DOI: 10.1055/s-00000131

Synfacts

Issue 03 · Volume 2010 · March 2010 DOI: 10.1055/s-002-20807

Editorial

I
editorial

Synform

A22
Zanda, Matteo: SYNFORM ISSUE 2010/03

Synthesis of Natural Products and Potential Drugs

z253
All PDFs of this category
0253
Guercio, G.; Bacchi et al., S.: Synthesis of the NK1 Receptor Antagonist GW597599
0254
Sato, S.; Shibuya, M.; Katoh, N.; Iwabuchi, Y.: Synthesis of the Gastrin/CCK-B Receptor Antagonist (+)-AG-041R
0255
Magnus, P.; Sane, N.; Fauber, B. P.; Lynch, V.: Synthesis of (-)-Galanthamine and (±)-Codeine
0256
Alimardanov et al., A.: Synthesis of a 3-Aryl-3-trifluoromethyl-2-aminopropanol Derivative
0257
Fu, R.; Zhao, B.; Shi, Y.: Synthesis of Substance P Receptor Antagonist (+)-CP-99,994
0258
Yoo, K.; Kim, H.; Yun, J.: Formal Synthesis of (+)-Indatraline
0259
Maimone, T. J.; Shi, J.; Ashida, S.; Baran, P. S.: Synthesis of Vinigrol
0260
Schmidt, Y.; Breit, B.: Synthesis of Vittatalactone
0261
Stang, E. M.; White, M. C.: Synthesis of 6-Deoxyerythronolide B
0262
Willot, M.; Radtke, L.; Könning, D.; Fröhlich, R.; Gessner, V. H.; Strohmann, C.; Christmann, M.: Synthesis of Engerlin A
0263
Garfunkle, J.; Kimball, F. S.; Trzupek, J. D.; Takizawa, S.; Shimamura, H.; Tomishima, [nl]M.; Boger, D. L.: Synthesis of Chloropeptin II
0264
Baschieri, A.; Bernardi, L.; Ricci, A.; Suresh, S.; Adamo, M. F. A.: Synthesis of (R)-(-)-Baclofen
0265
Carey et al., J. S.: Synthesis of a Glycine Antagonist
0266
Topczewski, J. J.; Callahan, M. P.; Neighbors, J. D.; Wiemer, D. F.: Synthesis of (+)-Angelichalcone
0267
Ohta, C.; Kuwabe, S.-i.; Shiraishi, T.; Shinohara, I.; Araki, H.; Sakuyama, S.; Makihara, T.; Kawanaka, Y.; Ohuchida, S.; Seko, T.: Synthesis of ONO-4819
0268
Li, N.; Chen, X.-H.; Song, J.; Luo, S.-W.; Fan, W.; Gong, L.-Z.: Synthesis of (S)-L-771688
0269
Tsuritani, T.; Mizuno, H.; Nonoyama, N.; Kii, S.; Akao, A.; Sato, K.; Yasuda, N.; Mase, T.: Synthesis of a Potential mGluR1 Antagonist
0270
Takahashi, Y.; Yoshimura, F.; Tanino, K.; Miyashita, M.: Synthesis of Zoanthenol
0271
Dowling, M. S.; Vanderwal, C. D.: Syntheses of (±)-Poitediol and (-)-Teucladiol
0272
Jakubec, P.; Cockfield, D. M.; Dixon, D. J.: Synthesis of (-)-Nakadomarin A
0273
Guinchard, X.; Roulland, E.: Synthesis of (+)-Neopeltolide

