DOI: 10.1055/s-00000131

Synfacts

Issue 12 · Volume 2009 · December 2009 DOI: 10.1055/s-002-20564

Synform

A76
Zanda, Matteo: SYNFORM ISSUE 2009/09

Synthesis of Natural Products and Potential Drugs

z1303
All PDFs of this category
1303
Hansen, K. B.; Hsiao, Y.; Xu, F.; Rivera, N.; Clausen, A.; Kubryk, M.; Krska, S.; Rosner, T.; Simmons, B.; Balsells, J.; Ikemoto, N.; Sun, Y.; Spindler, F.; Malan, C.; Grabowski, E. J. J.; Armstrong, III, J. D.: Synthesis of Sitagliptin
1304
Smith, III, A. B.; Dong, S.; Brenneman, J. B.; Fox, R. J.: Synthesis of (+)-Sorangicin A
1305
Movassaghi, M.; Tjandra, M.; Qi, J.: Synthesis of (-)-Himandrine
1306
Rano, T. A.; Kuo, G.-H.: Synthesis of a CETP Inhibitor
1307
Yoshimura, F.; Sasaki, M.; Hattori, I.; Komatsu, K.; Sakai, M.; Tanino, K.; Miyashita, M.: Synthesis of Zoanthamine
1308
Yun, S. Y.; Zheng, J.-C.; Lee, D.: Formal Synthesis of Platensimycin
1309
Sälinger, D.; Brückner, R.: Synthesis of (R)-Orphenadrine
1310
Mukherjee, S.; Lee, D.: Formal Synthesis of (-)-Cochleamycin A
1311
Jung, J. H.; Lee, E.: Synthesis of (-)-Amphidinolide X
1312
Schwartz, B. D.; Denton, J. R.; Lian, Y.; Davies, H. M. L.; Williams, C. M.: Synthesis of (-)-5-epi-Vibsanin E
1313
Wallace, G. A.; Gordon, T. D.; Hayes, M. F.; Konopacki, D. B.; Fix-Stenzel, S. R.; Zhang, X.; Grongsaard, P.; Cusack, K. P.; Schaffter, L. M.; Henry, R. F.; Stoffel, R. H.: Synthesis of S1P1 Receptor Agonists
1314
Hama, N.; Matsuda, T.; Sato, T.; Chida, N.: Synthesis of (-)-Agelastatin A
1315
Karpf, M.; Trussardi, R.: Synthesis of Tamiflu
1316
Czakó, B.; Kürti, L.; Mammoto, A.; Ingber, D. E.; Corey, E. J.: Synthesis of Cortistatin Analogues
1317
König, C. M.; Gebhardt, B.; Schleth, C.; Dauber, M.; Koert, U.: Synthesis of Phoslactomycin A

