DOI: 10.1055/s-00000131

Synfacts

Issue 01 · Volume 2005 · 2005 DOI: 10.1055/s-002-4363

Synthesis of Natural Products and Potential Drugs

0091
Herzon, S. B.; Myers, A. G.: Enantioselective Synthesis of Stephacidin B
0092
Arefolov, A.; Panek, J. S.: Total Synthesis of (+)-Discodermolide via Asymmetric Crotylation
0093
Mangion, I. K.; MacMillan, D. W. C.: Total Synthesis of (-)-Brasoside and (-)-Littoralisone
0094
Martinez, M. M.; Hoppe, D.: Total Synthesis of (-)-α-Kainic Acid
0095
Fujioka, H.; Ohba, Y.; Hirose, H.; Murai, K.; Kita, Y.: Total Synthesis of Rubrenolide
0096
Iwata, Y.; Maekawara, N.; Tanino, K.; Miyashita, M.: Total Synthesis of Tirandalydigin
0097
Chan, C.; Heid, R.; Zheng, S.; Guo, J.; Zhou, B.; Furuuchi, T.; Danishefsky, S. J.: Total Synthesis of Cribrostatin IV
0098
Holub, N.; Neidhöfer, J.; Blechert, S.: Total Synthesis of (+)-trans-195A
0099
Tsukano, C.; Ebine, M.; Sasaki, M.: Total Synthesis of Gymnocin-A
0100
Rozema, M. J.; Kruger, A. W.; Rohde, B. D.; Shelat, B.; Bhagavatula, L.; Tien, J. J.; Zhang, W.; Henry, R. F.: Synthesis of ABT-100, a Farnesyl Transferase Inhibitor
0101
Paterson, I.; Delgado, O.; Florence, G. J.; Lyothier, I.; O’Brien, M.; Scott, J. P.; Sereinig, N.: Synthesis of Discodermolide Using Solely Substrate-Based Stereocontrol
0102
Trost, B. M.; Fandrick, D. R.: Total Synthesis of (+)-Pseudodistomin D
0103
Baran, P. S.; Guerrero, C. A.; Ambhaikar, N. B.; Hafensteiner, B. D.: Total Synthesis of Stephacidin A
0104
Danner, P.; Bauer, M.; Phukan, P.; Maier, M. E.: Total Synthesis of Cryptophycin 3
0105
Feldman, K. S.; Skoumbourdis, A. P.: Synthesis of ()-Dibromophakellstatin

