DOI: 10.1055/s-00000131

Synfacts

Issue 01 · Volume 2010 · January 2010 DOI: 10.1055/s-002-20656

Synform

A1
Zanda, Matteo: SYNFORM ISSUE 2010/01

Synthesis of Natural Products and Potential Drugs

z1
All PDFs of this category
0001
Nicolaou, K. C.; Dalby, S. M.; Li, S.; Suzuki, T.; Chen, D. Y.-K.: Synthesis of (+)-Haplophytine
0002
Pospíšil, J.; Müller, C.; Fürstner, A.: Synthesis of Aspercyclide B
0003
Ueda, H.; Satoh, H.; Matsumoto, K.; Sugimoto, K.; Fukuyama, T.; Tokuyama, H.: Synthesis of (+)-Haplophytine
0004
Mori, K.; Ohmori, K.; Suzuki, K.: Synthesis of Antibiotic TAN-1085
0005
Kim, K.; Cha, J. K.: Synthesis of Cyathin A3 and Cyathin B2
0006
Ghosh, A. K.; Shurrush, K.; Kulkarni, S.: Synthesis of (-)-Tetrahydrolipstatin
0007
Trenkle, J. D.; Jamison, T. F.: Synthesis of Gloeosporone
0008
Bender, C. F.; Yoshimoto, F. K.; Paradise, C. L.; De Brabander, J. K.: Synthesis of Berkelic Acid
0009
Ueda, M.; Yamaura, M.; Ikeda, Y.; Suzuki, Y.; Yoshizato, K.; Hayakawa, I.; Kigoshi, H.: Synthesis of Haterumalide NA
0010
Pesti, J.; Chen, C.-K.: Synthesis of Ravuconazole
0011
Boggs, S.; Elitzin, V. I.; Gudmundsson, K.; Martin, M. T.; Sharp, M. J.: CXCR4 Antagonist (GSK812397)
0012
Steinhuebel, D.; Sun, Y.; Matsumura, K.; Sayo, N.; Saito, T.: Synthesis of (R)-Sitagliptin
0013
Liu, W.-J.; Lv, B.-D.; Gong, L.-Z.: Synthesis of (-)-Bestatin
0014
Dong, J.-Q.; Wong, H. N. C.: Synthesis of (±)-Pallavicinolide
0015
Kong, K.; Romo, D.; Lee, C.: Synthesis of (-)-Gymnodimine
0016
Ogawa, S.; Urabe, D.; Yokokura, Y.; Arai, H.; Arita, M.; Inoue, M.: Synthesis of Resolvin E2
0017
Magauer, T.; Martin, H. J.; Mulzer, J.: Synthesis of Kendomycin
0018
Nicolaou, K. C.; Ortiz, A.; Zhang, H.: Synthesis of Vannusal B
0019
Campbell, M. J.; Johnson, J. S.: Synthesis of (+)-Polyanthellin A
0020
Ghosh, A. K.; Xi, K.: Formal Synthesis of (±)-Platencin

Synthesis of Heterocycles

z21
All PDFs of this category
0021
Ueda, S.; Nagasawa, H.: Copper-Catalyzed Synthesis of 1,2,4-Triazoles
0022
Liang, Z.; Hou, W.; Du, Y.; Zhang, Y.; Pan, Y.; Mao, D.; Zhao, K.: FeCl3-Mediated Synthesis of Benzo[b]furans from α-Aryl Ketones
0023
Lage, S.; Martínez-Estíbalez, U.; Sotomayor, N.; Lete, E.: Palladium-Catalyzed Synthesis of Pyrroloisoquinolines and Isoindoles
0024
Yasmin, N.; Ray, J. K.: Cs2CO3-Promoted Synthesis of Substituted Oxazoles
0025
Mizuno, A.; Kusama, H.; Iwasawa, N.: Rhodium-Catalyzed Synthesis of Pyrroles by [4+1] Cycloaddition
0026
Qiu, J.-W.; Zhang, X.-G.; Tang, R.-Y.; Zhong, P.; Li, J.-H.: Iron-Catalyzed Synthesis of 2-Aminobenzo-thiazoles
0027
Yadav, J. S.; Reddy, B. V. S.; Narasimhulu, G.; Chandrakanth, D.; Satheesh, G.: Cerium(III)-Catalyzed Synthesis of N-Arylpyrrolidines
0028
Phan, D. H. T.; Kim, B.; Dong, V. M.: Rhodium-Catalyzed Enantioselective Synthesis of Phthalides
0029
Rizk, T.; Bilodeau, E. J.-F.; Beauchemin, A.: Hydroamination Route to Pyridines and Pyrazines
0030
Praveen, C.; Jegatheesan, S.; Perumal, P. T.: Gold-Catalyzed Synthesis of Quinolines
0031
Pi, S.-S.; Zhang, X.-G.; Tang, R.-Y.; Li, J.-H.: CuBr-Catalyzed Synthesis of 2-Aminobenzo-thiazoles
0032
Contiero, F.; Jones, K. M.; Matts, E. A.; Porzelle, A.; Tomkinson, N. C. O.: Acid-Mediated Synthesis of Benzofurans from Arylhydroxylamines
0033
Ahmad, O. K.; Hill, M. D.; Movassaghi, M.: One-Step Synthesis of Polysubstituted Pyrimidines
0034
Parvatkar, P. T.; Parameswaran, P. S.; Tilve, S. G.: Iodine-Catalyzed One-Pot Synthesis of 6H-Indoloquinoline Derivatives
0035
Egi, M.; Azechi, K.: Gold-Catalyzed Synthesis of Pyrroles and Furans

