DOI: 10.1055/s-00000084

Synthesis

Ausgabe 10 · Volume 2007 · Mai 2007 DOI: 10.1055/s-002-6704

review

1439
Domínguez de María, Pablo; García-Burgos, Carlos A.; Bargeman, Gerrald; van Gemert, Robert W.: Pig Liver Esterase (PLE) as Biocatalyst in Organic Synthesis: From Nature to Cloning and to Practical Applications
https://www.thieme-connect.de/bilder/synthesis/200710/e177_ga

short paper

1453
Kurz, Thomas; Thimann, Wolfgang; Geffken, Detlef: Synthesis of 3-Alkoxy-5,6-dihydro-4H-1,2,5-oxadiazines from Alkyl α-Aminohydroximates
https://www.thieme-connect.de/bilder/synthesis/200710/t010_ga
1456
Kuik, Árpád; Skoda-Földes, Rita; Jánosi, László; Kollár, László: Facile Synthesis of Unsymmetrical 1,n′-Disubstituted Ferrocenoyl Amino Acid Derivatives by Palladium-Catalyzed Aminocarbonylation
https://www.thieme-connect.de/bilder/synthesis/200710/t024_ga

paper

1459
Jiang, Yan; Zhou, Guo-Chuan; He, Guang-Li; He, Ling; Li, Ju-Lian; Zheng, Shi-Long: Ruthenium(II)-Porphyrin Catalyzed Selective N-Imidation of Aromatic Nitrogen Heterocycles
https://www.thieme-connect.de/bilder/synthesis/200710/f015_ga
1465
Guan, Zheng-Hui; Zuo, Wei; Zhao, Lian-Biao; Ren, Zhi-Hui; Liang, Yong-Min: An Economical and Convenient Synthesis of Vinyl Sulfones
https://www.thieme-connect.de/bilder/synthesis/200710/f030_ga
1471
Nery, Marcelo S.; Azevedo, Mariangela S.; Cardoso, Jari N.; Slana, Glaucia B. C.; Lopes, Rosangela S. C.; Lopes, Cláudio C.: A New Chemoselective Synthesis of Brombuterol
https://www.thieme-connect.de/bilder/synthesis/200710/m072_ga
1475
Paliakov, Ekaterina; Elleboe, Thomas; Boykin, David W.: New Synthons for the Preparation of Arylimidazolines and Tetrahydro­pyrimidine Analogues
https://www.thieme-connect.de/bilder/synthesis/200710/m074_ga
1481
Thomas, James B.; Brieaddy, Lawrence E.; Boldt, Karl G.; Perretta, Carin; Carroll, F. Ivy: Synthesis and Resolution of the Benzomorphan-Based Kappa Opioid Agonist Bremazocine
https://www.thieme-connect.de/bilder/synthesis/200710/m077_ga
1485
Kumara Swamy, K. C.; Pavan Kumar, K. V. P.; Rama Suresh, R.; Satish Kumar, N.: Easy and Stereoselective Synthesis of Cyclopropyl-Substituted Phosphonates via α-Chlorophosphonates
https://www.thieme-connect.de/media/synthesis/200710/p006_ga.gif
1491
Tyrrell, Elizabeth; Hunie Tesfa, Kibur; Mann, Alastair; Singh, Kuldip: Enantioselective Alkynylation Reactions to Substituted Benzaldehyde and Salicylaldehyde Derivatives: The Effect of Substituents upon the Efficiency and Enantioselectivity
https://www.thieme-connect.de/bilder/synthesis/200710/p146_ga
1499
Schobert, Rainer; Wicklein, André: Short Syntheses of (-)-(R)-Pyrrolam A and (1S)-1-Hydroxyindolizidin-3-one
https://www.thieme-connect.de/bilder/synthesis/200710/t013_ga
1503
Kulik, Svetlana N.; Kobko, Alexander S.; Tolmachev, Andrey A.; Tverdokhlebov, Anton V.; Shishkin, Oleg V.; Chernega, Alexander N.: A New Approach to Pyrazino[2,1-b]quinazolines and Pyrazino[1,2-a]thi­eno[3,2-d]pyrimidines
https://www.thieme-connect.de/bilder/synthesis/200710/z035_ga
1509
Chandrasekhar, Srivari; Basu, Debjit; Raji Reddy, Ch.: Palladium-Catalyzed Reduction of N-(tert-Butoxycarbonyl)indoles by Polymethylhydrosiloxane
https://www.thieme-connect.de/bilder/synthesis/200710/z042_ga
1513
Alizadeh, Abdolhamid; Nematollahi, Davood; Hbibi, Davood; Hesari, Mahdi: Domino Oxidation-Michael Reactions of Catechols with Barbituric Acid Derivatives in Water: An Efficient Synthesis of Polycyclic Pyrimidinones
https://www.thieme-connect.de/bilder/synthesis/200710/z044_ga
1517
Woschek, Anna; Mahout, Marek; Mereiter, Kurt; Hammerschmidt, Friedrich: Synthesis of 2-Heptyl-1-hydroxy-4(1H)-quinolone - Unexpected Rearrangement of 4-(Alkoxycarbonyloxy)quinoline N-Oxides to 1-(Alkoxycarbonyloxy)-4(1H)-quinolones
https://www.thieme-connect.de/bilder/synthesis/200710/t183_ga
1523
Blair, Michael; Andrews, Philip C.; Fraser, Benjamin H.; Forsyth, Craig M.; Junk, Peter C.; Massi, Massimiliano; Tuck, Kellie L.: Facile Methods for the Separation of the cis- and trans-Diastereomers of Limonene­ 1,2-Oxide and Convenient Routes to Diequatorial and Diaxial 1,2-Diols
https://www.thieme-connect.de/bilder/synthesis/200710/p004_ga
1528
Fukuhara, Tsuyoshi; Hasegawa, Chihiro; Hara, Shoji: A Facile Synthesis of Oxazolines, Thiazolines, and Imidazolines Using α,α-Difluoroalkylamines
https://www.thieme-connect.de/bilder/synthesis/200710/f014_ga
1535
Tang, Shi; Li, Jin-Heng; Xie, Ye-Xiang; Wang, Nai-Xing: Halogenation of Indoles with Copper(II) Halides: Selective Synthesis of 2-Halo-, 3-Halo-, and 2,3-Dibromoindoles
https://www.thieme-connect.de/bilder/synthesis/200710/f023_ga
1542
Yoshida, Masanori; Osafune, Kanako; Hara, Shoji: Facile Synthesis of Iodonium Salts by Reaction of Organotrifluoroborates with p-Iodotoluene Difluoride
https://www.thieme-connect.de/bilder/synthesis/200710/f031_ga
1547
Sulima, Agnieszka; Folk, John; Jacobson, Arthur E.; Rice, Kenner C.: A New Approach to the Synthesis of the Nonpeptide NOP Receptor Antagonist J-113397
https://www.thieme-connect.de/bilder/synthesis/200710/m004_ga
1554
Rybáčková, Markéta; Bělohradský, Martin; Holý, Petr; Pohl, Radek; Dekoj, Václav; Závada, Jiří: Synthesis of Highly Symmetrical Triptycene Tetra- and Hexacarboxylates
https://www.thieme-connect.de/bilder/synthesis/200710/t019_ga
1559
Soley, Roger; Albericio, Fernando; Álvarez, Mercedes: Novel Synthesis of Arylethynyl Heterocycles
https://www.thieme-connect.de/bilder/synthesis/200710/t028_ga
1566
Prado, Soizic; Toum, Valérie; Saint-Joanis, Brigitte; Michel, Sylvie; Koch, Michel; Cole, Stewart T.; Tillequin, François; Janin, Yves L.: Antimycobacterial Benzofuro[3,2-f]chromenes from a 5-Bromochromen-6-ol
https://www.thieme-connect.de/bilder/synthesis/200710/t177_ga
1571
Hesse, Stéphanie; Kirsch, Gilbert: Buchwald-Hartwig Amination of β-Chloroacroleins by Lactams and Heteroarylamines
https://www.thieme-connect.de/bilder/synthesis/200710/z052_ga

