DOI: 10.1055/s-00000131

Synfacts

Issue 02 · Volume 2009 · February 2009 DOI: 10.1055/s-002-15179

Synform

A1
Zanda, Matteo: SYNFORM ISSUE 2009/01

Synthesis of Natural Products and Potential Drugs

0117
Canales, E.; Corey, E. J.: Synthesis of Estrone Methyl Ether
0118
Evans, P. A.; Andrews, W. J.: Synthesis of (+)-Leucascandrolide A Macrolactone
0119
Burgey, C. S.; Paone, D. V.; Shaw, A. W.; Deng, J. Z.; Nguyen, D. N.; Potteiger, C. M.; Graham, S. L.; Vacca, J. P.; Williams, T. M.: Synthesis of Telcagepant (MK-0974)
0120
Yao, Y.-S.; Yao, Z.-J.: Syntheses of Cassiarins A and B
0121
Ebner, D. C.; Trend, R. M.; Genet, C.; McGrath, M. J.; O’Brien, P.; Stoltz, B. M.: Synthesis of (-)-Amurensinine
0122
Tiefenbacher, K.; Mulzer, J.: Formal Synthesis of (-)-Platencin
0123
Paterson, I.; Razzak, M.; Anderson, E. A.: Synthesis of Saliniketal B
0124
Navarro, I.; Basset, J.-F.; Hebbe, S.; Major, S. M.; Werner, T.; Howsham, C.; Bräckow, J.; Barrett, A. G. M.: Synthesis of 15G256β
0125
Takahashi, K.; Midori, M.; Kawano, K.; Ishihara, J.; Hatakeyama, S.: Synthesis of (-)-Salinosporamide A
0126
Varin, M.; Barré, E.; Iorga, B.; Guillou, C.: Synthesis of (±)-Codeine
0127
Sakakura, A.; Umemura, S.; Ishihara, K.: Synthesis of Fluvibactin
0128
Yun, S. Y.; Zheng, J.-C.; Lee, D.: Formal Synthesis of Platencin
0129
Fleck, M.; Bach, T.: Synthesis of ()-Punctaporonin C
0130
Cheung, L. L.; Marumoto, S.; Anderson, C. D.; Rychnovsky, S. D.: Synthesis of SCH 351448
0131
Guo, H.; Mortensen, M. S.; O’Doherty, G. A.: Formal Synthesis of RK-397

Synthesis of Heterocycles

0133
Shaabani, A.; Maleki, A.; Mofakham, H.: One-Pot Three-Component Synthesis of Tetrahydro-1H-1,5-benzodiazepines
0134
Shaaban, M. R.: Microwave-Assisted Synthesis of Trifluoromethyl-Containing Heterocycles
0135
Lv, X.; Liu, Y.; Qian, W.; Bao, W.: Cu-Catalyzed Heteroannulation Route to 2-Iminobenzo-1,3-oxathioles
0136
Samanta, S.; Mohapatra, H.; Jana, R.; Ray, J. K.: Intramolecular Heck Route to 5-, 6-, and 7-Membered O-Containing Heterocycles
0137
Fischer, D.; Tomeba, H.; Pahadi, N. K.; Patil, N. T.; Huo, Z.; Yamamoto, Y.: Synthesis of Isoquinolines by I2-Mediated Electrophilic Heteroannulation
0138
Feroci, M.; Chiarotto, I.; Rossi, L.; Inesi, A.: The Gewald Synthesis of 2-Aminothiophenes using Activated Sulfur
0139
Grigg, R.; Sridharan, V.; Shah, M.; Mutton, S.; Kilner, C.; MacPherson, D.; Milner, P.: Pd-Catalyzed Three-Component Synthesis of Isoindolones and Phthalazones
0140
Melkonyan, F.; Topolyan, A.; Yurovskaya, M.; Karchava, A.: Concise Cu-Catalyzed Synthesis of 3-Carboxyl-N-Aminoindoles
0141
Jordan-Hore, J. A.; Johansson, C. C. C.; Gulias, M.; Beck, E. M.; Gaunt, M. J.: Oxidative Pd(II)-Catalyzed C-H Bond Activation Route to Carbazoles
0142
Teimouri, M. B.; Mansouri, F.: One-Pot Three-Component Synthesis of 7H-Phenaleno[1,2-b]furan-7-ones
0143
Wang, Y.-F.; Toh, K. K.; Chiba, S.; Narasaka, K.: Mn(III)-Catalyzed Synthesis of Pyrroles from 1,3-Dicarbonyls and Vinyl Azides
0144
Khankischpur, M.; Kurz, T.: Microwave-Assisted Synthesis of 1,2,4-Triazolium Ylides
0145
Han, B.; Li, J.-L.; Ma, C.; Zhang, S.-J.; Chen, Y.-C.: Organocatalytic Asymmetric Inverse-Electron-Demand Aza-Diels-Alder Reaction
0146
Ghosh, D.; Thander, L.; Ghosh, S. K.; Chattopadhyay, S. K.: Aza-Claisen-RCM Route to 1-Benzazepine Derivatives
0147
Cheng, X.; Vellalath, S.; Goddard, R.; List, B.: Direct Catalytic Asymmetric Synthesis of Cyclic Aminals from Aldehydes

