DOI: 10.1055/s-00000131

Synfacts

Issue 04 · Volume 2011 · April 2011 DOI: 10.1055/s-002-21773

Synform

A28
Zanda, Matteo: SYNFORM ISSUE 2011/04

Synthesis of Natural Products and Potential Drugs

z349
All PDFs of this category
0349
Lau, S. Y. W.: Syntheses of (±)-Hamigeran B and (±)-4-Bromohamigeran B
0350
Humphrey, G. R.; Pye, P. J.; Zhong et al., Y.-L.: Synthesis of the HIV Integrase Inhibitor Raltegravir Potassium
0351
Taylor, B. L. H.; Swift, E. C.; Waetzig, J. D.; Jarvo, E. R.: Asymmetric Synthesis of 1,1-Diarylethane Drugs
0352
Wang, B.; Ramirez, A. P.; Slade, J. J.; Morken, J. P.: Synthesis of (-)-Sclerophytin A
0353
Nishimura, T.; Unni, A. K.; Yokoshima, S.; Fukuyama, T.: Synthesis of (+)-Lyconadin A
0354
Graham, J. P.; Langlade, N.; Northall, J. M.; Roberts, A. J.; Whitehead, A. J.: Synthesis of Glycine Transporter Inhibitor GSK2137305
0355
Deschamps, N. M.; Elitzin, V. I.; Liu, B.; Mitchell, M. B.; Sharp, M. J.; Tabet, E. A.: Synthesis of Triple Reuptake Inhibitor GSK1360707F
0356
Zhang, Z.; Chen, J.; Yang, Z.; Tang, Y.: Biomimetic Synthesis of (±)-Rossinone B
0357
Ding, H.; Chen, D. Y.-K.: Formal Synthesis of (-)- and (+)-Phalarine
0358
Narjes et al., F.: Synthesis of MK-3281
0359
Clark, J. S.; Berger, R.; Hayes, S. T.; Thomas, L. H.; Morrison, A. J.; Gobbi, L.: Synthesis of Three of the Cladiellins
0360
Milburn et al., R. R.: Synthesis of a p38 MAP Kinase Inhibitor
0361
Gu, Z.; Zakarian, A.: Synthesis of Sintokamides A, B and E

Synthesis of Heterocycles

z363
All PDFs of this category
0363
Balamurugan, K.; Jeyachandran, V.; Perumal, S.; Menéndez, J. C.: One-Pot Synthesis of Tetrahydroisoquinolines via Benzene Ring Annulation
0364
Trost, B. M.; Lumb, J.-P.; Azzarelli, J. M.: Palladium-Catalyzed Atom-Economical Synthesis of Pyrroles
0365
Rai, A.; Singh, A. K.; Singh, S.; Yadav, L. D. S.: Organocatalytic Cascade Synthesis of Decahydroquinolines
0366
Cież, D.; Svetlik, J.: Synthesis of Imidazolin-5-ones by Thermolysis of α-Azido Esters
0367
Lei, Y.; Wang, Z.-Q.; Xie, Y.-X.; Yu, S.-C.; Tang, B.-X.; Li, J.-H.: Base-Mediated Synthesis of 4,5-Disub-stituted Furan-2(5H)-ones
0368
Yu, X.; Pan, X.; Wu, J.: Synthesis of Pyrazoloisoquinolines via a Multicomponent Suzuki Reaction Sequence
0369
Attanasi, O. A.; De Crescentini, L.; Favi, G.; Nicolini, S.; Perrulli, F. R.; Santeusanio, S.: Synthesis of 1,3,5-Trisubstituted Hydantoin via a Three-Component Reaction
0370
Světík, J.; Kettmann, V.: Unexpected Products from the Biginelli Reactions of 3-Amino-1,2,4-triazole
0371
Liang, F.; Lin, S.; Wei, Y.: Synthesis of Furo[3,2-c]pyridinones via an Aza-Oxy-Carbanion Relay Strategy
0372
D’Souza, A. M.; Spiccia, N.; Basutto, J.; Jokisz, P.; Wong, L. S.-M.; Meyer, A. G.; Holmes, A. B.; White, J. M.; Ryan, J. H.: 1,3-Dipolar Cycloaddition Route to 1,3-Benzodiazepinones
0373
Kumar, P. M.; Kumar, K. S.; Poreddy, S. R.; Mohakhud, P. K.; Mukkanti, K.; Pal, M.: Extending the Scope of the Biginelli Reaction Using Palladium Catalysis
0374
Gainer, M. J.; Bennett, N. R.; Takahashi, Y.; Looper, R. E.: Rhodium(II)-Catalyzed Hydroamination of Propargylguanidines
0375
Dell’Acqua, M.; Facoetti, D.; Abbiati, G.; Rossi, E.: Sonogashira-Heteroannulative Route to Dihydroisobenzofurans
0376
Wang, W.; Ollio, S.; Herdtweck, E.; Dömling, A.: Combined Ugi-Pictet-Spengler Synthesis of Polycyclic Ketopiperazines
0377
Jen, T.; Mendelsohn, B. A.; Ciufolini, M. A.: Oxidative Approach to Isoxazolines

