DOI: 10.1055/s-00000131

Synfacts

Issue 01 · Volume 2009 · January 2009 DOI: 10.1055/s-002-14460

Synthesis of Natural Products and Potential Drugs

0001
Zutter, U.; Iding, H.; Spurr, P.; Wirz, B.: Synthesis of Tamiflu
0002
Fuwa, H.; Sasaki, M.: Synthesis of (-)-Attenol A
0003
Lumb, J.-P.; Choong, K. C.; Trauner, D.: Synthesis of Rubioncolin B
0004
Zeng, W.; Chemler, S. R.: Synthesis of (S)-(+)-Tylophorine
0005
Yamada, H.; Nagao, K.; Dokei, K.; Kasai, Y.; Michihata, N.: Synthesis of (-)-Corilagin
0006
Miyashita, K.; Tsunemi, T.; Hosokawa, T.; Ikejiri, M.; Imanashi, T.: Synthesis of Leustroducsin B
0007
Yang, H.; Carter, R. G.; Zakharov, L. N.: Synthesis of (-)-Lycopodine
0008
Li, Z.; Gao, Y.; Tang, Y.; Dai, M.; Wang, G.; Wang, Z.; Yang, Z.: Synthesis of Crisamicin A
0009
Kienzler, M. A.; Suseno, S.; Trauner, D.: Synthesis of (-)-Halenaquinone
0010
Hayashi, Y.; Miyakoshi, N.; Kitagaki, S.; Mukai, C.: Synthesis of a Jatropha Sesquiterpenoid
0011
Liu, K.; Chougnet, A.; Woggon, W.-D.: Synthesis of α-Tocopherol
0012
Shie, J.-J.; Fang, J.-M.; Wong, C.-H.: Synthesis of Tamiphosphor
0013
Cong, H.; Ledbetter, D.; Rowe, G. T.; Caradonna, J. P.; Jr., J. A. Porco,: Synthesis of Nicolaioidesin C
0014
Yamagishi, H.; Matsumoto, K.; Iwasaki, K.; Miyazaki, T.; Yokoshima, S.; Tokuyama, [nl]H.; Fukuyama, T.: Synthesis of Eudistomin E

Synthesis of Heterocycles

0015
Wipf, P.; Maciejewski, J. P.: Ti-Catalyzed Synthesis of Indolines
0016
Cikotiene, I.; Morkunas, M.; Rudys, S.; Buksnaitiene, R.; Brukstus, A.: Thermal Heteroannulation Route to Pyrido[4,3-d]pyrimidines
0017
Fu, Z.; Wang, M.; Ma, Y.; Liu, Q.; Liu, J.: Ketene Thioacetals in Furan Ring Construction
0018
Hashimoto, T.; Uchiyama, N.; Maruoka, K.: Asymmetric Synthesis of Aziridines from Diazoacetamides and N-Boc Imines
0019
Chan, Y.; Guthmann, H.; Brimble, M. A.; Barker, D.: Diastereoselective Mannich-Based Synthesis of Piperidones
0020
Arnott, G.; Brice, H.; Clayden, J.; Blaney, E.: Synthesis of Spirocyclic Piperidines from
N-Arylisonicotinamides
0021
Kaim, L. El; Gizzi, M.; Grimaud, L.: Synthesis of Highly Substituted Indoles via an Intramolecular Heck Cyclization
0022
Chang, J. H.; Shin, H.: Large Scale One-Pot Synthesis of 4-Substituted-1H-Pyrrole-3-Carboxylates
0023
Wasa, M.; Yu, J.-Q.: Synthesis of β-, γ-, and δ-Lactams via Pd(II)-Catalyzed C-H Activation
0024
Shanthi, G.; Perumal, P. T.: Three-Component Synthesis of Substituted Chromenes
0025
Andersson, H.; Gustafsson, M.; Olsson, R.; Almqvist, F.: Synthesis of 2-Substituted Pyridine N-Oxides via Directed ortho-Metalation
0026
Imase, H.; Noguchi, K.; Hirano, M.; Tanaka, K.: Au-Catalyzed Cycloisomerization of
N-Alkenyl Alkynylamides to 2-Pyridones
0027
Horneff, T.; Chuprakov, S.; Chernyak, N.; Gevorgyan, V.; Fokin, V. V.: Rh(II)-Catalyzed Transannulation of
1,2,3-Triazoles with Nitriles
0028
Yang, D.; Fu, H.; Hu, L.; Jiang, Y.; Zhao, Y.: Cu-Catalyzed Heterannulation Route to Benzimidazoles from ortho-Haloacetanilides
0029
Veitch, G. E.; Bridgwood, K. L.; Rands-Trevor, K.; Ley, S. V.: Magnesium Nitride as a Source of Ammonia for the Paal-Knorr Synthesis of Pyrroles