Synthesis of Heterocycles

z1319
All PDFs of this category
1319
González-Gómez, Á.; Domínguez, G.; Pérez-Castells, J.: Gold-Catalyzed Synthesis of Benzazepines
1320
Gruit, M.; Michalik, D.; Tillack, A.; Beller, M.: Platinum-Catalyzed Synthesis of Pyrrolo[3,2-c]azepin-4-ones
1321
Gao, L.; Hwang, G.-S.; Lee, M. Y.; Ryu, D. H.: Catalytic Enantioselective Synthesis of 2-Pyrazolines
1322
Li, H.; Hsung, R. P.: Rh-Catalyzed Synthesis of 2-Amido-furans via Cyclopropenation of Ynamides
1323
Wang, J.-Y.; Wang, X.-P.; Yu, Z.-S.; Yu, W.: Lewis Acid Catalyzed Synthesis of Multisubstituted Pyrroles
1324
Ueno, S.; Ohtsubo, M.; Kuwano, R.: Palladium-Catalyzed Synthesis of Tetrahydroisoquinolines
1325
Cantagrel, G.; de Carné-Carnavalet, B.; Meyer, C.; Cossy, J.: FeCl3-Promoted Cyclization of o-Alkylaryl Isocyanates to Oxindoles
1326
Mosslemin, M. H.; Anary-Abbasinejad, M.; Anaraki-Ardakani, H.: Multicomponent Synthesis of 2-Aminofurans
1327
Hodgkinson, R. C.; Schulz, J.; Willis, M. C.: Cascade N-Annulation Route to 7-Azaindoles
1328
Bernini, R.; Fabrizi, G.; Sferrazza, A.; Cacchi, S.: Copper-Catalyzed C-H Activation to Polysubstituted Indoles
1329
Pati, K.; Liu, R.-S.: Ruthenium-Catalyzed Synthesis of Pyridones and Isoquinolones
1330
Yamashita, M.; Horiguchi, H.; Hirano, K.; Satoh, T.; Miura, M.: Construction of Carbazoles via Pd-Catalyzed Oxidative Coupling of Alkynes
1331
Kazmaier, U.; Schmidt, C.: One-Pot Stereoselective Synthesis of Furanoid Amino Acids
1332
Chen, D.; Shen, G.; Bao, W.: Copper-Catalyzed Synthesis of 2H-1,4-Benzoxazin-3-(4H)-ones
1333
Murru, S.; Ghosh, H.; Sahoo, S. K.; Patel, B. K.: Synthesis of Arylthiobenzothiazoles via a Copper(I)-Catalyzed S-Arylation

Synthesis of Materials and Unnatural Products

z1335
All PDFs of this category
1335
Kissel, P.; Schlüter, A. D.; Sakamoto, J.: Molecular Chain Mail
1336
Deshpande, R.; Jiang, L.; Schmidt, G.; Rakovan, J.; Wang, X.; Wheeler, K.; Wang, H.: Tandem Heck Reaction/6π-Electrocyclization for the Synthesis of opp-Dibenzoporphyrins
1337
Filippone, S.; Maroto, E. E.; Martín-Domenech, A.; Suarez, M.; Martín, N.: Catalytic Enantioselective Synthesis of Fullerene Derivatives
1338
Hilt, G.; Paul, A.; Hengst, C.: Cobalt-Catalyzed [6+2] Cycloadditions with Cycloheptatriene
1339
Dale, T. J.; Rebek Jr., J.: Nerve Agent Sensor and Antidote in One Molecule
1340
Zhu, X.; Mitsui, C.; Tsuji, H.; Nakamura, E.: Indenes and Indacenes
1341
Yao, J. H.; Chi, C.; Wu, J.; Loh, K.-P.: Bianthryl Diimides
1342
Barluenga, J.; Campos-Gómez, E.; Minatti, A.; Rodríguez, D.; González, J. M.: Iodonium Ion Triggered Arene Functionalization
1343
Suzuki, T.; Ishigaki, Y.; Iwai, T.; Kawai, H.; Fujiwara, K.; Ikeda, H.; Kano, Y.; Mizuno, K.: A Redox Approach to Molecular Logic Operators
1344
Bolz, I.; Schaarschmidt, D.; Rüffer, T.; Lang, H.; Spange, S.: A New Record for Negative Solvatochromism
1345
Zhao, Z.; Wang, Z.; Lu, P.; Chan, C. Y. K.; Liu, D.; Lam, J. W. Y.; Sung, H. H. Y.; Williams, I. D.; Ma, Y.; Tang, B. Z.: Aggregation-Induced Emission
1346
Furukawa, S.; Kobayashi, J.; Kawashima, T.: Synthesis of Dibenzosiloles
1347
Shefer, N.; Harel, T.; Rozen, S.: Fast Oxidation to Sulfones
1348
Baik, C.; Hudson, Z.; Amarne, H.; Wang, S.: Photoisomerization
1349
Takagi, K.; Sugihara, K.; Isomura, T.: Large Shifts from Proton Transfer

