DOI: 10.1055/s-00000131

Synfacts

Issue 01 · Volume 2006 · January 2006 DOI: 10.1055/s-002-4566

Synthesis of Natural Products and Potential Drugs

0001
Porco, J. A.; Zhu, J.; Grigoriadis, N. P.; Lee, J. P.: Copper-Mediated Synthesis of Azaphilones
0002
Paterson, I.; Chen, D. Y.-K.; Coster, M. J.; Aceña, J. L.; Bach, J.; Wallace, D. J.: Synthesis of Spongistatin 1
0003
King, H. D.; Meng, Z.; Denhart, D.; Mattson, R.; Kimura, R.; Wu, D.; Gao, Q.; Macor, J. E.: Synthesis of BMS-594726
0004
Nishiyama, T.; Isobe, M.; Ichikawa, Y.: Synthesis of Glycocinnaspermicin D
0005
Enders, D.; Lenzen, A.; Raabe, G.: Synthesis of 1-epi-Cripowellin A and B Aglycone
0006
Loh, T.-P.; Lee, C.-L. K.: Synthesis of (-)-Epibatidine
0007
Trost, B. M.; Dong, L.; Schroeder, G. M.: Synthesis of (+)-Allocyathin
0008
Nicolaou, K. C.; Montagnon, T.; Vassilikogiannakis, G.; Mathison, C. J. N.: Synthesis of Coleophomone B
0009
Wilson, R. M.; Jen, W. S.; MacMillan, D. W. C.: Synthesis of Solanopyrone A
0010
Yu, S. H.; Ferguson, M. J.; McDonald, R.; Hall, D. G.: Synthesis of Eupomatilone-6
0011
Pollex, A.; Millet, A.; Müller, J.; Hiersemann, H.; Abraham, L.: Synthesis of Viridiofungin A
0012
Strand, D.; Rein, T.: Synthesis of Pyragonicin
0013
Bolshakov, S.; Leighton, J. L.: Synthesis of (+)-SCH 351338
0014
Nicolaou, K. C.; Safina, B. S.; Zak, M.; Lee, S. H.; Navalainen, M.; Bella, M.; Estrada, A. A.; Funke, C.; Zecri, F. J.; Bulat, S.: Synthesis of Thiostrepton
0015
Paquette, L. A.; Tian, Z.; Seekamp, C. K.; Wang, T.: Synthesis of (-)-Neplanocin A

Synthesis of Heterocycles

0017
Zhao, J.; Larock, R. C.: A Benzyne Route to Xanthones and Thioxanthones
0018
González-Vera, J. A.; García-López, M. T.; Herranz, R.: Synthesis of Pyrrolo-imidazoindoles from Tryptophan Methyl Ester
0019
Ney, J. E.; Hay, M. B.; Yang, Q.; Wolfe, J.-P.: Palladium-Catalyzed Stereoselective Synthesis of 2-Allylpyrrolidines
0020
Clochard, M.; Grundy, J.; Donnadieu, B.; Mathey, F.: Synthesis of 3-Acylphospholes
0021
Yanada, R.; Obika, S.; Kobayashi, Y.; Inokuma, T.; Oyama, M.; Yanada, K.; Takemoto, Y.: Synthesis of 3-Benzylideneoxindoles
0022
Larquetoux, L.; Ouhamou, N.; Chiaroni, A.; Six, Y.: Titanium(IV)-Catalyzed Synthesis of 3-Azabicyclo[3.1.0]hexane Derivatives
0023
Rosas, N.; Sharma, P.; Arellano, I.; Ramírez, M.; Pérez, D.; Hernández, S.; Cabera, A.: Fe(II)-Mediated Synthesis of 5-Carboxy-3-pyrrolin-2-ones
0024
Frisch, K.; Landa, A.; Saaby, S.; Jørgensen, K. A.: Enantioselective Synthesis of 1,2-Dihydroisoquinolines and 1,2-Dihydrophthalazines
0025
Kaloko Jr, J.; Hayford, A.: Synthesis of Indolizine Derivatives by Electrocyclization
0026
Hiramatsu, N.; Takahashi, N.; Noyori, R.; Mori, Y.: Stereoselective Synthesis of Fused Tetrahydropyrans
0027
Markgraf, J. H.; Dowst, A. A.; Hensley, L. A.; Jakobsche, C. E.; Kaltner, C. J.; Webb, P. J.; Zimmerman, P. W.: A Versatile Synthesis of Benzacanthinones by Intramolecular Radical Coupling
0028
Ahmed, M. S. Mohamed; Kobayashi, K.; Mori, A.: Palladium-Catalyzed Multicomponent Synthesis of Pyrazoles and Isoxazoles
0029
Welter, C.; Moreno, R. M.; Streiff, S.; Helmchen, G.: Synthesis of (+)(R)- and (-)(S)-Nicotine via Enantioselective Ir-Catalyzed Allylic Amination
0030
Dziedzic, M.; Lipner, G.; Illangua, J. M.; Furman, B.: Synthesis of Dihydropyridinones and Hexahydroindolizin-7(1H)-one Derivatives
0031
Adamo, M. F. A.; Donati, D.; Duffy, E. F.; Sarti-Fantoni, P.: Diastereoselective Synthesis of Spiroisoxazolines

