Synlett

Ausgabe 05 · Volume 2010 · März 2010 DOI: 10.1055/s-002-20856

• Accepted Manuscripts
• eFirst
• Ausgabe
• Meistgelesen

account

675

Shapiro, Nathan D.; Toste, F. Dean: A Reactivity-Driven Approach to the Discovery and Development of Gold-Catalyzed Organic Reactions

• Volltext
• HTML
• PDF (429 kb)

692

Wang, Shaozhong; Zhang, Guozhu; Zhang, Liming: Gold-Catalyzed Reaction of Propargylic Carboxylates via an Initial 3,3-Rearrangement

• Volltext
• HTML
• PDF (547 kb)

letter

707

Wei, Shengwei; Stingl, Kerstin A.; Weiß, Katharina M.; Tsogoeva, Svetlana B.: Thieme Chemistry Journal Awardees - Where Are They Now? Bifunctional Organocatalysis with N-Formyl-l-Proline: A Novel Approach to Epoxide Ring Opening and Sulfide Oxidation

• Volltext
• HTML
• PDF (126 kb)

712

Yadav, Ashok K.; Kumar, Manoj; Yadav, Tripti; Jain, Renuka: (1R,5R)-1-(1′-Dimethylaminoethyl)-2-isopropylidene-5-methylcyclohexanol as a Chiral Ligand in the Enantioselective Addition of Diethylzinc to Aldehydes

• Volltext
• HTML
• PDF (80 kb)

715

Sureshbabu, Vommina V.; Chennakrishnareddy, Gundala; Hemantha, Hosahalli P.: Synthesis of Thioureido-Linked Peptidomimetics, Glycosylated Amino Acids, and Neoglycoconjugates Using Bis(benzotriazolyl)methanethione as Thioacylating Agent

• Volltext
• HTML
• PDF (135 kb)

721

Sreeramamurthy, Kintali; Ashok, Ettam; Mahendar, Velisoju; Santoshkumar, Gourishetti; Das, Parthasarathi: Direct Synthesis of N-Aryl Derivatives of Quinazolin-4(3H)-ones Employing Arylboronic Acids in the Presence of Cu(OAc)₂

• Volltext
• HTML
• PDF (114 kb)

725

Schleiss, Julie; Cerniauskaite, Deimante; Gueyrard, David; Iori, Renato; Rollin, Patrick; Tatibouët, Arnaud: Thioimidate N-Oxides: From Nature to Synthetic Pathways

• Volltext
• HTML
• PDF (102 kb)

729

Frigerio, Fabio; Haseler, Claire A.; Gallagher, Timothy: Synthesis of (+)-Kuraramine

• Volltext
• HTML
• PDF (68 kb)

Supporting Information

731

Ali, Asad; Khera, Rasheed Ahmad; Ibad, Muhammad Farooq; Hussain, Munawar; Langer, Peter: Synthesis of Bis(diaryl)sulfones by Site-Selective Suzuki-Miyaura Reactions of 2,4′-Bis(trifluoromethylsulfonyloxy)diphenylsulfone

• Volltext
• HTML
• PDF (91 kb)

735

Majumdar, K. C.; Taher, Abu; Ponra, Sudipta: Unusual Product from Condensative Cyclization: Pyrano[3,2-f]quinolin-3,10-diones from 6-Amino-5-[(trimethylsilyl)ethynyl]-2H-chromen-2-one and Aryl Aldehydes

• Volltext
• HTML
• PDF (126 kb)

Supporting Information

741

Hajipour, Abdol R.; Ghayeb, Yosof; Sheikhan, Nafisehsadat; Ruoho, Arnold E.: Brønsted Acidic Ionic Liquid as an Efficient and Reusable Catalyst for Synthesis of 14-Aryl- or 14-Alkyl-14H-dibenzo[a,j]xanthenes under Solvent-Free Conditions

• Volltext
• HTML
• PDF (75 kb)

745

Borkin, Dmitry; Carlson, Alena; Török, Béla: K-10-Catalyzed Highly Diastereoselective Synthesis of Aziridines

• Volltext
• HTML
• PDF (224 kb)

749

Baumann, Marcus; Baxendale, Ian R.; Ley, Steven V.: Synthesis of 3-Nitropyrrolidines via Dipolar Cycloaddition Reactions Using a Modular Flow Reactor

• Volltext
• HTML
• PDF (142 kb)

753

Vitoriano, Bruno C.; Carvalho, Luísa C. R.; Estevão, Mónica S.; Sekera, Michael H.; Marques, M. Manuel B.: A Simple Route Toward New Clomiphene Metabolites

• Volltext
• HTML
• PDF (90 kb)

Supporting Information

757

Ramesh, Subburethinam; Gaddam, Vikram; Nagarajan, Rajagopal: A Flexible Approach to the Chromenoquinolines under Copper/Lewis Acid Catalysis

• Volltext
• HTML
• PDF (140 kb)

Supporting Information

761

Hanessian, Stephen; Mi, Xueling: An Organocatalytic Approach to Enantiopure 2,6-Disubstituted Tetrahydropyranols

• Volltext
• HTML
• PDF (92 kb)

765

Niu, Liang-Feng; Xin, Yang-Chun; Wang, Ren-Lin; Jiang, Fan; Xu, Peng-Fei; Hui, Xin-Ping: Asymmetric Aza-Friedel-Crafts Reaction of 2-Naphthol with Tosylimines Catalyzed by a Dinuclear Zinc Complex

• Volltext
• HTML
• PDF (306 kb)

