DOI: 10.1055/s-00000131

Synfacts

Issue 07 · Volume 2006 · June 2006 DOI: 10.1055/s-002-4958

Synthesis of Natural Products and Potential Drugs

0633
Aggarwal, V. K.; Charmant, J. P. H.; Fuentes, D.; Harvey, J. N.; Hynd, G.; Ohara, D.; Picoul, W.; Robiette, R.; Smith, C.; Vasse, J.-L.; Winn, C. L.: Synthesis of SK&F 104353
0634
Motoyoshi, H.; Horigome, M.; Watanabe, H.; Kitahara, T.: Synthesis of FR901464
0635
Fukuda, N.; Sasaki, K.; Sastry, T. V. R. S.; Kanai, M.; Shibasaki, M.: Synthesis of (+)-Lactacystin
0636
Crimmins, M. T.; Brown, B. H.; Plake, H. R.: Syntheses of Ophirin B and Astrogorgin
0637
Tonogaki, K.; Itami, K.; Yoshida, J.-I.: Synthesis of (±)-Rolipram
0638
Coleman, R. S.; Lu, X.: Synthesis of Strobilurin B
0639
Nising, C. F.; Ohnemüller, U. K.; Bräse, S.: Synthesis of Diversonol
0640
Davies, H. M. L.; Dai, X.; Long, M. S.: Synthesis of (-)-Colombiasin A and(-)-Elisapterosin B
0641
Kawasaki, T.; Shinada, M.; Kamimura, D.; Ohzono, M.; Ogawa, A.: Synthesis of (-)-Flustramine B and(-)-Flustramide B
0642
Reisman, S. E.; Ready, J. M.; Hasuoka, A.; Smith, C. J.; Wood, J. L.: Synthesis of (±)-Welwitindolinone A Isonitrile
0643
Hart, A. C.; Phillips, A. J.: Synthesis of (+)-Cylindramide A
0644
Zhang, Y.; Liebeskind, L. S.: Synthesis of (-)-Bao Gong Teng A
0645
Kano, T.; Hashimoto, T.; Maruoka, K.: Synthesis of Manzacidin A
0646
Cohen, F.; Overman, L. E.: Synthesis of Batzelladine F
0647
Dirat, O.; Elliott, J. M.; Jelley, R. A.; Jones, A. B.; Reader, M.: Synthesis of NK1 Antagonists

Synthesis of Heterocycles

0649
Yang, X.; Luo, S.; Fang, F.; Liu, P.; Lu, Y.; He, M.; Zhai, H.: Intramolecular [3+2] Cycloaddition Approach to Nicotine Analogues
0650
Neogi, A.; Majhi, T. P.; Mukhopadhyay, R.; Chattopadhyay, P.: Benzoxazocines by Palladium-Catalyzed Intramolecular Amination
0651
Toffano, M.; Dobrota, C.; Fiaud, J.-C.: Catalytic Pd-Mediated Approach to Enantiopure Phosphorus Ligands
0652
Couty, S.; Meyer, C.; Cossy, J.: Combined Heck-Suzuki Reactions in a Synthesis of Lennoxamine
0653
Zhoa, A.; Njogu, M. N.; Pittman, C. U.: Synthesis of Chiral Oxazolo and Thiazolo Isoquinolinones
0654
Deprez, N. R.; Kalyani, D.; Krause, A.; Sanford, M. S.: 2-Arylation of Indoles using Diaryliodonium Salts
0655
IJsselstijn, M.; Cintrat, J. C.: Synthesis of 4-Amino Triazoles by Huisgen [3+2] Cycloaddition
0656
Lee, C. K. Y.; Herlt, A. J.; Simpson, G. W.; Willis, A. C.; Easton, C. J.: Asymmetric Synthesis of Δ2-Isoxazolines
0657
Williams, J. T.; Bahia, P. S.; Kariuki, B. M.; Spencer, N.; Philp, D.; Snaith, J. S.: Synthesis of cis- or trans-3,4-Disubstituted Piperidines
0658
Lesma, G.; Danieli, B.; Saccheti, A.; Silvani, A.: Synthesis of Cyclic β-Amino Acids by RCM
0659
Denmark, S. E.; Fan, Y.: Diastereoselective Approach to Non-racemic Bipyridine bis-N-Oxides
0660
Movassaghi, M.; Hill, M. D.: Pyridine and Quinoline Derivatives via Ru-Catalyzed Cyclization of Azadienynes
0661
Langlois, N.; Nguyen, B. K. Le; Retailleau, P.; Tarnus, C.; Salomon, E.: Synthesis of Indolizidines Bearing Quaternary Stereocenters
0662
Pastre, J. C.; Correia, C. R. D.: Heck Reaction of Acrylates with Arenediazonium Tetrafluoroborates
0663
Herrera, A.; Martínez-Alvarez, R.; Ramiro, P.; Molero, D.; Almy, J.: Synthesis of 2,5- and 2,4,5-Substituted 1,3-Oxazoles