Synthesis of Heterocycles

z275
All PDFs of this category
0275
Tejedor, D.; Méndez-Abt, G.; García-Tellado, F.: Substituted Dihydropyridines from Propargyl Enol Ethers
0276
Wu, T.; Yin, G.; Liu, G.: Pd-Catalyzed Synthesis of Fluoropiperidines
0277
Staben, S. T.; Blaquiere, N.: Pd-Catalyzed Synthesis of 1,2,4-Triazoles
0278
Wong, Y.-C.; Parthasarathy, K.; Cheng, C.-H.: Cobalt-Catalyzed Synthesis of Pyrrolidinones from Nitriles and Acrylamides
0279
Baxendale, I. R.; Schou, S. C.; Sedelmeier, J.; Ley, S. V.: General Syntheses of Heterocycles Using Modular Flow Reactors
0280
Xu, X.; Li, H.; Xie, X.; Li, Y.: Iron-Catalyzed Synthesis of 9-Substituted Xanthenes
0281
Yang, X.; Liu, H.; Fu, H.; Qiao, R.; Jiang, Y.; Zhao, Y.: Copper-Catalyzed Synthesis of Quinazolines From 2-Bromobenzonitriles
0282
Jiang, H.; Mai, R.; Cao, H.; Zhu, Q.; Liu, X.: l-Proline-Catalyzed Synthesis of Highly Substituted 1,4-Dihydropyridines
0283
Okamoto, N.; Miwa, Y.; Minami, H.; Takeda, K.; Yanada, R.: Platinum-Catalyzed Synthesis of Indoles and Isoquinolines from 2-Alkynylarylamides
0284
Chernyak, N.; Tilly, D.; Li, Z.; Gevorgyan, V.: Palladium-Catalyzed Synthesis of Fused Heterocycles
0285
Gao, H.; Zhao, X.; Yu, Y.; Zhang, J.: Gold-Catalyzed Synthesis of Furo[3,4-c]-azepines
0286
Queffélec, C.; Montchamp, J.-L.: Synthesis of Diverse P,N-Containing Heterocycles
0287
Han, X.; Lu, X.: Pd-Catalyzed Synthesis of Dihydrocoumarins
0288
Shen, Z.; Lu, X.: Copper-Mediated Halocyclization Route to 3-Haloindoles
0289
Chouhan, G.; Alper, H.: Synthesis of 1,4-Benzo- and Pyrido-oxazepinones via a Domino Process

Synthesis of Materials and Unnatural Products

z291
All PDFs of this category
0291
Kaul, E.; Senkovskyy, V.; Tkachov, R.; Bocharova, V.; Komber, H.; Stamm, M.; Kiri, A.: A Bifunctional Initiator for Block Copolymer Synthesis
0292
Juárez-Pérez, E. J.; Viñas, C.; Teixidor, F.; Santillan, R.; Farfán, N.; Abreu, A.; Yépez, R.; Núñez, R.: A Resourceful Synthesis of Metallodendrimers
0293
Bharat; Bhola, R.; Bally, T.; Valente, A.; Cyrański, M. K.; Dobrzycki, Ł.; Spain, S. M.; Rempała, P.; Chin, M. R.; King, B. T.: Encircling the Square: Synthesis of Quadrannulene
0294
Tsuchikama, K.; Kasagawa, M.; Endo, K.; Shibata, T.: Iridium-Catalyzed Cascade Formation of Benzofulvenes
0295
Pemberton, B. C.; Barooah, N.; Srivatsava, D. K.; Sivaguru, J.: Cucurbituril-Catalyzed Photodimerization of Coumarins
0296
Miura, T.; Higashino, T.; Saito, S.; Osuka, A.: Expanded Isophlorins
0297
Schenck, C. L.; Nadeau, J. M.: An Axially Chiral Monomer
0298
Zeng, Z.; Spiccia, L.: Thymidine Nucleotide Sensor
0299
Zhang, X.; Jiang, X.; Luo, J.; Chi, C.; Chen, H.; Wu, J.: 2D Organic Semiconductor
0300
Wu, D.; Pisula, W.; Haberecht, M. C.; Feng, X.; Müllen, K.: Heteroatom-Containing Polycyclic Aromatics
0301
Goldup, S. M.; Leigh, D. A.; McGonigal, P. R.; Ronaldson, V. E.; Slawin, A. M. Z.: Templated Threading to [3]Rotaxanes
0302
Albright, T. A.; Dosa, P. I.; Grossmann, T. N.; Khrustalev, V. N.; Oloba, O. A.; Padilla, R.; Paubelle, R.; Stanger, A.; Timofeeva, T. V.; Vollhardt, K. P. C.: Photo-Activated Metal Migration
0303
Colquhoun, H. M.; Greenland, B. W.; Zhu, Z.; Shaw, J. S.; Cardin, C. J.; Burattini, S.; Elliott, J. M.; Basu, S.; Gasa, T. B.; Stoddart, J. F.: Macrocyclic Polycations Made to Order
0304
Gopalsamuthiram, V.; Predeus, A. V.; Huang, R. H.; Wulff, W. D.: Chiral Calixarenes
0305
Vivat, J. F.; Adams, H.; Harrity, J. P. A.: N-B Directed Cycloadditions