Synthesis of Materials and Unnatural Products

0031
Song, S.; Jin, Y.; Kim, S. H.; Moon, J.; Kim, K.; Kim, J. Y.; Park, S. H.; Lee, K.; Suh, H.: Indenoindene Polymers
0032
Dergunov, S. A.; Pinkhassik, E.: Nanopores with a Defined Chemical Environment
0033
Jing, F.; Hillmyer, M. A.: A Bifunctional Monomer for Toughening Polylactide
0034
Zhang, K.; Tieke, B.: Highly Fluorescent Polymers with a Large Stokes Shift
0035
Feng, J.; Liang, B.; Wang, D.; Xue, L.; Li, X.: Fluorescent Dyes Containing Perylene and BODIPY Analogues
0036
Guthrie, D. A.; Tovar, J. D.: A Conformational Protecting Group
0037
Balija, A. M.; Kohman, R. E.; Zimmerman, S. C.: Degradable Dendrimers
0038
Sreejith, S.; Divya, K. P.; Ajayaghosh, A.: NIR Squaraine Dye Detects Aminothiols
0039
Geramita, K.; McBee, J.; Tao, Y.; Segalman, R. A.; Tilley, T. D.: Fluorinated Heterofluorenes
0040
Liu, Z.; Li, C.; Wagner, M.; Avlasevich, Y.; Herrmann, A.; Müllen, K.: Novel Rylene NIR Dyes
0041
Shimizu, M.; Nagao, I.; Tomioka, Y.; Hiyama, T.: Polycyclic Aromatics via Cross-Coupling
0042
Mori, S.; Nambo, M.; Chi, L.-C.; Bouffard, J.; Itami, K.: Pd(II)-Catalyzed Hydroarylation of Fullerene
0043
Werz, D. B.; Fischer, F. R.; Kornmayer, S. C.; Rominger, F.; Gleiter, R.: Sulfur- and Selenium-Containing Cyclophanes