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

0033
Drago, C.; Caggiano, L.; Jackson, R. F. W.: Chiral Sulfoxide Synthesis via Vanadium-Catalyzed Oxidation of Sulfides
0034
Rainka, M. P.; Milne, J. E.; Buchwald, S. L.: Dynamic Kinetic Resolution in Cu-Catalyzed Conjugate Hydride Addition
0035
Wang, X.; Shi, L.; Li, M.; Ding, K.: Heterogeneous Catalyst for Enantioselective Epoxidation of α,β-Unsaturated Ketones
0036
Wadamoto, M.; Yamamoto, H.: Ag(I)-Catalyzed Allylation of Ketones with Allyltrimethoxysilanes
0037
Clark, J. S.; Roche, C.: Asymmetric Copper-Catalyzed Allylic Amination and Oxidation Reactions
0038
Lee, E. E.; Batey, R. A.: Stereoselective Synthesis of Allylic Alcohols via [3,3]-Sigmatropic Rearrangement
0039
Becht, J.-M.; Bappert, E.; Helmchen, G.: N-Heterocyclic Carbenes for Conjugate Additions of Arylboronic Acids
0040
Trost, B. M.; Ball, Z. T.; Kang, E.-J.: Synthesis of Tertiary Silanes by Diastereoselective Rearrangement-Addition
0041
Takita, R.; Yakura, K.; Oshima, T.; Shibasaki, M.: Asymmetric Propargyl Alcohols via Aldehyde Alkynylation
0042
Langner, M.; Rémy, P.; Bolm, C.: C1-Aminosulfoximines in Copper-Catalyzed Asymmetric Mukaiyama-Aldol Reactions
0043
Hansen, K. B.; Rosner, T.; Kubryk, M.; Dormer, P. G.; Armstrong III, J. D.: Asymmetric Catalytic Hydrogenation of Enamines
0044
Tanaka, K.; Hagiwara, Y.; Noguchi, K.: Rh-Catalyzed Enantioselective [4+2] Cyclization of 4-Alkynals and Acrylamides
0045
Minami, K.; Saito, H.; Tsutsui, H.; Nambu, H.; Anada, M.; Hashimoto, S.: 1,2-Disubstituted Cyclopentanes by Catalyzed C-H Insertion Reactions of α-Diazo Esters
0046
Trost, B. M.; Fandrick, D. R.; Dinh, D. C.: Dynamic Kinetic Asymmetric Allylic Alkylations of Allenes
0047
Lipshutz, B. H.; Frieman, B. A.: CuH in a Bottle: A Convenient Reagent for Asymmetric Hydrosilylations
0048
Shibata, T.; Arai, Y.; Tahara, Y.-K.: Enantioselective [2+2+2] Cycloaddition of 1,6-Enynes and Alkynes
0049
Kong, J.-R.; Cho, C.-W.; Krische, M. J.: Synthesis of Unnatural Amino Acids via Reductive C-C Bond Forming Hydrogenation
0050
Nakamura, M.; Hajra, A.; Endo, K.; Nakamura, E.: Enantioselective Synthesis of Quaternary α-Fluoroketones via Decarboxylation
0051
Zeng, W.; Zhou, Y.-G.: AgOAc-Catalyzed Asymmetric [3+2] Cycloaddition of Azomethine Ylides
0052
Yamagiwa, N.; Qin, H.; Matsunaga, S.; Shibasaki, M.: (S,S,S)-REMB-Catalyzed Enantioselective Aza-Michael Reactions
0053
Mohr, J. T.; Behenna, D. C.; Harned, A. M.; Stoltz, B. M.: Quaternary Carbon Center Formation by Decarboxylation of Allyl β-Ketoesters
0054
Vasse, J.-L.; Joosten, A.; Denhez, C.; Szymoniak, J.: Stereoselective Synthesis of Pyrrolidines via Hydrozirconation-Cyclization