Synthesis of Materials and Unnatural Products

0149
Briquel, R.; Mazzolini, J.; Bris, T. Le; Boyron, O.; Boisson, F.; Delolme, F.; D’Agosto, F.; Boisson, C.; Spitz, R.: Functional End-Capping for PE
0150
Loudet, A.; Bandichhor, R.; Burgess, K.; Palma, A.; McDonnell, S. O.; Hall, M. J.; O’Shea, D. F.: Design and Synthesis of Near-IR Fluorophores
0151
Walker, W.; Veldman, B.; Chiechi, R.; Patil, S.; Bendikov, M.; Wudl, F.: Antiaromatic Lowering of the HOMO-LUMO Gap
0152
Shimizu, M.; Mochida, K.; Hiyama, T.: Silicon-Bridged Biaryls
0153
Finke, A. D.; Moore, J. S.: 1,3,5-Polyphenylene Dendron Synthesis by C-H Activation
0154
Feng, X.; Feng, F.; Yu, M.; He, F.; Xu, Q.; Tang, H.; Wang, S.; Li, Y.; Zhu, D.: Tyrosinase Activity Sensor
0155
Gug, S.; Bolze, F.; Specht, A.; Bourgogne, C.; Goeldner, M.; Nicoud, J.-F.: A Protecting Group for Two-Photon Uncaging
0156
Matsuo, Y.; Iwashita, A.; Abe, Y.; Li, C.-Z.; Matsuo, K.; Hashiguchi, M.; Nakamura, E.: Efficient Regioselective 1,4-Substitution of [60]Fullerenes
0157
Velasco, V. M.; Zolotukhin, M. G.; Guzmán-Gutiérrez, M. T.; Morales, S. L.; Fomine, S.; Carreón-Castro, M. P.; Salmón, M.; Scherf, U.: Aromatic Polymers with Pentafluorophenyl Groups
0158
Wu, L.; Burgess, K.: Everything’s Coming Up Rosamine
0159
Ralli, P.; Zhang, Y.; Lemal, D. M.: Perfluorobarrelene
0160
Neelakandan, P. P.; Ramaiah, D.: DNA-Assisted Long-Lived Excimer Formation in a Cyclophane
0161
Riehm, T.; De Paoli, G.; Wadepohl, H.; De Cola, L.; Gade, L. H.: A Handle for Perylene Dyes

