DOI: 10.1055/s-00000131

Synfacts

Issue 01 · Volume 2011 · January 2011 DOI: 10.1055/s-002-21566

Synform

A1
Zanda, Matteo: SYNFORM ISSUE 2011/01

Synthesis of Natural Products and Potential Drugs

z1
All PDFs of this category
0001
Marsini, M. A.; Reider, P. J.; Sorensen, E. J.: Synthesis of PA-824
0002
Burns, A. R.; McAllister, G. D.; Shanahan, S. E.; Taylor, R. J. K.: Synthesis of (+)-Dictyosphaeric Acid A
0003
Valenta, P.; Carroll, P. J.; Walsh, P. J.: Synthesis of PRC200-SS
0004
Breyer, S.; Effenberger-Neidnicht, K.; Schobert, R.: Synthesis of (-)-Thespesone
0005
Tatsuta, K.; Tanaka, H.; Tsukagoshi, H.; Kashima, T.; Hosokawa, S.: Synthesis of Lactonamycin
0006
Zuo, Z.; Xie, W.; Ma, D.: Synthesis of (-)-Communesin F
0007
Ko, J. S.; Keum, J. E.; Ko, S. Y.: Synthesis of Oseltamivir
0008
Zhu, Y.; Loudet, A.; Burgess, K.: Synthesis of (-)-Spongidepsin
0009
Flyer, A. N.; Si, C.; Myers, A. G.: Synthesis of Cortistatins A, J, K and L
0010
Gu, Z.; Zakarian, A.: Synthesis of Rhazinilam
0011
Li, H.; Xu, R.; Cole, D.; Clader, J. W.; Greenlee, W. J.; Nomeir, A. A.; Song, L.; Zhang, L.: Synthesis of a γ-Secretase Inhibitor
0012
Bezençon et al., O.: Synthesis of ACT-178882 (MK-1597)
0013
Duthion, B.; Pardo, D. Gomez; Cossy, J.: Synthesis of LY503430

Synthesis of Heterocycles

z15
All PDFs of this category
0015
Álvarez, R.; Martínez, C.; Madich, Y.; Denis, J. G.; Aurrecoechea, J. M.; de Lera, Á. R.: Benzofurans, Indoles, and Isoquinolones via Castro-Stephens and Heck Reactions
0016
Dong, C.; Xie, L.; Mou, X.; Zhong, Y.; Su, W.: Palladium-Catalyzed Synthesis of 1,3,4-Benzotriazepines and Indazoles
0017
Li, R.-J.; Pi, S.-F.; Liang, Y.; Wang, Z.-Q.; Song, R.-J.; Chen, G.-X.; Li, J.-H.: Palladium-Catalyzed Annulation Route to 6H-Benzo[c]chromenes
0018
Muthusaravanan, S.; Perumal, S.; Yogeeswari, P.; Sriram, D.: Substituted Indolizines via a Multicomponent 1,3-Dipolar Cycloaddition Strategy
0019
Liu, C.; Zhang, X.; Wang, R.; Wang, W.: Synthesis of 4H-Chromenes by an Enantio-selective Oxa-Michael-Aldol Reaction
0020
Chen, J.; Ma, S.: Regioselective Synthesis of 2-Alkoxyfurans from Cyclopropenyl Carboxylates
0021
Ballini, R.; Gabrielli, S.; Palmieri, A.; Petrini, M.: Metal-Free Synthesis of 1,4-Disubstituted Carbazoles from Sulfonylindoles
0022
Morin, M. S. T.; St-Cyr, D. J.; Arndtsen, B. A.: Horner-Wadsworth-Emmons Reagent as 1,3-Dipolar Cycloaddition Precursor
0023
Ouizem, S.; Cheramy, S.; Botuha, C.; Chemla, F.; Ferreira, F.; Pérez-Luna, A.: Cyclization of Zincated Homoallylamino Nitriles to Methanopyrrolidines
0024
Lourdusamy, E.; Yao, L.; Park, C.-M.: Synthesis of Pyrroles by [3+2] Cycloaddition of α-Diazo Oxime Ethers with Alkenes
0025
Patil, N. T.; Raut, V. S.: Metal/Amine Cooperative Catalysis. Heteroannulation Route to Quinolines
0026
Jacq, J.; Bessières, B.; Einhorn, C.; Einhorn, J.: 1,3-Diaryl Isobenzofurans from Arylboronic Acids and ortho-Keto Aldehydes
0027
Yagoubi, M.; Cruz, A. C. F.; Nichols, P. L.; Elliott, R. L.; Willis, M. C.: Palladium-Catalyzed Heteroannulation Route to Indoles and Benzofurans
0028
Seki, H.; Georg, G. I.: Synthesis of Dihydropyridin-4(1H)-ones via Wolff Rearrangement
0029
Zeng, L.-Y.; Cai, C.: Multicomponent Synthesis of Azaphenanthreneamides