Synthesis of Materials and Unnatural Products

0665
Xu, R.; Gramlich, V.; Frauenrath, H.: Solid-State Organization Enables Copolymerization
0666
Zhang, S.; Lukoyanova, O.; Echegoyen, L.: An Orthogonal Protection-Deprotection Route to Antipodal Fullerene Derivatives
0667
Kamplain, J. W.; Bielawski, C. W.: Dynamic Covalent Polymers Based upon Carbene Dimerization
0668
Ammann, M.; Rang, A.; Schalley, C. A.; Bäuerle, P.: Interlocked Oligothiophene Macrocycles
0669
Han, F. S.; Osajima, H.; Cheung, M.; Tokoyama, H.; Fukuyama, T.: Chiral, Macrocyclic Oligothiazolines
0670
Itami, K.; Tonogaki, K.; Nokami, T.; Ohashi, Y.; Yoshida, J.-I.: Fully Conjugated PPV Dendrimers
0671
Liu, Y.; Nishiura, M.; Wang, Y.; Hou, Z.: A Single-Molecule White-Light Emitter
0672
Chen, Y.-L.; Hau, C.-K.; Wang, H.; He, H.; Wong, M.-S.; Lee, A. W. M.: Stable Isobenzofurans
0673
Collins, S. K.; Grandbois, A.; Vachon, M. P.; Côté, J.: RCM Helicene Synthesis
0674
Dohi, T.; Morimoto, K.; Maruyama, A.; Kita, Y.: Regioselective Pyrrole Oxidative Dimerization

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

0675
Hedberg, C.; Källström, K.; Brandt, P.; Hansen, L. K.; Andersson, P. G.: Hydrogenation of Trisubstituted Olefins with Ir-Phosphine Thiazole Complexes
0676
Szõri, K.; Szöllõsi, G.; Bartók, M.: Dynamic Kinetic Resolution of Racemic Ethyl 2-Fluoroacetoacetate
0677
Nakhla, J. S.; Kampf, J. W.; Wolfe, J. P.: Intramolecular Pd-Catalyzed Carboetherification and Carboamination
0678
Trost, B. M.; Zhang, Y.: Mo(0)-Catalyzed Allylic Alkylation of 3-Alkyloxindole
0679
Wu, J.; Wang, F.; Ma, Y.; Cui, X.; Cun, L.; Zhu, J.; Deng, J.; Yu, B.: Asymmetric Transfer Hydrogenation of Cyclic Imines and Iminiums
0680
Xu, W.; Kong, A.; Lu, X.: Pd-Catalyzed Asymmetric Synthesis ofα-Alkylidene-γ-butyrolactams
0681
Tanaka, K.; Takeishi, K.; Noguchi, K.: Synthesis of Axially Chiral Aromatic Amides via [2+2+2] Cycloaddition
0682
Colombo, F.; Benaglia, M.; Orlandi, S.; Usuelli, F.; Celentano, G.: Enantioselective Synthesis of Propargylamines
0683
Janka, M.; He, W.; Haedicke, I. E.; Fronczek, F. R.; Frontier, A. J.; Eisenberg, R.: Ir(III)-Catalyzed Tandem Nazarov Cyclization/Michael Addition
0684
Tonogaki, K.; Itami, K.; Yoshida, J.-I.: Three-Component Cyclization with Allenylboronate Platform
0685
Cho, C.-W.; Krische, M. J.: Reductive Coupling of Alkynes and α-Keto Aldehydes
0686
Shintani, R.; Yashio, K.; Nakamura, T.; Okamoto, K.; Shimada, T.; Hayashi, T.: Development of a New ‘Axially Chiral’ Bisphosphine Ligand
0687
Gao, X.; Hall, D. G.; Deligny, M.; Favre, A.; Carreaux, F.; Carboni, B.: Three-Component Hetero-[4+2] Cycloaddition/Allylboration
0688
Itoh, T.; Miyazaki, M.; Fukuoka, H.; Nagata, K.; Ohsawa, A.: (-)-Emetine Synthesis via Asymmetric Allylation of Cyclic Imines
0689
Maier, T. C.; Fu, G. C.: Enantioselective α-Oxygenation ofα-Diazoesters
0690
Blanc, A.; Toste, F. D.: Cyclic Ethers through a Catalyzed Resolution/Oxidative Cyclization
0691
Chu, Y.; Shan, Z.; Liu, D.; Sun, N.: Spiroborate Ether Mediated Enantioselective Reduction of Oxime Ethers
0692
Trost, B. M.; Jaratjaroonphong, J.; Reutrakul, V.: Direct Catalytic Asymmetric Mannich Reaction via a Dinuclear Zinc Catalyst
0693
Weis, M.; Waloch, C.; Seiche, W.; Breit, B.: Self-Assembly of Ligands for Combinatorial Homogeneous Catalysis
0694
Mazet, C.; Roseblade, S.; Köhler, V.; Pfaltz, A.: Kinetic Resolution of Diols and Pyridyl Alcohols
0695
Lipshutz, B. H.; Tanaka, N.; Taft, B. R.; Lee, C.-T.: Access to Chiral Silanes via Asymmetric Hydrosilylation
0696
Kikuchi, S.; Sato, H.; Fukuzawa, S.-I.: Asymmetric Conjugate Addition ofO-Benzylhydroxylamine
0697
Rauniyar, V.; Hall, D. G.: Asymmetric Additions of Allyl- and Crotylboronates to Aldehydes
0698
Cozzi, P. G.: Mn-Catalyzed Reformatsky Reaction with Ketones
0699
Shintani, R.; Inoue, M.; Hayashi, T.: Rh-Catalyzed Asymmetric Arylation and Alkenylation of Isatins
0700
Chan, V. S.; Sterwart, I. C.; Bergman, R. G.; Toste, F. D.: Synthesis of P-Stereogenic Phosphines
0701
Scriban, C.; Glueck, D. S.: Synthesis of P-Stereogenic Phosphines
0702
Lu, S.-F.; Du, D.-M.; Xu, J.: Enantioselective Friedel-Crafts Alkylation of Indoles with Nitroalkenes
0703
Romero, A.; Woerpel, K. A.: Stereoselective Synthesis of Highly Substituted γ-Lactams
0704
Evans, D. A.; Aye, Y.; Wu, J.: anti-Selective Sc(III)-Catalyzed Sakurai Additions to Glyoxyamide
0705
Llamas, T.; Arrayás, R. G.; Carretero, J. C.: 1,3-Dipolar Cycloaddition of Azomethine Ylides with Vinyl Sulfones
0706
Liu, L.; Montgomery, J.: Synthesis of Cyclopentanes via Cyclopropane Ring Opening
0707
Shi, W.-J.; Zhang, Q.; Xie, J.-H.; Zhu, S.-F.; Hou, G.-H.; Zhou, Q.-L.: Hydrovinylation of α-Alkyl Vinylarenes
0708
Kinder, R. E.; Widenhoefer, R. A.: Asymmetric Cyclization-Hydroboration of 1,6-Enynes