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

0163
Kim, D. E.; Lee, B. H.; Rajagopalasarma, M.; Genêt, J.-P.; Ratovelomanana-Vidal, V.; Jeong, N.: Desymmetrization of Diallyl Acetals of Alkynals by Rodium Catalysis
0164
Yang, D.; Long, Y.; Wang, H.; Zhang, Z.: Iridium-Catalyzed Ring-Opening Reactions with Secondary Amines
0165
Shintani, R.; Park, S.; Shirozu, F.; Murakami, M.; Hayashi, T.: Palladium-Catalyzed Synthesis of Chiral Lactams from Racemic Lactones
0166
Aydin, J.; Conrad, C. S.; Szabó, K. J.: Mild Protocol for the Synthesis of syn-1,2-Aminonitriles
0167
Seiser, T.; Cramer, N.: Cyclohexenones via C-C Bond Activation of Allenyl Cyclobutanes
0168
Tan, C.; Liu, X.; Wang, L.; Wang, J.; Feng, X.: Asymmetric Aza-Henry Reaction of Ketoimines
0169
Zheng, K.; Shi, J.; Liu, X.; Feng, X.: Carbonyl-Ene Reaction Catalyzed by N,N′-Dioxide-Nickel(II) Complex
0170
Qiu, M.; Hu, X.-P.; Huang, J.-D.; Wang, D.-Y.; Deng, J.; Yu, S.-B.; Duan, Z.-C.; Zheng, Z.: A New Phosphine-Aminophosphine Ligand for Enantioselective Hydrogenation
0171
Thu, H.-Y.; Tong, G. S.-M.; Huang, J.-S.; Chan, S. L.-F.; Deng, Q.-H.; Che, C.-M.: Selective Carbene Insertion into Primary C-H Bonds
0172
Yue, T.; Wang, M.-X.; Wang, D.-X.; Zhu, J.: Aluminum Salen Passerini-Type Synthesis of 5-(1-Hydroxyalkyl)tetrazoles
0173
Xu, X.; Zhou, J.; Yang, L.; Hu, W.: Rhodium-Catalyzed Enantioselective Multicomponent Reaction
0174
Li, Z.-W.; Wang, T.-L.; He, Y.-M.; Wang, Z.-J.; Fan, Q.-H.; Pan, J.; Xu, L.-J.: Synthesis of Chiral Tetrahydroquinolines by Asymmetric Hydrogenation
0175
Jautze, S.; Peters, R.: Bimetallic Palladium Catalyzed Michael Addition of α-Cyanoacetates
0176
Chen, I.-H.; Oisaki, K.; Kanai, M.; Shibasaki, M.: Copper(I)-Catalyzed Hetero-Diels-Alder Reaction of Ketones
0177
Du, Y.; Xu, L.-W.; Shimizu, Y.; Oisaki, K.; Kanai, M.; Shibasaki, M.: Copper-Catalyzed Asymmetric Reductive Mannich Reaction
0178
Morimoto, H.; Yoshino, T.; Yukawa, T.; Lu, G.; Matsunaga, S.; Shibasaki, M.: Lewis Base Assisted Brønsted Base: Phosphine Oxides and La-Aryloxides
0179
Hernández-Toribio, J.; Arrayás, R. G.; Carretero, J. C.: Copper-Catalyzed Mannich Reaction of Glycinate Schiff Bases with Imines
0180
Trost, B. M.; Ferreira, E. M.; Gutierrez, A. C.: Metal-Catalyzed Syntheses of cis- or trans-Fused Bicyclic Compounds
0181
Hénon, H.; Mauduit, M.; Alexakis, A.: 1,4- versus 1,6-Selective Asymmetric Copper-Catalyzed Conjugate Addition
0182
Reynolds, T. E.; Binkley, M. S.; Scheidt, K. A.: Addition to Sulfinylimines via Brook Rearrangement of Hydroxypropargylsilanes
0183
Ito, H.; Sasaki, Y.; Sawamura, M.: Copper(I)-Catalyzed Substitution of Propargylic Carbonates with Diboron
0184
Adachi, S.; Harada, T.: Oxazaborolidione-Catalyzed Asymmetric Mukaiyama Aldol Reaction of Ketones
0185
Bercot, E. A.; Caille, S.; Bostick, T. M.; Ranganathan, K.; Jensen, R.; Faul, M. M.: Quaternary Center Formation via Diastereoselective Arylation of Enolates
0186
Cho, H. Y.; Morken, J. P.: Ni-Catalyzed Diastereoselective Coupling of Dienes and Aldehydes
0187
Zhao, J.-F.; Tsui, H.-Y.; Wu, P.-J.; Lu, J.; Loh, T.-P.: In(III)-PyBox Complex Catalyzed Enantioselective Carbonyl-ene Reaction
0188
Li, Z.; Gao, Y.; Jiao, Z.; Wu, N.; Wang, D. Z.; Yang, Z.: A Protocol for Palladium(II)-Mediated Alkoxycarbonylation