Metal-Mediated Synthesis

0055
Shimizu, H.; Kobayashi, S.: Tantalum-Promoted Synthesis of α-Amino Amides from Imines and Isocyanates
0056
Felpin, F.-X.: Pd/C-Catalyzed Cross-Coupling of Arylboronic Acids with 2-Iodoenones
0057
Hatakeyama, T.; Ito, S.; Nakamura, M.; Nakamura, E.: Alkylation of Magnesium Enamides with Alkyl Chlorides and Fluorides
0058
Pozzi, D.; Scanlan, E. M.; Renaud, P.: A Mild Reduction of Alkenes to Alkanes via Alkylcatecholboranes
0059
Maifeld, S. V.; Lee, D.: Tandem Alkynylation-Hydrosilylation of Carbonyl Compounds
0060
Hlavinka, M. L.; Greco, J. F.; Hagadorn, J. R.: A Direct Zincation of Amides, Phosphonates and Phosphine Oxides
0061
Estevam, I. H. S.; da Silva, M. F.; Bieber, L. W.: Zinc-Promoted Aminomethylation of Organic Halides
0062
McLaughlin, M.: Cross-Coupling of Benzyl Phosphates with Arylboronic Acids
0063
Ikeda, Z.; Oshima, K.; Matsubara, S.: Preparation and Reactions of 2-Aryl-3-silyl-1,3-butadienes
0064
Shintani, R.; Okamoto, K.; Hayashi, T.: Rh/Chiral Diene-Catalyzed Enantioselective 1,4-Addition to β-Silyl Enones
0065
Flaherty, A.; Trunkfield, A.; Barton, W.: Cross-Coupling of B-Benzyl-9-BBN with Aryl Halides and Triflates
0066
Sakuma, D.; Togo, H.: Synthesis of Cyclopropanes from Homoallylic Iodides and 1,3-Dihalopropanes
0067
Itoh, Y.; Mikami, K.: Radical α-Trifluoromethylation of Ketones via Lithium Enolates

Organo- and Biocatalysis

0069
Akiyama, T.; Saitoh, Y.; Morita, H.; Fuchibe, K.: TADDOL-Derived Phosphoric Acid Catalyst
0070
Fini, F.; Sgarzani, V.; Pettersen, D.; Herrera, R. P.; Bernardi, L.; Ricci, A.: Highly Enantioselective Phase-Transfer-Catalyzed Aza-Henry Reaction
0071
Weinstein, R.; Lerner, R. A.; Barbas, C. F.; Shabat, D.: Antibody-Catalyzed Asymmetric Intramolecular Michael Reaction
0072
Hoffmann, S.; Seayad, A. M.; List, B.: Brønsted Acid Catalyzed Highly Enantioselective Transfer Hydrogenation of Ketimines
0073
Hayashi, Y.; Gotoh, H.; Tamura, T.; Yamaguchi, H.; Masui, R.; Shoji, M.: Cysteine-Derived Organocatalyst for Enantioselective Michael Reactions
0074
Kano, T.; Yamaguchi, Y.; Tokuda, O.; Maruoka, K.: Organocatalytic anti-Selective Direct Mannich Reaction
0075
Raheem, I. T.; Jacobsen, E. N.: Thiourea Derivative Catalyzed Asymmetric Aza-Baylis-Hillman Reaction
0076
Krafft, M. E.; Seibert, K. A.; Haxell, T. F. N.; Hirosawa, C.: Intramolecular Morita-Baylis-Hillman-type Alkylation of Enones
0077
McCooey, S. H.; Connon, S.: Bifunctional Organocatalysts for the Asymmetric Addition of Malonate to Nitroalkenes
0078
Reynolds, N. T.; Rovis, T.: Organocatalytic Asymmetric Synthesis of α-Chloroesters
0079
Gondi, V. B.; Gravel, M.; Rawal, V. H.: Organocatalytic Asymmetric Vinylogous Mukaiyama Aldol Reaction

Polymer-Supported Synthesis

0081
Bertini, V.; Lucchesini, F.; Pocci, M.; Alfei, S.: Polymeric 1,3-Dithiane Reagents
0082
Tajima, T.; Fuchigami, T.: Anodic Methoxylation Using Recyclable Solid-Supported Bases
0083
Koo, D. H.; Kim, M.; Chang, S.: WO3 Nanoparticles on MCM-48 for the Oxidation of Olefins
0084
Li, P.; Wang, L.; Li, H.: Ligand-, Copper- and Amine-Free Sonogashira Reaction with Pd Nanoparticles
0085
Pontrello, J. K.; Allen, M. J.; Underbakke, E. S.; Kiessling, L. L.: Solid-Phase Functionalization of Soluble Polymers
0086
Helms, B.; Guillaudeu, S. J.; Xie, Y.; McMurdo, M.; Hawker, C. J.; Fréchet, J. M. J.: Multiarm Star Polymer-Supported Acid and Base Catalyst
0087
Margathe, J.-F.; Shipman, M.; Smith, S. C.: Polymer-Supported Methyleneaziridines for Multicomponent Reactions
0088
Shanmugasundaram, M.; Garcia-Martinez, I.; Li, Q.; Estrada, A.; Martinez, N. E.; Martinez, L. E.: Microwave-Assisted Solid-Phase Dötz Benzannulation Reaction
0089
Maki, T.; Ishihara, K.; Yamamoto, H.: N-Alkyl-4-boronopyridinium Salts for Dehydrative Condensations
0090
Dambruoso, P.; Massi, A.; Dondoni, A.: Polymer-Assisted Solution-Phase Synthesis of the Isotetronic Acid
0091
Guinó, M.; Hii, K. K(M): Recyclable Polymer-Supported Pd Catalysts for Aryl Amination Reactions
0092
Chung, W.-J.; Kim, D.-K.; Lee, Y.-S.: Alcohol Oxidation with Polymer-Supported IBX
0093
Guinó, M. G.; Hii, K. K(M): Polymer-Supported Phosphines as Palladium Scavenger