Synthesis of Materials and Unnatural Products

z37
All PDFs of this category
0037
Ma, X.; Tang, J.; Shen, Y.; Fan, M.; Tang, H.; Radosz, M.: One Pot per Generation
0038
Lee, Y.-G.; Koyama, Y.; Yonekawa, M.; Takata, T.: High Degree of Functionality from Click Chemistry Polymers
0039
Mayerhöffer, U.; Deing, K.; Gruß, K.; Braunschweig, H.; Meerholz, K.; Würthner, F.: Very High Short-Circuit Currents in Squaraine Solar Cells
0040
Yanagisawa, S.; Ueda, K.; Sekizawa, H.; Itami, K.: Programmable Tetraarylthiophenes
0041
Nambo, M.; Wakamiya, A.; Yamaguchi, S.; Itami, K.: Fullerene Allylation
0042
Park, S.; Kwon, J. E.; Kim, S. H.; Seo, J.; Chung, K.; Park, S.-Y.; Jang, D.-J.; Medina, B. M.; Gierschner, J.: And ”Then There Was White"
0043
Ito, S.; Iida, T.; Kawakami, J.; Okujima, T.; Morita, N.: Packing-In Negative Charge with Azulenes
0044
Jiao, C.; Huang, K.-W.; Luo, J.; Zhang, K.; Chi, C.; Wu, J.: High Fluorescent Quantum Yield Bis-N-Annulated Quatterylenebis(dicarboximide)
0045
Ooyama, Y.; Kagawa, Y.; Fukuoka, H.; Ito, G.; Harima, Y.: Mechanofluorochromism in Organic Donor-Acceptor Dyes
0046
Zenkina, O. V.; Karton, A.; Shimon, L. J. W.; Martin, J. M. L.; van der Boom, M. E.: Reversing the Trend in Oxidative Addition
0047
Krohn, K.; Aslan, A.; Ahmed, I.; Pescitelli, G.; Funaioli, T.: Quinone-ly You
0048
Ferry, A.; Billard, T.; Langlois, B. R.; Bacqué, E.: An Easy Way to Trifluoromethanesulfanyls
0049
Janich, S.; Fröhlich, R.; Wakamiya, A.; Yamaguchi, S.; Würthwein, E.-U.: Ring Around the Porphyrins
0050
Zhang, K.; Huang, K.-W.; Li, J.; Luo, J.; Chi, C.; Wu, J.: Synthesis of a Quinoidal Bisanthene
0051
Pillekamp, M.; Alachraf, W.; Oppel, I. M.; Dyker, G.: Small Hydrocarbon Cages