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

0045
Lu, S.-M.; Bolm, C.: Iridium-Catalyzed Hydrogenation of Enones
0046
Toullec, P. Y.; Chao, C.-M.; Chen, Q.; Gladiali, S.; Genêt, J.-P.; Michelet, V.: Enantioselective Hydroarylation-Cycloisomerization of 1,6-Enynes
0047
Yan, X.-X.; Peng, Q.; Li, Q.; Zhang, K.; Yao, J.; Hou, X.-L.; Wu, Y.-D.: Copper-Catalyzed Diastereoselective Switch in Mannich Reactions
0048
Nakao, Y.; Ebata, S.; Yada, A.; Hiyama, T.; Ikawa, M.; Ogoshi, S.: Nickel-Catalyzed Intramolecular Arylcyanation of Alkenes
0049
Hawner, C.; Li, K.; Cirriez, V.; Alexakis, A.: Construction of Aryl-Substituted Quaternary Centers by Conjugate Addition
0050
Álvarez-Dorta, D.; León, E. I.; Kennedy, A. R.; Riesco-Fagundo, C.; Suárez, E.: Sequential Photoelimination and Aldol Cyclization of 1,2-Diketones
0051
Haak, R. M.; Berthiol, F.; Jergphagnon, T.; Gayet, A. J. A.; Tarabiono, C.; Postema, [nl]C. P.; Ritleng, V.; Pfeffer, M.; Janssen, D. B.; Minnaard, A. J.; Feringa, [nl]B. L.; de Vries, J. G.: Chemo-Enzymatic Resolution of
β-Haloalcohols
0052
Tadpetch, K.; Rychnovsky, S. D.: Stereocontrolled Synthesis of Highly Substituted Tetrahydropyrans
0053
Young, A. J.; White, M. C.: Diastereoselective, Catalytic Pd(II)-Based Allylic Alkylation
0054
Ischay, M. A.; Anzovino, M. E.; Du, J.; Yoon, T. P.: Visible Light Photocatalysis for
[2+2] Cycloadditions
0055
Zhang, Y.-Z.; Zhu, S.-F.; Wang, L.-X.; Zhou, Q.-L.: Enantioselective Carbene Insertion into
Si-H Bonds
0056
Marcé, P.; Díaz, Y.; Matheu, M. I.; Castillón, S.: Enantioselective Hydroacylation Applied to the Synthesis of Nucleoside Analogues
0057
Lee, S.; Kim, S.: Zinc-Catalyzed Conjugate Radical Addition of Phosphoric Enones
0058
Yang, Y.; Zhu, S.-F.; Zhou, C.-Y.; Zhou, Q.-L.: Nickel-Catalyzed Coupling of Alkynes and Aldehydes
0059
Lipshutz, B. H.; Amorelli, B.; Unger, J. B.: Copper-Catalyzed Asymmetric Conjugate Reduction/Aldol Reaction
0060
Evans, P. A.; Inglesby, P. A.: Diastereoselective Carbocyclization of Alkenylidenecyclopropanes
0061
Träff, A.; Bogár, K.; Warner, M.; Bäckvall, J.-E.: Synthesis of Chiral Chlorohydrin Acetates by Combined Enzyme and Metal Catalysis
0062
Yazaki, R.; Nitabaru, T.; Kumagai, N.; Shibasaki, M.: Cu/Li-Catalyzed Asymmetric Addition of Allylic Cyanides to Ketoimines
0063
Xu, H.; Zhang, W.; Shu, D.; Werness, J. B.; Tang, W.: Stereospecific and Regioselective Ring Expansion of Cyclopropanes
0064
Du, H.; Zhao, B.; Yuan, W.; Shi, Y.: Copper(I)/Chiral Bisphosphine Catalyzed Diamination of Conjugated Dienes
0065
Trost, B. M.; Thaisrivongs, D. A.: Palladium-Catalyzed Asymmetric Allyic Alkylation of Unstabilized Nucleophiles
0066
Okamoto, K.; Hayashi, T.; Rawal, V. H.: New Chiral Diene Ligands for Rhodium-Catalyzed Conjugate Additions
0067
Wang, L.; Liu, X.; Dong, Z.; Fu, X.; Feng, X.: Nickel(II)/Chiral Nitrogen Oxide Catalyzed Oxa-Michael Addition
0068
Bos, P. H.; Minnaard, A. J.; Feringa, B. L.: Conjugate Addition of Grignard Reagents to α,β-Unsaturated Sulfones
0069
Gonzalez, A. S.; Arrayas, R. G.; Rivero, M. R.; Carretero, J. C.: Copper-Catalyzed Vinylogous Mannich Reaction of Sulfonylimines
0070
Li, C.; Wang, C.; Villa-Marcos, B.; Xiao, J.: Iridium-Catalyzed Counteranion-Induced Asymmetric Hydrogenation of Imines
0071
Lee, C.-T.; Lipshutz, B. H.: Copper-Catalyzed Enantioselective Reduction of Ketones
0072
Wang, C.-J.; Gao, F.; Liang, G.: Application of a New Biphenyl Diamine Ligand in Enantioselective Hydrogenation
0073
Schneider, U.; Ueno, M.; Kobayashi, S.: Indium(0)-Catalyzed Allylations of Ketones in Water
0074
Zhu, S.; Perman, J. A.; Zhang, X. P.: Cobalt-Catalyzed Asymmetric Cyclopropanation

