DOI: 10.1055/s-00000131

Synfacts

Issue 12 · Volume 2008 · December 2008 DOI: 10.1055/s-002-13901

Synform

A116
Zanda, Matteo: SYNFORM ISSUE 2008/11

Synthesis of Natural Products and Potential Drugs

1241
Martin, C. L.; Overman, L. E.; Rohde, J. M.: Synthesis of (±)-Actinophyllic Acid
1242
Miller, K. A.; Shanahan, C. S.; Martin, S. F.: Synthesis of (-)-Alstonerine
1243
Scott, J. P.; Ashwood, M. S.; Brands, K. M. J.; Brewer, S. E.; Cowden, C. J.; Dolling, U.-H.; Emerson, K. M.; Gibb, A. D.; Goodyear, A.; Oliver, S. F.; Stewart, G. W.; Wallace, D. J.: Synthesis of an Estrogen Receptor-β Agonist
1244
Liverton, N. J.: Synthesis of Potent Inhibitor of HCV NS3/4A Protease
1245
Szpilman, A. M.; Manthorpe, J. M.; Carreira, E. M.: Synthesis of 35-Deoxy Amphotericin B Methyl Ester
1246
Margalef, I. V.; Rupnicki, L.; Lam, H. W.: Formal Synthesis of Salinosporamide A
1247
Liu, P.; Hong, S.; Weinreb, S. M.: Synthesis of (-)-Secu’amamine
1248
Qin, H.-L.; Panek, J. S.: Synthesis of Geldanamycin
1249
Selig, P.; Bach, T.: Synthesis of (+)-Meloscine
1250
Teske, J. A.; Deiters, A.: Synthesis of Cannabinoids
1251
Bisai, A.; West, S. P.; Sarpong, R.: Synthesis of (±)-Lyconadin A
1252
Fürstner, A.; Ackerstaff, J.: Formal Synthesis of (-)-Haouamine
1253
Wu, Y.-C.; Liron, M.; Zhu, J.: Synthesis of (-)-Quinocarcin
1254
Tsai, A. S.; Bergman, R. G.; Ellman, J. A.: Synthesis of (-)-Incarvillateine
1255
Fuwa, H.; Naito, S.; Goto, T.; Sasaki, M.: Synthesis of (+)-Neopeltolide

Synthesis of Heterocycles

1257
Grant, D.; Dahl, R.; Cosford, N. D. P.: Microreactor Synthesis of 1,2,4-Oxadiazoles
1258
Paone, D. V.; Shaw, A. W.: Synthesis of Highly Substituted Imidazoles from 1,2-Amino Alcohols and Thioamides
1259
Bray, C. D.: A Diels-Alder Approach to Benzannulated [5,6]-Spiroketals
1260
Willy, B.; Dallos, T.; Rominger, F.; Schönhaber, J.; Müller, T. J. J.: Three-Component Synthesis of 1,5-Benzo-
diazepines
1261
Mamedov, V. A.; Saifina, D. F.; Gubaidullin, A. T.; Saifina, A. F.; Rizvanov, I. K.: One-Pot Synthesis of 2-(Indolizin-2-yl)benz-imidazoles from Quinoxalinones
1262
Barluenga, J.; Riesgo, L.; Vicente, R.; López, L. A.; Tomás, M.: Cu(I)-Catalyzed Synthesis of Polysubstituted Furans
1263
Batchelor, D. V.; Beal, D. M.; Brown, T. B.; Ellis, D.; Gordon, D. W.; Johnson, P. S.; Mason, H. J.; Ralph, M. J.; Underwood, T. J.; Wheeler, S.: Acid-Mediated Synthesis of 3-N,N-Dialkyl-amino-1,2,4-Triazoles
1264
Rudkin, M. E.; Joensuu, P. M.; MacLachlan, W. S.; Lam, H. W.: Synthesis of β-Hydroxylactams via Co-Catalyzed Alkylative Aldol Cyclization
1265
Gasiecki, A. F.; Cross, J. L.; Henry, R. F.; Gracias, V.; Djuric, S. W.: Synthesis of Spiro Pyrrolidines from Tetrahydropyridinium Salts
1266
Gabriele, B.; Mancuso, R.; Salerno, G.: Synthesis of Functionalized Benzofurans via Pd-Catalyzed Cycloisomerization
1267
Sasada, T.; Sakai, N.; Konakahara, T.: Three-Component Synthesis of Tetra-substituted Pyridines
1268
Eidamshaus, C.; Burch, J. D.: Pd-Catalyzed Enolate α-Arylation. Synthesis of Benzofurans
1269
Cui, S.-L.; Wang, J.; Wang, Y.-G.: Synthesis of Indoles from N-Aryl Amides and Ethyl Diazoacetate
1270
Horn, J.; Marsden, S. P.; Nelson, A.; House, D.; Weingarten, G. G.: Rh-Catalyzed Conjugate Addition of o-Amino-arylboronates. Synthesis of Quinolines
1271
Alizadeh, A.; Hosseinpour, R.; Rostamnia, S.: Synthesis of 4-Hydroxy-1H-pyrrole-2,3-dicarboxylic Acids

