Synthesis

Issue 10 · May 2007

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review
1439
Domínguez de María, Pablo; García-Burgos, Carlos A.; Bargeman, Gerrald; van Gemert, Robert W.: Pig Liver Esterase (PLE) as Biocatalyst in Organic Synthesis: From Nature to Cloning and to Practical Applications

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short paper
1453
Kurz, Thomas; Thimann, Wolfgang; Geffken, Detlef: Synthesis of 3-Alkoxy-5,6-dihydro-4H-1,2,5-oxadiazines from Alkyl α-Aminohydroximates

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1456
Kuik, Árpád; Skoda-Földes, Rita; Jánosi, László; Kollár, László: Facile Synthesis of Unsymmetrical 1,n′-Disubstituted Ferrocenoyl Amino Acid Derivatives by Palladium-Catalyzed Aminocarbonylation

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paper
1459
Jiang, Yan; Zhou, Guo-Chuan; He, Guang-Li; He, Ling; Li, Ju-Lian; Zheng, Shi-Long: Ruthenium(II)-Porphyrin Catalyzed Selective N-Imidation of Aromatic Nitrogen Heterocycles

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1465
Guan, Zheng-Hui; Zuo, Wei; Zhao, Lian-Biao; Ren, Zhi-Hui; Liang, Yong-Min: An Economical and Convenient Synthesis of Vinyl Sulfones

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1471
Nery, Marcelo S.; Azevedo, Mariangela S.; Cardoso, Jari N.; Slana, Glaucia B. C.; Lopes, Rosangela S. C.; Lopes, Cláudio C.: A New Chemoselective Synthesis of Brombuterol

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1475
Paliakov, Ekaterina; Elleboe, Thomas; Boykin, David W.: New Synthons for the Preparation of Arylimidazolines and Tetrahydropyrimidine Analogues

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1481
Thomas, James B.; Brieaddy, Lawrence E.; Boldt, Karl G.; Perretta, Carin; Carroll, F. Ivy: Synthesis and Resolution of the Benzomorphan-Based Kappa Opioid Agonist Bremazocine

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1485
Kumara Swamy, K. C.; Pavan Kumar, K. V. P.; Rama Suresh, R.; Satish Kumar, N.: Easy and Stereoselective Synthesis of Cyclopropyl-Substituted Phosphonates via α-Chlorophosphonates

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1491
Tyrrell, Elizabeth; Hunie Tesfa, Kibur; Mann, Alastair; Singh, Kuldip: Enantioselective Alkynylation Reactions to Substituted Benzaldehyde and Salicylaldehyde Derivatives: The Effect of Substituents upon the Efficiency and Enantioselectivity

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1499
Schobert, Rainer; Wicklein, André: Short Syntheses of (-)-(R)-Pyrrolam A and (1S)-1-Hydroxyindolizidin-3-one

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1503
Kulik, Svetlana N.; Kobko, Alexander S.; Tolmachev, Andrey A.; Tverdokhlebov, Anton V.; Shishkin, Oleg V.; Chernega, Alexander N.: A New Approach to Pyrazino[2,1-b]quinazolines and Pyrazino[1,2-a]thieno[3,2-d]pyrimidines

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1509
Chandrasekhar, Srivari; Basu, Debjit; Raji Reddy, Ch.: Palladium-Catalyzed Reduction of N-(tert-Butoxycarbonyl)indoles by Polymethylhydrosiloxane

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1513
Alizadeh, Abdolhamid; Nematollahi, Davood; Hbibi, Davood; Hesari, Mahdi: Domino Oxidation-Michael Reactions of Catechols with Barbituric Acid Derivatives in Water: An Efficient Synthesis of Polycyclic Pyrimidinones

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1517
Woschek, Anna; Mahout, Marek; Mereiter, Kurt; Hammerschmidt, Friedrich: Synthesis of 2-Heptyl-1-hydroxy-4(1H)-quinolone - Unexpected Rearrangement of 4-(Alkoxycarbonyloxy)quinoline N-Oxides to 1-(Alkoxycarbonyloxy)-4(1H)-quinolones