Synthesis of Heterocycles

0107
Chung, J. Y. L.; Cvetovich, R.; Amato, J.; McWilliams, J. C.; Reamer, R.; DiMichele, L.: Enantioselective Pyrrolidine Synthesis
0108
Cutri, S.; Diez, A.; Bonin, M.; Micouin, L.; Husson, H.-P.: Regio- and Stereoselective Synthesis of Structurally Diverse Polycyclic Indolyldiamines
0109
Yi, C. S.; Yun, S. Y.; Guzei, I. A.: Regioselective Hydroamination for the Synthesis of Tricyclic Quinolines
0110
Denmark, S. E.; Montgomery, J. I.: Synthesis of a Highly Strained Heterocycle Involving a Nitro Acetal to Aminal Rearrangement
0111
Lin, Y. S.; Liu, C. W.; Tsai, T. Y. R.: A Heterocyclic N-Oxide-Mediated Morita-Baylis-Hillman Reaction
0112
Ohno, H.; Miyamura, K.; Mizutani, T.; Kadoh, Y.; Takeoka, Y.; Hamaguchi, H.; Tanaka, T.: Tandem Cyclization of Allenenes to Tri- and Tetracyclic Heterocycles
0113
Grimster, N. P.; Gauntlett, C.; Godfrey, C. R. A.; Gaunt, M. J.: Palladium-Catalyzed Regioselective Direct C-2 and C-3 Functionalization of Indoles
0114
Wang, Z.; Bao, W.; Jiang, Y.: Synthesis of Aza-Stilbenes via an Ullmann C-N Coupling Reaction in Ionic Liquids
0115
Cottineau, B.; O’Shea, D. F.: Carbolithiation of Vinyl Pyridines as a Route to 7-Azaindoles
0116
Soderberg, B. C. G.; Hubbard, J. W.; Rector, S. R.; O’Neil, S. N.: Synthesis of Fused Indoles by Sequential Heck Reaction and N-Heteroannulation
0117
Kim, M. S.; Kim, Y.-W.; Hahm, H. S.; Jang, J. W.; Lee, W. K.; Ha, H.-J.: A Stereospecific Synthesis of Imidazolidin-2-ones from Aziridine-2-carboxylates and Isocyanates
0118
Zhao, J.; Hartwig, J. F.: Ruthenium-Catalyzed Cyclization of Diols to Lactones
0119
Sommen, G. L.; Linden, A.; Heimgartner, H.: Cycloaddition of Carbodiimides to Selenazetidines
0120
Zhuang, W.; Hazell, R. G.; Jørgensen, K. A.: Enantioselective Synthesis of Tryptamines and Tetrahydro-β-carbolines
0121
Nakao, Y.; Imanaka, H.; Sahoo, A. K.; Yada, A.; Hiyama, T.: Tetraorganosilicon Reagents for Cross-Coupling Reactions

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

0123
Shibata, N.; Kohno, J.; Takai, K.; Ishimaru, T.; Nakamura, S.; Toru, T.; Kanemasa, S.: Enantioselective Fluorination and Chlorination of Compounds Capable of Two-Point Binding
0124
Moreau, X.; Bazán-Tejeda, B.; Campagne, J.-M.: Enantioenriched α,β-Unsaturated Lactones via Vinylogous Mukaiyama Aldol
0125
Magdziak, D.; Lalic, G.; Lee, H. M.; Fortner, K. C.; Aloise, A. D.; Shair, M. D.: Protic Functionality-Tolerant Decarboxylative Thioester syn-Aldol Reactions
0126
Zhang, W.; Basak, A.; Kosugi, Y.; Hoshino, Y.; Yamamoto, H.: Vanadium-Catalyzed Enantioselective Epoxidation of Allylic Alcohols
0127
Dounay, A. B.; Overman, L. E.; Wrobleski, A. D.: Sequential Catalytic Asymmetric Heck-Iminium Ion Cyclization
0128
Hayashi, T.; Yamamoto, S.; Tokunaga, N.: Rhodium-Catalyzed Asymmetric 1,6-Addition of Aryl Zinc Reagents to Dienones
0129
Evans, M. A.; Morken, J. P.: Synthesis of Furans by the Pd-Catalyzed Oshima-Utimoto Reaction
0130
Donohoe, D. J.; Butterworth, S.: OsO4-Catalyzed Diastereoselective Formation of cis-Tetrahydrofurans
0131
Ohkuma, T.; Sandoval, C. A.; Srinivasan, R.; Lin, Q.; Wei, Y.; Muñiz, K.; Noyori, R.: Asymmetric Hydrogenation of tert-Alkyl Ketones
0132
Jagt, R. B. C.; de Vries, J. G.; Feringa, B. L.; Minnaard, A. J.: Enantioselective Synthesis of 2-Aryl-4-piperidones
0133
Martin-Matute, B.; Edin, M.; Bogár, K.; Kaynak, F. B.; Bäckvall, J.-E.: Dual Ru(II)/Lipase-Catalyzed Dynamic Kinetic Resolution of Secondary Alcohols
0134
Ng, S.-S.; Jamison, T. F.: Enantioenriched Allylic Alcohols via sp-Carbon Coupling of Allenes
0135
Schaefer, C.; Fu, G. C.: Asymmetric Couplings of Ketenes with Aldehydes to Generate Enol Esters
0136
Luanphaisarnnont, T.; Ndubaku, C. O.; Jamison, T. F.: anti-1,2-Diols via a Ni-Catalyzed Reductive Coupling
0137
Knöpfel, T. F.; Zarotti, P.; Ichikawa, T.; Carreira, E. M.: Catalytic, Enantioselective, Conjugate Alkyne Addition
0138
Ward, D. E.; Souweha, M. S.: Enantioselective Diels-Alder Using a Bimetallic Catalyst
0139
Kakei, H.; Tsuji, R.; Ohshima, T.; Shibasaki, M.: Asymmetric Epoxidation of α,β-Unsaturated Esters With Yttrium-Biphenyldiol Complex
0140
Davies, H. M. L.; Jin, Q.: Enantioselective Double C-H Activation of Dihydronaphthalenes
0141
Anderson, J. C.; Howell, G. P.; Lawrence, R. M.; Wilson, C. S.: Copper-Catalyzed Asymmetric Nitro-Mannich Reactions
0142
Evans, D. A.; Wu, J.: Sc(III)-Catalyzed Syn-Selective Enantioselective Carbonyl Ene Reactions
0143
Harada, S.; Handa, S.; Matsunaga, S.; Shibasaki, M.: N-(2-Hydroxyacetyl)pyrrole as an Ester Surrogate in Asymmetric Mannich Reactions
0144
Hamashima, Y.; Suzuki, T.; Takano, H.; Shimura, Y.; Sodeoka, M.: Catalytic Enantioselective Fluorination of Oxindoles
0145
Zhu, S.-F.; Yang, Y.; Wang, L.-X.; Liu, B.; Zhou, Q.-L.: Pd-Catalyzed Asymmetric Allylation of Aldehydes using Allylic Alcohols
0146
Evans, D. A.; Fandrick, K. R.; Song, H.: Enantioselective Friedel-Crafts Alkylations of α,β-Unsaturated 2-Acyl Imidazoles
0147
Boxer, M. B.; Yamamoto, H.: Diastereoselective [2+2] Cyclizations

Metal-Mediated Synthesis

0149
Takeda, T.; Ozaki, M.; Kuroi, S.; Tsubochi, A.: Cyclopropanation and Carbonyl Olefination of Alkynylsilyldithianes via Titanium Alkynyl­-carbenes
0150
Burgos, C.; Canales, E.; Matos, K.; Soderquist, J. A.: A Robust and Versatile Allyl- and Crotylboration with a Recyclable Auxiliary
0151
Chen, C.; Yang, L.-M.: Ni(II)-Catalyzed Arylation of Diarylamines
0152
Barbero, A.; Castreño, P.; Pulido, F. J.: One-Pot Synthesis of Spiro-Cyclopropanes from Oxoallylsilanes
0153
Cook, G. R.; Kargbo, R.; Maity, B.: Enantioselective Allylation of Hydrazones by Allylindium Complexes
0154
Black, D. A.; Arndsten, B. A.: A New Synthesis of Amides from Imines, Acid Chlorides and Organostannanes
0155
Lysén, M.; Kelleher, S.; Begtrup, M.; Kristensen, J. L.: Pd-Catalyzed Coupling of Arylboronic Esters with Carbamoyl Chlorides
0156
Yamato, S.; Yamamura, G.; Komatsu, M.; Arai, M.; Fukuyama, T.; Ryu, I.: Multicomponent Reactions Based on Dilithio Ketone α,β-Dianions
0157
Barrero, A. F.; Herrador, M. Mar; Moral, J. F. Quílez del; Arteaga, P.; Arteaga, J.; Piedra, M.; Sánchez, E. M.: Ti-Catalyzed Reductive Coupling of Terpenic Allylic Halides
0158
Ueura, K.; Satoh, T.; Miura, M.: Rh-Catalyzed Cross-Coupling Reactions and Arylation of Benzonitrile
0159
Macklin, T. K.; Snieckus, V.: Directed Metalation and Cross-Coupling of N,N-Dialkyl Aryl O-Sulfamates
0160
Yamashita, M.; Yamada, K.; Tomioka, K.: Asymmetric Conjugate Addition of Arylalkynes to Nitroolefins
0161
Moessner, C.; Bolm, C.: Copper-Catalyzed Arylation of Sulfoximines with Arylboronic Acids
0162
Hodgson, D. M.; Bray, C. D.; Kindon, N. D.: Base-Promoted Dimerization of Terminal Epoxides
0163
De, S.; Welker, M. E.: BF3-Substituted 1,3-Dienes and Their Diels-Alder/Cross-Coupling Reactions