Metal-Mediated Synthesis

0709
Guram, A. S.; King, A. O.; Allen, J. G.; Wang, X.; Schenkel, L. B.; Chan, J.; Bunel, E. E.; Faul, M. M.; Larsen, R. D.; Martinelli, M. J.; Reider, P. J.: New Catalysts for Cross-Coupling of Heteroaryl Chlorides
0710
Dai, Q.; Gao, W.; Liu, D.; Kapes, L. M.; Zhang, X.: New Triazolyl Phosphines for Cross-Coupling of Aryl Chlorides
0711
Montel, F.; Beaudegnies, R.; Kessabi, J.; Martin, B.; Muller, E.; Wendeborn, S.; Jung, P. M. J.: Cu-Catalyzed Preparation of 1,4-Diynes from TMS Alkynes
0712
Black, D. A.; Arndtsen, B. A.: Cu-Promoted Coupling of Imines, Acid Chlorides and Organoindium Reagents
0713
Lee, D.; Kim, D.; Yun, J.: Enantioselective Conjugate Reduction of Unsaturated Nitriles
0714
Hama, T.; Culkin, D. A.; Hartwig, J. F.: Pd-Catalyzed α-Arylation of Zinc Amide Enolates
0715
Cozzi, P. G.; Kostrusz, P.: Enantioselective Addition of Me2Zn to Aldehydes Catalyzed by ClCr(Salen)
0716
Beenen, M. A.; Weix, D. J.; Ellman, J. A.: Enantioselective Synthesis of Arylglycines from Arylboronic Acids
0717
Jagt, R. B.; Toullec, P. Y.; Geerdink, D.; de Vries, J. G.; Feringa, B. L.; Minnaard, A. J.: Rh-Catalyzed Asymmetric Arylation ofN-Sulfamoyl Aldimines
0718
Lee, K.; Maleczka, R. E.: Pd(0)-Catalyzed Reduction of Aromatic Acid Chlorides to Aldehydes
0719
Molander, G. A.; Ham, J.: Synthesis of Functionalized Organotrifluoroborates from Halomethyltrifluoroborates
0720
Krasovskiy, A.; Krasovskaya, V.; Knochel, P.: Highly Efficient Magnesiation of Functionalized Arenes and Heteroarenes
0721
González-Bobes, F.; Fu, G. C.: Nickel-Catalyzed Suzuki Reaction of Unactivated Alkyl Halides