Synthesis of Materials and Unnatural Products

1273
Xu, R.; Schweizer, W. B.; Frauenrath, H.: Poly(diacetylene)s from Preorganized Monomers
1274
Yang, C.-W.; Hsia, T.-H.; Chen, C.-C.; Lai, C.-K.; Liu, R.-S.: BINOL-Based Columnar Fluorescent Liquid Crystals
1275
Schwertfeger, H.; Würtele, C.; Serafin, M.; Hausmann, H.; Carlson, R. M. K.; Dahl, J. E. P.; Schreiner, P. R.: Monoprotection of Diamondoid Diols
1276
Davis, N. K. S.; Pawlicki, M.; Anderson, H. L.: Anthracene-Fused Porphyrins
1277
Sadhu, K. K.; Bharadwaj, P. K.: Cu(I)/Cu(II) Fluorescence Switch
1278
Li, L.; Brennessel, W. W.; Jones, W. D.: Polycyclic Isoquinoline Salts
1279
Zhang, X.; Matsuo, Y.; Nakamura, E.: Bright Light from C60 Chromophores
1280
Matano, Y.; Miyajima, T.; Fukushima, T.; Kaji, H.; Kimura, Y.; Imahori, H.: Fusing Phosphole and Thiophene
1281
Jiang, W.; Qian, H.; Li, Y.; Wang, Z.: Addition of Heteroatoms to Perylenes
1282
Alam, M. A.; Tsuda, A.; Sei, Y.; Yamaguchi, K.; Aida, T.: Helical Polymer of Porphyrin and a Chiral Pd(II) Complex
1283
Otero, G.; Biddau, G.; Sánchez-Sánchez, C.; Caillard, R.; López, M. F.; Rogero, C.; Palomares, F. J.; Cabello, N.; Basanta, M. A.; Ortega, J.; Méndez, J.; Echavarren, A. M.; Pérez, R.; Gómez-Lor, B.; Martín-Gago, J. A.: Facile Synthesis of Fullerenes
1284
Kim, E.; Koh, M.; Ryu, J.; Park, S. B.: A Full-Color-Tunable Fluorophore
1285
Asadi, A.; Patrick, B. O.; Perrin, D. M.: An H-Bond Tetrameric Rosette