Synthesis of Materials and Unnatural Products

z379
All PDFs of this category
0379
Jiao, C.; Huang, K.-W.; Chi, C.; Wu, J.: Donor-Acceptor Type Fused Porphyrin-Perylene Monoimides
0380
Venkataramani, S.; Jana, U.; Dommaschk, M.; Sönnichsen, F. D.; Tuczek, F.; Herges, R.: Lights, Magnets, Action!
0381
Rong, L.; Liu, Q.; Shi, Y.; Tang, J.: New 7b-Arylfluoradenes
0382
Gramage-Doria, R.; Armspach, D.; Matt, D.; Toupet, L.: A Chelating Diphosphane Ligand on a β-Cyclodextrin Backbone
0383
Frensch, L. K.; Pröpper, K.; John, M.; Demeshko, S.; Brückner, C.; Meyer, F.: Twist with Twin Porphyrin
0384
Wang, F.; Zhang, W.; Zhu, J.; Li, H.; Huang, K.-W.; Hu, J.: New Precursor for Difluorocarbenes
0385
Liu, J.; Lam, J. W. Y.; Jim, C. K. W.; Ng, J. C. Y.; Shi, J.; Su, H.; Yeung, K. F.; Hong, Y.; Faisal, M.; Yu, Y.; Wong, K. S.; Tang, B. Z.: Click it!
0386
Li, H.; Liu, J.; Sun, C.-L.; Li, B.-J.; Shi, Z.-J.: Cross-Coupling Made Easy
0387
Birsa, M. L.; Jones, P. G.; Hopf, H.: [2,2]Paracyclophanes with New Bridges
0388
Fukumoto, S.; Nakashima, T.; Kawai, T.: Photon-Quantitative Cyclization of Dithiazolylarylene
0389
Auzias, M.; Häussinger, D.; Neuburger, M.; Wegner, H. A.: Photoinduced Rearrangements of 3,3′-Bis(arylbenzofurans)
0390
Davis, N. K. S.; Thompson, A. L.; Anderson, H. L.: Extended Porphyrins
0391
Bojase, G.; Nguyen, T. V.; Payne, A. D.; Willis, A. C.; Sherburn, M. S.: Ivyanes from Dendralenes