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z307
All PDFs of this category
0307
Tian, G.-Q.; Kaiser, T.; Yang, J.: Diastereoselective Alkyne-Aldehyde Reductive Coupling
0308
Sakakura, A.; Kondo, R.; Matsumura, Y.; Akakura, M.; Ishihara, K.: Rational Design of Diels-Alder Catalysts
0309
Baktharaman, S.; Afagh, N.; Vandersteen, A.; Yudin, A. K.: Synthesis and Application of Vinyl Aziridines
0310
Lu, L.-Q.; Li, F.; An, J.; Zhang, J.-J.; An, X.-L.; Hua, Q.-L.; Xiao, W.-J.: Diastereoselective Domino Synthesis of Tricyclic Heterocycles
0311
Malkov, A. V.; Gordon, M. R.; Stončius, S.; Hussain, J.; Kočovský, P.: Desymmetrization of Medium-Ring Cyclic Epoxides with SiCl4 and Chiral Mono-N-Oxide Lewis Base
0312
Seayad, A. M.; Ramalingam, B.; Yoshinaga, K.; Nagata, T.; Chai, C. L. L.: Protocol for the Titanium-Catalyzed Asymmetric Cyanation of Imines
0313
Sun, Y.-J.; Li, N.; Zheng, Z.-B.; Liu, L.; Yu, Y.-B.; Qin, Z.-H.; Fu, B.: Copper-Catalyzed Enantioselective Friedel-Crafts Alkylation of Indoles
0314
Bandini, M.; Eichholzer, A.: Gold-Catalyzed Friedel-Crafts Allylic Alkylation of Indoles with Alcohols
0315
Akiyama, K.; Gao, F.; Hoveyda, A. H.: Copper-Catalyzed Allylic Alkylation of Trisubstituted Vinylaluminum Reagents
0316
Iwata, M.; Yazaki, R.; Suzuki, Y.; Kumagai, N.; Shibasaki, M.: Synthesis of 1,3-Polyols via Direct Aldol Reactions of Thioamides
0317
Shigeno, M.; Yamamoto, T.; Murakami, M.: Stereoselective Restructuring of 3-Arylcyclobutanols into 1-Indanols
0318
Lassauque, N.; Franciò, G.; Leitner, W.: Nickel-Catalyzed Asymmetric Hydrovinylation at Room Temperature
0319
Boussonnière, A.; Dénès, F.; Lebreton, J.: Radical Cyclization of α-Bromo Aluminum Acetals
0320
Jensen, K. H.; Pathak, T. P.; Zhang, Y.; Sigman, M. S.: Enantioselective Difunctionalization of Alkenes Catalyzed by Palladium(II)
0321
Yoshino, T.; Morimoto, H.; Lu, G.; Matsunaga, S.; Shibasaki, M.: Magnesium Schiff Base Catalyzed Direct Asymmetric Aldol Reaction
0322
Li, W.; Hou, G.; Chang, M.; Zhang, X.: Iridium-Catalyzed Asymmetric Hydrogenation of N-Arylimines
0323
Da, C.-S.; Wang, J.-R.; Yin, X.-G.; Fan, X.-Y.; Liu, Y.; Yu, S.-L.: Asymmetric Addition of Deactivated Grignard Reagents to Aldehydes
0324
Watanabe, Y.; Washio, T.; Shimada, N.; Anada, M.; Hashimoto, S.: Rhodium(II) Carboxamidate Catalyzed Hetero-Diels-Alder Reaction of Rawal’s Diene
0325
Takimoto, M.; Usami, S.; Hou, Z.: Stereospecific Synthesis of Tetrasubstituted Alkenes via Sc-Catalyzed Methylalumination
0326
Zhang, W.; Huang, W.; Hu, J.: Synthesis of Fluoroalkenes from Fluorosulfoximines and Nitrones
0327
Huang, X.-R.; Chen, C.; Lee, G.-H.; Peng, S.-M.: Enantioselective Allylation of Ketones Using a Spirocyclic Chiral Borate
0328
Lei, B.-L.; Ding, C.-H.; Yang, X.-F.; Wan, X.-L.; Hou, X.-L.: Kinetic Resolution of the Nucleophile in Palladium-Catalyzed Allylic Alkylation
0329
Komeyama, K.; Saigo, N.; Miyagi, M.; Takaki, K.: Stereospecific Intramolecular Alkynylcyclopropanation of Olefins
0330
Evanno, L.; Ormala, J.; Pihko, P. M.: New Protocols for Noyori Transfer Hydrogenation
0331
Lee, Y.; Jang, H.; Hoveyda, A. H.: Synthesis of Vicinal Diboronates by Cu(I)-Catalyzed B-Cu Addition to Alkynes
0332
Liang, G.; Tong, M.-C.; Wang, C.-J.: endo-Selective and Enantioselective 1,3-Dipolar Cycloaddition of Azomethine Ylides