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

1287
Watson, M. P.; Jacobsen, E. N.: Nickel-Catalyzed C-CN Bond Activation and Asymmetric Arylcyanation
1288
Zani, L.; Eriksson, L.; Adolfsson, H.: Amino Acid Derived Sulfinamide Ligands for Transfer Hydrogenation
1289
Walz, I.; Togni, A.: Nickel-Catalyzed Asymmetric Nazarov Cyclization
1290
Goossen, L. J.; Blanchot, M.; Salih, K. S. M.; Karch, R.; Rivas-Nass, A.: Stereodivergent Synthesis of (Z)- and (E)-Thioenamides
1291
Watkins, A. L.; Hashiguchi, B. G.; Landis, C. R.: Asymmetric Hydroformylation: Synthesis of α-Branched Aryl Aldehydes
1292
Khiar, N.; Navas, R.; Suárez, B.; Álvarez, E.; Fernández, I.: New Phosphinite Thioglycosides for Asymmetric Hydrogenation
1293
Vázquez-Romero, A.; Rodríguez, J.; Lledó, A.; Verdaguer, X.; Riera, A.: Application of an Enantioselective Cyclopentenone Synthesis
1294
Komanduri, V.; Grant, C. D.; Krische, M. J.: Rhodium-Catalyzed Reductive Coupling of 2-Vinyl Pyridines and Imines
1295
Harada, H.; Thalji, R. K.; Bergman, R. G.; Ellman, J. A.: Enantioselective Hydroarylation of Alkenes via C-H Activation
1296
García-Fortanet, J.; Buchwald, S. L.: Palladium-Catalyzed Asymmetric α-Arylation of Aldehydes
1297
Zhou, J.; Hartwig, J. F.: Highly Efficient Intermolecular Hydroamination of Bicyclic Alkenes
1298
Sudo, Y.; Shirasaki, D.; Harada, S.; Nishida, A.: Ytterbium-Catalyzed Enantioselective Diels-Alder Reaction
1299
Gendrineau, T.; Chuzel, O.; Eijsberg, H.; Genêt, J.-P.; Darses, S.: New C1-Symmetric Diene Ligands in Rhodium-Catalyzed 1,2-Addition
1300
Ito, H.; Kosaka, Y.; Nonoyama, K.; Sasaki, Y.; Sawamura, M.: Copper-Catalyzed Cyclopropanation of Allylic Carbonates with Diboron
1301
Bondzic, B. P.; Farwick, A.; Liebich, J.; Eilbracht, P.: Iridium-Catalyzed Allylic Substitution Reactions in Tryptamine Synthesis
1302
Yang, X.; Zhou, X.; Lin, L.; Chang, L.; Liu, X.; Feng, X.: Michael Addition of Nitroalkanes to Nitroolefins
1303
Spiess, S.; Welter, C.; Franck, G.; Taquet, J.-P.; Helmchen, G.: Air-Stable Iridium Catalyst in Asymmetric Allylic Substitution
1304
Smith, S. W.; Fu, G. C.: Nickel-Catalyzed Asymmetric Negishi Cross-Couplings
1305
Arai, N.; Azuma, K.; Nii, N.; Okhuma, T.: Hydrogenation of Ketones to Provide Aryl Allylic Alcohols
1306
Godineau, E.; Schenk, K.; Landais, Y.: Diastereoselective Radical Cyclization Towards Piperidinones
1307
Toussaint, A.; Pfaltz, A.: Borobox Ligands for Asymmetric Henry Reactions
1308
Li, C.; Xiao, J.: Rhodium-Catalyzed Asymmetric Hydrogenation of Cyclic Imines
1309
Sabot, C.; Bérard, D.; Canesi, S.: Oxidative Aromatic Umpolung Strategy Applied to Tetrahydrofuran Synthesis
1310
Fernández-Pérez, H.; Pericàs, M. A.; Vidal-Ferran, A.: Novel P-O-P Ligands for Highly Efficient Hydrogenation of Alkenes

Metal-Mediated Synthesis

1311
Bahde, R. J.; Rychnovsky, S. D.: Cyclization of α-Amino Alkyllithium Reagents via Carbolithiation
1312
Martinelli, J. R.; Watson, D. A.; Freckmann, D. M. M.; Barder, T. E.; Buchwald, S. L.: Pd-Catalyzed Carbonylation of Aryl Bromides at Atmospheric Pressure
1313
Shen, Q.; Hartwig, J. F.: Efficient Amination of Heteroaryl and Aryl Halides Using [(CyPF-t-Bu)PdCl2]
1314
Zhou, G.; Lim, D.; Coltart, D. M.: Versatile Crossed-Claisen Rearrangement by Soft Enolization of Thioesters
1315
Xu, H.; Ekoue-Kovi, K.; Wolf, C.: Efficient Cross-Coupling Using Pd-Phosphinous Acid Catalysts
1316
Lipshutz, B. H.; Chung, D. W.; Rich, B.: Sonogashira Couplings of Aryl Bromides at Room Temperature in Water
1317
Niu, J.; Zhou, H.; Li, Z.; Xu, J.; Hu, S.: An Efficient Ullmann-Type Cu-Catalyzed C-O Bond Formation
1318
Molander, G. A.; Gormisky, P. E.: Coupling of Cyclopropyl- and Cyclobutyl-trifluoroborates with Aryl Chlorides
1319
Brunner, G.; Eberhard, L.; Oetiker, J.; Schröder, F.: Tandem Cyclopropanation with CH2Br2 under Grignard Conditions
1320
Watson, D. A.; Fan, X.; Buchwald, S. L.: Carboxylic Acid Derivatives through Carbonylation of Aryl Chlorides
1321
Kantchev, E. A. B.; Peh, G.-R.; Zhang, C.; Ying, J. Y.: Practical Heck-Mizoroki Coupling Mediated by a Novel Palladacycle
1322
Trost, B. M.; Livingston, R. C.: Ru-Catalyzed Selective Redox Isomerization of Propargylic Alcohols
1323
Yamada, K.-i; Nakano, M.; Maekawa, M.; Akindele, T.; Tomioka, K.: Sn-Free Radical Addition of Acyloxymethyl to Imines
1324
Chuzel, O.; Roesch, A.; Genêt, J.-P.; Darses, S.: Rh-Catalyzed Synthesis of Sterically Hindered Diarylketones
1325
Gong, H.; Gagné, M. R.: Saturated C-Glycosides via Ni-Catalyzed Diastereoselective Cross-Coupling