Metal-Mediated Synthesis

0075
Bull, J. A.; Charette, A. B.: Improved Synthesis of gem-Diiodoalkanes
0076
Guo, D.; Huang, H.; Xu, J.; Jiang, H.; Liu, H.: Iron-Catalyzed N-Arylation of Aryl Halides with Amines
0077
Wunderlich, S.; Knochel, P.: Microwave-Enhanced Zincation of Arenes and Heteroarenes
0078
Caron, L.; Campeau, L.-C.; Fagnou, K.: Pd-Catalyzed ortho-Arylation of Nitroaromatics with Aryl Halides
0079
Gunanathan, C.; Milstein, D.: Direct Synthesis of Primary Amines from Alcohols and Ammonia
0080
Li, H.; Yang, H.; Liebeskind, L. S.: Mild Enantiopure Synthesis of α-Amino Ketones from Thiol Esters
0081
Pericas, À; Shafir, A.; Vallribera, A.: ZnO-Catalyzed Transesterification of
β-Keto Esters
0082
Sugiura, M.; Sato, N.; Kotani, S.; Nakajima, M.: Trichlorosilane-Mediated Conjugate Reduction and Reductive Aldol Reaction
0083
Martin, R.; Buchwald, S. L.: α-Arylation of Aldehydes Using Electron-Rich Aryl Halides
0084
Ogata, T.; Hartwig, J. F.: Mild Pd-Catalyzed Amination of Aryl and Heteroaryl Tosylates
0085
Goossen, L. J.; Salih, K. S. M.; Blanchot, M.: Diastereoselective Synthesis of Secondary Enamides
0086
Chen, S.-N.; Wu, W.-Y.; Tsai, F.-Y.: Pd(II)-Catalyzed Hiyama Cross-Coupling Using a Water-Soluble Ligand System
0087
Fors, B. P.; Watson, D. A.; Biscoe, M. R.; Buchwald, S. L.: Pd/BrettPhos: A Highly Active Catalyst for
C-N Cross-Coupling Reactions
0088
Chen, G.; Wang, Z.; Wu, J.; Ding, K.: In-Catalyzed Direct Cyanation of Alcohols using TMSCN
0089
Guo, J.; Harling, J. D.; Steel, P. G.; Woods, T. M.: Cross-Coupling Reactions with Enol Phosphinates

Organo- and Biocatalysis

0091
Xie, J.; Yoshida, K.; Takasu, K.; Takemoto, Y.: Enantioselective [3+2] Cycloadditions of Azomethine Ylides and Nitroolefins
0092
Gianelli, C.; Sambri, L.; Carlone, A.; Bartoli, G.; Melchiorre, P.: anti-Mannich Reaction of Aldehydes with in situ Generated N-Cbz and N-Boc Imines
0093
Koszelewski, D.; Levandera, I.; Clay, D.; Guebitz, G. M.; Rozzell, D.; Kroutil, W.: Formal Enzymatic Reductive Amination with Ammonia
0094
Malerich, J. P.; Hagihara, K.; Rawal, V. H.: Chiral Squaramide Organocatalysis
0095
Mandal, T.; Zhao, C.-G.: Self-Assembled Organocatalysts
0096
Guin, J.; De Sarkar, S.; Grimme, S.; Studer, A.: Biomimetic Aldehyde Oxidation Catalyzed by NHCs
0097
Gui, Y.; Li, J.; Guo, C.-S.; Li, X.-L.; Lu, Z.-F.; Huang, Z.-Z.: A New Catalyst for the Enantioselective Sulfur Ylide Epoxidation
0098
He, R.; Wang, X.; Hashimoto, T.; Maruoka, K.: Tetraalkylphosphonium Salts as Chiral Phase-Transfer Catalysts
0099
Burda, E.; Hummel, W.; Gröger, H.: Combination of Metals and Enzymes:
A Chemoenzymatic Approach
0100
Pesciaioli, F.; De Vincentiis, F.; Galzerano, P.; Bencivenni, G.; Bartoli, G.; Mazzanti, [nl]A.; Melchiorre, P.: Asymmetric Aziridination of Enones