Metal-Mediated Synthesis

0189
Cahiez, G.; Gager, O.; Lecomte, F.: Mn-Catalyzed Cross-Coupling of Aryl Grignard Reagents with Alkenyl Halides
0190
Fu, Y.; Wang, J.-X.; Wang, K.; Hu, Y.: Efficient Ni(II)-Catalyzed Dialkylation of Aromatic Aldehydes
0191
Wilson, D. A.; Wilson, C. J.; Rosen, B. M.; Percec, V.: Ni-Catalyzed One-Pot Neopentylglycol-borylation
0192
Do, H.-Q.; Khan, R. M. Kashif; Daugulis, O.: Efficient Cu/Phenanthroline-Catalyzed Arylation of sp² C-H Bonds
0193
Herzon, S. B.; Hartwig, J. F.: Ta(V)-Catalyzed Hydroaminoalkylation of Olefins with Dialkylamines
0194
Williams, C. M.; Johnson, J. B.; Rovis, T.: Ni-Catalyzed Reductive Carboxylation of Styrenes Using CO2
0195
Berman, A. M.; Lewis, J. C.; Bergman, R. G.; Ellman, J. A.: Direct Arylation of α-Substituted Pyridines and Quinolines
0196
Rodríguez-Solla, H.; Simal, C.: Addition of LiCH2I to Imines: An Efficient Synthesis of Aziridines
0197
Alacid, E.; Nájera, C.: Cross-Coupling of Aryltrifluoroborates with Organic Chlorides in Aqueous Media
0198
Yasui, E.; Wada, M.; Takamura, N.: Synthesis of Aryl Hydrazones from α-Diazo Esters
0199
Yuda, S. S.; Kuninobu, Y.; Takai, K.: Re-Catalyzed Cycloaddition of β-Keto Esters to Aliphatic Allenes
0200
Quasdorf, K. W.; Tian, X.; Garg, N. K.: Ni-Catalyzed Cross-Coupling of Aryl Pivalates with Arylboronic Acids
0201
Augustine, J. K.; Naik, Y. A.; Vairaperumal, V.; Narasimhan, S.: Di-tert-butyl Dicarbonate: A Versatile Carboxylating Agent
0202
Zhang, W.-X.; Nishiura, M.; Hou, Z.: Rare Earth Metal Catalyzed Cross-Coupling of Isocyanides
0203
Zhang, L.; Qing, J.; Yang, P.; Wu, J.: Hiyama Cross-Coupling of Aryl Mesylates