feature article

1576
Restorp, Per; Dressel, Martina; Somfai, Peter: Synthesis of Functionalized Pyrrolidines by a Highly Stereoselective [3+2]-Annulation Reaction of N-Tosyl-α-Amino Aldehydes and 1,3-Bis(silyl)propenes
https://www.thieme-connect.de/bilder/synthesis/200710/t016_ga

practical synthetic procedures

1584
Ward, Dale E.; Rasheed, M. Abdul; Gillis, H. Martin; Beye, Garrison E.; Jheengut, Vishal; Achonduh, George T.: Simple and Efficient Preparation of Reagents for Thiopyran Introduction:
Methyl Tetrahydro-4-oxo-2H-thiopyran-3-carboxylate, Tetrahydro-4H-thiopyran-4-one, and 3,6-Dihydro-4-trimethylsilyloxy-2H-thiopyran
https://www.thieme-connect.de/bilder/synthesis/200710/m061_ga
1587
Bandini, Marco; Eichholzer, Astrid; Tommasi, Simona; Umani-Ronchi, Achille: Practical Aspects in the Gram-Scale Synthesis of Chiral Diamino-Bithiophene ‘DAT2’ Ligand
https://www.thieme-connect.de/bilder/synthesis/200710/z024_ga

addenda and errata

e1
Ward, Dale E.; Rasheed, M. Abdul; Gillis, H. Martin; Beye, Garrison E.; Jheengut, Vishal; Achonduh, George T.: Simple and Efficient Preparation of Reagents for Thiopyran Introduction: Methyl Tetrahydro-4-oxo-2H-thiopyran-3-carboxylate, Tetrahydro-4H-thiopyran-4-one, and 3,6-Dihydro-4-trimethylsilyloxy-2H-thiopyran