Synthesis of Materials and Unnatural Products

z31
All PDFs of this category
0031
Matsuda, T.; Yamaguchi, Y.; Ishida, N.; Murakami, M.: A Versatile Synthetic Method for Silaindenes
0032
Roznyatovskiy, V.; Lynch, V.; Sessler, J. L.: Dinaphthoporphycenes Made Easy
0033
Ito, A.; Yokoyama, Y.; Aihara, R.; Fukui, K.; Eguchi, S.; Shizu, K.; Sato, T.; Tanaka, K.: Polyaniline Rings
0034
Lesbani, A.; Kondo, H.; Sato, J.-i.; Yamanoi, Y.; Nishihara, H.: A New Method for Hypersilyl Aromatic Compounds
0035
Pei, B.-J.; Chan, W.-H.; Lee, A. W. M.: Oxadisilole Groups as a Benzyne Precursor and a Route to Triptycenes
0036
Nelson, T. L.; Young, T. M.; Liu, J.; Mishra, S. P.; Belot, J. A.; Balliet, C. L.; Javier, A. E.; Kowalewski, T.; McCullough, R. D.: Tailor-Made Donor-Acceptor Polymer for OFETs
0037
Sugiyasu, K.; Honsho, Y.; Harrison, R. M.; Sato, A.; Yasuda, T.; Seki, S.; Takeuchi, M.: Threaded Polythiophene
0038
Li, F.-B.; You, X.; Wang, G.-W.: Fullerene-Fused Lactones
0039
Kobayashi, M.; Matsuo, T.; Fukunaga, T.; Hashizume, D.; Fueno, H.; Tanaka, K.; Tamao, K.: Stable Conjugated Disilenes
0040
Simkowa, I.; Latos-Graźyński, L.; Stępień, M.: π Conjugation Through a Ferrocenothia-porphyrin Macrocycle
0041
Wei, J.; Han, B.; Guo, Q.; Shi, X.; Wang, W.; Wei, N.: 1,5,9-Triazacoronenes
0042
Ando, S.; Facchetti, A.; Marks, T. J.: Overcoming Insolubility Towards Thin Films
0043
Portius, P.; Filippou, A. C.; Schnakenburg, G.; Davis, M.; Wehrstedt, K.-D.: Taming the Silicon Tetraazide Beast
0044
Pardo, E.; Ferrando-Soria, J.; Dul, M.-C.; Lescouëzec, R.; Journaux, Y.; Ruiz-García, R.; Cano, J.; Julve, M.; Lloret, F.; Cañadillas-Delgado, L.; Pasán, J.; Ruiz-Pérez, C.: Double-Stranded Copper(II) meso-Helicates

