DOI: 10.1055/s-00000131

Synfacts

Issue 06 · Volume 2010 · June 2010 DOI: 10.1055/s-002-21046

Synform

A48
Zanda, Matteo: SYNFORM ISSUE 2010/06

Synthesis of Natural Products and Potential Drugs

z619
All PDFs of this category
0619
Hobson, L. A.; Parsons, R. L.: Synthesis of BMS-644950
0620
Campbell, E. L.; Zuhl, A. M.; Lui, C. M.; Boger, D. L.: Synthesis of (+)-Fendleridine and (+)-1-Acetylaspidoalbidine
0621
Xu, F.; Corley, E.; Zacuto, M.; Conlon, D. A.; Pipik, B.; Humphrey, G.; Murry, J.; Tschaen, D.: Synthesis of a Dipeptidyl Peptidase IV Inhibitor
0622
Mai, C.-K.; Sammons, M. F.; Sammakia, T.: Formal Synthesis of Diazonamide A
0623
Trost, B. M.; Osipov, M.; Dong, G.: Synthesis of (-)-Ranirestat
0624
Deng, X.; Liang, J. T.; Peterson, M.; Rynberg, R.; Cheung, E.; Mani, N. S.: Synthesis of a Cathepsin S Inhibitor
0625
Gemma, S.; Gabellieri, E.; Coccone, S. S.; Marti, F.; Taglialatela-Scafati, O.; Novellino, E.; Campiani, G.; Butini, S.: Synthesis of Dihydroplakortin
0626
Burke, C. P.; Haq, N.; Boger, D. L.: Synthesis of Phostriecin and Sultriecin
0627
Yoshinari, T.; Ohmori, K.; Schrems, M. G.; Pfaltz, A.; Suzuki, K.: Synthesis of (+)-Macrocidin A
0628
Smith, B. J.; Sulikowski, G. A.: Synthesis of (±)-Haliclonacyclamine
0629
Marchart, S.; Gromov, A.; Mulzer, J.: Synthesis of Branimycin

Synthesis of Heterocycles

z631
All PDFs of this category
0631
Yasmin, N.; Ray, J. K.: Efficient Heteroannulation Route for the Synthesis of Isoindoles and Pyrroles
0632
Lorion, M.; Agouridas, V.; Couture, A.; Deniau, E.; Grandclaudon, P.: Synthesis of Benzosultams from Cyclic Sulfamidates
0633
Ding, C.; Tu, S.; Yao, Q.; Li, F.; Wang, Y.; Hu, W.; Zhang, A.: Radical-Mediated Decarboxylative Route to Naphtho[2,3-a]carbazoles
0634
Guan, Z.-H.; Yan, Z.-Y.; Ren, Z.-H.; Liu, X.-Y.; Liang, Y.-M.: Synthesis of Indoles via Iron-Catalyzed Heteroannulative Oxidative Coupling
0635
Adib, M.; Ansari, S.; Feizi, S.; Bijanzadeh, H. R.: Multicomponent Synthesis of Triazoloquinazolines
0636
Cai, Q.; Li, Z.; Wei, J.; Fu, L.; Ha, C.; Pei, D.; Ding, K.: Copper-Catalyzed Synthesis of Aza-Fused Polycyclic Quinolines
0637
Lu, H.; Tao, J.; Jones, J. E.; Wojtas, L.; Zhang, X. P.: Synthesis of Cyclophosphoramidates by Intramolecular C-H Amination
0638
Kondoh, A.; Yorimitsu, H.; Oshima, K.: Palladium-Catalyzed Heteroannulation Route to 2-Indolylphosphines
0639
Zeng, F.; Alper, H.: Synthesis of 2-Heteroquinazolin-4-(3H)-ones via Palladium Catalysis
0640
Ye, L.; Cui, L.; Zhang, G.; Zhang, L.: Gold-Catalyzed Synthesis of Dihydrofuran-3-ones from Homopropargylic Alcohols
0641
Huo, Z.; Gridnev, I. D.; Yamamoto, Y.: Electrophile-Induced Cyclization of ortho-Azido Propynyl Benzenes to Quinolines
0642
Majumder, S.; Odom, A. L.: Pyrimidine Synthesis via a Titanium-Catalyzed Multicomponent Reaction
0643
Dubrovskiy, A. D.; Larock, R. C.: Synthesis of Benzisoxazoles by [3+2] Cycloaddition of Nitrile Oxides with Arynes
0644
Liu, Y.; Wang, M.; Yuan, H.; Liu, Q.: Copper(II) Bromide/BoronTrifluoride Cocatalyzed Synthesis of Benzofurans
0645
Liu, Y.; Qian, J.; Lou, S.; Zhu, J.; Xu, Z.: Gold(III)-Catalyzed Synthesis of 4H-Chromenes

