DOI: 10.1055/s-00000131

Synfacts

Issue 09 · Volume 2009 · September 2009 DOI: 10.1055/s-002-20326

Synthesis of Natural Products and Potential Drugs

z939
All PDFs of this category
0939
Synthesis of Sporolide B
0940
Synthesis of a Polychlorinated Sulpholipid Cytotoxin
0941
Synthesis of Ciguatoxin
0942
Synthesis of (-)-FR182877
0943
Synthesis of Norsertraline
0944
Synthesis of Vinblastine
0945
Synthesis of (+)-Peloruside A
0946
Synthesis of (+)-Serratezomine A
0947
Synthesis of Antiostatin B2
0948
Synthesis of (+)-11-Hydroxyerythratidine
0949
Synthesis of Lysergic Acid Methyl Ester
0950
Synthesis of (-)-PNU-286607
0951
Synthesis of µ-Opioid Selective Ligands
0952
Synthesis of (-)-Spicigerolide
0953
Synthesis of Bacilosarcin A

Synthesis of Heterocycles

z955
All PDFs of this category
0955
Synthesis of Spiro β-Lactams and Oxoindoles by Oxidative Dearomatization
0956
Ring-Closing Metathesis Approach to Quinolizinium Salts
0957
Chemoselective Synthesis of Naphthyridines and Pyrano[3,2-c]pyridines
0958
Photostimulated Intramolecular SRN1 Reaction of Diarylamines to Carbazoles
0959
Copper-Catalyzed C-H Activation for the Synthesis of Benzoxazoles
0960
Synthesis of Pyrroloindoles and Dipyrrolo-pyridines by a Hydroamination Route
0961
General Synthesis of Hantzsch Esters in 2,2,2-Trifluoroethanol
0962
Synthesis of 1,3-Benzothiazines by Catalytic Generation of Cesium Acetylide
0963
Synthesis of 2-Aminobenzothiazoles via Oxidative C-H Functionalization
0964
Synthesis of 4,4-Difluorodihydrofuran-3(2H)-ones
0965
Organocatalytic Synthesis of Benzo[b]thiepines
0966
An Improved Synthesis of Dichloro-pyrazinones
0967
Silver-Catalyzed Synthesis of 2,3-Dihydro-pyrroles
0968
Piperidines from Organocatalytic Inverse-Demand Aza-Diels-Alder Reaction
0969
One-Pot Synthesis of 2-Sulfanylindoles

Synthesis of Materials and Unnatural Products

z971
All PDFs of this category
0971
Synthesis of Push-Pull Pyrroles and their Oxidative Anellation Reaction
0972
Conjugated Borasiloxane Cages
0973
Functional Fullerenes for Electronics
0974
Rapid Access to Diphenyl- and Acenaphthoquinoline Derivatives
0975
Fluorine-Containing Semiconducting Polymers
0976
Benzonaphthyridines from Morita-Baylis-Hillman Adduct Acetates
0977
Synthesis of ortho-Linked Oligo-9,9′-spirobifluorenes
0978
Azulene Photochromes
0979
Graft Copolymers from a Double ROMP
0980
Azulenated Cyanine Dyes
0981
A Breakdown in Communication
0982
Planar Polyselenophenes
0983
Giving a Use to Triazoles
0984
Selective Dimerization of Indolocarbazoles
0985
A Highly Selective Cyanide Sensor

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z987
All PDFs of this category
0987
Ir-Catalyzed Cross-Coupling of Styrene Derivatives with Allylic Carbonates
0988
Platinum-Catalyzed Asymmetric 1,4-Dihydroxylation of 1,3-Dienes
0989
Lanthanum(III)-Binaphthyldisulfonate Complex Catalyzed Strecker Reaction
0990
Synthesis of Quaternary Stereocenters through a Radical Cyclization
0991
Co-Salen Complexes Catalyzed Kinetic Resolution of Terminal Epoxides
0992
Synthesis of α-Hydroxyallenes by SN2′ of Propargylic Dioxolanones
0993
Copper-NHC Catalysts for Asymmetric Conjugate Addition
0994
Rhodium-Catalyzed 1,4-Addition of Arylboronic Acids
0995
Chiral Dinuclear Palladium Complexes in Ring-Opening Reactions
0996
Asymmetric Addition of Terminal Alkynes to Imines Catalyzed by Copper(I)
0997
Iridium-Catalyzed Stereoselective Two-Directional Elongation of 1,3-Polyols
0998
Oxidative Addition of Nucleophiles to Vinyl Oxazolidinones
0999
Titanium-Mediated Cross-Coupling of Aldimines and Allylic Alcohols
1000
Asymmetric Isomerization of Primary Allylic Alcohols
1001
Metal-Mediated Isomerization of Terminal Olefins
1002
Generation and Applications of α-Chiral Allylic Stannanes
1003
Iridium-Catalyzed Hydrogenation of
α,β-Unsaturated Amides
1004
Transfer Hydrogenation in Iterative Elongation of Alcohols
1005
Diastereoselective Hydroarylation for the Synthesis of Dihydrocoumarins
1006
Divergent Cyclization towards Cyclopropanes and Oxetanes
1007
Catalytic Asymmetric α-Addition of Isocyanoacetamides to Aldehydes
1008
H8BINOL-Catalyzed Enantioselective Alkyl Propiolate Addition to Aliphatic Aldehydes
1009
Titanium Superoxide Catalyzed Aminobromination of Olefins
1010
Cyclobutanones via Ring Expansion of Allenylcyclopropanols
1011
A Sterically Demanding NHC Ligand
1012
Ketene Silyl Acetal Addition to Alkynes Gives Alkenylindiums
1013
Nucleophilic Addition of Samarium Enolates to Imines
1014
Chiral β-Hydroxy Ethers from Spiroborate Ester Mediated Reductions

