dahl, J. E. P.; Liu, S.; Carlson, R. M. K.: Functionalization of Nanodiamond

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0036
Bai, J.; Shea, K.: Synthesis of TMS-Modified Polymethylenes

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0037
Chisholm, M. H.; Gallucci, J. C.; Yin, H.: A Reusable Ring-Enlarging Catalyst

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0038
Licandro, E.; Rigamonti, C.; Ticozzelli, M. T.; Monteforte, M.; Baldoli, C.; Giannini, C.; Maiorana, S.: Preparation of Novel Tetrathia[7]helicenes

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0039
Knoblock, K. M.; Silvestri, C. J.; Collard, D. M.: Stacked Conjugated Oligothiophenes

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0040
Silva, A. M. G.; Lacerda, P. S. S.; Tomé, A. C.; Neves, M. G. P. M. S.; Silva, A. M. S.; Cavaleiro, J. A. S.; Makarova, E. A.; Lukyanets, E. A.: Porphyrin-Chlorin Dyads by 1,3-Dipolar Cycloaddition

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0041
Yamazaki, D.; Nishinaga, T.; Tanino, N.; Komatsu, K.: Bent Radical Cation Dimers from Bicyclooctene-Substituted Terthiophenes

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0042
Benniston, A. C.; Rewinska, D. B.: Fluorophore Formed in Ambient Light by two Ring Closures

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0043
Jousselme, B.; Sonmez, G.; Wudl, F.: New Fullerene Electronic Acceptors and Acids

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0044
Lemieux, V.; Gauthier, S.; Branda, N. R.: Molecular Switches for Photorelease

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0045
Dong, Z.; Karpowicz Jr, R. J.; Bai, S.; Yap, G. P. A.; Fox, J. M.: Control of Helicity in a Metal Complex

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0046
Ie, Y.; Umemoto, Y.; Kaneda, T.; Aso, Y.: Synthesis of a Hexafluorocyclopentene-Annelated Thiophene Monomer

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Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions
0047
Ohmura, T.; Taniguchi, H.; Suginome, M.: Asymmetric Silylboronation of Allenes

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0048
Toullec, P. Y.; Genin, E.; Leseurre, L.; Genêt, J.-P.; Michelet, V.: Au(I)-Catalyzed Diastereoselective Tandem Addition/Carbocyclization

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0049
Hu, A.; Ogasawara, M.; Sakamoto, T.; Okada, A.; Nakajima, K.; Takahashi, T.; Lin, W.: Intermolecular Asymmetric Hydroamination

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0050
Cozzi, P. G.: Catalytic Enantioselective Imino-Reformatsky Reaction

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0051
Sibi, M. P.; Zimmerman, J.: Enantioselective Radical Additions to Acyloxy Pyrones

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0052
Tosaki, S.-y; Hara, K.; Gnanadesikan, V.; Morimoto, H.; Harada, S.; Sugita, M.; Yamagiwa, N.; Matsunaga, S.; Shibasaki, M.: Enantioselective Resolution of Ketone Nitroaldol Products

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0053
Tsuchiya, Y.; Hamashima, Y.; Sodeoka, M.: Palladium-Catalyzed Enantioselective Conjugate Reduction of Enones

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0054
Bolm, C.; Whelligan, D. K.: New Ligands: Hydroxyoxazolinyl[2.2]paracyclophanes in Asymmetric Catalysis

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0055
Maheswaran, H.; Prasanth, K. L.; Krishna, G. G.; Ravikumar, K.; Sridhar, B.; Kantam, M. L.: Enantioselective Copper-Catalyzed Nitroaldol Reaction

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0056
Gnanadesikan, V.; Corey, E. J.: Enantioselective Synthesis of β-Lactone Catalyzed by a Chiral Oxazaborolidine

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0057
Morita, N.; Krause, N.: Au(I)-Catalyzed Formal Hydroamination of Chiral Allenes to 3-Pyrrolines

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0058
Bew, S. P.; Hughes, D. L.; Palmer, N. J.; Savic, V.; Soapi, K. M.; Wilson, M. A.: Stereoselective Synthesis of N-Alkylaziridines from N-Chloroamines

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0059
Li, P.; Forbeck, E. M.; Evans, C. D.; Joullié, M. M.: Cu(I)-Catalyzed Stereoselective Formation of Tertiary Alkyl-Aryl Ethers

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0060
Belokon, Y. N.; Maleev, V. I.; North, M.; Usanov, D. L.: Role of the X Anion in the VO(salen) (X)-Mediated Cyanohydrin Synthesis