Synthesis of Materials and Unnatural Products

z647
All PDFs of this category
0647
Miyagawa, N.; Watanabe, M.; Matsuyama, T.; Koyama, Y.; Moriuchi, T.; Hirao, T.; Furusho, Y.; Takata, T.: Rotaxane Structure Specific Palladium-Catalyzed Rearrangement
0648
Zhen, Y.; Wang, C.; Wang, Z.: Preparation of N-Type Graphitic Nanoribbons
0649
Shinozaki, S.; Hamura, T.; Ibusuki, Y.; Fujii, K.; Uekusa, H.; Suzuki, K.: Radialene Synthesis
0650
Huang, X.-h.; Lu, Y.; He, Y.-b.; Chen, Z.-h.: Phosphate Ion Sensing in an Aqueous Environment
0651
Uoyama, H.; Kim, K. S.; Kuroki, K.; Shin, J.-Y.; Nagata, T.; Okujima, T.; Yamada, H.; Ono, N.; Kim, D.; Uno, H.: Cruciform Porphyrin Pentamers
0652
Zhang, X.; Fan, S.; He, C.-Y.; Wan, X.; Min, Q.-Q.; Yang, J.; Jiang, Z.-X.: Olefination of Perfluoroarenes
0653
Kooistra, F. B.; Leuning, T. M.; Martinez, E. M.; Hummelen, J. C.: Conjugated Fullerenes
0654
Ehm, C.; Lentz, D.: A Hyper-Reactive Tetrafluorinated Cumulene
0655
Rogness, D. C.; Larock, R. C.: Gentle One-Step Synthesis of Acridines
0656
Kryger, M. J.; Ong, M. T.; Odom, S. A.; Sottos, N. R.; White, S. R.; Martinez, T. J.; Moore, J. S.: You Break It, You Fix It
0657
Hiraoka, H.; Hisanaga, Y.; Shiro, M.; Shionoya, M.: Assembly with a New Twist
0658
Uehara, K.; Wagner, C. B.; Vogler, T.; Luftmann, H.; Studer, A.: Boron Group Transfer Polymerization
0659
Crawford, S. M.; Thompson, A.: De-Boronation of BODIPY
0660
Dong, D.-J.; Li, H.-H.; Tian, S.-K.: Stereoselective Olefination
0661
Chen, W.-C.; Lee, Y.-W.; Chen, C.-T.: Dual-Mode Switching