Organo- and Biocatalysis

0723
Purkarthofer, T.; Gruber, K.; Gruber-Khadjawi, M.; Waich, K.; Skranc, W.; Mink, D.; Griengl, H.: Biocatalytic Asymmetric Henry Reaction
0724
Chi, Y.; Gellman, S. H.: Enantioselective Organocatalytic Aminomethylation of Aldehydes
0725
Takikawa, H.; Hachisu, Y.; Bode, J. W.; Suzuki, K.: Asymmetric Intramolecular Crossed Aldehyde-Ketone Benzoin Cyclization
0726
Sakakura, A.; Suzuki, K.; Nakano, K.; Ishihara, K.: Asymmetric Diels-Alder Reaction Catalyzed by a Chiral Diammonium Salt
0727
Huang, H.; Jacobsen, E. N.: Chiral Amine-Thiourea Catalyst for the Asymmetric Michael Addition
0728
Mossé, S.; Laars, M.; Kriis, K.; Kanger, T.; Alexakis, A.: Michael Addition Catalyzed by a Chiral Bimorpholine
0729
Ting, A.; Lou, S.; Schaus, A. E.: Quaternary Carbon Centers by Cinchonine-Catalyzed Mannich Reactions
0730
Liu, Y.-H.; Chen, L.-H.; Shi, M.: Asymmetric Aza-Morita-Baylis-Hillman Reaction Catalyzed by a Phenol-Bearing Phosphine
0731
Rueping, M.; Antonchick, A. P.; Theissmann, T.: Highly Enantioselective Organocatalytic Transfer Hydrogenation of Quinolines

Polymer-Supported Synthesis

0733
Levin, Y.; Hamza, K.; Abu-Reziq, R.; Blum, J.: One-Pot Bromination and Dehydrobromination
0734
Shokouhimehr, M.; Kim, J.-H.; Lee, Y.-S.: Heck Reaction Catalyzed by Polymer-Supported Carbene-Palladium Complex
0735
Girard, C.; Önen, E.; Aufort, M.; Beauière, S.; Samson, E.; Herscovici, J.: [3+2] Cycloaddition Using Reusable Polymer-Supported Catalyst
0736
Takahashi, T.; Watahiki, T.; Kitazume, S.; Yasuda, H.; Sakakura, T.: Synergistic Hybrid Catalyst for Cyclic Carbonate Synthesis
0737
Ferrand, Y.; Daviaud, R.; Maux, P. Le; Simonneaux, G.: Asymmetric Oxidation Using Polymer-Supported Chiral Metalloporphyrins
0738
Shore, G.; Morin, S.; Organ, M. G.: Microwave-Assisted Microreactor for Suzuki and Heck Reactions
0739
Byk, G.; Kabha, E.: A Solid-Supported Stereoselective Multicomponent Reaction
0740
Ménand, M.; Blais, J.-C.; Valéry, J.-M.; Xie, J.: Synthesis of Sugar-Aza-Crown Ethers
0741
Bianco, A.; Fournel, S.; Wieckowski, S.; Hoebeke, J.; Guichard, G.: Solid-Phase Synthesis of CD40L Mimetics
0742
Zhang, H.; Piacham, T.; Drew, M.; Patek, M.; Mosbach, K.; Ye, L.: MIP for Regioselective Huisgen 1,3-Dipolar Cycloaddition Reaction
0743
König, H. M.; Abbel, R.; Schollmeyer, D.; Kilbinger, A. F. M.: Solid-Phase Synthesis of Oligo(p-benzamide) Foldamers
0744
Abu-Reziq, R.; Alper, H.; Wang, D.; Post, M. L.: Silica-Coated Magnetite Nanoparticles Supported Rhodium Catalyst
0745
Motokura, K.; Fujita, N.; Mori, K.; Mizugaki, T.; Ebitani, K.; Kaneda, K.: Solid Acid Catalyzed Addition Reaction of 1,3-Dicarbonyl Compounds onto Alkenes
0746
Grunlan, M. A.; Regan, K. R.; Bergbreiter, D. E.: Liquid-Liquid Separation of Polysiloxane-Supported Quinine Catalysts