Organo- and Biocatalysis

1327
Uraguchi, D.; Ueki, Y.; Ooi, T.: Cooperative Catalysis of Chiral Tetraaminophosphonium Carboxylates
1328
Ju, Y.-D.; Xu, L.-W.; Li, L.; Lai, G.-Q.; Qiu, H.-Y.; Jiang, J.-X.; Lu, Y.: Noyori Ligand as Organocatalyst
1329
Oh, S. H.; Rho, H. S.; Lee, J. W.; Youk, S. H.; Chin, J.; Song, C. E.: A New Catalyst for the Desymmetrization of Cyclic Anhydrides
1330
Zhao, G.-L.; Rios, R.; Vesely, J.; Eriksson, L.; Córdova, A.: An Atom-Economic Domino Reaction Process
1331
Voss, C. V.; Gruber, C. C.; Faber, K.; Knaus, T.; Macheroux, P.; Kroutil, W.: Four Enzymatic Reactions in One Pot
1332
Procuranti, B.; Connon, S. J.: Pyridinium Salts as New Organocatalysts for Acetalizations
1333
Kim, S. M.; Lee, J. H.; Kim, D. Y.: A New Bifunctional Catalyst: The Direct Amination of α-Cyanoketones
1334
Martin, N. J. A.; Cheng, X.; List, B.: Asymmetric Transfer Hydrogenation of β-Nitroacrylates
1335
Rabalakos, C.; Wulff, W. D.: Enantioselective Michael Addition of Nitroalkanes to Nitroolefines
1336
Lombardo, M.; Pasi, F.; Easwar, S.; Trombini, C.: Imidazolium-Tagged Hydroxyproline
1337
Zhou, J.; Wakchaure, V.; Kraft, P.; List, B.: Desymmetrizing Aldol Cyclodehydration

Polymer-Supported Synthesis

1339
Lipshutz, B. H.; Nihan, D. M.; Vinogradova, E.; Taft, B. R.; Bokovi, Z. V.: A Bimetallic, Heterogeneous, Multifunctional Catalyst
1340
Jun, B.-H.; Kim, J.-H.; Park, J.; Kang, H.; Lee, S.-H.; Lee, Y.-S.: Dihydroxylation of Olefins with Polymer-Supported Osmium Catalyst
1341
Amali, A. J.; Rana, R. K.: Pd Nanoparticles in Assembled Silica Microcapsules
1342
Yamada, Y. M. A.; Guo, H.; Uozumi, Y.: Oxidative Cyclization of Alkenols Using Convoluted Polymeric Tungsten Catalysts
1343
Krishnan, G. R.; Sreekumar, K.: Organocatalysis with Polystyrene-Supported PAMAM Dendrimers
1344
Sirion, U.; Bae, Y. J.; Lee, B. S.; Chi, D. Y.: Huisgen 1,3-Dipolar Cycloaddition with an Ionic Polymer-Supported Copper(I) Catalyst
1345
Sanna, M.; White, P. D.; Chan, W. C.: Efficient Removal of Amines Using Polymer-Supported Cyclic Anhydride
1346
Likhar, P. R.; Roy, M.; Roy, S.; Subhas, M. S.; Kantam, M. L.; Sreedhar, B.: Oxidative Heck Reaction with Polyaniline-Supported Pd Catalyst
1347
Lucchesi, C.; Inasaki, T.; Miyamura, H.; Matsubara, R.; Kobayashi, S.: Aerobic Oxidation of Alcohols with Gold Nanoparticles
1348
Hagiwara, H.; Okunaka, N.; Hoshi, T.; Suzuki, T.: Olefin Metathesis with Immobilized Grubbs Catalyst
1349
Schätz, A.; Grass, R. N.; Stark, W. J.; Reiser, O.: TEMPO-Immobilized on Magnetic C/Co Nanoparticles for Alcohol Oxidation
1350
Ishida, T.; Nagaoka, M.; Akita, T.; Haruta, M.: Au/PCPs-Catalyzed Aerobic Oxidation of Alcohols
1351
Wang, X.; Kawanami, H.; Islam, N. M.; Chattergee, M.; Yokoyama, T.; Ikushima, Y.: Aerobic Oxidation of Alcohols with Gold Nanoparticles
1352
Uozumi, Y.; Suzuka, T.: π-Allylic Sulfonylation in Water with PS-PEG Pd-Phosphine Complexes