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z663
All PDFs of this category
0663
Mukherjee, P.; Widenhoefer, R. A.: Gold-Catalyzed γ-Selective Amination of Allylic Alcohols
0664
Yoshida, S.; Fukui, K.; Kikuchi, S.; Yamada, T.: Silver-Catalyzed Desymmetrization via Carbon Dioxide Incorporation
0665
Oura, I.; Shimizu, K.; Ogata, K.; Fukuzawa, S.-i.: Azomethine Ylide Cycloadditions with ThioClickFerrophos Ligands
0666
Martín-Rodríguez, M.; Nájera, C.; Sansano, J. M.; Costa, P. R. R.; de Lima, E. C.; Dias, A. G.: Enantioselective 1,3-Dipolar Cycloaddition of Azomethine Ylides and Alkenes
0667
Lang, F.; Li, D.; Chen, J.; Li, L.; Cun, L.; Zhu, J.; Deng, J.; Liao, J.: New Ligands for Rhodium-Catalyzed Asymmetric 1,4-Additions
0668
Chen, W.-W.; Zhao, Q.; Xu, M.-H.; Lin, G.-Q.: Asymmetric Ullmann Coupling of Biaryl Dials Catalyzed by Nickel
0669
Bechem, B.; Patman, R. L.; Hashmi, A. S. K.; Krische, M. J.: Asymmetric Allylation, Crotylation, and tert-Prenylation of Furan Methanols and Furfurals
0670
Schotes, C.; Mezzetti, A.: Ruthenium-Catalyzed Enantioselective Diels-Alder Reaction of β-Keto Esters
0671
Li, Q.; Jiang, G.-J.; Jiao, L.; Yu, Z.-X.: Rhodium(I)-Catalyzed Intramolecular [3+2] Cycloaddition of α-Ene-Vinylcyclopropanes
0672
Sharma, R. K.; RajanBabu, T. V.: Asymmetric Hydrovinylation of 1,3-Dienes
0673
Kalow, J. A.; Doyle, A. G.: Asymmetric Synthesis of Fluorohydrins
0674
Lv, J.; Li, X.; Zhong, L.; Luo, S.; Cheng, J.-P.: Binary Acid Catalysis in Enantioselective Friedel-Crafts Reactions
0675
Tang, W.; Capacci, A. G.; White, A.; Ma, S.; Rodriguez, S.; Qu, B.; Savoie, J.; Patel, N. D.; Wei, X.; Haddad, N.; Grinberg, N.; Yee, N. K.; Krishnamurthy, D.; Senanayake, C. H.: Chiral Biphosphorous Ligands for Rhodium-Catalyzed Asymmetric Hydrogenation
0676
Zupančič, B.; Mohar, B.; Stephan, M.: P-Stereogenic Diphosphine Ligands for Asymmetric Hydrogenation
0677
Ward, A. F.; Wolfe, J. P.: Synthesis of Tetrahydrofurans by Diastereoselective Carboetherification
0678
Reddy, V. J.; Douglas, C. J.: Palladium-Catalyzed Asymmetric Intramolecular Cyanoamidation
0679
Endo, K.; Ogawa, M.; Shibata, T.: Catalytic Asymmetric Conjugate Addition of Organozinc Reagents
0680
Hu, X.; Cao, Z.; Liu, Z.; Wang, Y.; Du, H.: Synthesis and Applications of Acyclic Chiral Diene Ligands
0681
Hashimoto, T.; Maeda, Y.; Omote, M.; Nakatsu, H.; Maruoka, K.: Enantioselective 1,3-Dipolar Cycloaddition of Azomethine Imines
0682
Pigza, J. A.; Molinski, T. F.: A Concise Synthesis of (S)-β-Methylisoleucine
0683
Donohoe, T. J.; Lindsay-Scott, P. J.; Parker, J. S.; Callens, C. K. A.: Synthesis of Pyrrolidines by Osmium-Catalyzed Oxidative Cyclization
0684
Huang, Y.; Tokunage, E.; Suzuki, S.; Shiro, M.; Shibata, N.: Zinc-Catalyzed Enantioselective Friedel-Crafts Alkylation
0685
Streuff, J.; White, D. E.; Virgil, S. C.; Stoltz, B. M.: Palladium-Catalyzed Asymmetric Alkylation of β-Keto Esters
0686
Hata, T.; Bannai, R.; Otsuki, M.; Urabe, H.: Iron(II)-Catalyzed Selective Grignard Addition to Vinyl Oxiranes
0687
Li, Q.; Ding, C.-H.; Hou, X.-L.; Dai, L.-X.: Copper-Catalyzed Asymmetric Michael Reaction of Glycines to Nitroalkenes
0688
Wang, J.; Li, W.; Liu, Y.; Chu, Y.; Lin, L.; Liu, X.; Feng, X.: Enantioselective Conjugate Addition of Cyanide
0689
Ito, T.; Overman, L. E.; Wang, J.: Dynamic Kinetic Resolution via Aza-Cope Rearrangement
0690
Teller, H.; Flügge, S.; Goddard, R.; Fürstner, A.: Phosphoramidite Ligands with an Acyclic TADDOL Backbone for Gold Catalysis
0691
Zhu, Y.; Zhai, C.; Yang, L.; Hu, W.: Copper-Catalyzed Three-Component Reactions: Access to Furan Derivatives
0692
Shepherd, N. E.; Tanabe, H.; Xu, Y.; Matsunaga, S.; Shibasaki, M.: Nickel-Catalyzed Vinylogous Mannich and Michael Reactions