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z393
All PDFs of this category
0393
Waibel, M.; Cramer, N.: Rhodium(I)-Catalyzed Asymmetric Desymmetrization by Retro-Allylation
0394
Drouet, F.; Lalli, C.; Liu, H.; Masson, G.; Zhu, J.: Calcium-Catalyzed Enantioselective Electrophilic Amination of Enamides
0395
May, T. L.; Dabrowski, J. A.; Hoveyda, A. H.: Enantioselective Conjugated Addition of Vinylaluminums to Cyclic Enones
0396
Clavier, H.; Jeune, K. Le; de Riggi, I.; Tenaglia, A.; Buono, G.: [6+2] Cycloadditions between Cyclohepta-triene and Allenes
0397
Garayalde, D.; Krüger, K.; Nevado, C.: Gold-Catalyzed Cyclopenta- and Cyclo-heptannulation
0398
Tenaglia, A.; Jeune, K. Le; Giordano, L.; Buono, G.: Palladium-Catalyzed Synthesis of Alkynylcyclopropanes
0399
DeAngelis, A.; Shurtleff, V. W.; Dmitrenko, O.; Fox, J. M.: Rhodium(II)-Catalyzed Enantioselective C-H Functionalization of Indoles
0400
Murai, M.; Hatano, R.; Kitabata, S.; Ohe, K.: Regio- and Stereoselective Bromocyanation of Alkynes
0401
Daka, P.; Xu, Z.; Alexa, A.; Wang, H.: Direct Aldol Reaction Catalyzed by a Chiral Bifunctional Catalyst System
0402
Mazet, C.; Gérard, D.: Catalytic Asymmetric Hydroboration of α-Substituted Styrenyl Derivatives
0403
Rueping, M.; Koenigs, R. M.: Brønsted Acid Differentiated Metal Catalysis by Kinetic Discrimination
0404
Lee, J. Y.; You, Y. S.; Kang, S. H.: Desymmetrization of 2,2-Disubstituted
1,3-Propanediols
0405
Geng, H.; Huang, K.; Sun, T.; Li, W.; Zhang, X.; Zhou, L.; Wu, W.: Asymmetric Rhodium-Catalyzed Hydrogenation of β-Amino Ketones
0406
Yang, G.; Shen, Y.; Li, K.; Sun, Y.; Hua, Y.: Highly Regio- and Diastereoselective [3+2] Cycloadditions
0407
Sladojevich, F.; Trabocchi, A.; Guarna, A.; Dixon, D. J.: Cinchona-Derived Amino Phosphine Precatalysts for Cooperative Catalysis
0408
Cambeiro, X. C.; Pericàs, M. A.: Chiral Aminotriazole Ligands in Ruthenium-Catalyzed Transfer Hydrogenation
0409
Ratjen, L.; García-García, P.; Lay, F.; Beck, M. E.; List, B.: Catalytic Asymmetric Vinylogous and Bisvinylogous Aldol Reactions
0410
Fujisaki, J.; Matsumoto, K.; Katsuki, T.: Highly Selective Aluminum-Catalyzed Oxidation of Cyclic Dithioacetals
0411
Yang, Z.; Wang, Z.; Bai, S.; Liu, X.; Lin, L.; Feng, X.: Enantioselective Addition of Pyrazolones to Dialkyl Azodicarboxylates
0412
Antczak, M. I.; Cai, F.; Ready, J. M.: Chiral Auxiliary Controlled Asymmetric Synthesis of Tertiary Alcohols
0413
Zhao, J.-F.; Tan, B.-H.; Loh, T.-P.: Enantioselective Mukaiyama Aldol Reactions with Glyoxylates
0414
Junge, K.; Wendt, B.; Addis, D.; Zhou, S.; Das, S.; Fleischer, S.; Beller, M.: Asymmetric Ketone Hydrogenation Catalyzed by Copper-Phosphine Complexes
0415
Zhou, X.-Y.; Bao, M.; Zhou, Y.-G.: Brønsted Acid Activated Palladium-Catalyzed Hydrogenation of Ketimines
0416
Jiao, Y.; Cao, C.; Zhou, Z.: Synthesis of 1,3-Diols through Grignard Addition to Isopropenyl Acetate
0417
Aikawa, K.; Mimura, S.; Numata, Y.; Mikami, K.: Asymmetric Ene and Aldol Reactions of Isatins, Diketones, and Keto Esters
0418
Vincent, G.; Guillot, R.; Kouklovsky, C.: Sequential Addition of Nucleophiles to Bicyclic Isoxazololactams
0419
Teichert, J. F.; Fañanás-Mastral, M.; Feringa, B. L.: Iridium-Catalyzed Asymmetric Intramolecular Allylic Amidation
0420
Chen, F.; Wang, T.; He, Y.; Ding, Z.; Li, Z.; Xu, L.; Fan, Q.-H.; Xu, M.-H.: Asymmetric Hydrogenation of Ketimines