Organo- and Biocatalysis

0205
Uraguchi, D.; Asai, Y.; Ooi, T.: Organocatalytic Peptide Modification
0206
Nakayama, K.; Maruoka, K.: Opposite Catalyst Selectivities Using a Common Chiral Source
0207
Hatano, M.; Maki, T.; Moriyama, K.; Arinobe, M.; Ishihara, K.: Chiral Brønsted Acid-Base Pyridinium Disulfonate Catalysts
0208
Lakhdar, S.; Tokuyasu, T.; Mayr, H.: Insights into Iminium Catalysis
0209
Graham, T. H.; Jones, C. M.; Jui, N. T.; MacMillan, D. W. C.: α-Alkylation of Aldehydes with Styrenes
0210
Rueping, M.; Antonchick, A. P.: Catalytic Asymmetric Aza-Cope Rearrangement
0211
Hayashi, Y.; Samanta, S.; Itoh, T.; Ishikawa, H.: Catalytic Asymmetric ”Aldol" Reaction
0212
Yang, Y.-Q.; Zhao, G.: Primary-Secondary Diamine Catalysts for Malonate Additions to Enones
0213
Hahn, B. T.; Fröhlich, R.; Harms, K.; Glorius, F.: Proline Catalyzed anti-Selective Mannich Reaction
0214
Jang, D. O.; Kim, S. Y.: Radical Addition to C=N Bonds Mediated by Chiral Ammonium Salts
0215
Ganesh, M.; Seidel, D.: Highly Active Catalyst for the Addition of Indoles to Nitroalkenes
0216
Rommel, M.; Fukuzumi, T.; Bode, J. W.: NHC-Catalyzed Annulation of Enals to Cyclic Ketimines
0217
Chi, Y.; Scroggins, S. T.; Boz, E.; Fréchet, J. M. J.: Biomimetic Chemoselectivity Control of Aldol Reactions
0218
Huang, X.-L.; He, L.; Shao, P.-L.; Ye, S.: NHC-Catalyzed [4+2] Cycloaddition of Ketenes with N-Benzoyldiazenes

Polymer-Supported Synthesis

0219
Ceylan, S.; Friese, C.; Lammel, C.; Mazac, K.; Kirschning, A.: Magnetic Nanoparticles as Inductive Heating Elements in Microreactors
0220
Motoyama, Y.; Abe, M.; Kamo, K.; Kosako, Y.; Nagashima, H.: Isomerization of Allyl Ethers with [Ru3]@SiEGcap
0221
Carrera, N.; Gutiérrez, E.; Benavente, R.; Villavieja, M. M.; Albéniz, A. C.; Espinet, P.: Clean Stille Reaction with Recyclable Stannylated Polynorbornenes
0222
Trilla, M.; Borja, G.; Pleixats, R.; Man, M. W. C.; Bied, C.; Moreau, J. J. E.: Silica-Supported Palladium Catalysts for Suzuki-Miyaura Reactions
0223
Kantam, M. L.; Chakravarti, R.; Chintareddy, V. R.; Sreedhar, B.; Bhargava, S.: Sequential Heck Coupling and Hydrogenation
0224
Motokura, K.; Tada, M.; Iwasawa, Y.: Synthesis of 1,3-Dinitroalkanes with Immobilized Amines
0225
Monguchi, Y.; Kitamoto, K.; Ikawa, T.; Maegawa, T.; Sajiki, H.: C-N Coupling Reaction Catalyzed by Palladium on Carbon
0226
García, J. I.; Lópes-Sánchez, B.; Mayoral, J. A.: A Self-Assembled Coodination Polymer as a Homo- and Heterogeneus Catalyst
0227
Kiasat, A. R.; Badri, R.; Zargar, B.; Sayyahi, S.: Regioselective Azidolysis of Epoxides in Water Using PEG-Grafted Dowex Resin
0228
Kim, J. W.; Yamaguchi, K.; Mizuno, N.: Oxygenation of Primary Amines to Amides by Ru(OH)x/Al2O3
0229
Pande, S.; Saha, A.; Jana, S.; Sarkar, S.; Basu, M.; Pradhan, M.; Sinha, A. K.; Saha, S.; Pal, A.; Pal, T.: Alcohol Oxidation with Resin-Immoblized Cu Nanocomposites
0230
Jiang, H.-y; Yang, C.-f; Li, C.; Fu, H.-y; Chen, H.; Li, R.-x; Li, X.-j: Asymmetric Hydrogenation of Ketones Using Ir/SiO2/Ph3P/Diamine Catalysts
0231
Sakai, H.; Tsutsumi, K.; Morimoto, T.; Kakiuchi, K.: Silica-Supported Palladium-Catalyzed Synthesis of Indole Derivatives
0232
Wiles, C.; Watts, P.: Strecker Reaction in Microreactor