Metal-Mediated Synthesis

z693
All PDFs of this category
0693
Wasa, M.; Engle, K. M.; Yu, J.-Q.: Amide-Directed Olefination of sp³ C-H Bonds
0694
Ackermann, L.; Barfüsser, S.; Pospech, J.: Direct C-H Functionalization of Oxazoles Using Sulfamates and Phosphates
0695
Huang, J.; Chan, J.; Chen, Y.; Borths, C. J.; Baucom, K. D.; Larsen, R. D.; Faul, M. M.: A Highly Efficient Cocatalytic System for Direct Arylation of Heteroarenes
0696
Anbarasan, first article: P.; Neumann, H.; Beller, M.; Yamada, second article: S.; Gavryushin, A.; Knochel, P.: Two Expedient Protocols for the Electrophilic Fluorination of Grignard Reagents
0697
Yao, M.-L.; Reddy, M. Srinivasa; Yong, L.; Walfish, I.; Blevins, D. W.; Kabalka, G. W.: Chemoselective Bromodeboronation of Organotrifluoroborates
0698
Kim, S.-H.; Rieke, R. D.: 2-Pyridyl- and 3-Pyridylzincs: Direct Preparation and Coupling Reaction
0699
Zhang, F.; Greaney, M. F.: Decarboxylative C-H Cross-Coupling of Azoles
0700
Han, X.; Zhang, Y.; Wu, J.: Two-Step Transition-Metal-Free Allylation of Grignard Reagents
0701
Chen, M.; Zheng, X.; Li, W.; He, J.; Lei, A.: Palladium-Catalyzed Aerobic Cross-Coupling of Alkylzincs to Terminal Alkynes
0702
Schneider, C. C.; Caldeira, H.; Gay, B. M.; Back, D. F.; Zeni, G.: Transmetalation of (Z)-Telluroenynes: Stereoselective Synthesis of (Z)-Enynols
0703
Yan, G.; Kuang, C.; Zhang, Y.; Wang, J.: Palladium-Catalyzed Direct Cyanation of Indoles with K4[Fe(CN)6]
0704
Zhou, Y.; Lecourt, T.; Micouin, L.: 1,4-Disubstituted 5-Alumino-1,2,3-triazoles from Aluminum Acetylides and Azides
0705
Blümke, T.; Chen, Y.-H.; Peng, Z.; Knochel, P.: Direct Insertion of Aluminum to Functionalized Unsaturated Halides
0706
Wu, H.; Hynes, J.: Copper-Catalyzed Chlorination of Arylboronic Acids
0707
Tan, Y.; Hartwig, J. F.: Direct Amination of Aromatic C-H Bonds Using Oxime Esters