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0061
Muthusamy, S.; Krishnamurthi, J.; Suresh, E.: Chemodivergent Formation of Furanones and Piperidines

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0062
Šebesta, R.; Almassy, A.; Císařová, I.; Toma: Ferrocenophane Diphosphine Ligands for Pd-Catalyzed Allylic Substitution

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0063
Whitehead, A.; McParland, J. P.; Hanson, P. R.: Regioselective Cuprate Additions to Tethered Allylic Phosphates

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0064
Aikawa, K.; Akutagawa, S.; Mikami, K.: Rhodium-Catalyzed Intramolecular [4+2] Cycloaddition

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0065
Restorp, P.; Fischer, A.; Somfai, P.: [3+2] Annulation of N-Ts-α-Amino Aldehydes and 1,3-Bis(silyl)propenes

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0066
Trost, B. M.; Stambuli, J. P.; Silverman, S. M.; Schwörer, U.: Asymmetric Palladium-Catalyzed [3+2] Cycloaddition

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0067
Hajra, A.; Yoshikai, N.; Nakamura, E.: N,O,P-Ligand for Cu(II)-Catalyzed Enantioselective Conjugate Additions

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0068
Ohmura, T.; Furukawa, H.; Suginome, M.: Complementary Stereoselectivity in Pt-Catalyzed Silaboration of Alkenes

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0069
Shibata, T.; Tahara, Y.-k: Chiral Quaternary Carbon Stereocenters via Diene-yne [2+2+2] Cycloaddition FREE ACCESS

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0070
Hoyos, P.; Fernández, M.; Sinisterra, J. V.; Alcántara, A. R.: Dynamic Kinetic Resolution of Benzoins by Lipase-Ru Catalysis

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0071
Kwiatkowski, P.; Majer, J.; Chaadaj, W.; Jurczak, J.: 2,5-Disubstituted Furans via Diastereoselective Friedel-Crafts Reaction

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0072
Abraham, C. J.; Paull, D. H.; Scerba, M. T.; Grebinski, J. W.; Lectka, T.: Bifunctional Inverse Electron Demand Hetero-Diels-Alder Reactions

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0073
Bazán-Tejeda, B.; Bluet, G.; Broustal, G.; Campagne, J.-M.: Cu-Catalyzed Asymmetric Synthesis of α,β-Unsaturated δ-Lactones

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0074
Sibi, M. P.; Manyem, S.; Palencia, H.: Achiral Additives for Enhancing the Stereoselectivity of Cycloadditions

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0075
Hargrave, J. D.; Bish, G.; Frost, C. G.: Rh-Catalyzed Asymmetric Synthesis of 2-Substituted Pyrrolizidinones

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Metal-Mediated Synthesis
0077
Durandetti, M.; Périchon, J.: Iron-Catalyzed Allylation of Ketones

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0078
Mata, Y.; Diéguez, M.; Pàmies, O.; Woodward, S.: Asymmetric Ni Phosphite Catalyzed Trialkylaluminum Addition to Aldehydes

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0079
Krasovskiy, A.; Malakhov, V.; Gavryushin, A.; Knochel, P.: Direct LiCl-Promoted Insertion of Zinc into Organic Iodides and Bromides FREE ACCESS

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0080
Saito, T.; Nishimoto, Y.; Yasuda, M.; Baba, A.: Direct Lewis Acid Promoted C-Allylation of Alcohols with Allylsilanes

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0081
Murphy, J. M.; Lawrence, J. D.; Kawamura, K.; Incarvito, C.; Hartwig, J. F.: Ru-Catalyzed Regiospecific Borylation of Methyl C-H Bonds

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0082
Berkessel, A.; Sebastian-Ibarz, M. L.; Müller, T.: Lipase/Aluminum-Catalyzed Dynamic Kinetic Resolution of Alcohols

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0083
Nimmagadda, R. D.; McRae, C.: Reduction of Oxygen Functionalities to Alkanes with Alkylsilanes

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0084
Zhao, B.; Lu, X.: Pd(II)-Catalyzed Addition of Boronic Acids to Nitriles

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0085
Herath, A.; Montgomery, J.: Ni-Catalyzed Intramolecular Enal-Alkyne [3+2] Reductive Cycloaddition

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0086
Tsubouchi, A.; Onishi, K.; Takeda, T.: Stereoselective Preparation of Silyloxy-Alkenylcopper Species from Acylsilanes

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0087
Novak, A.; Humphreys, L. D.; Walker, M. D.; Woodward, S.: AlMe₃-DABCO-Promoted Synthesis of Amides