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z1351
All PDFs of this category
1351
Stanley, L. M.; Hartwig, J. F.: Iridium-Catalyzed N-Allylation of Indoles
1352
Murarka, S.; Deb, I.; Zhang, C.; Seidel, D.: Catalytic Enantioselective Synthesis of Ring-Fused Tetrahydroquinolines
1353
Parsons, A. T.; Johnson, J. S.: Synthesis of Tetrahydropyrans through Formal [4+2] Cycloaddition
1354
Mercier, A.; Yeo, W. C.; Chou, J.; Chaudhuri, P. D.; Bernardinelli, G.; Kündig, E. P.: Synthesis of Planar Chiral Ru Complexes through Asymmetric Hydrogenolysis
1355
Yu, R. T.; Friedman, R. K.; Rovis, T.: Synthesis of Bicyclic Azocine Rings via Rh-Catalyzed [4+2+2] Cycloaddition
1356
Zhang, P.; Morken, J. P.: Catalytic Enantioselective Allylation of Dienals
1357
Soltani, O.; Ariger, M. A.; Carreira, E. M.: Asymmetric Transfer Hydrogenation of Nitroalkenes
1358
Yaji, K.; Shindo, M.: Scandium-Catalyzed Stereoselective Nazarov Reaction
1359
Prévost, M.; Woerpel, K. A.: Diastereoselective Reaction of Silylene with Epoxides and Aldehydes
1360
Hermange, P.; Dau, M. E. T. H.; Retailleau, P.; Dodd, R. H.: Diastereoselective Three-Component Vinylogous Mannich Reaction
1361
Rankic, D. A.; Hopkins, J. M.; Parvez, M.; Keay, B. A.: Rhodium-Catalyzed Asymmetric Hydrogenation
1362
Saito, T.; Kikuchi, T.; Tanabe, H.; Yahiro, J.; Otani, T.: Stereoselective Construction of β-Lactams with Cu(II) Complexes
1363
Liu, X.-Y.; Che, C.-M.: Synthesis of Chiral Secondary Amines by Gold(I)-Chiral Brønsted Acid Catalysis
1364
Shibata, T.; Uchiyama, T.; Endo, K.: Rhodium-Catalyzed [2+2+2] Cycloaddition of Branched Triynes
1365
Suematsu, H.; Katsuki, T.: Enantioselective Aliphatic C-H Bond Functionalization
1366
Kliman, L. T.; Mlynarski, S. N.; Morken, J. P.: Platinum-Catalyzed Asymmetric Diboration of Terminal Alkenes
1367
Sibi, M. P.; Kawashima, K.; Stanley, L. M.: Kinetic Resolution of Pyrazolidinones by a Cu(II)-Catalyzed Diels-Alder Reaction
1368
Zhao, J.; Burgess, K.: Selective Syntheses of Vicinal Dimethyl Chirons by Hydrogenation
1369
Smith, A. J.; Abbott, L. K.; Martin, S. F.: Heteroaryl Titanates and Zinc Reagents in Enantioselective Conjugate Addition
1370
Matsumoto, K.; Oguma, T.; Katsuki, T.: Epoxidation of Styrenes Catalyzed by Titanium(Salan) Complexes
1371
Eloi, A.; Rose-Munch, F.; Rose, E.: Resolution of Arene-Manganese Complexes Using a Camphor Auxiliary
1372
Zhang, Y.-Z.; Zhu, S.-F.; Cai, Y.; Mao, H.-X.; Zhou, Q.-L.: Copper Bisoxazoline Catalyzed Enantioselective S-H Insertion
1373
Friestad, G. K.; Lee, H. J.: Titanium-Induced Ring Opening of a Strained Bicyclic Acetal
1374
Chen, J.; Lang, F.; Li, D.; Cun, L.; Zhu, J.; Deng, J.; Liao, J.: Pd-Catalyzed Allylic Alkylation and Amination Reactions with Sulfinylphosphines
1375
Cai, Q.; Zhao, Z.-A.; You, S.-L.: Asymmetric Construction of Polycyclic Indoles via Sequential Catalysis
1376
Shintani, R.; Tsutsumi, Y.; Nagaosa, M.; Nishimura, T.; Hayashi, T.: Synthesis of All-Carbon Quaternary Stereocenters
1377
Wang, X.-N.; Shao, P.-L.; Lv, H.; Ye, S.: NHC-Catalyzed Enantioselective Synthesis of β-Trifluoromethyl-β-lactones
1378
Hui, Y.; Zhang, Q.; Jiang, J.; Lin, L.; Liu, X.; Feng, X.: Scandium Catalyzed Friedel-Crafts Alkylation of Indoles
1379
Giampietro, N. C.; Kampf, J. W.; Wolfe, J. P.: Enantioselective Synthesis of α-Alkyl-α,β-dihydroxy Esters
1380
Shibata, Y.; Tanaka, K.: Rhodium-Catalyzed Hydroacylation of Alkenes with Aldehydes
1381
Kim, H. Y.; Shih, H.-J.; Knabe, W. E.; Oh, K.: Reversal of Enantioselectivity in the Synthesis of Pyrrolidines