Metal-Mediated Synthesis

z421
All PDFs of this category
0421
Miyasaka, M.; Hirano, K.; Satoh, T.; Kowalczyk, R.; Holm, C.; Miura, M.: Copper-Catalyzed Direct Sulfoximination
0422
Lin, B.; Wu, Z.-H.; Gu, Y.-F.; Sun, C.-L.; Wang, B.-Q.; Shi, Z.-J.: Co-Catalyzed Cross-Coupling of C-H Bonds with Grignard Reagents
0423
Tsai, A. S.; Brasse, M.; Bergman, R. G.; Ellman, J. A.: Rh(III)-Catalyzed C-H Activation and Oxidative Coupling with Alkenes
0424
Jithunsa, M.; Ueda, M.; Miyata, O.: CuCl2-Mediated Cyclization of N-Alkoxy-ortho-alkynylbenzamides
0425
Pintori, D. G.; Greaney, M. F.: Pd-Catalyzed Oxidative Intramolecular C-H Coupling for Medium-Ring Synthesis
0426
Cao, J.; Yang, X.; Hua, X.; Deng, Y.; Lai, G.: Polysequential Synthesis of 2-Azaanthra-cenes from Ethynylbenzenes
0427
Wang, Z.-Q.; Lei, Y.; Zhou, M.-B.; Chen, G.-X.; Song, R.-J.; Xie, Y.-X.; Li, J.-H.: Iron-Mediated Tandem Annulation for the Synthesis of Various Chromenes
0428
Miyoshi, T.; Miyakawa, T.; Ueda, M.; Miyata, O.: Polarity Inversion of Ketones: Umpolung Reaction at the α-Position
0429
Wang, G.-W.; Yuan, T.-T.; Li, D.-D.: Palladium-Catalyzed One-Pot C-C and C-N Bond Formation by Dual C-H Activation
0430
Beng, T. K.; Gawley, R. E.: Asymmetric Synthesis of 2-Aryl and 2-Vinyl Piperidines by Dynamic Resolution
0431
Xiao, Q.; Xia, Y.; Li, H.; Zhang, Y.; Wang, J.: Copper(I)-Catalyzed Coupling of N-Tosyl-hydrazones with Terminal Alkynes
0432
Barluenga, J.; Florentino, L.; Aznar, F.; Valdés, C.: Palladium-Catalyzed Cross-Coupling of Tosylhydrazones and Aryl Nonaflates
0433
Chen, Q.; Ilies, L.; Nakamura, E.: Cobalt-Catalyzed ortho-Alkylation through Directed C-H Bond Activation
0434
Selander, N.; Paasch, J. R.; Szabó, K. J.: Palladium-Catalyzed Synthesis of Functionalized Allylsilanes and Allylboronates

