Synthesis

Issue 23/2014

Nguyen, Thanh Binh; Ermolenko, Ludmila; Al-Mourabit, Ali: Three-Component Reaction between Isocyanides, Aliphatic Amines and Elemental Sulfur: Preparation of Thioureas under Mild Conditions with Complete­ Atom Economy

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Issue 22/2014

Takemoto, Yuki; Yoshida, Hiroto; Takaki, Ken: Facile Access to vic-Borylstannylalkanes via Copper-Catalyzed Three-Component Borylstannylation of Alkenes

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Issue 21/2014

Pace, Vittorio; Castoldi, Laura; Mamuye, Ashenafi Damtew; Holzer, Wolfgang: Homologation of Isocyanates with Lithium Carbenoids: A Straightforward Access to α-Halomethyl- and α,α-Dihalomethylamides

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Issue 20/2014

Wang, Ruzhi; Jiang, Heng; Cheng, Yuanzheng; Kadi, Adnan A.; Fun, Hoong-Kun; Zhang, Yan; Yu, Shouyun: Somophilic Isocyanide Insertion: Synthesis of 6-Arylated and 6-Trifluoro­methylated Phenanthridines

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Issue 18/2014

Yu, Xiaoqiang; Huang, Nan; Feng, Xiujuan; Yamamoto, Yoshinori; Bao, Ming: Synthesis of 1,3,5-Trisubstituted Pyrazoles by the Cope-Type Hydroamination of 1,3-Dialkynes with Alkylhydrazines

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Issue 17/2014

Haraguchi, Ryosuke; Matsubara, Seijiro: Preparation of the Zinc Enolate Equivalent of Amides by Zinciomethylation of Isocyanates: Catalytic Asymmetric Reformatsky-Type Reaction

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Issue 16/2014

Liu, Lu; Zhang, Junliang: Product Selectivity Control in the Domino Cyclization of 2-(2-Alkynylarylidene)-1,3-dicarbonyl Compounds Catalyzed by Metal Lewis Acids

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Issue 15/2014

Gao, Ke; Yamakawa, Takeshi; Yoshikai, Naohiko: Cobalt-Catalyzed Chelation-Assisted Alkylation of Arenes with Primary and Secondary Alkyl Halides

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Issue 09/2014

Pan, Feng-Feng; Yu, Wei; Qi, Zheng-Hang; Qiao, Chunhua; Wang, Xing-Wang: Efficient Construction of Chiral Spiro[benzo[g]chromene-oxindole] Derivatives via Organocatalytic Asymmetric Cascade Cyclization

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Issue 07/2014

Schmid, Fabian; Bernasconi, Maurizio; Jessen, Henning J.; Pfaltz, Andreas; Gademann, Karl: Catalytic Enantioselective Total Synthesis of (–)-Pyridovericin

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Issue 06/2014

Beck, Thorsten M.; Haller, Heike; Streuff, Jan; Riedel, Sebastian: Brominations with Pr₄NBr₉ as a Solid Reagent with High Reactivity and Selectivity­

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Issue 24/2013

Inomata, Sotaro; Harada, Yusuke; Nakamura, Yuya; Nakamura, Taisuke; Ishizone, Takashi: Synthesis of 1,3-Dehydroadamantanes Possessing Alkyl, Phenyl, and Alkoxy Substituents by Intramolecular Wurtz-Type Coupling Reaction of 1,3-Dibromoadamantanes

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Issue 23/2013

Reekie, Tristan A.; Kavanagh, Madeline E.; Longworth, Mitchell; Kassiou, Michael: Synthesis of Biologically Active Seven-Membered-Ring Heterocycles

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Issue 21/2013

Di Franco, Thomas; Boutin, Nicolas; Hu, Xile: Suzuki–Miyaura Cross-Coupling Reactions of Unactivated Alkyl Halides Catalyzed by a Nickel Pincer Complex

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Issue 19/2013

Hepburn, Hamish B.; Chotsaeng, Nawasit; Luo, Yunfei; Lam, Hon Wai: Enantioselective Rhodium-Catalyzed Allylation of Cyclic Imines with Potassium Allyltrifluoroborates

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Issue 18/2013

Rulli, Giuseppe; Fredriksen, Kim A.; Duangdee, Nongnaphat; Bonge-Hansen, Tore; Berkessel, Albrecht; Gröger, Harald: Asymmetric Organocatalytic Aldol Reaction in Water: Mechanistic Insights and Development of a Semi-Continuously Operating Process

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Issue 17/2013

Barsoum, David N.; Brassard, Christopher J.; Deeb, Jason H. A.; Okashah, Najeah; Sreenath, Kesavapillai; Simmons, J. Tyler; Zhu, Lei: Synthesis of 5-Iodo-1,2,3-triazoles from Organic Azides and Terminal Alkynes­: Ligand Acceleration Effect, Substrate Scope, and Mechanistic Insights

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Issue 16/2013

Wouters, Ana D.; Bessa, Adrieli B.; Sachini, Maraísa; Wessjohann, Ludger A.; Lüdtke, Diogo S.: Boron–Zinc Exchange in The Diastereoselective Arylation of Sugar-Based Aldehydes­: Stereoselective Synthesis of (+)-7-epi-Goniofufurone and Analogues

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Issue 15/2013

Harthong, Steven; Bach, Renaud; Besnard, Céline; Guénée, Laure; Lacour, Jérôme: Ring-Expansion Reactions of Binaphthyl Azepines and Ferrocenophanes through Metal-Catalyzed [1,2]-Stevens Rearrangements

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Issue 14/2013

Xu, Changming; Zhang, Long; Zhou, Pengxin; Luo, Sanzhong; Cheng, Jin-Pei: A Practical Protocol for Asymmetric Synthesis of Wieland–Miescher and Hajos–Parrish Ketones Catalyzed by a Simple Chiral Primary Amine

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Issue 13/2013

Keene, Craig; Kürti, László: Regiospecific Synthesis of Novel Cyclic Nitrostyrenes and 3-Substituted 2-Nitronaphthalenes

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Richers, Matthew T.; Deb, Indubhusan; Platonova, Alena Yu.; Zhang, Chen; Seidel, Daniel: Facile Access to Ring-Fused Aminals via Direct α-Amination of Secondary Amines with o-Aminobenzaldehydes: Synthesis of Vasicine, Deoxyvasicine, Deoxyvasicinone, Mackinazolinone, and Ruteacarpine

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Issue 12/2013

An, Qianjin; Shen, Jiefeng; Butt, Nicholas; Liu, Delong; Liu, Yangang; Zhang, Wanbin: Asymmetric Domino Double Michael Addition of Nitroolefins and Aldehyde Esters with trans-Perhydroindolic Acid as an Organocatalyst

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Issue 11/2013

Fleck, Carsten; Franzmann, Elisa; Claes, Dorith; Rickert, Aljona; Maison, Wolfgang: Synthesis of Functionalized Adamantane Derivatives: (3 + 1)-Scaffolds for Applications in Medicinal and Material Chemistry

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Issue 10/2013

Lu, Jin-Yong; Riedrich, Matthias; Wojtas, K. Philip; Arndt, Hans-Dieter: Assembly of the Nosiheptide A-Ring: A Fruitful Lesson

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Issue 08/2013

Marqués-López, Eugenia; Herrera, Raquel P.; Marks, Timo; