DOI: 10.1055/s-00000131

Synfacts

Issue 10 · Volume 2010 · October 2010 DOI: 10.1055/s-002-21347

Synthesis of Natural Products and Potential Drugs

z1093
All PDFs of this category
1093
al., A. Ribecai et: Synthesis of a Corticotropin-Releasing Factor Antagonist
1094
Nicolaou, K. C.; Kang, Q.; Ng, S. Y.; Chen, D. Y.-K.: Synthesis of Englerins A and B
1095
Tudge, M.; Savarin, C. G.; DiFelice, K.; Maligres, P.; Humphrey, G.; Reamer, B.; Tellers, D. M.; Hughes, D.: Synthesis of Prostaglandin D2 Receptor Antagonist
1096
Csatayová, K.; Davies, S. G.; Lee, J. A.; Ling, K. B.; Roberts, P. M.; Russell, A. J.; Thomson, J. E.: Synthesis of trans-SCH-A
1097
Binanzer, M.; Fang, G. Y.; Aggarwal, V. K.: Synthesis of (-)-Decarestrictine D
1098
Nicolaou, K. C.; Sun, Y.-P.; Korman, H.; Sarlah, D.: Synthesis of Cylindrocyclophane F
1099
Trzupek, J. D.; Lee, D.; Crowley, B. M.; Marathias, V. M.; Danishefsky, S. J.: Synthesis of (-)-Phalarine
1100
Johnston, E. V.; Bogár, K.; Bäckvall, J.-E.: Synthesis of (R)-Bufuralol
1101
Whiting, M.; Harwood, K.; Hossner, F.; Turner, P. G.; Wilkinson, M. C.: Synthesis of EP1 Antagonist GSK269984B
1102
Zi, W.; Yu, S.; Ma, D.: Synthesis of Galbulimima Alkaloid (-)-GB 13
1103
Mei, T.-S.; Wang, D.-H.; Yu, J.-Q.: Synthesis of Diclofenac and Lumiracoxib
1104
Elitzin, V. I.; Harvey, K. A.; Kim, H.; Salmons, M.; Sharp, M. J.; Tabet, E. A.; Toczko, M. A.: Synthesis of Triple Reuptake Inhibitor (-)-GSK1360707
1105
Lawrence, A. L.; Adlington, R. M.; Baldwin, J. E.; Lee, V.; Kershaw, J. A.; Thompson, A. L.: Biomimetic Synthesis of Guajadial and Psidial A
1106
Yun, S. Y.; Hansen, E. C.; Volchkov, I.; Cho, E. J.; Lo, W. Y.; Lee, D.: Synthesis of (-)-Dactylolide
1107
Matsuo, J.-i.; Okada, R.; Ishibashi, H.: Synthesis of (±)-Bremazocine
1108
al., G. W. Stewart et: Synthesis of a c-Met Kinase Inhibitor
1109
Jiang, X.; Lee, G. T.; Villhauer, E. B.; Prasad, K.; Prashad, M.: Synthesis of a Phosphodiesterase-4 Inhibitor

Synthesis of Heterocycles

z1111
All PDFs of this category
1111
Fordyce, E. A. F.; Morrison, A. J.; Sharp, R. D.; Paton, R. M.: Synthesis of 1,2,4-Thiadiazoles and Isothiazoles
1112
Kim, J.; Song, H.; Park, S. B.: Regioselective Synthesis of N-Alkyl-3-substituted Tetrahydroindazolones
1113
Ye, L.; He, W.; Zhang, L.: Gold-Catalyzed Synthesis of Oxetan-3-ones from Propargylic Alcohols
1114
Bonnamour, J.; Piedrafita, M.; Bolm, C.: Effect of Fe and Cu Salts in the Heteroannulative Synthesis of Benzo[b]furans
1115
Awasthi, C.; Yadav, L. D. S.: NHC-Mediated [2+2] Cycloaddition Route to Nitro-β-thiolactams
1116
Yu, H.; Jin, W.; Sun, C.; Chen, J.; Du, W.; He, S.; Yu, Z.: Synthesis of Bicyclic Pyridones from 1,3-Butadienes
1117
Li, S.; Yuan, Y.; Zhu, J.; Xie, H.; Chen, Z.; Wu, Y.: Copper-Catalyzed Annulative Synthesis of 2-Fluoromethylated Quinolines
1118
Liu, C.-C.; Parthasarathy, K.; Cheng, C.-H.: Nickel-Catalyzed Heteroannulative Route to Isoquinolones
1119
Parsons, A. T.; Smith, A. G.; Neel, A. J.; Johnson, J. S.: Mg-Catalyzed Dynamic Asymmetric Synthesis of Chiral Pyrrolidines
1120
Xi, J.; Dong, Q.-L.; Liu, G.-S.; Wang, S.; Chen, L.; Yao, Z.-J.: Bischler-Napieralski Synthesis of Phenanthridines
1121
Tobisu, M.; Fujihara, H.; Koh, K.; Chatani, N.: Copper-Catalyzed Borylative and Silylative Cyclization of Isocyanides to Indoles
1122
Spiteri, C.; Keeling, S.; Moses, J. E.: 1H-Indazoles via Huisgen [3+2] Cycloaddition of Benzynes with Nitrile Imines
1123
Malakar, C. C.; Merisor, E.; Conrad, J.; Beifuss, U.: Molybdenum Complex Catalyzed Reductive Cyclization of ω-Nitro Alkenes
1124
Polivanova, A. G.; Shkavrov, S. V.; Churakov, A. V.; Lermontov, A. S.; Lermontov, S. A.: Synthesis of 1,5-Disubstituted Fluorinated Tetrazoles
1125
Brenzovich Jr., W. E.; Benitez, D.; Lackner, A. D.; Shunatona, H. P.; Tkatchouk, E.; III, W. A. Goddard; Toste, F. D.: Gold-Catalyzed Intramolecular Aminoarylation to Pyrrolidines

Synthesis of Materials and Unnatural Products

z1127
All PDFs of this category
1127
Hiorns, R. C.; Cloutet, E.; Ibarboure, E.; Khoukh, A.; Bejbouji, H.; Vignau, L.; Cramail, H.: Fullerene as a Repeat Unit in a Novel Donor-Acceptor Polymer
1128
Diev, V. V.; Hanson, K.; Zimmerman, J. D.; Forrest, S. R.; Thompson, M. E.: Soluble Fused Pyrene-Diporphyrins via Oxidative Ring Closure
1129
Rieger, R.; Beckmann, D.; Pisula, W.; Kastler, M.; Müllen, K.: An Extended Polythiophene with Interesting Core Synthesis
1130
Sinha, M. K.; Reany, O.; Parvari, G.; Karmakar, A.; Keinan, E.: When Bipy Met Cucurbit[6]uril
1131
Hu, R.; Feng, J.; Hu, D.; Wang, S.; Li, S.; Li, Y.; Yang, G.: Fluoride Sensing in Water
1132
Tam, T. L.; Li, H.; Wei, F.; Tan, K. J.; Kloc, C.; Lam, Y. M.; Mhaisalkar, S. G.; Grimsdale, A. C.: One-Pot (Synthesis) Feeds Many Chemists
1133
Esser-Kahn, A. P.; Sottos, N. R.; White, S. R.; Moore, J. S.: Triggered Microcapsule Depolymerization
1134
Tzirakis, M. D.; Orfanopoulos, M.: Crowning of the Fullerene
1135
Fukuhara, G.; Inoue, Y.: Amplified Chiral Sensing
1136
Miyasaka, M.; Pink, M.; Rajca, S.; Rajca, A.: Spiro Oligothiophenes
1137
Fischer, G. M.; Jüngst, C.; Isomäki-Krondahl, M.; Gauss, D.; Möller, H. M.; Daltrozzo, E.; Zumbusch, A.: Break Symmetry, and Get Benefits
1138
Tsuchimoto, T.; Igarashi, M.; Aoki, K.: Catalytic β-Alkylation of Pyrroles
1139
Berná, J.; Alajarín, M.; Orenes, R.-A.: A Dynamic Molecular Shuttle
1140
Yoshida, H.; Mukae, M.; Ohshita, J.: Renaissance of Diels-Alder Reaction of Borylalkenes

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z1141
All PDFs of this category
1141
Nörder, A.; Herrmann, P.; Herdtweck, E.; Bach, T.: Diastereoselective Catalytic C-H Amination
1142
Yazaki, R.; Kumagai, N.; Shibasaki, M.: Enantioselective Conjugate Addition of Alkynes to Thioamides
1143
Zhu, S.-F.; Cai, Y.; Mao, H.-X.; Xie, J.-H.; Zhou, Q.-L.: Iron-Catalyzed Asymmetric OH Bond Insertions
1144
Moro, A. Venturini; Tiekink, E. R. T.; Zuckerman-Schpector, J.; Lüdtke, D. S.; Correia, C. R. D.: New Ligand for Asymmetric Arylation of Aldehydes
1145
Schwab, R. S.; Soares, L. C.; Dornelles, L.; Rodrigues, O. E. D.; Paixão, M. W.; Godoi, M.; Braga, A. L.: Chiral Chalcogen Peptides as Ligands for Aryl Transfer to Aldehydes
1146
Reddy, R. S.; Chouthaiwale, P. V.; Suryavanshi, G.; Chavan, V. B.; Sudalai, A.: Cobalt-Catalyzed HKR of Alkoxy- and Azido Epoxides
1147
Pullmann, T.; Engendahl, B.; Zhang, Z.; Hölscher, M.; Zanotti-Gerosa, A.; Dyke, A.; Franciò, G.; Leitner, W.: New Quinaphos Ligands for Asymmetric Hydrogenation
1148
Müslehiddinoğlu, J.; Li, J.; Tummala, S.; Deshpande, R.: Diastereoselective Hydrogenation of Imines
1149
Ager, B. J.; Bourque, L. E.; Buchner, K. M.; Woerpel, K. A.: Synthesis of Silacyclobutanes
1150
Hamed, O.; Henry, P. M.; Becker, D. P.: Palladium(II)-Catalyzed Dicarboxylation of Chiral Allylic Alcohols
1151
Naik, A.; Maji, T.; Reiser, O.: Iron(II)-Bis(isonitrile) Catalyzed Asymmetric Transfer Hydrogenation
1152
Liu, L.; Floreancig, P. E.: Stereoselective Synthesis of Cyclic Ethers
1153
Tambar, U. K.; Lee, S. K.; Leighton, J. L.: Enantioselective Aza-Diels-Alder Reactions
1154
Yang, C.-M.; Jeganmohan, M.; Parthasarathy, K.; Cheng, C.-H.: Regio- and Stereoselective Three-Component Reaction towards 1,3-Dienes
1155
Woodmansee, D. H.; Müller, M.-A.; Neuburger, M.; Pfaltz, A.: Iridium-Catalyzed Asymmetric Hydrogenation of Trisubstituted Olefins
1156
Bădoiu, A.; Bernardinelli, G.; Kündig, E. P.: Enantioselective 1,3-Dipolar Cycloadditions of N-Methylnitrones and Enals
1157
McDonald, R. I.; Stahl, S. S.: Palladium-Catalyzed Oxidative Cyclization of Allylic Sulfamides
1158
Blay, G.; Hernández-Olmos, V.; Pedro, J. R.: Preparation of Chiral Building Blocks via Enantioselective Henry Reaction
1159
Cartigny, D.; Püntener, K.; Ayad, T.; Scalone, M.; Ratovelomanana-Vidal, V.: Enantio- and Diastereoselective Synthesis of syn-1,2-Diol Derivatives
1160
Verendel, J. J.; Zhou, T.; Li, J.-Q.; Paptchikhine, A.; Lebedev, O.; Andersson, P. G.: Synthesis of Chiral Pyrrolidines, Piperidines, and Azepanes
1161
Xu, Q.-L.; Liu, W.-B.; Dai, L.-X.; You, S.-L.: Iridium-Catalyzed Asymmetric Allylic Substitution
1162
Pelphrey, P.; Hansen, J.; Davies, H. M. L.: Enantioselective Cyclopropanation at ppm Catalyst Loading
1163
Stanley, L. M.; Bai, C.; Ueda, M.; Hartwig, J. F.: Kinetic Asymmetric Substitution of Racemic Allylic Esters
1164
Fan, X.-Y.; Yang, Y.-X.; Zhuo, F.-F.; Yu, S.-L.; Li, X.; Guo, Q.-P.; Du, Z.-X.; Da, C.-S.: Lewis Acid/Lewis Base Assisted Asymmetric Grignard Reaction
1165
Soltani, O.; Ariger, M. A.; Vázquez-Villa, H.; Carreira, E. M.: Catalytic Enantioselective Transfer Hydrogenation in Water
1166
Franck, G.; Brödner, K.; Helmchen, G.: Enantioselective Synthesis of Cyclohexenones
1167
Guo, C.; Song, J.; Luo, S.-W.; Gong, L.-Z.: Asymmetric Dehydrogenative Cross-Coupling
1168
Liu, Z.; Du, H.: New Ligands for Palladium-Catalyzed Asymmetric Allylic Substitutions
1169
Marié, J.-C.; Xiong, Y.; Min, G. K.; Yeager, A. R.; Taniguchi, T.; Berova, N.; Schaus, S. E.; Porco Jr., J. A.: Lewis Acid Catalyzed Asymmetric Rearrangement of 3-Allyloxyflavones