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z45
All PDFs of this category
0045
Usanov, D. L.; Yamamoto, H.: Asymmetric Propargylation of Benzaldehydes
0046
Arai, T.; Yokoyama, N.; Mishiro, A.; Sato, H.: Stereoselective [3+2] Cycloaddition of Imino Esters with Nitroalkenes
0047
Denmark, S. E.; Kalyani, D.; Collins, W. R.: Lewis Base Catalyzed Asymmetric Selenoetherification
0048
Liang, G.; Tong, M.-C.; Tao, H.; Wang, C.-J.: Synthesis of Chiral α,β-Diamino Acids Using Copper(I)/TF-BiphamPhos
0049
Rankic, D. A.; Lucciola, D.; Keay, B. A.: Modification of BINAP Ligand has Profound Effect in Intramolecular Heck Reactions
0050
Uraguchi, D.; Ito, T.; Nakamura, S.; Ooi, T.: Asymmetric Hydrophosphonylation of Ynones
0051
Trost, B. M.; Czabaniuk, L. C.: Asymmetric Benzylation of 3-Aryl Oxindoles
0052
Fang, Y.-Q.; Bio, M. M.; Hansen, K. B.; Potter, M. S.; Clausen, A.: Magnesium-Promoted N-Selective Alkylation of Amides and Carbamates
0053
Chen, J.-P.; Ding, C.-H.; Liu, W.; Hou, X.-L.; Dai, L.-X.: Acylsilanes as Pronucleophiles in Palladium-Catalyzed Asymmetric Allylic Alkylation
0054
Worthy, A. D.; Joe, C. L.; Lightburn, T. E.; Tan, K. L.: Substrate-Binding Phosphine Ligand in Enantioselective Hydroformylation
0055
Trost, B. M.; Osipov, M.; Dong, G.: Pd-Catalyzed Asymmetric Allylic Alkylation of Heterocycles with Vinyl Aziridines
0056
Zhou, X.; Zhang, Q.; Hui, Y.; Chen, W.; Jiang, J.; Lin, L.; Liu, X.; Feng, X.: Asymmetric Hydrophosphonylation of Trifluoromethyl Ketones
0057
Hartog, T. den; Rudolph, A.; Maciá, B.; Minnaard, A. J.; Feringa, B. L.: Enantioselective Synthesis of trans-1-Alkyl-
2-Substituted Cyclopropanes
0058
Kim, H.; Yun, J.: Copper-Catalyzed 1,4-Hydroboration of Coumarins with Pinacolborane
0059
Sakakura, A.; Hori, M.; Fushimi, M.; Ishihara, K.: Enantioselective Cycloaddition of Nitrones with Propioloyl- and Acryloylpyrazoles
0060
Gourdet, B.; Lam, H. W.: Asymmetric Dihydroxylation of Enamides to Give Quaternary Alcohols
0061
Pattison, G.; Piraux, G.; Lam, H. W.: Asymmetric Rhodium-Catalyzed Addition of Arylboronic Acids to Alkenylheteroarenes
0062
Zhao, J.-F.; Tjan, T.-B. W.; Loh, T.-P.: Improved Reactivity in the Carbonyl-Ene Reaction Due to Counterion Effects
0063
Tamura, K.; Sugiya, M.; Yoshida, K.; Yanagisawa, A.; Imamoto, T.: Rhodium-Catalyzed Asymmetric Hydrogenation with a P-Stereogenic Ligand
0064
Tian, F.; Yao, D.; Liu, Y.; Xie, F.; Zhang, W.: Iridium-Catalyzed Asymmetric Hydrogenation of Exocyclic Ketones, Lactones, and Lactams
0065
Tran, D. N.; Cramer, N.: Rhodium-Catalyzed Domino C-H Activation-Intramolecular Allylation of Imines
0066
Ramachandran, P. V.; Parthasarathy, G.; Gagare, P. D.: Stereoselective Enolboration of α-Trifluoro-methylpropionates
0067
Huang, Y.; Pullarkat, S. A.; Li, Y.; Leung, P.-H.: Palladium(II)-Catalyzed Asymmetric Hydrophosphination of Enones
0068
Cheon, C. H.; Imahori, T.; Yamamoto, H.: Lewis Acid Assisted Brønsted Acid Catalyzed Asymmetric Protonation Reaction
0069
Zhou, S.; Fleischer, S.; Junge, K.; Das, S.; Addis, D.; Beller, M.: Iron-Catalyzed Enantioselective Transfer Hydrogenation of Imines
0070
Wencel-Delord, J.; Alexakis, A.; Crévisy, C.; Mauduit, M.: Copper-Catalyzed 1,6-Conjugate Addition to Cyclic Dienones
0071
Zhao, J.-F.; Tan, B.-H.; Zhu, M.-K.; Tjan, T.-B. W.; Loh, T.-P.: Indium-Catalyzed Enantioselective Carbonyl-Ene Reaction of Trifluoropyruvate
0072
Sasaki, K.; Hayashi, T.: Asymmetric Conjugate Addition to Borylalkenes
0073
Hasegawa, Y.; Gridnev, I. D.; Ikariya, T.: Bifunctional Catalysts for Asymmetric Conjugate Addition
0074
Gou, F.-R.; Li, W.; Zhang, X.; Liang, Y.-M.: Iridium-Catalyzed Enantioselective Hydrogenation of Quinoline Derivatives