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z53
All PDFs of this category
0053
Kister, J.; DeBaillie, A. C.; Lira, R.; Roush, W. R.: cis-Selective Hydroboration of Allenes
0054
Kim, H.; Chin, J.: Asymmetric Diaza-Cope Rearrangement Employing α-Keto Esters
0055
Gregg, T. M.; Farrugia, M. K.; Frost, J. R.: Enantioselective Cyclopropanation of Allenes Catalyzed by a Rhodium(II) Complex
0056
Hattori, G.; Yoshida, A.; Miyake, Y.; Nishibayashi, Y.: Enantioselective Ring Opening of Propargyl Epoxides
0057
Blay, G.; Fernández, I.; Monleón, A.; Muñoz, M. C.; Pedro, J. R.; Vila, C.: Zr- and Hf-Catalyzed Asymmetric Friedel-Crafts Alkylation of Indoles with Endiones
0058
Masarwa, A.; Fürstner, A.; Marek, I.: Synthesis of Chiral Cyclobutenes with All-Carbon Quaternary Stereocenters
0059
Tadaoka, H.; Cartigny, D.; Nagano, T.; Gosavi, T.; Ayad, T.; Genêt, J.-P.; Ohshima, T.; Ratovelomanana-Vidal, V.; Mashima, K.: Ir-Catalyzed Asymmetric Hydrogenation of 2-Aryl- and 2-Alkylquinolinium Salts
0060
Asikainen, M.; Krause, N.: Chiral 2,5-Dihydrofurans Via Tandem Lipase/Gold Catalysis
0061
Seki, K.; Yu, R.; Yamazaki, Y.; Yamashita, Y.; Kobayashi, S.: Zirconium-Catalyzed Enantioselective Ring Opening of meso-Aziridines
0062
Yoshida, M.; Higuchi, M.; Shishido, K.: Palladium-Catalyzed Stereoselective Construction of Chromans
0063
Chen, M.; Handa, M.; Roush, W. R.: Stereoselective Synthesis of 2-Methyl-3-butene-1,2-diols
0064
Colobert, F.; Valdivia, V.; Choppin, S.; Leroux, F. R.; Fernández, I.; Álvarez, E.; Khiar, N.: Diastereoselective Synthesis of Axially Chiral Biaryls
0065
Ma, S.; Han, X.; Krishan, S.; Virgil, S. C.; Stoltz, B. M.: Asymmetric Stereoablative Alkylation of 3-Halooxindoles
0066
Mršić, N.; Jerphagnon, T.; Minnaard, A. J.; Feringa, B. L.; de Vries, J. G.: Enantioselective Reduction of Quinoxalines
0067
Valdez, S. C.; Leighton, J. L.: Tandem Asymmetric Aza-Darzens/Ring-Opening Reactions
0068
Parmar, D.; Duffy, L. A.; Sadasivam, D. V.; Matsubara, H.; Bradley, P. A.; II, R. A. Flowers; Procter, D. J.: Reduction of Lactones with Samarium Iodide
0069
Hao, X.; Kuriyama, M.; Chen, Q.; Yamamoto, Y.; Yamada, K.-i.; Tomioka, K.: Rhodium-Catalyzed Addition of Arylboroxines to N-Phosphinoyl Aldimines
0070
Fillion, E.; Zorzitto, A. K.: Rhodium-Catalyzed Conjugate Alkynylation with TMS-acetylene
0071
Yu, X.; Lu, X.: Palladium-Catalyzed Tandem Annulation of 2-Formylarylboronic Acids with Allenoates
0072
Ghosh, P.; Cusick, J. R.; Inghrim, J.; Williams, L. J.: Addressing Selectivity in the Formation and Reactions of Spirodiepoxides
0073
Guthrie, D. B.; Geib, S. J.; Curran, D. P.: Asymmetric Synthesis of Chiral 3,4-Dihydro-quinolin-2-ones
0074
Abell, J. P.; Yamamoto, H.: Aluminum-Catalyzed Asymmetric Strecker Reaction
0075
Pelletier, S. M.-C.; Ray, P. C.; Dixon, D. J.: Three-Component Diastereoselective Synthesis of Pyrrolidinones
0076
Suzuki, T.; Ghozati, K.; Katoh, T.; Sasai, H.: Catalytic Oxidative Desymmetrization of meso-Secondary Diols
0077
Selim, K. B.; Matsumoto, Y.; Yamada, K.-i.; Tomioka, K.: Copper-Catalyzed Asymmetric Allylic Arylation with Grignard Reagents
0078
Nishimura, T.; Sawano, T.; Hayashi, T.: Rhodium-Catalyzed Asymmetric Conjugate Alkynylation
0079
Du, J.; Yoon, T. P.: [2+2] Cycloadditions by Visible Light Photocatalysis
0080
Shiomi, T.; Adachi, T.; Toribatake, K.; Zhou, L.; Nishiyama, H.: Rhodium-Catalyzed β-Boration of α,β-Unsaturated Carbonyl Compounds
0081
Hojo, D.; Noguchi, K.; Tanaka, K.: Cationic Rh(I)/Ag(I) Complexes Catalyzed the Synthesis of Tetrasubstituted Alkenes
0082
Aikawa, K.; Hioki, Y.; Mikami, K.: Dicationic Pd(II)-Catalyzed Alkenylation of Glyoxylate with Vinylsilanes