Metal-Mediated Synthesis

z1383
All PDFs of this category
1383
Vechorkin, O.; Barmaz, D.; Proust, V.: Ni-Catalyzed Sonogashira Coupling of Nonactivated Alkyl Halides
1384
Metzger, A.; Melzig, L.; Despotopoulou, C.; Knochel, P.: Cross-Coupling of Organozinc Reagents with Thiomethylated Heterocycles
1385
Bhayana, B.; Fors, B. P.; Buchwald, S. L.: A Versatile Ligand for Suzuki-Miyaura Coupling of Tosylates and Mesylates
1386
Lapointe, D.; Fagnou, K.: Pd(II)-Catalyzed Direct Benzylation of Heteroarenes
1387
McNulty, J.; Das, P.: One-Pot Method for the Homologation of Aldehydes to Carboxylic Acids
1388
Fors, B. P.; Buchwald, S. L.: Palladium-Catalyzed Synthesis of Nitroarenes Using Sodium Nitrite
1389
Tobisu, M.; Hyodo, I.; Chatani, N.: Ni-Catalyzed Arylation of Arylzinc Reagents with N-Aromatic Heterocycles
1390
Bouffard, J.; Itami, K.: Nickel-Catalyzed Addition of Organo-boronates to Aldehydes and Ketones
1391
Nishikata, T.; Lipshutz, B. H.: Allylic Ethers as Educts for Aqueous Suzuki-Miyaura Couplings
1392
Ma, X.; Wang, J.-X.; Li, S.; Wang, K.-H.; Huang, D.: Zn-Cu Mediated Regioselective Addition of Propargyl Bromide to Carbonyls
1393
Berini, C.; Brayton, D. F.; Mocka, C.; Navarro, O.: (NHC)-Pd or -Ni-Catalyzed Oxidation of Secondary Alcohols by Chlorobenzene
1394
Ravikumar, P. C.; Yao, L.; Fleming, F. F.: NbCl5/NbBr5-Mediated Alkoxide Rearrangements to Allylic and Allenic Halides
1395
Ito, S.; Fujiwara, Y.-i.; Nakamura, E.; Nakamura, M.: Iron-Catalyzed Cross-Coupling of Alkyl Sulfonates with Arylzinc Reagents
1396
Wu, J. Y.; Moreau, B.; Ritter, T.: Fe-Catalyzed 1,4-Hydroboration of 1,3-Dienes

