DOI: 10.1055/s-00000131

Synfacts

Issue 08 · Volume 2010 · August 2010 DOI: 10.1055/s-002-21206

Synform

A64
SYNFORM ISSUE 2010/08

Synthesis of Natural Products and Potential Drugs

z851
All PDFs of this category
0851
Synthesis of (±)-Clivonine
0852
Synthesis of a Tamoxifen Homologue
0853
Synthesis of (S)-Rivastigmine
0854
Formal Synthesis of Eurylene
0855
Synthesis of ent-Abudinol B
0856
Synthesis of MK-5596
0857
Synthesis of Oseltamivir
0858
Synthesis of (+)-Complanadine A
0859
Synthesis of RO5114436
0860
Synthesis of (-)-Cubebol
0861
Synthesis of (S)-Profens
0862
Synthesis of (-)-Actinophyllic Acid
0863
Synthesis of (+)-Complanadine A
0864
Synthesis of the Core Structure of P2X7 Receptor Antagonists
0865
Synthesis of BMS-587101

Synthesis of Heterocycles

z867
All PDFs of this category
0867
Copper-Catalyzed Synthesis of Pyridine N-Oxides from α,β-Unsaturated Oximes
0868
Copper-Catalyzed One-Pot Synthesis of Benzimidazo[1,2-b]isoquinolin-11-ones
0869
CuI/La(OTf)3-Catalyzed Synthesis of Isomeric Ellipticine
0870
One-Step Synthesis of Annulated Hydroquinolines
0871
Copper-Catalyzed Cascade Synthesis of Triazoloquinoxalines
0872
Osmium-Catalyzed Synthesis of 3-Benzoxepines
0873
Rhodium-Catalyzed Synthesis of 3-Aryl and 3-Alkenyl Phthalides
0874
Synthesis of 1,2-Benzisoxazoles via a 1,3-Dipolar Cycloaddition
0875
A Lactonization Route to 5-(Trifluoromethyl)-2(5H)-furanones
0876
Synthesis of 1,4-Benzodioxanes via Epoxide Opening and Cyclization
0877
Synthesis of Substituted Indoles Using Flow Microreactors
0878
Synthesis of Pyrroles via [3,3]-Rearrangement and Paal-Knorr Reaction
0879
One-Step Synthesis 3-Nitroisoxazoles
0880
Synthesis of 2H-Indazoles via [3+2]-Dipolar Cycloaddition
0881
Synthesis of Trisubstituted Isoxazoles via Gold-Catalyzed Domino Reaction

Synthesis of Materials and Unnatural Products

z883
All PDFs of this category
0883
Turn-On Labeling in Living Cells
0884
Incorporation of π-Conjugated Molecules within Peptide Backbones
0885
Naturally Renewable Polymers from an Innovative Living Polymerization
0886
Stable Borepin Rings
0887
Emergent Self-Assembly
0888
Novel Cyclyne via Mild Reductive Aromatization
0889
C-H Activation Directed Multicomponent Assembly of Macrocycles
0890
Simple Perfluoroalkylation
0891
A Cyclic [4]Rotaxane
0892
Trifluoromethylation of Terminal Alkynes
0893
Porphyrin-Based Molecular Turnstiles
0894
Benzo[k]fluoranthenes
0895
Sticky Caps for Polymers
0896
A Stable Fullerene Anion

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z897
All PDFs of this category
0897
Diastereoselective Synthesis of Axially Chiral Bis-sulfoxide Ligands
0898
Gold-Catalyzed Synthesis of E-α-Haloenones from Propargyl Acetates
0899
Regiocontrol in the Nickel-Catalyzed Aldehyde-Alkyne Reductive Coupling
0900
Chiral Bis(oxazolinyl)phenyl Ruthenium(II) Catalysts for Asymmetric Cyclopropanation
0901
Nickel-Catalyzed Reductive Coupling of Dienes with Aldehydes
0902
Construction of Chiral Tetrasubstituted Olefins Using Ring-Closing Metathesis
0903
E-Selective Allylboration of α-Substituted Allylboronates
0904
Synthesis and Application of C2-Bridged Diphosphine Palladium Complexes
0905
Modular Synthesis of P-OP Ligands and Application in Asymmetric Hydrogenation
0906
Copper-Catalyzed Selective Aryl-Allyl Coupling
0907
Zirconium-Mediated Enantioselective Darzens Reaction
0908
Friedel-Crafts Alkylation of Indoles with Diphenylamine Bis(imidazoline) Ligands
0909
Ir-Catalyzed Asymmetric Allylic Amination and Pt-Catalyzed Cycloisomerization
0910
Scandium-Catalyzed Asymmetric α-Amination of 3-Substituted 2-Oxindoles
0911
Selective Domino Synthesis of Heterocycles through Cooperative Catalysis
0912
Synthesis of Chiral Sulfonimidamides and Application in Asymmetric Henry Reaction
0913
Chromium-Catalyzed Enantioselective Synthesis of 1,3-Butadien-2-ylcarbinols
0914
Asymmetric Rh(II)- and Cu(I)-Catalyzed Si-H Insertion Leading to Chiral Crotylsilanes
0915
Synthesis of 1,3-syn-Diol Acetals via Re-Catalyzed Allylic Alcohol Transposition
0916
Addition of Trialkylaluminium Regents to Extended Michael Acceptors
0917
Valine-Derived Ruthenium Complex for Catalytic Metathesis Desymmetrization
0918
Friedel-Crafts Alkylation of Indoles via Combinatorial Transition-Metal Catalysis
0919
Enantioselective Propargylation of Aldehydes by Copper Catalysis
0920
MIDA and BF3K in Rhodium-Catalyzed Stereoselective Addition to Aldimines
0921
A Novel Tetraoxazoline Ligand for Asymmetric Hydrosilylation
0922
Sterospecific Copper-Catalyzed Formation of Cyclobutyl- and Cyclopentylboronates
0923
Chemo- and Enantioselective Synthesis of 3-Allyl-3-aryl Oxindoles
0924
Synthesis of Heterobicycles by Intramolecular Aza-Prins Reaction
0925
Enantioselective Hydrogenation of α-Dehydroamino Acid Esters
0926
C-C Coupling of Ethanol and Dienes

