DOI: 10.1055/s-00000131

Synfacts

Issue 08 · Volume 2009 · August 2009 DOI: 10.1055/s-002-19445

Synform

A50
Zanda, Matteo: SYNFORM ISSUE 2009/06

Synthesis of Natural Products and Potential Drugs

z817
All PDFs of this category
0817
Sattely, E. S.; Meek, S. J.; Malcolmson, S. J.; Schrock, R. R.; Hoveyda, A. H.: Synthesis of (+)-Quebrachamine
0818
al., H. Li et: Synthesis of a Hepatitis C Polymerase Inhibitor
0819
Kim, H.; Baker, J. B.; Lee, S.-U.; Park, Y.; Bolduc, K. L.; Park, H.-B.; Dickens, M. G.; Lee, D.-S.; Kim, Y.; Kim, S. H.; Hong, J.: Synthesis of Subglutinol A
0820
Crimmins, M. T.; Christie, H. S.; Long, A.; Chaudhary, K.: Synthesis of Apoptolidin A
0821
Imagawa, H.; Saijo, H.; Kurisaki, T.; Yamamoto, H.; Kubo, M.; Fukuyama, Y.; Nishizawa, M.: Synthesis of ()-Neovibsanin B
0822
Li, Y.; Nawrat, C. C.; Pattenden, G.; Winne, J. M.: Synthesis of ()-Anthecularin
0823
Hyodo, T.; Kiyotsuka, Y.; Kobayashi, Y.: Synthesis of the Active Form of Loxoprofen
0824
Bitar, A. Y.; Frontier, A. J.: Formal Synthesis of ()-Roseophilin
0825
Wu, X.; Zhou, J.; Snider, B. B.: Synthesis of (-)-Berkelic Acid
0826
Macklin, T. K.; Micalizio, G. C.: Synthesis of (+)-Phorbasin C
0827
Dickson, D. P.; Wardrop, D. J.: Synthesis of ()-Agelastatin A
0828
Isaacson, J.; Kobayashi, Y.: Synthesis of Dysibetaine
0829
Dong, S.; Hamel, E.; Bai, R.; Covell, D. G.; Beutler, J. A.; Jr., J. A. Porco: Synthesis of (+)-Chamaecypanone C
0830
Murata, Y.; Yamashita, D.; Kitahara, K.; Minasako, Y.; Nakazaki, A.; Hikage, N.; Takao, K.-i.; Kobayashi, S.: Synthesis of (-)-Norzoanthamine
0831
Qiu, X.-L.; Zhu, J.; Wu, G.; Lee, W.-H.; Chamberlain, A. R.: Synthesis of IBR2 Analogues

Synthesis of Heterocycles

z833
All PDFs of this category
0833
Yoshino, Y.; Kurahashi, T.; Matsubara, S.: Ni-Catalyzed Synthesis of 4-Quinolones from Alkynes and Isatoic Anhydrides
0834
Heravi, M. M.; Baghernejad, B.; Oskooie, H. A.: Three-Component Synthesis of Benzothiazines
0835
Lechel, T.; Möhl, S.; Reissig, H.-U.: Synthesis of 5-Alkoxy Pyrimidines via Enamides
0836
Ackermann, L.; Barfüßer, S.; Potukuchi, H. K.: Copper-Catalyzed Domino Synthesis of Indoles
0837
Komine, Y.; Kamisawa, A.; Tanaka, K.: Synthesis of Dibenzofurans by Rhodium-Catalyzed [2+2+2] Cycloaddition
0838
Heim-Riether, A.; Gipson, K. R.: One-Pot Synthesis of Imidazo[2,1-a]phthal-azines
0839
Coulter, M. M.; Dornan, P. K.; Dong, V. M.: Rh-Catalyzed Synthesis of Benzoxapinones and Benzothiapinones
0840
Rahanyan, N.; Linden, A.; Baldridge, K. K.; Siegel, J. S.: Diazafluoranthene Derivatives via Diels-Alder Reaction
0841
Rao, R. K.; Naidu, A. B.; Sekar, G.: Synthesis of 1,4-Benzoxazines by Domino SN2 and Goldberg Coupling
0842
Zhang, J.; Zhang, M.; Cao, W.; Song, L.; Qian, Q.; Tan, J.; Shao, M.: Synthesis of Trifluoromethyl-Substituted Tetrahydropyrans
0843
Spitz, C.; Lohier, J.-F.; Santos, J. Sopkova-de Oliveira; Reboul, V.; Metzner, P.: 1,4-Benzothiazepines via Nucleophilic Catalysis
0844
Engstrom, K. M.; Baize, A. L.; Franczyk, T. S.; Kallemeyn, J. M.; Mulhern, M. M.; Rickert, R. C.; Wagaw, S.: Friedel-Crafts, Thermal or Reductive Cyclization Route to Thienopyridines
0845
Merkul, E.; Boersch, C.; Frank, W.; Müller, T. J. J.: Three-Component Synthesis of Substituted N-Boc-4-iodopyrroles
0846
Shi, Z.; Zhang, C.; Li, S.; Pan, D.; Ding, S.; Cui, Y.; Jiao, N.: Dioxygen as Oxidant for the Synthesis of Indoles by Pd-Catalyzed C-H Activation
0847
Greszler, S. N.; Johnson, J. S.: Diastereoselective Synthesis of γ-Butyro-lactones