Polymer-Supported Synthesis

0101
Komáromi, A.; Novák, Z.: Copper-Free Sonogashira Coupling of Aryl Chlorides with Pd/C
0102
Zhang, J.; Zhang, Z.; Wang, Y.; Zheng, X.; Wang, Z.: Coupling of Phenols and Aryl Halides with Nano-Copper Oxide
0103
Arakawa, Y.; Haraguchi, N.; Itsuno, S.: Polymer-Supported Chiral Quaternary Ammonium Salts
0104
Li, P.; Wang, L.; Zhang, Y.; Wang, M.: Synthesis of Propargylamines Catalyzed by PS-Supported NHC-Ag(I)
0105
Arakawa, Y.; Chiba, A.; Haraguchi, N.; Itsuno, S.: Asymmetric Hydrogen-Transfer Reaction with Polymer-Supported Ru Catalysts
0106
Abe, Y.; Hirakawa, T.; Nakajima, S.; Okano, N.; Hayase, S.; Kawatsura, M.; Hirose, Y.; Itoh, T.: Activation of Lipase by Chiral Imidazolium Cetyl-PEG10-Sulfate
0107
Kawamorita, S.; Hamasaka, G.; Ohmiya, H.; Hara, K.; Fukuoka, A.; Sawamura, M.: Hydrogenation of Hindered Ketones with a Silica-Supported Rh complex
0108
Choi, M. K.-W.; Yu, W.-Y.; So, M.-H.; Zhou, C.-Y.; Deng, Q.-H.; Che, C.-M.: Polymer-Supported Ruthenium Catalyst for Carbenoid Transfer Reactions
0109
Van Berlo, B.; Houthoofd, K.; Sels, B. F.; Jacobs, P. A.: Silica-Immobilized Second-Generation Hoveyda-Grubbs Catalyst
0110
Sharghi, H.; Aberi, M.; Doroodmand, M. M.: Reusable Cobalt(III)-Salen Complex Immobilized on Activated Carbon
0111
Proch, S.; Herrmannsdörfer, J.; Kempe, R.; Kern, C.; Jess, A.; Seyfarth, L.; Senker, [nl]J.: Solvent- and Base-Free Aerobic Oxidation with Pt@MOF-177
0112
Pérez-Faginas, P.; Aranda, M. T.; Coady, L.; García-López, M. T.; González-Muñiz, R.: Tetrasubstituted β-Lactams from Amino Acids
0113
Gupta, H. K.; Mazumder, A.; Garg, P.; Gutch, P. K.; Dubey, D. K.: Synthesis of Dialkyl Chlorophosphates Using PS-DVB Bound Reagent
0114
Neau, F.; Li, Z.; Richards, R.; Toullec, P. Y.; Genêt, J.-P.; Dumbuya, K.; Gottfried, [nl]J. M.; Steinrück, H.-P.; Pârvulescu, V. I.; Michelet, V.: Synthesis of Functionalized Lactones with Heterogeneous Gold Catalyst

Addenda and Errata

0115
Cu(I)-Promoted Synthesis of Chloromethyl Ketones from CCl3-Carbinols