Metal-Mediated Synthesis

z83
All PDFs of this category
0083
Tarselli, M. A.; Micalizio, G. C.: Titanium-Mediated Reductive Cross-Coupling of Aliphatic Imines
0084
Moldoveanu, C.; Wilson, D. A.; Wilson, C. J.; Corcoran, P.; Rosen, B. M.; Percec, V.: Ni-Catalyzed Neopentylglycolborylation of Aryl Chlorides
0085
Watson, D. A.; Su, M.; Teverovskiy, G.; Zhang, Y.; García-Fortanet, J.; Kinzel, T.; Buchwald, S. L.: Palladium-Catalyzed Conversion of Aryl Triflates to Aryl Fluorides
0086
Zhang, S.-Y.; Tu, Y.-Q.; Fan, C.-A.; Zhang, F.-M.; Shei, L.: Fe-Catalyzed C-H Functionalization and Coupling of Alcohols with Alkenes
0087
Harvey, J. N.; Jover, J.; Lloyd-Jones, G. C.; Moseley, J. D.; Murray, P.; Renny, J. S.: Palladium-Catalyzed Newman-Kwart Rearrangement of Thiocarbamates
0088
Gøgsig, T. M.; Lindhardt, A. T.; Skrydstrup, T.: Heteroarylsulfonates in Iron-Catalyzed Coupling with Alkyl Grignard Reagents
0089
Hatakeyama, T.; Nakagawa, N.; Nakamura, M.: Iron-Catalyzed sp²-sp³ Cross-Coupling of Alkenylzinc Compounds
0090
Miura, K.; Inoue, G.; Sasagawa, H.; Kinoshita, H.; Ichikawa, J.; Hosomi, A.: Nucleophilic Addition of Alenylsilanes at the β-Position
0091
Xiao, Q.; Ma, J.; Yang, Y.; Zhang, Y.; Wang, J.: C=C Double Bond Formation via Coupling of N-Tosylhydrazones with Benzyl Halides
0092
Pridmore, S. J.; Slatford, P. A.; Taylor, J. E.; Whittlesey, M. K.; Williams, J. M. J.: Ru-Catalyzed Isomerization of Alkynediols and in situ Cyclization
0093
Aponick, A.; Li, C.-Y.; Malinge, J.; Marques, E. F.: A Facile Gold-Catalyzed Synthesis of Heterocycles from Propargyl Alcohols
0094
Thommes, K.; Kiefer, G.; Scopelliti, R.; Severin, K.: Olefin Cyclopropanation by Sequential Radical Addition/Dechlorination
0095
Isogai, Y.; Menggenbateer; Khan, F. N.; Asao, N.: CuX2-Mediated [4+2] Benzannulation for the Synthesis of Haloaromatic Compounds
0096
Tlili, A.; Xia, N.; Monnier, F.; Taillefer, M.: A Simple Cu-Catalyzed Synthesis of Phenols from Aryl Halides
0097
Brand, G. J.; Studte, C.; Breit, B.: ZnCl2-Catalyzed Enantiospecific C(sp³)-C(sp³) Cross-Coupling Giving (Oligo)deoxypropionates