Organo- and Biocatalysis

0165
Akiyama, T.; Morita, H.; Itoh, J.; Fuchibe, K.: Chiral Brønsted Acid Catalyzed Hydrophosphonylation of Imines
0166
Traverse, J. F.; Zhao, Y.; Hoveyda, A. H.; Snapper, M. L.: Proline-Based N-Oxides as Modular Chiral Catalysts for Allylation

Polymer-Supported Synthesis

0167
Cornejo, A.; Fraíle, J. M.; García, J. I.; Gil, M. J.; Luis, S. V.; Martínez-Merino, V.; Mayoral, J. A.: Immobilization of Bis(oxazolinyl)pyridines
0168
Weisberg, A.; Halak, B.; Portnoy, M.: The First Solid-Phase Synthesis of Bis(oxazolinyl)pyridine Ligands
0169
Houghten, R. A.; Yu, Y.: ‘Volatilizable’ Supports for High-Throughput Organic Synthesis
0170
Arseniyadis, S.; Subhash, P. V.; Valleix, A.; Wagner, A.; Mioskowski, C.: Polymer-Supported Acetylating Agent for the Kinetic Resolution of Amines
0171
Severinsen, R.; Kilburn, J. P.; Lau, J. F.: Solid Phase Synthesis of Small Heterocyclic Scaffolds
0172
Brenelli, E. C. S.; Brenelli, J. A.; Pinto, R. C. L.: Synthetic Procedure for Azidoalcohols Utilizing Polymer-Supported Reagent
0173
Hamamoto, H.; Suzuki, Y.; Yamada, Y. M. A.; Tabata, H.; Takahashi, H.; Ikegami, S.: A Thermomorphic Polymeric Catalyst for Alcoholic Oxidation
0174
Guinó, M.; Hii, K. K(M): Solid Phase Synthesis of α,α-Disubstituted Amino Acid Derivatives
0175
Uozumi, Y.; Kikuchi, M.: Selective Monoarylation of Dibromoarenes with Polymeric Palladium Catalyst
0176
Thomas, K. M.; Naduthambi, D.; Tririya, G.; Zondlo, N. J.: Proline Editing: A New Strategy for the Diversity-Oriented Peptide Synthesis
0177
Davies, H. M. L.; Walji, A. M.: Universal Strategy for the Immobilization of Chiral Dirhodium Catalysts
0178
Porzelle, A.; Fessner, W.-D.: Reversible Substrate Anchoring in Solid-Supported Organic Synthesis
0179
Li, Y.; Li, Z.; Li, F.; Wang, Q.; Tao, F.: Asymmetric Reduction of Ketones Catalyzed by a Polymeric Chiral Ru Complex
0180
Nakano, H.; Takahashi, K.; Fujita, R.: Asymmetric Diels-Alder Reaction Using a Polymer-Supported N-P Type Ligand
0181
Basso, A.; Ebert, C.; Gardossi, L.; Linda, P.; Phuong, T. T.; Zhu, M.; Wessjohann, L.: PGA-Catalyzed Hydrolysis of Phenylacetic Hydrazides on a Solid Phase