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0088
Sato, T.; Watanabe, S.; Kiuchi, H.; Oi, S.; Inoue, Y.: Rh-Catalyzed Hydrogenation of Olefins with Zn Metal and Water

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0089
Mun, S.; Lee, J.-E.; Yun, J.: Cu-Catalyzed β-Boration of Michael Acceptors with Bis(pinacolato)diboron

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Organo- and Biocatalysis
0091
Arp, F. O.; Fu, G. C.: Nonenzymatic Kinetic Resolution of Indolines

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0092
Wolfer, J.; Bekele, T.; Abraham, C. J.; Dogo-Isonagie, C.; Lectka, T.: Highly Enantioselective Synthesis of 1,4-Benzoxazinones and α-Amino Acids

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0093
Chen, X.-H.; Xu, X.-Y.; Liu, H.; Cun, L.-F.; Gong, L.-Z.: First Organocatalytic Asymmetric Biginelli Reaction FREE ACCESS

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0094
Li, H.; Wang, J.; E-Nunu, T.; Zu, L.; Jiang, W.; Wei, S.; Wang, W.: Chiral Chromenes via Domino Oxa-Michael-Aldol Reaction

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0095
Kirschner, A.; Bornscheuer, U. T.: Enzymatic Kinetic Resolution of β-Hydroxy Ketones

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0096
Brandau, S.; Maerten, E.; Jørgensen, K. A.: Highly Enantioselective Organocatalytic Michael-Aldol Domino Reactions

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0097
Rueping, M.; Azap, C.: Asymmetric Synthesis of Isoquinuclidines

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0098
Cho, D. H.; Jang, D. O.: Enantioselective Radical Addition of Alkyl Halides to Glyoxylate Oxime Ether

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0099
Fini, F.; Bernardi, L.; Herrera, R. P.; Pettersen, D.; Ricci, A.; Sgarzani, V.: Phase-Transfer-Catalysis of Direct Mannich Reaction of Malonates with N-Carbamoylimines

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0100
He, M.; Uc, G. J.; Bode, J. W.: Chiral N-Heterocyclic Carbene Catalyzed Oxodiene Diels-Alder Reactions

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0101
Shen, Y.-M.; Zhao, M.-X.; Xu, J.; Shi, Y.: Aziridination of Chalcones Using Tertiary Amine Catalysts

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Polymer-Supported Synthesis
0103
Arai, T.; Watanabe, M.; Fujiwara, A.; Yokoyama, N.; Yanagisawa, A.: CD-Monitored HTS of Chiral Catalysts FREE ACCESS

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0104
Testero, S. A.; Mata, E. G.: Solid-Phase Synthesis of β-Lactam Analogues

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0105
Uozumi, Y.; Suzuka, T.; Kawade, R.; Takenaka, H.: Allylic Azidation in Water

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0106
Abid, M.; Spaeth, A.; Török, B.: An Efficient Synthesis of Five-Membered N-Heterocycles

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0107
Yuan, X.-Y.; Li, H.-Y.; Hodge, P.; Kilner, M.; Tastard, C. Y.; Zhang, Z.-P.: A Facile One-Pot Synthesis of Polymer-Supported 1,1′-Bi(2-naphthol)s

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0108
Chai, L.; Chen, H.; Li, Z.; Wang, Q.; Tao, F.: Enantioselective Hydrogenation Using a PEG-Supported Biphep-Ru Complex

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0109
Wu, Y.; Zhang, Y.; Yu, M.; Zhao, G.; Wang, S.: Asymmetric Aldol Reaction in Water Using Dendrimer-Supported Proline

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0110
Sommer, W. J.; Weck, M.: Poly(norbornene)-Supported N-Heterocyclic Carbenes

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0111
Uozumi, Y.; Suzuka, T.: Safety Asymmetric π-Allylic C1-Substitution with Nitromethane in Water

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0112
Wang, J.; Yan, L.; Qian, G.; Yang, K.; Liu, H.; Wang, X.: Heteropolyacid-Functionalized Silica Catalyst for the Acylal Formation

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0113
Ribière, P.; Declerck, V.; Nédellec, Y.; Yadav-Bhatnagar, N.; Martinez, J.; Lamaty, F.: Synthesis of Poly(ethylene glycol) Supported Benzazepines

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0114
Motokura, K.; Fujita, N.; Mori, K.; Mizugaki, T.; Ebitani, K.; Jitsukawa, K.; Kaneda, K.: α-Alkylation of Nitriles Promoted by Hydrotalcite-Supported Catalysts

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0115
Schuster, C.; Knollmüller, M.; Gärtner, P.: Polymer-Supported m-Hydrobenzoin-Derived Chiral Auxiliary

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