Metal-Mediated Synthesis

z1171
All PDFs of this category
1171
Yoshida, Y.; Murakami, K.; Yorimitsu, H.; Oshima, K.: Stereoselective Rhodium-Catalyzed Arylzincation of Terminal Allenes
1172
Iwai, T.; Fujihara, T.; Terao, J.; Tsuji, Y.: Iridium-Catalyzed Annulation of Carbamoyl Chlorides with Internal Alkynes
1173
Ishida, N.; Shimamoto, Y.; Murakami, M.: Oligo(arylenevinylene)s Containing Tetrasubstituted Vinylene Units
1174
Houlden, C. E.; Lloyd-Jones, G. C.; Booker-Milburn, K. I.: Transient Urea as Directing Group: Synthesis of ortho-Functionalized Anilines
1175
Chernyak, D.; Skontos, C.; Gevorgyan, V.: Two-Component Cyclization to N-Fused Pyrroles
1176
Whittaker, A. M.; Rucker, R. P.; Lalic, G.: Catalytic SN2′-Selective Substitution of Allylic Chlorides with Arylboronic Esters
1177
Torregrosa, R. R. P.; Ariyarathna, Y.; Chattopadhyay, K.; Tunge, J. A.: Decarboxylative Benzylation of Alkynes and Substituted Ketones
1178
Liang, Z.; Yao, B.; Zhang, Y.: Palladium-Catalyzed Regioselective Arylation of Indoles with Arylsiloxanes
1179
Park, J. H.; Cho, Y.; Chung, Y. K.: Rhodium-Catalyzed Pauson-Khand-Type Reaction
1180
Wu, X.-F.; Neumann, H.; Beller, M.: Preparation of Chalcones by Carbonylative Heck Reaction
1181
Melhado, A. S.; Brenzovich Jr., W. E.; Lackner, A. D.; Toste, F. D.: Gold-Catalyzed Oxidative Oxyarylation of Alkenes
1182
Štefane, B.: Selective Addition of Organolithium Reagents to BF2-Chelates
1183
Simon, M.-O.; Genêt, J.-P.; Darses, S.: RuCl3-Catalyzed Hydroarylation
1184
Rakshit, S.; Patureau, F. W.; Glorius, F.: Rhodium-Catalyzed Allylic sp³ C-H Activation of Enamines in the Synthesis of Pyrroles