Synthesis of Materials and Unnatural Products

z849
All PDFs of this category
0849
Zhou, X.-H.; Luo, J.; Huang, S.; Kim, T.-D.; Shi, Z.; Cheng, Y.-J.; Jang, S.-H.; Jr., D. B. Knorr; Overney, R. M.; Jen, A. K. Y.: Non-Covalent Assembly of Nonlinear Optical Chromophores
0850
Li, H.; Jäkle, F.: Mild Approach to Organoboron Quinolate Polymers
0851
Levi, Z. U.; Tilley, T. D.: Homocoupling for Pentalenes Synthesis
0852
Sun, Z.-N.; Wang, H.-L.; Liu, F.-Q.; Chen, Y.; Tam, P. K. H.; Yang, D.: BODIPY-Based Nitrite Detection
0853
Schneider, T. F.; Kaschel, J.; Dittrich, B.; Werz, D. B.: Iterative Synthesis of Fused Oligofurans
0854
Huang, K.; Rzayev, J.: Copolymer-Derived Nanotubes
0855
Werner, C.; Hopf, H.; Grunenberg, J.; Ernst, L.; Jones, P. G.; Köhler, F.; Herges, R.: Sondheimer’s Chemistry Gets 3D
0856
Kitazawa, K.; Kochi, T.; Sato, M.; Kakiuchi, F.: C-H Activation to Make Highly Functionalized Anthracenes
0857
Miao, S.; Appleton, A. L.; Berger, N.; Barlow, S.; Marder, S. R.; Hardcastle, K. I.; Bunz, U. H. F.: Azapentacenes
0858
Matano, Y.; Nakashima, M.; Imahori, H.: Oligophospholes
0859
Ohmura, T.; Kijima, A.; Suginome, M.: Isoindoles Made to Order by an Additive
0860
Kaiser, T. E.; Stepanenko, V.; Würthner, F.: Perylene Bisimide J-Aggregates
0861
Donuru, V. R.; Vegesna, G. K.; Velayudham, S.; Green, S.; Liu, H.: Conjugated Poly(BODIPY)