Metal-Mediated Synthesis

z333
All PDFs of this category
0333
Quasdorf, K. W.; Riener, M.; Petrova, K. V.; Garg, N. K.: Nickel-Catalyzed Suzuki-Miyaura Coupling of Aryl Carbamates, Carbonates, and Sulfamates
0334
Kim, S. Y.; Park, Y.; Chung, Y. K.: Pt-Catalyzed Tandem Cycloisomerization and Cope Rearrangement of Dienynes
0335
Mitchell, T. A.; Bode, J. W.: BF3-Mediated Coupling of Organotrifluoro-borates and Acetals
0336
Denichoux, A.; Fukuyama, T.; Doi, T.; Horiguchi, J.; Ryu, I.: Ruthenium Hydride Catalyzed Coupling of α,β-Unsaturated Aldehydes with Primary Alcohols
0337
Nishihara, Y.; Saito, D.; Inoue, E.; Okada, Y.; Miyazaki, M.; Inoue, Y.; Takagi, K.: Ynones via Copper-Mediated Cross-Coupling of Alkynylboronates and Acid Chlorides
0338
Lu, P.; Sanchez, C.; Cornella, J.; Larrosa, I.: Silver(I)-Catalyzed Decarboxylation of Aromatic Carboxylic Acids
0339
Wunderlich, S. H.; Knochel, P.: Direct Ferration and Nickel-Catalyzed Alkylation of Aromatic Compounds
0340
Cherkupally, P.; Beier, P.: Nucleophilic Trifluoromethylation Using Diethyl Trifluoromethanephosphonate
0341
Urkalan, K. B.; Sigman, M. S.: Csp³-Csp³ Bond Formation via Palladium-Catalyzed Hydroalkylation of Styrenes
0342
Fandrick, D. R.; Reeves, J. T.; Tan, Z.; Lee, H.; Song, J. J.; Yee, N. K.; Senanayake, C. H.: Allene Synthesis and Propargylations with Stable Propargyl Boronates
0343
Martínez-Asencio, A.; Ramón, D. J.; Yus, M.: Alkylation of Amines and Sulfonamides by Copper(II)-Catalyzed Hydrogen Transfer
0344
Kosal, A. D.; Ashfeld, B. L.: Titanocene-Catalyzed 1,4-Reduction of α,β-Unsaturated Carbonyl Compounds
0345
Ankner, T.; Hilmersson, G.: SmI2/H2O/Amine Promoted Cleavage of Benzyl-Heteroatom Bonds
0346
Okamoto, S.; He, J.-Q.; Ohno, C.; Oh-iwa, Y.; Kawaguchi, Y.: Ti/Mg-Mediated McMurry Coupling of Aryl Aldehydes and Imino Pinacol Coupling
0347
López-Pérez, A.; Adrio, J.; Carretero, J. C.: Pd-Catalyzed Coupling of sec-Benzylic Bromides with Grignard Reagents