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1523
Blair, Michael; Andrews, Philip C.; Fraser, Benjamin H.; Forsyth, Craig M.; Junk, Peter C.; Massi, Massimiliano; Tuck, Kellie L.: Facile Methods for the Separation of the cis- and trans-Diastereomers of Limonene 1,2-Oxide and Convenient Routes to Diequatorial and Diaxial 1,2-Diols

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1528
Fukuhara, Tsuyoshi; Hasegawa, Chihiro; Hara, Shoji: A Facile Synthesis of Oxazolines, Thiazolines, and Imidazolines Using α,α-Difluoroalkylamines

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1535
Tang, Shi; Li, Jin-Heng; Xie, Ye-Xiang; Wang, Nai-Xing: Halogenation of Indoles with Copper(II) Halides: Selective Synthesis of 2-Halo-, 3-Halo-, and 2,3-Dibromoindoles

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1542
Yoshida, Masanori; Osafune, Kanako; Hara, Shoji: Facile Synthesis of Iodonium Salts by Reaction of Organotrifluoroborates with p-Iodotoluene Difluoride

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1547
Sulima, Agnieszka; Folk, John; Jacobson, Arthur E.; Rice, Kenner C.: A New Approach to the Synthesis of the Nonpeptide NOP Receptor Antagonist J-113397

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1554
Rybáčková, Markéta; Bělohradský, Martin; Holý, Petr; Pohl, Radek; Dekoj, Václav; Závada, Jiří: Synthesis of Highly Symmetrical Triptycene Tetra- and Hexacarboxylates

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1559
Soley, Roger; Albericio, Fernando; Álvarez, Mercedes: Novel Synthesis of Arylethynyl Heterocycles

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1566
Prado, Soizic; Toum, Valérie; Saint-Joanis, Brigitte; Michel, Sylvie; Koch, Michel; Cole, Stewart T.; Tillequin, François; Janin, Yves L.: Antimycobacterial Benzofuro[3,2-f]chromenes from a 5-Bromochromen-6-ol

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1571
Hesse, Stéphanie; Kirsch, Gilbert: Buchwald-Hartwig Amination of β-Chloroacroleins by Lactams and Heteroarylamines

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feature article
1576
Restorp, Per; Dressel, Martina; Somfai, Peter: Synthesis of Functionalized Pyrrolidines by a Highly Stereoselective [3+2]-Annulation Reaction of N-Tosyl-α-Amino Aldehydes and 1,3-Bis(silyl)propenes

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practical synthetic procedures
1584
Ward, Dale E.; Rasheed, M. Abdul; Gillis, H. Martin; Beye, Garrison E.; Jheengut, Vishal; Achonduh, George T.: Simple and Efficient Preparation of Reagents for Thiopyran Introduction:
Methyl Tetrahydro-4-oxo-2H-thiopyran-3-carboxylate, Tetrahydro-4H-thiopyran-4-one, and 3,6-Dihydro-4-trimethylsilyloxy-2H-thiopyran

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1587
Bandini, Marco; Eichholzer, Astrid; Tommasi, Simona; Umani-Ronchi, Achille: Practical Aspects in the Gram-Scale Synthesis of Chiral Diamino-Bithiophene ‘DAT2’ Ligand

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addenda and errata
e1
Ward, Dale E.; Rasheed, M. Abdul; Gillis, H. Martin; Beye, Garrison E.; Jheengut, Vishal; Achonduh, George T.: Simple and Efficient Preparation of Reagents for Thiopyran Introduction: Methyl Tetrahydro-4-oxo-2H-thiopyran-3-carboxylate, Tetrahydro-4H-thiopyran-4-one, and 3,6-Dihydro-4-trimethylsilyloxy-2H-thiopyran FREE ACCESS

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