Supporting Information

769

Phillips, David J.; Graham, Andrew E.: Guanidine Bases in Synthesis: Extending the Scope of the Corey-Chaykovsky Epoxidation

• Volltext
• HTML
• PDF (112 kb)

774

Friedmann, Christian; Bräse, Stefan: Synthesis of Paracyclophane Thiols via an Unprecedented Reduction-Deprotection Sequence: Direct Conversion of tert-Butyl Sulfoxides into Thiols with Boron Tribromide

• Volltext
• HTML
• PDF (192 kb)

777

Praveen, C.; Kalyanasundaram, A.; Perumal, P. T.: Gold(III)-Catalyzed Synthesis of Isoxazoles by Cycloisomerization of α,β-Acetylenic Oximes

• Volltext
• HTML
• PDF (103 kb)

782

Körber, Nadine; Rominger, Frank; Müller, Thomas J. J.: Enantioselective One-Pot Rhodium-Catalyzed Cycloisomerization-Wittig Sequence to Chiral Functionalized 4-Alkyl 3-Alkylidene Tetrahydrofuran(on)es

• Volltext
• HTML
• PDF (123 kb)

787

Weisbrod, Samuel H.; Marx, Andreas: Synthesis of Water-Soluble Phosphinophenol for Traceless Staudinger Ligation

• Volltext
• HTML
• PDF (78 kb)

790

Silveira, Claudio C.; Mendes, Samuel R.; Líbero, Francieli M.: Solvent-Free Anti-Markovnikov Addition of Thiols to Alkenes Using Anhydrous Cerium(III) Chloride as Catalyst

• Volltext
• HTML
• PDF (80 kb)

793

Wilding, Emily E.; Gregg, John J.; Mullins, Richard J.: Asymmetric Conjugate Addition of Crotylstannane: Synthesis of (-)-Lasiol

• Volltext
• HTML
• PDF (83 kb)

796

Johnson, Sarah; Drowns, Matt; Tatlock, John; Linton, Angelica; Gonzalez, Javier; Hoffman, Robert; Jewell, Tanya; Patel, Leena; Blazel, Julie; Tang, Mingnam; Li, Hui: Synthetic Route Optimization of PF-00868554, An HCV Polymerase Inhibitor in Clinical Evaluation

• Volltext
• HTML
• PDF (97 kb)

801

Yano, Tomotake; Hoshino, Masakatsu; Kuroboshi, Manabu; Tanaka, Hideo: A Practical One-Pot Transformation of Triphenylphosphine Oxide to Triphenylphosphine by Reduction of in situ Generated Triphenylphosphine Dichloride

• Volltext
• HTML
• PDF (177 kb)

804

Tang, Zhi Yong; Zhang, Yuan; Wang, Tao; Wang, Wei: Rhodium(I)-Catalyzed Synthesis of Aryltriethoxysilanes from Arenediazonium Tosylate Salts with Triethoxysilane

• Volltext
• HTML
• PDF (239 kb)

Supporting Information

809

Cui, Dong-Mei; Zheng, Jin-Zhou; Yang, Liu-Yang; Zhang, Chen: (PPh₃)AuCl/AgOTf-Catalyzed Intermolecular Hydroamination of Alkynes with Sulfonamides To Form N-Sulfonyl Imines

• Volltext
• HTML
• PDF (71 kb)

Supporting Information

812

Barge, Alessandro; Occhiato, Ernesto G.; Prandi, Cristina; Scarpi, Dina; Tabasso, Silvia; Venturello, Paolo: A New, Practical and Efficient Method for Protecting Alcohols as tert-Butyl Ethers

• Volltext
• HTML
• PDF (92 kb)

817

Mukherjee, Sabuj; Sivappa, Rasapalli; Yousufuddin, Muhammed; Lovely, Carl J.: An Approach to the Oxazoline-Containing Fragments of the Oroidin Dimers Nagelamide R and T

• Volltext
• HTML
• PDF (168 kb)

822

Fujitani, Manabu; Tsuchiya, Masami; Okano, Kentaro; Takasu, Kiyosei; Ihara, Masataka; Tokuyama, Hidetoshi: Total Synthesis of (±)-Lepadiformine A via Radical Translocation-Cyclization Reaction

• Volltext
• HTML
• PDF (166 kb)

827

Sakai, Yuki; Ikeuchi, Kazutada; Yamada, Yuji; Wakimoto, Toshiyuki; Kan, Toshiyuki: Modified Julia-Kocienski Reaction Promoted by Means of m-NPT (Nitro­phenyltetrazole) Sulfone

• Volltext
• HTML
• PDF (82 kb)

830

Song, Liping; Li, Xianfu; Xing, Chunhui; Li, Dongmei; Zhu, Shizheng; Deng, Hongmei; Shao, Min: Fluorine-Containing Furan Derivatives from the Michael Addition of Ethyl 4,4,4-Trifluoro-3-oxobutanoate with β-Nitrostyrenes

• Volltext
• HTML
• PDF (130 kb)

Supporting Information

spotlight

835

Yella, Ramesh: Chloroacetylchloride: A Versatile Reagent in Heterocyclic Synthesis

• Volltext
• HTML
• PDF (77 kb)

837

Li, Yanchun: Trimethylsilyl Chloride (TMSCl)

• Volltext
• HTML
• PDF (71 kb)

addenda and errata

839

Chemistry of Lactam-Derived Vinyl Phosphates: Stereoselective Synthesis of (+)-Fagomine

• Volltext
• HTML
• PDF (29 kb)

840

A Practical Synthesis of (S)-Cyclopent-2-enol

• Volltext
• HTML
• PDF (27 kb)