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z863
All PDFs of this category
0863
Buchner, K. M.; Clark, T. B.; Loy, J. M. N.; Nguyen, T. X.; Woerpel, K. A.: Diastereo- and Regioselective Silacyclopropanation of Allenes
0864
Yu, M.; Skouta, R.; Zhou, L.; Jiang, H.-f.; Yao, X.; Li, C.-J.: Silver-Catalyzed Cascade Reaction of Terminal Alkynes with Salicylaldehydes
0865
Pignataro, L.; Lynikaite, B.; Cvengro, J.; Marchini, M.; Piarulli, U.; Gennari, C.: Combination of Acidic and Basic Phosphites in Rhodium-Induced Hydrogenations
0866
Tsoglin, E.; Chechik, H.; Karseboom, G.; Chinkov, N.; Stanger, A.; Marek, I.: Zirconium-Mediated Synthesis of Cyclobutyl Derivatives
0867
Hou, X. L.; Zheng, B. H.: Palladium-Catalyzed Kinetic Resolution of Nitrogen Nucleophiles
0868
Meyer, N.; Lough, A. J.; Morris, R. H.: Iron-Catalyzed Transfer Hydrogenation of Ketones
0869
Yoshikai, N.; Miura, K.; Nakamura, E.: Copper/Aminohydroxyphosphine-Catalyzed Allylic Substitution of Cinnamyl Phosphates
0870
Alamsetti, S. Kumar; Muthupandi, P.; Sekar, G.: Oxidative Kinetic Resolution of Racemic Benzoins
0871
Nakamura, I.; Chan, C. S.; Araki, T.; Terada, M.; Yamamoto, Y.: Platinum-Catalyzed Carboalkoxylation of 6-(1-Alkoxyethoxy)-hex-2-ynoates
0872
Michel, B. W.; Camelio, A. M.; Cornell, C. N.; Sigman, M. S.: Palladium/Quinox-Catalyzed Wacker-Type Oxidation of Terminal Olefins
0873
Peruncheralathan, S.; Teller, H.; Schneider, C.: Titanium-Catalyzed Asymmetric Ring Opening of meso-Aziridines
0874
Hardee, D. J.; Lambert, T. H.: Lanthanum(III)-Catalyzed Cyclopropanation
0875
Iwai, T.; Fujihara, T.; Terao, J.; Tsuji, Y.: Coupling without Decarbonylation
0876
Alnasleh, B. K.; Sherrill, W. M.; Rubina, M.; Banning, J.; Rubin, M.: Formal Nucleophilic Substitution of Bromocyclopropanes
0877
Zhou, S.; Wu, K.-H.; Chen, C.-A.; Gau, H.-M.: AlArEt2(THF) as Arylation Reagents for Aldehydes and Ketones
0878
Ward, A. F.; Wolfe, J. P.: Palladium-Catalyzed Etherification in the Synthesis of bis-Tetrahydrofurans
0879
Li, C.; Villa-Marcos, B.; Xiao, J.: Cocatalyzed Asymmetric Reductive Amination
0880
Senapati, B. K.; Hwang, G.-S.; Lee, S.; Ryu, D. H.: Enantioselective Morita-Baylis-Hillman Reaction
0881
Yao, M.-L.; Quick, T. R.; Wu, Z.; Quinn, M. P.; Kabalka, G. W.: Stereoselective Coupling of Alkoxides and Alkynes
0882
Marcoux, D.; Azzi, S.; Charette, A. B.: TfNH2 Additive Enhances Selectivity of a Rhodium-Catalyzed Reaction
0883
Cortez, N. A.; Aguirre, G.; Parra-Hake, M.; Somanathan, R.: Heterogeneous Asymmetric Transfer Hydrogenation
0884
Malkov, A. V.; Czemerys, L.; Malyshev, D. A.: Asymmetric Epoxidation of Allylic Alcohols in Water
0885
Yamamoto, Y.; Kurihara, K.; Miyaura, N.: Enantioselective Ruthenium(II)-Catalyzed Aldehyde Arylations
0886
Yokoyama, N.; Arai, T.: A Copper-Imidazoline-Aminophenol Complex for Asymmetric 1,4-Additions
0887
García-Fortanet, J.; Kessler, F.; Buchwald, S. L.: Palladium-Catalyzed Asymmetric Dearomatization
0888
Tomita, D.; Yamatsugu, K.; Kanai, M.; Shibasaki, M.: Synthesis of 3-Hydroxy-2-oxindoles via Cu(I)F-Catalyzed Protocols
0889
Ovaska, T. V.; Sullivan, J. A.; Ovaska, S. I.; Winegrad, J. B.; Fair, J. D.: Synthesis of Chiral Seven-Membered Bicycles through Sigmatropic Rearrangements
0890
Chen, S.; Hou, Z.; Zhu, Y.; Wang, J.; Lin, L.; Liu, X.; Feng, X.: Scandium-Catalyzed Enantioselective Multicomponent Mannich Reaction
0891
Wang, H.; Wang, Z.; Ding, K.: Epoxidation of α,β-Unsaturated Ketones with a Self-Supported BINOL-Zn Complex
0892
Egami, H.; Katsuki, T.: Iron-Catalyzed Oxidative Coupling to Provide Enantioenriched BINOLS