Metal-Mediated Synthesis

z75
All PDFs of this category
0075
Tsvelikhovsky, D.; Buchwald, S. L.: Pd-Ligand Controlled Cyclization for the Preparation of Heteroaromatics
0076
Ball, L. T.; Green, M.; Lloyd-Jones, G. C.; Russell, C. A.: Gold-Catalyzed Oxyarylation of Alkenes
0077
Brenzovich, Jr., W. E.; Brazeau, J.-F.; Toste, F. D.: Gold-Catalyzed Oxidative Coupling Reactions
0078
Chu, L.; Qing, F.-L.: Copper-Catalyzed Oxidative Trifluoromethylation of Boronic Acids
0079
Werner, E. W.; Sigman, M. S.: A Selective and General Palladium Catalyst for the Oxidative Heck Reaction
0080
Nakao, Y.; Yamada, Y.; Kashihara, N.; Hiyama, T.: Selective C4 Alkylation of Pyridines Using Nickel/Lewis Acid Catalysis
0081
Molander, G. A.; Hiebel, M.-A.: Synthesis and Reactions of Amidomethyl-trifluoroborates
0082
Barluenga, J.; Escribano, M.; Aznar, F.; Valdés, C.: Arylation of α-Chiral Ketones via
Cross-Coupling of Tosylhydrazones
0083
Kinzel, T.; Zhang, Y.; Buchwald, S. L.: A New Palladium Precatalyst for the Suzuki Coupling of Unstable Boronic Acids
0084
Tran, L. D.; Daugulis, O.: Iron-Catalyzed Deprotonative Alkylation of (Hetero)Arenes
0085
Custar, D. W.; Le, H.; Morken, J. P.: Palladium-Catalyzed Carbonylative Conjugate Addition of Dialkylzinc Reagents
0086
Hirone, N.; Sanjiki, H.; Tanaka, R.; Hata, T.; Urabe, H.: Substitution of Silanes with Grignard Reagents
0087
Barker, G.; O’Brien, P.; Campos, K. R.: Diamine-Free Lithiation of N-Boc Hetero-cycles in THF
0088
Tsubouchi, A.; Enatsu, S.; Kanno, R.; Takeda, T.: Regio- and Stereoselective Silyl Enol Ethers
0089
Ely, R. J.; Morken, J. P.: Nickel(0)-Catalyzed 1,4-Diborylation of Conjugated Dienes