Organo- and Biocatalysis

z1185
All PDFs of this category
1185
Lu, M.; Lu, Y.; Zhu, D.; Zeng, X.; Li, X.; Zhong, G.: Enantioselective α-Aminoxylation of Enecarbamates
1186
Zheng, W.; Wojtas, L.; Antilla, J. C.: Catalytic Asymmetric Peroxidation of Imines
1187
Jain, P.; Antilla, J. C.: Allylboration of Aldehydes
1188
Matoba, K.; Kawai, H.; Furukawa, T.; Kusuda, A.; Tokunaga, E.; Nakamura, S.; Shiro, M.; Shibata, N.: Trifluoromethyl-2-Isoxazoles via Phase-Transfer Catalysis
1189
Li, N.; Chen, X.-H.; Zhou, S.-M.; Luo, S.-W.; Song, J.; Ren, L.; Gong, L.-Z.: Precipitation Induced Nonlinear Effects in Phosphoric Acid Catalysis
1190
Liu, W.; Cao, H.; Zhang, H.; Chung, K. H.; He, C.; Wang, H.; Kwong, F. Y.; Lei, A.: DMEDA-Catalyzed Cross-Coupling of Unactivated Benzene
1191
Van Humbeck, J. F.; Simonovich, S. P.; Knowles, R. R.; MacMillan, D. W. C.: A Closed-Shell Mechanism Alternative for Sibi’s α-Oxyamination of Aldehydes
1192
Kano, T.; Mii, H.; Maruoka, K.: Organocatalytic Asymmetric α-Aminoxylation of Aldehydes
1193
Sparr, C.; Gilmour, R.: Using Fluorine to ‘Freeze Out’ Catalyst Conformations
1194
Pousse, G.; Cavelier, F. Le; Humphreys, L.; Rouden, J.; Blanchet, J.: Chiral Phosphoric Acid Catalyzed Direct Aldol Reactions of Glyoxylates
1195
Dong, S.; Liu, X.; Chen, X.; Mei, F.; Zhang, Y.; Gao, B.; Lin, L.; Feng, X.: An Unexpected Chiral Bisguanidine Catalyzed Hetero-Diels-Alder Reaction
1196
Li, J.-L.; Kang, T.-R.; Zhou, S.-L.; Li, R.; Wu, L.; Chen, Y.-C.: Crotonaldehyde-Derived Dienamine as Dienophile in IEDDA Reaction
1197
Savile, C. K.; Janey, J. M.; Mundorff, E. C.; Moore, J. C.; Tam, S.; Jarvis, W. R.; Colbeck, J. C.; Krebber, A.; Fleitz, F. J.; Brands, J.; Devine, P. N.; Huisman, G. W.; Hughes, G. J.: A Manufactured Enzyme for the Synthesis of Chiral Amines

Polymer-Supported Synthesis

z1199
All PDFs of this category
1199
O’Brien, M.; Baxendale, I. R.; Ley, S. V.: Flow Ozonolysis Using a Semipermeable Teflon AF-2400 Membrane
1200
Zhang, J.; Yu, C.; Wang, S.; Wan, C.; Wang, Z.: Synthesis of Quinazolines with Supported Copper Oxide Nanoparticles
1201
Karimi, B.; Elhamifar, D.; Clark, J. H.; Hunt, A. J.: Suzuki-Miyaura Coupling in Water Using Pd@PMO-IL
1202
Ito, S.; Hayashi, A.; Komai, H.; Kubota, Y.; Asami, M.: Sakurai Allylation and Mukaiyama Aldol Reaction with Al-MCM-41
1203
Hornung, C. H.; Hallmark, B.; Mackley, M. R.; Baxendale, I. R.; Ley, S. V.: EVOH Capillary Supported Palladium Catalyst for Flow Transfer Hydrogenation
1204
Tagata, T.; Nishida, M.; Nishida, A.: Continuous Flow C-H Borylation of Arenes
1205
Akkilagunta, V. K.; Reddy, V. P.; Rao, K. R.: C-S Cross-Coupling with Iron/Graphite
1206
Piscopo, C. G.; Loebbecke, S.; Maggi, R.; Sartori, G.: Supported Sulfonic Acid as a Catalyst for Baeyer-Villiger Oxidation with H2O2
1207
Mori, S.; Takubo, M.; Yanase, T.; Maegawa, T.; Monguchi, Y.; Sajiki, H.: Pd/C-Catalyzed Oxidation of 1,2-Diarylalkynes with DMSO and O2
1208
Dhakshinamoorthy, A.; Alvaro, M.; Garcia, H.: Regioselective Ring Opening of Epoxides with [Fe(BTC)]
1209
Fall, A.; Sene, M.; Gaye, M.; Gómez, G.; Fall, Y.: Oxidation of Alcohols with TEMPO Immobilized on an Ionic Liquid
1210
Kawamorita, S.; Ohmiya, H.; Sawamura, M.: Regioselective C-H Borylation of Heteroarenes with Silica-SMAP-Ir