Metal-Mediated Synthesis

z893
All PDFs of this category
0893
Xu, H.; Wolf, C.: Copper(I)-Catalyzed Amination of Aryl Halides with Aqueous Ammonia
0894
Molander, G. A.; Sandrock, D. L.: Ionic Ethane-1,2-diboron Species as a Synthetically Useful Dianion Equivalent
0895
Fernández-Mateos, A.; Madrazo, S. Encinas; Teijón, P. Herrero; González, R. Rubio: Ti(III)-Promoted Couplings of Epoxides with Nitriles
0896
Phipps, R. J.; Gaunt, M. J.: A meta-Selective Copper-Catalyzed C-H Bond Arylation
0897
Wen, Y.; Zhao, B.; Shi, Y.: Cu(I)-Catalyzed Diamination of Disubstituted Terminal Alkenes
0898
Lee, K.-s.; Zhugralin, A. R.; Hoveyda, A. H.: NHC-Catalyzed Boron Conjugate Additions to α,β-Unsaturated Carbonyl Compounds
0899
Lemonnier, G.; Zoute, L.; Dupas, G.; Quirion, J.-C.; Jubault, P.: One-Pot Stereoselective Synthesis of α-Fluoroacrylates from Aldehydes and Ketones
0900
Seomoon, D.; A, J.; Lee, P. H.: Indium-Mediated Butadienylation of Imines
0901
Peh, G.-R.; Kantchev, E. A. B.; Zhang, C.; Ying, J. Y.: An NHC-Ligated Palladacycle as an Active Catalyst for Heck-Mizoroki Reaction
0902
Chu, L.; Zhang, X.; Qing, F.-L.: CuBr-Catalyzed Oxidative Difluoromethylation of Tertiary Amines
0903
Cazorla, C.; Métay, E.; Andrioletti, B.; Lemaire, M.: Simple Electrophilic Fluorination of Organoboron Compounds
0904
Knapp, D. M.; Gillis, E. P.; Burke, M. D.: MIDA Boronates: A New Stable Form of Boronic Acids for Coupling Reactions
0905
Nishikata, T.; Lipshutz, B. H.: Amination of Allylic Alcohols in Water
0906
Hu, P.; Kan, J.; Su, W.; Hong, M.: Palladium Trifluoroacetate/Benzoquinone: A Versatile Olefination Catalyst
0907
Coste, A.; Karthikeyan, G.; Couty, F.; Evano, G.: Synthesis of Ynamides via Coupling of 1,1-Dibromo-1-alkenes with Amides