Organo- and Biocatalysis

z435
All PDFs of this category
0435
Schrittwieser, J. H.; Resch, V.; Sattler, J. H.; Lienhart, W.-D.; Durchschein, K.; Winkler, A.; Gruber, K.; Macheroux, P.; Kroutil, W.: Biocatalytic Formation of C-C Bonds
0436
Belmessieri, D.; Morrill, L. C.; Simal, C.; Slawin, A. M. Z.; Smith, A. D.: Asymmetric Michael Addition-Lactonization of Carboxylic Acids
0437
Cohen, D. T.; Cardinal-David, B.; Scheidt, K. A.: NHC-Catalyzed Addition of Homoenolate Equivalents to Unsaturated Keto Esters
0438
Kwiatkowski, P.; Beeson, T. D.; Conrad, J. C.; MacMillan, D. W. C.: Asymmetric α-Fluorination of Cyclic Ketones
0439
So, S. S.; Burkett, J. A.; Mattson, A. E.: Internal Lewis Acid Activation of Ureas
0440
Haibach, M. C.; Deb, I.; De, C. K.; Seidel, D.: Indole Annulation via an Internal Redox Cascade
0441
Hayashi, M.; Nakamura, S.: Enantioselective Protonation by Cinchona Alkaloids via Phospha-Brook Rearrangement
0442
Han, X.; Wang, Y.; Zhong, F.; Lu, Y.: Dipeptide-Based Phosphine Catalyst for Cycloaddition of Allenes to Acrylates
0443
Fang, X.; Jiang, K.; Xing, C.; Hao, L.; Chi, Y. R.: A Cascade Annulation of Enals and Dienones
0444
Sakakura, A.; Ohkubo, T.; Yamashita, R.; Akakura, M.; Ishihara, K.: Dehydrative Condensation of Dicarboxylic Acids with Aminoboronic Acids
0445
Luo, J.; Wang, H.; Han, X.; Xu, L.-W.; Kwiatkowski, J.; Huang, K.-W.; Lu, Y.: Asymmetric Vinylogous Aldol Reactions of Furanones and α-Keto Esters
0446
Jousseaume, T.; Wurz, N. E.; Glorius, F.: NHC-Catalyzed Intermolecular Stetter Reaction with Asymmetric Protonation
0447
Brazier, J. B.; Jones, K. M.; Platts, J. A.; Tomkinson, N. C. O.: Solvent-Dependance in Organocatalyzed Diels-Alder Reactions

Polymer-Supported Synthesis

z449
All PDFs of this category
0449
Bogdan, A. R.; James, K.: Flow Macrocyclization Using Copper Tubing
0450
Firouzabadi, H.; Iranpoor, N.; Ghaderi, A.; Ghavami, M.; Hoseini, S. J.: Heck and Suzuki Reactions Using Supported Palladium Nanoparticles
0451
Cui, X.; Zhang, Y.; Shi, F.; Deng, Y.: Alkylation with Alcohols Catalyzed by Ag/Mo Hybrid Metal
0452
Verma, S.; Jain, S. L.; Sain, B.: Synthesis of Dihydropyrimidinones with PEG-Supported Thiourea Dioxide
0453
Motoyama, Y.; Nishikata, T.; Nagashima, H.: Asymmetric Cyclopropanation with [Cu(OTf)2(t-Bu2-DABox)][Pt]@Si
0454
Massi, A.; Cavazzini, A.; De Zoppo, L.; Pandoli, O.; Costa, V.; Pasti, L.; Giovannini, P. P.: Aldol and α-Amination Reactions with Proline-Functionalized Reactors
0455
Chen, J. M.; Zeng, X. M.; Zhdankin, V. V.: Polystyrene-Supported Iodosylbenzene Sulfate as an Oxidizing Agent
0456
Lubinu, M. C.; De Luca, L.; Giacomelli, G.; Porcheddu, A.: Mono-N-Alkylation of Anilines with R3N Using Pd/C under Microwave Irradiation
0457
Chan-Thaw, C. E.; Villa, A.; Prati, L.; Thomas, A.: Triazine-Based Polymer/Nano-Pd: Oxidation of Alcohols
0458
Qureshi, Z. S.; Deshmukh, K. M.; Tambade, P. J.; Bhanage, B. M.: Carbonylative Suzuki-Miyaura Coupling Using PS-Pd-NHC
0459
Keivanloo, A.; Bakherad, M.; Bahramian, B.; Rahmani, M.; Taheri, S. A. N.: Synthesis of α,β-Acetylenic Ketones with Polystyrene-Supported ZnBr2
0460
Li, J.; Cao, J.-j.; Wei, J.-f.; Shi, X.-y.; Zhang, L.-h.; Feng, J.-j.; Chen, Z.-g.: A Silica-Supported Imidazolium Salt for Nucleophilic Substitution in Water