Organo- and Biocatalysis

z349
All PDFs of this category
0349
Piccinini, A.; Kavanagh, S. A.; Connon, P. B.; Connon, S. J.: Catalytic Synthesis of Terminal Epoxides via Methylene Transfer to Aldehydes
0350
Uehara, H.; III, C. F. Barbas: anti-Selective Michael Reaction of Aldehydes
0351
Lovick, H. M.; Michael, F. E.: Intramolecular Oxyamination of Alkenes
0352
Vedachalam, S.; Zeng, J.; Gorityala, B. Kishan; Antonio, M.; Liu, X.-W.: NHC-Catalyzed Intramolecular Cross-Coupling of Aldehydes and Nitriles
0353
Moss, T. A.; Alonso, B.; Fenwick, D. R.; Dixon, D. J.: Phase-Transfer-Catalyzed Alkylations by Ring-Opening of Sulfamidates
0354
Pansare, S. V.; Lingampally, R.; Kirby, R. L.: Michael Addition for the Synthesis of Octahydroindole Natural Products
0355
Zheng, Z.; Perkins, B. L.; Ni, B.: Enantioselective Michael Addition Using Recyclable and Water-Soluble Catalysts
0356
Gu, L.; Zhang, Y.: N-Heterocyclic Carbene Catalyzed Oxidation of Aldehydes Using CO2 as Oxidant
0357
Sun, F.-G.; Huang, X.-L.; Ye, S.: Synthesis of 4-Hydroxytetralones via a Cascade Stetter-Aldol Reaction
0358
Liang, X.; Yang, J.: An Efficient Ionic Liquid Catalyst for the Synthesis of Biodiesel
0359
De Sarkar, S.; Grimme, S.; Studer, A.: Oxidative Acylation of Alcohols in the Presence of Amines
0360
Polshettiwar, V.; Varma, R. S.: A Magnetic Multi-Purpose Organocatalyst

Polymer-Supported Synthesis

z361
All PDFs of this category
0361
Metzger, A.; Qin, L.-Y.; Cole, A. G.; Saionz, K. W.; Brescia, M.-R.; Gstach, H.; Wareing, J. R.; Zimmermann, J.; Brill, W. K.-D.; Baldwin, J. J.; Dolle, R. E.; Henderson, I.: Solid-Phase Synthesis of 2-Amino-7,8-dihydropteridin-6(5H)-ones
0362
Ackermann, L.; Vicente, R.: Palladium-Catalyzed Arylation in Polyethylene Glycol under Air
0363
He, J.; Kim, J. W.; Yamaguchi, K.; Mizuno, N.: Synthesis of Amines from Alcohols and Urea with Ru(OH)x/TiO2
0364
Bakherad, M.; Keivanloo, A.; Bahramian, B.; Rajaie, M.: A Coupling Reaction of Acid Chlorides with Alkynes Using a PS-Pd Complex
0365
Wu, X.-J.; Jiang, R.; Wu, B.; Su, X.-M.; Xu, X.-P.; Ji, S.-J.: Nano Iron Oxide Catalyst for Intramolecular C-N Coupling Reaction
0366
Yinghuai, Z.; Kuijin, L.; Huimin, N.; Chuanzhao, L.; Stubbs, L. P.; Siong, C. F.; Muihua, T.; Peng, S. C.: Metathesis of Unsaturated Fatty Acid Esters with a Reusable Ruthenium Catalyst
0367
Rosario-Amorin, D.; Wang, X.; Gaboyard, M.; Clérac, R.; Nlate, S.; Heuzé, K.: Suzuki Coupling with Palladium Dendron Complex Grafted on MNPs
0368
Jiang, Z.; She, J.; Lin, X.: C-S Cross-Coupling with Palladium on Charcoal
0369
Alza, E.; Pericàs, M. A.: Michael Addition with a Polymer-Supported Organocatalyst
0370
Chen, C.-K.; Chen, Y.-W.; Lin, C.-H.; Lin, H.-P.; Lee, C.-F.: Reaction of Thiols with Aryl Iodides with CuO on Mesoporous Silica
0371
Lee, C.-T.; Huang, S.; Lipshutz, B. H.: Tandem One-Pot Diazo Transfer-Click Reactions Using Cu/C as a Catalyst
0372
He, L.; Wang, L.-C.; Sun, H.; Ni, J.; Cao, Y.; He, H.-Y.; Fan, K.-N.: A Gold-Catalyzed Reduction of Nitro Compounds with CO and H2O
0373
Schweizer, S.; Becht, J.-M.; Drian, C. Le: Suzuki-Miyaura Coupling of Aryl Chlorides with Supported Palladium Catalyst