Organo- and Biocatalysis

z1397
All PDFs of this category
1397
Boeckmann Jr., R. K.; Miller, J. R.: Direct Hydroxymethylation Using Formaldehyde
1398
Guo, Q.-X.; Peng, Y.-G.; Zhang, J.-W.; Song, L.; Feng, Z.; Gong, L.-Z.: Brønsted Acid Catalyzed Alkylation of Enamides
1399
Nodes, W. J.; Nutt, D. R.; Chippindale, A. M.; Cobb, A. J. A.: Efficient Intramolecular Michael Addition of a Nitroalkane into a Conjugated Ester
1400
Zhang, Q.-W.; Fan, C.-A.; Zhang, H.-J.; Tu, Y.-Q.; Zhao, Y.-M.; Gu, P.; Chen, Z.-M.: Brønsted Acid Catalyzed Enantioselective Semipinacol Rearrangement
1401
Chen, Y.; Lie, F.; Li, Z.: Enantioselective Hydroxylations of Benzylic C-H Bonds Using Biocatalysis
1402
Luo, R.-S.; Weng, J.; Ai, H.-B.; Lu, G.; Chan, A. S. C.: Bicyclic Prolinol Silyl Ether Catalysts
1403
Zhang, E.; Fan, C.-A.; Tu, Y.-Q.; Zhang, F.-M.; Song, Y.-L.: Vinylogous α-Ketol Rearrangement
1404
Hirano, K.; Biju, A. T.; Piel, I.; Glorius, F.: NHC-Catalyzed Intramolecular Hydroacylation of Unactivated Double Bonds
1405
Ryan, S. J.; Candish, L.; Lupton, D. W.: NHC-Catalyzed Conjugate Addition Involving α,β-Unsaturated Acyl Azoliums
1406
Bew, S. P.; Fairhurst, S. A.; Hughes, D. L.; Legentil, L.; Liddle, J.; Pesce, P.; Nigudkar, S.; Wilson, M. A.: Fluoronium Organocatalysis
1407
Smith, S. W.; Fu, G. C.: Nucleophilic Addition γ to the Carbonyl Group
1408
Uraguchi, D.; Ueki, Y.; Ooi, T.: Supramolecular Chiral Organic Ion Pair Catalyst

Polymer-Supported Synthesis

z1409
All PDFs of this category
1409
Tanabe, K. K.; Cohen, S. M.: Mukaiyama Aldol Reaction Catalyzed by a MOF-Based Fe³+ Complex
1410
Molander, G. A.; Cavalcanti, L. N.; Canturk, B.; Pan, P.-S.; Kennedy, L. E.: Hydrolysis of Organotrifluoroborates with Silica Gel and Water
1411
Hagiwara, H.; Sekifuji, M.; Tsubokawa, N.; Hoshi, T.; Suzuki, T.: Knoevenagel Reaction Catalyzed by Dendrimeric Nano-Silica PAMAM
1412
Mitsudome, T.; Noujima, A.; Mizugaki, T.; Jitsukawa, K.; Kaneda, K.: Oxidation of Silanes with AuHAP in Water
1413
Swapna, K.; Kumar, A. V.; Reddy, V. P.; Rao, K. R.: C-N Cross-Coupling with Fe/Carbon Graphite
1414
Kitahara, H.; Kamiya, I.; Sakurai, H.: Au:PVP-Catalyzed Intramolecular Addition of Sulfonamide to Alkenes
1415
Oishi, T.; Katayama, T.; Yamaguchi, K.; Mizuno, N.: Alkyne-Alkyne Homocoupling with Cu(OH)X/TiO2
1416
Xu, J.-F.; Huang, X.: Solid-Phase Synthesis of 2-Pyridones, 1,4-Diazepines, and 1,4-Oxazepines
1417
Crich, D.; Sana, K.: Peptidyl Thioacid Synthesis with 9-Fluorenylmethyl Thiol-Linked Resin
1418
Yamada, Y. M. A.; Watanabe, T.; Torii, K.; Uozumi, Y.: Catalytic Membrane-Installed Microchannel Reactors for Allylic Arylation
1419
Osako, T.; Uozumi, Y.: Bipyridyl-Palladium Catalyst for Aerobic Oxidation of Alcohols
1420
Kim, J. Y.; Jo, Y.; Lee, S.; Choi, H. C.: Hydrodehalogenation of Aryl Halides with Pd-CNT Nanocomposites
1421
Kim, J. W.; He, J.; Yamaguchi, K.; Mizuno, N.: Synthesis of Aldimines from Alcohols and Amines with Ru(OH)x/TiO2