Metal-Mediated Synthesis

z1015
All PDFs of this category
1015
Coupling of Secondary Alkylzinc Halides with Aryl Bromides and Chlorides
1016
CuBr-Mediated Oxyalkylation of Styrenes by Cyclic Ethers
1017
Pd(OTf)2˙2H2O-Catalyzed ortho-Fluorination of Benzyl Triflamides
1018
Cu-Catalyzed Aerobic Oxidative Coupling of Alkynes to H-Phosphonates
1019
Copper(I)-Catalyzed Room-Temperature Borylation of Aryl Halides
1020
2-Pyrazol-5-ylaniline as ortho-Directing Agent for Arylboronic Acids in C-H Silylation
1021
Allylation and Crotylation of Carbonyls Using Organotrifluoroborates
1022
Practical Arene Hydrogenation by Heterogeneous Catalysts
1023
Chemoselective Chemical and Electrochemical Deprotections of Toluates
1024
AgOTf-Mediated Fluorination of Boronic Acids
1025
Synthesis of Diarylmethanes via Pd-Catalyzed α-Arylation of Benzylketones
1026
Ruthenium-Catalyzed Oxidation of Primary Alcohols into Amides
1027
Direct C-H Arylation of Benzene, Naphthalene, and Pyridine
1028
Gold-Catalyzed Synthesis of Piperidin-4-ones
1029
Ni-Catalyzed C-N Bond Formation at the β-Position of Saturated Ketones

Organo- and Biocatalysis

z1031
All PDFs of this category
1031
A Highly Enantioselective α-Bromination?
1032
One-Step Synthesis of Furofuranes
1033
N-Allylic Alkylation of Indoles
1034
One-Pot Synthesis of Bicyclic Isoxazolidines with Five Stereogenic Centers
1035
Enantioselective Aziridination Using Chiral Phosphoric Acids
1036
Enantioselective Ring Opening of meso-Aziridines with TMS-Protected Thiophenol
1037
Formal Alkynylation and Alkenylation of α,β-Unsaturated Aldehydes
1038
Highly Enantioselective Michael Addition to Nitroolefins in Water
1039
Formal [3+2] Cycloaddition with in situ Generated N-Carbamoyl Nitrones
1040
Lewis Base Catalysts Containing Axial Chirality of Allenes
1041
Asymmetric Epoxidation of Electron-Deficient α,β-Enones
1042
NHC-Catalyzed Redox Amidation of α-Hydroxyenones
1043
Highly Selective Formal [3+3] Cyclohexenone Annulation
1044
Enzymatic Control over Self- and Cross-Aldol Reactions

Polymer-Supported Synthesis

z1045
All PDF of this category
1045
Optical Resolution with Immobilized Enzymes on Nanoparticles
1046
Tandem Condensation Reactions with H-mont-NH2
1047
Benzylidene Diacetate Formation with Silica-Bonded S-Sulfonic Acid
1048
Solid-Phase Synthesis of Isocoumarins via Halocyclization
1049
A Gold-Immobilized Capillary Column Reactor for Oxidation of Alcohols
1050
Asymmetric Cyclopropanation with Immobilized Ru(II)-Salen-Py2
1051
Suzuki-Miyaura Coupling with NHC-Palladium Polymer
1052
One-Pot Oxidation-Wittig Reaction with Ruthenium Catalyst
1053
MonoSil Microreactor for Knoevenagel Reaction and Transesterification
1054
Asymmetric Hydrosilylation of Ketones by Copper Ferrite Nanoparticles
1055
Cyanosilylation and Hydrosilylation with Poly-NHC Particles
1056
Suzuki-Miyaura Cross-Coupling of Aryl Bromides with Pd-CNT
1057
Solid-Supported 2-Imidazolidinone Chiral Auxiliary for Alkylation

Addenda and Errata

1058
Synthesis of BYK 405879