Organo- and Biocatalysis

z99
All PDFs of this category
0099
Baer, K.; Kraußer, M.; Burda, E.; Hummel, W.; Berkessel, A.; Gröger, H.: Combining Organo- and Biocatalysis
0100
De, C. K.; Klauber, E. G.; Seidel, D.: A New Approach to Asymmetric DMAP Catalysis
0101
Markert, M.; Scheffler, U.; Mahrwald, R.: Cross-Aldol Reactions of Enolizable Aldehydes
0102
Han, X.; Kwiatkowski, J.; Xue, F.; Huang, K.-W.; Lu, Y.: A Highly Efficient Chiral Amine-Thiourea Catalyst
0103
Larson, S. E.; Baso, J. C.; Li, G.; Antilla, J. C.: Desymmetrization of meso-Aziridines with Thiols
0104
Baschieri, A.; Bernardi, L.; Ricci, A.; Suresh, S.; Adamo, M. F. A.: Styrylisoxazoles as Cinnamate Equivalents
0105
Belot, S.; Vogt, K. A.; Besnard, C.; Krause, N.; Alexakis, A.: Combining Gold- and Organocatalysis
0106
He, R.; Shirakawa, S.; Maruoka, K.: Enantioselective Base-Free Phase-Transfer Reaction
0107
Lindner, J.-P.; Röben, C.; Studer, A.; Stasiak, M.; Ronge, R.; Greiner, A.; Wendorff, H.-J.: Catalysts in a Bottle
0108
Zuend, S. J.; Coughlin, M. P.; Lalonde, M. P.; Jacobsen, E. N.: Gram-Scale Strecker Synthesis of Unnatural α-Amino Acids
0109
Joannesse, C.; Johnston, C. P.; Concellón, C.; Simal, C.; Philp, D.; Smith, A. D.: Enantioselective Steglich Rearrangement Using Isothiourea Catalysts
0110
Hili, R.; Yudin, A. K.: Cascade Reactions of Amphoteric Amino Aldehydes
0111
Barnett, D. S.; Moquist, P. N.; Schaus, S. E.: Mechanistic Insight in an Improved Allylboration of Ketones
0112
Fiori, K. W.; Puchlopek, A. L. A.; Miller, S. J.: Enantioselective Sulfonylation of Polyols

Polymer-Supported Synthesis

z113
All PDFs of this category
0113
Olmos, A.; Alix, A.; Sommer, J.; Pale, P.: Mukaiyama Aldol Reaction with Sc(III)-USY
0114
Yamaguchi, K.; Oishi, T.; Katayama, T.; Mizuno, N.: Huisgen Reaction of Organic Azides and Alkynes with Cu(OH)x/TiO2
0115
Spivey, A. C.; Tseng, C.-C.; Jones, T. C.; Kohler, A. D.; Ellames, G. J.: Parallel Solid-Phase Synthesis of Iodinated Analogues of Rimonabant
0116
Bhadra, S.; Sreedhar, B.; Ranu, B. C.: Base-Controlled Sequential C-S Bond Formation by CuSO4/Al2O3 Catalyst
0117
Motokura, K.; Tanaka, S.; Tada, M.; Iwasawa, Y.: Silica-Alumina-Supported Catalysts for Efficient 1,4-Addition Reactions
0118
Shimizu, K.-s.; Ohshima, K.; Satsuma, A.: Amide Synthesis from Alcohols and Amines with Ag/Al2O3
0119
Banerjee, S.; Sereda, G.: Three-Component Synthesis of Substituted Pyridines with Silica Nanoparticles
0120
Gruttadauria, M.; Salvo, A. M. P.; Giacalone, F.; Agrigento, P.; Noto, R.: Asymmetric Aldol Reaction with Polystyrene-Supported Proline-Based Catalysts
0121
Karimi, B.; Esfahani, F. K.: Aerobic Oxidation of Alcohols with Gold Nanoparticles Supported on Cs2CO3
0122
Dhakshinamoorthy, A.; Alvaro, M.; Garcia, H.: Carbon-Carbon Multiple Bond Reduction by MOF with Hydrazine
0123
Taher, A.; Kim, J.-B.; Jung, J.-Y.; Ahn, W.-S.; Jin, M.-J.: Suzuki Coupling in Water with Pd-NHC Immobilized on Fe3O4/Ionic Liquid
0124
Sreedhar, B.; Arundhathi, R.; Reddy, P. L.; Kantam, M. L.: C-N/C-O Bond Formation with CuI Nanoparticles
0125
Chandrasekhar, V.; Narayanan, R. S.; Thilagar, P.: Suzuki-Miyaura Coupling with Sn6O6-Pd Nanocomposites
0126
Mori, S.; Takubo, M.; Makida, K.; Yanase, T.; Aoyagi, S.; Maegawa, T.; Monguchi, Y.; Sajiki, H.: Aerobic Oxidation of Alcohols with Ruthenium on Carbon

Addenda and Errata

0127
Ni-Catalyzed Sonogashira Coupling of Nonactivated Alkyl Halides
0127
Synthesis of Kapakahines B and F
0127
Biaryl Cross Coupling Catalyzed by Fe/Co/Ni-Fluorides and NHC Ligands