Organo- and Biocatalysis

z909
All PDFs of this category
0909
Armstrong, A.; Bhonoah, Y.; White, A. J. P.: Constrained Bicyclic β-Proline Analogues in Aldol Reaction
0910
Cassani, C.; Bernardi, L.; Fini, F.; Ricci, A.: Mannich Reaction of Sulfonylacetates
0911
Litvinas, N. D.; Brodsky, B. H.; Bois, J. Du: Organocatalytic C-H Hydroxylation
0912
Bui, T.; Syed, S.; III, C. F. Barbas: Additions of Oxindoles to Nitroolefins: An Entry to Pyrrolidinoindolines
0913
Uraguchi, D.; Nakashima, D.; Ooi, T.: Asymmetric Aza-Michael Reaction Catalyzed by a Charged Brønsted Acid
0914
Jiang, H.; Elsner, P.; Jensen, K. L.; Falcicchio, A.; Marcos, V.; Jørgensen, K. A.: Molecular Complexity by Organocatalytic One-Pot Strategies
0915
Simmons, B.; Walji, A. M.; MacMillan, D. W. C.: Cycle-Specific Aminocatalysis Cascades
0916
Kimmel, K. L.; Robak, M. T.; Ellman, J. A.: Enantioselective Conjugate Addition of Thioacetic Acid to Nitroalkenes
0917
García-García, P.; Lay, F.; Rabalakos, C.; List, B.: Disulfonimides as a New Key Structure in Organocatalysis
0918
Lakhdar, S.; Appel, R.; Mayr, H.: Strong Directed Electrostatic Activation
0919
Müller, C.; Bauer, A.; Bach, T.: Intramolecular [2+2] Photocycloaddition
0920
Andrus, M. B.; Harper, K. C.; Christiansen, M. A.; Binkley, M. A.: Phase-Transfer-Catalyzed Asymmetric α-Alkylation of Esters
0921
Wanner, M. J.; Boots, R. N. A.; Eradus, B.; de Gelder, R.; van Maarseveen, J. H.; Hiemstra, H.: An Organocatalytic Pictet-Spengler Reaction in Total Synthesis
0922
Amatore, M.; Beeson, T. D.; Brown, S. P.; MacMillan, D. W. C.: SOMO Activation/α-Chlorination: From Aldehydes to Terminal Epoxides
0923
Verkade, J. M. M.; van der Pijl, F.; Willems, M. M. J. H. P.; Quaedflieg, P. J. L. M.; van Delft, F. L.; Rutjes, F. P. J. T.: An Organocatalytic Route to Both Enantiomers of Lasubine II

Polymer-Supported Synthesis

z925
All PDF of this category
0925
Iijima, Y.; Munakata, A.; Shin-ya, K.; Ganesan, A.; Doi, T.; Takahashi, T.: A Solid-Phase Total Synthesis of Spiruchostatin A
0926
Chuan, Y.; Chen, G.; Peng, Y.: Asymmetric Michael Reaction in Water Using MPS-Supported Prolinol Catalyst
0927
Shimizu, K.-i.; Sato, R.; Satsuma, A.: C-C Cross-Coupling of Alcohols Catalyzed by Ag/Al2O3
0928
Harju, K.; Vesterinen, J.; Yli-Kauhaluoma, J.: Traceless Synthesis of N-Unsubstituted Pyrazoles on a Solid Support
0929
Gilles, A.; Martinez, J.; Cavelier, F.: Polymer-Supported Synthesis of an Apratoxin Analogue
0930
Zhi, H.; Lü, C.; Zhang, Q.; Luo, J.: Synthesis of Benzopyrans with PEG-Based Dicationic Ionic Liquid
0931
Baxendale, I. R.; Ley, S. V.; Mansfield, A. C.; Smith, C. D.: Preparation of Alkynes and Triazoles Using Modular Flow Reactors
0932
Sun, H.; Su, F.-Z.; Ni, J.; Cao, Y.; He, H.-Y.; Fan, K.-N.: Gold Supported on Hydroxyapatite as a Tandem Catalyst
0933
Chattopadhyay, K.; Dey, R.; Ranu, B. C.: Suzuki Coupling and Cyanation with CuO/Pd
0934
Kassaee, M. Z.; Movahedi, F.; Masrouri, H.: One-Pot Synthesis of α-Amino Phosphonates with ZnO Nanoparticles
0935
Fujihara, T.; Yoshida, S.; Terao, J.; Tsuji, Y.: A Phosphine Ligand Bearing EG12 for the Suzuki-Miyaura Coupling
0936
Yoshida, M.; Hedberg, C.; Kaiser, M.; Waldmann, H.: Traceless Solid-Phase Synthesis of cis-Decalins
0937
Adak, L.; Chattopadhyay, K.; Ranu, B. C.: C-N Bond Formation with Palladium Nanoparticles

Addenda and Errata

0938
Iridium-Catalyzed Asymmetric Synthesis of 2,6-Disubstituted Piperidines
0938
Fully Fluorinated Pentaphenylborole
0938
Sonogashira Coupling and Construction of the Indole Ring with Palladium on Silica