Organo- and Biocatalysis

z91
All PDFs of this category
0091
Kanzian, T.; Lakhdar, S.; Mayr, H.: The Increased Reactivity of the Proline Carboxylate Derived Enamine
0092
Zhou, L.; Tan, C. K.; Jiang, X.; Chen, F.; Yeung, Y.-Y.: Cinchona Amino-Thiocarbamate Catalyzed Bromolactonization
0093
Murai, K.; Matsushita, T.; Nakamura, A.; Fukushima, S.; Shimura, M.; Fujioka, H.: Chiral Trisimidazoline Catalyzed Bromolactonization
0094
Liang, T.; Zhang, Z.; Antilla, J. C.: Brønsted Acid Catalyzed Asymmetric Pinacol Rearrangement
0095
Biju, A. T.; Glorius, F.: An Umpolung Reaction of Aldehydes with Arynes
0096
De Sarkar, S.; Studer, A.: NHC-Catalyzed Michael Addition to α,β-Unsaturated Aldehydes
0097
Liu, X.; Lu, Y.: Synthesis of Dihydroquinolones Using a Bifunctional Thiourea Catalyst
0098
Zhang, Z.; Xie, F.; Jia, J.; Zhang, W.: A Simple Lewis Base Catalyst for the Asymmetric Steglich Rearrangement
0099
Leverett, C. A.; Purohit, V. C.; Romo, D.: Organocatalytic Construction of Polycyclic Compounds
0100
Sohtome, S.; Tanaka, S.; Takada, K.; Yamaguchi, T.; Nagasawa, K.: Enantioswitching Catalysis with a Single Chiral Organocatalyst
0101
Bergonzini, G.; Vera, S.; Melchiorre, P.: γ-Alkylation of α-Branched Enals with Stable Carbocations
0102
Rossi, S.; Benaglia, M.; Genoni, A.; Benincori, T.; Celentano, G.: Diphosphine Oxide Catalyzed Direct Aldol Reactions
0103
Guo, Q.; Bhanushali, M.; Zhao, C.-G.: Quinidine Thiourea Catalyzed Aldol Reaction of Unactivated Ketones

Polymer-Supported Synthesis

z105
All PDFs of this category
0105
Dang, D.; Wu, P.; He, C.; Xie, Z.; Duan, C.: Asymmetric Catalysis with MOFs Prepared via Chiral Induction Effect
0106
Li, Y.; Wang, H.; Li, X.; Chen, T.; Zhao, D.: Coupling of Aryl Halides and Diaryl Diselenides with CuS/Fe
0107
Akagawa, K.; Fujiwara, T.; Sakamoto, S.; Kudo, K.: A One-Pot Tandem Reaction System Using Resin-Supported Peptide
0108
Wang, Y.; Ouyang, G.; Zhang, J.; Wang, Z.: Reduction of Nitrobenzenes and Oxidation of Alcohols with M-DNA
0109
Ranganath, K. V. S.; Kloesges, J.; Schäfer, A. H.; Glorius, F.: Asymmetric Arylation of Ketones with Chiral NHC Modified Fe3O4/Pd Nanoparticles
0110
Fujita, K.-i.; Yamazaki, M.; Ainoya, T.; Tsuchimoto, T.; Yasuda, H.: Dihydroxylation of Olefins with Dendric Osmium Complex
0111
Wang, Q.; Zhang, M.; Chen, C.; Ma, W.; Zhao, J.: Photocatalytic Aerobic Oxidation of Alcohols on TiO2
0112
Dimroth, J.; Keilitz, J.; Schedler, U.; Schomäcker, R.; Haag, R.: Asymmetric Transfer Hydrogenation of Ketones by Supported Rh-TsDPEN
0113
Pozo, C. del; Corma, A.; Iglesias, M.; Sánchez, F.: Asymmetric Hydrogenation with MCM-41-Supported Pincer Catalysts
0114
Miyamura, H.; Maehata, K.; Kobayashi, S.: In Situ Coupled Oxidation Cycle Catalyzed by Reusable Platinum Catalysts
0115
Yamada, Y. M. A.; Jin, C. K.; Uozumi, Y.: Oxidation of Alcohols by Polymeric Phosphotungstate with H2O2
0116
Palaniappan, S.; Rajender, B.: PANI-AgNO3-PTSA Salt Catalyzed Mannich Reaction
0117
Hu, F.-Q.; Xia, D.-X.; Lu, C.-F.; Chen, Z.-X.; Yang, G.-C.: Polystyrene-Supported Chiral Auxiliary for Asymmetric Alkylation