Metal-Mediated Synthesis

z927
All PDFs of this category
0927
Nickel-Catalyzed Arylative Ring Opening
0928
Atom-Efficient Coupling of Triarylbismuths with Bromide and Chloride Derivatives
0929
N-C Aryl Transfer via Umpolung Carbolithiation of Vinyl Ureas
0930
Copper-Catalyzed Direct Amination of Azoles with Chloroamines at Room Temperature
0931
A One-Pot Synthesis of (Z)-Acrylonitriles via an α-Diaminoboryl Carbanion
0932
Synthetic Equivalents for the Preparation of 1,2,3,4-Tetrahydroisoquinolines
0933
Stereoretentive Suzuki-Miyaura Coupling of Haloallenes
0934
Nickel-Catalyzed Synthesis of Poly-substituted Olefins from Alkenyl Acetates
0935
Arylsilane Oxidation - New Routes to Hydroxylated Aromatics
0936
Phosphorodiamidate-Directed Metalation of N-Heterocycles using Mg- and Zn-TMP
0937
Synthesis of 4,4′-Bipyridines via a Simple Dimerization Procedure
0938
Nickel-Catalyzed Allylic Substitution of Simple Alkenes
0939
La(CN)3-Catalyzed Acyl Silane-Ketone Benzoin Addition
0940
A P,N-Ligand for the Palladium-Catalyzed Arylation of Ammonia
0941
Difluoromethylation of Lithium Enolates with Trifluoromethyl Iodide

Organo- and Biocatalysis

z943
All PDFs of this category
0943
Michael Addition of Aldehydes to 2-Amino-1-nitroethenes
0944
Enantioselective One-Pot Synthesis of Substituted Cyclohexenones
0945
NMR Detection of the Enamine Intermediate in Proline-Catalyzed Aldol Reactions
0946
Catalytic Asymmetric Retro-Aldol Reaction
0947
Catalytic Asymmetric Transacetalization
0948
Asymmetric [3+2] Cycloaddition Catalyzed by 1,2-Aminophosphanes
0949
Aziridination of Cyclic Enones
0950
Inversion of Enantioselectivity in Proline Catalysis by Basic Additives
0951
NHC-Catalyzed Desymmetrization in Natural Product Synthesis
0952
Organocatalytic Vinylogous Mukaiyama Aldol Reactions
0953
Bifunctional Catalysts for Asymmetric Nazarov Cyclizations
0954
Cyclopropanation of α-Substituted α,β-Unsaturated Aldehydes
0955
Michael Reaction of α,α-Disubstituted Aldehydes and Maleimides
0956
Asymmetric Cyanosilylation of Nitroalkenes

Polymer-Supported Synthesis

z957
All PDFs of this category
0957
Solid-Phase Synthesis of Aminothiazoles
0958
Solid-Phase Synthesis of Peptides Using Cysteine Orthoesters
0959
Direct Borylation of Arenes Catalyzed by γ-Fe2O3
0960
Synthesis of Fused Quinolinium Salts Using Amberlite IRA 402(OH)
0961
5′-O-β,γ-Methylenetriphosphate Derivatives of Nucleosides
0962
Protein-Stabilized Palladium Nanoparticles for Biaryl Coupling
0963
Ligand-Free Ullmann Arylation of Indole Using PEG3400-Cu2O-Cs2CO3
0964
Silica-Based S-Sulfonic Acid for the Strecker Synthesis
0965
ZnCl2/Al2O3-Catalyzed Ferrier Azaglycosylation
0966
Microwave-Assisted Synthesis of Fused Quinoxalinones
0967
Oxidative Cyanation of Amines Using Heterogeneous Iron Phthalocyanines
0968
Simple Synthesis of Amides with Polymer-Supported Ph3P and Iodine
0969
Silica-Phase Synthesis of Kahalalide B and Its Analogues

Addenda and Errata

0970
Expedient Total Synthesis of Kinamycin F
0970
Enantioselective Synthesis of Substituted Indanones