Organo- and Biocatalysis

z709
All PDFs of this category
0709
Rendler, first article: S.; MacMillan, D. W. C.; Knowles, second article: R. R.; Lin, S.; Jacobsen, E. N.: Organocatalytic Carbocyclizations
0710
Holub, N.; Jiang, H.; Paixão, M. W.; Tiberi, C.; Jørgensen, K. A.: Asymmetric Synthesis of Bicyclo[2.2.2]oct-5-en-2-one by Using Organocatalysis
0711
Li, G.; Kaplan, M. J.; Wojtas, L.; Antilla, J. C.: TRIP-Catalyzed Asymmetric Addition of Dihydropyrans to N-Acyl Imines
0712
Takenaka, N.; Chen, J.; Captain, B.; Sarangthem, R. S.; Chandrakumar, A.: A Novel Hydrogen-Bonding Catalyst Class with Helical Chirality
0713
Li, D. R.; He, A.; Falck, J. R.: Enantioselective Reduction of Ketones - A New Alternative to the CBS Reduction?
0714
Lu, A.; Wu, R.; Wang, Y.; Zhou, Z.; Wu, G.; Fang, J.; Tang, C.: Asymmetric Michael Reaction Catalyzed by Chiral Thiophosphoramidate
0715
Hua, M.-Q.; Cui, H.-F.; Wang, L.; Nie, J.; Ma, J.-A.: Tuning the Conformational Flexibility of Catalysts
0716
Biju, A. T.; Wurz, N. E.; Glorius, F.: NHC-Catalyzed Hydroacylation of Unreactive Alkynes
0717
Jin, T.; Himuro, M.; Yamamoto, Y.: Brønsted Acid Catalyzed Cascade Cyclization of Enynes
0718
Albert, B. J.; Yamamoto, H.: Lewis Acid Assisted Triple-Aldol Cascades
0719
Sun, J.; Fu, G. C.: Phosphine-Catalyzed Carbon-Sulfur Bond Formation
0720
Mondal, M.; Ibrahim, A. A.; Wheeler, K. A.; Kerrigan, N. J.: BINAPHANE-Catalyzed Asymmetric Formal [2+2] Cycloaddition

Polymer-Supported Synthesis

z721
All PDFs of this category
0721
Dey, R.; Sreedhar, B.; Ranu, B. C.: Suzuki Coupling with Molecular Sieves Supported Palladium Catalyst
0722
Ando, K.; Suzuki, Y.: HWE Reaction with Polymer-Supported Phosphonate Reagents
0723
Goren, K.; Portnoy, M.: N-Alkylimidazole-Decorated Dendritic Catalysts for Baylis-Hillman Reaction
0724
Hagiwara, H.; Kuroda, T.; Hoshi, T.; Suzuki, T.: Diels-Alder Reaction with SiO2-Supported MacMillan Catalyst
0725
Sreedhar, B.; Kumar, A. S.; Reddy, P. S.: Synthesis of Propargylamines with Fe3O4 Nanoparticles
0726
Salvadori, J.; Balducci, E.; Zaza, S.; Petricci, E.; Taddei, M.: Microwave-Assisted Carbonylation of Aryl Iodides with Pd/C
0727
Zhou, S.; Johnson, M.; Veinot, J. G. C.: Fe@FexOy/Pd for Suzuki-Miyaura Cross-Coupling
0728
Dhakshinamoorthy, A.; Alvaro, M.; Garcia, H.: Claisen-Schmidt Condensation Catalyzed by MOF Composites
0729
Duplais, C.; Forman, A. J.; Baker, B. A.; Lipshutz, B. H.: Sonogashira Coupling with UC Pd under Copper-Free Conditions
0730
Motoyama, Y.; Kamo, K.; Yuasa, A.; Nagashima, H.: Atom-Transfer Radical Cyclization with [Cu/bipy]@Si
0731
Bacsa, B.; Bősze, S.; Kappe, C. O.: Direct Solid-Phase Synthesis of the β-Amyloid (1-42) Peptide
0732
Tsukamoto, D.; Shiraishi, Y.; Hirai, T.: Mg(II)/Zeolite Y Assisted Photoreaction of Olefins with Acetone
0733
Roche, D.; Lardy, C.; Tournier, L.; Prunier, M.; Valeur, E.: A Polymer-Supported Nitrosation Reagent of Amines
0734
El Kadib, A.; Molvinger, K.; Bousmina, M.; Brunel, D.: Chitosan/Titania-Promoted Carbon-Carbon Bond Forming Reactions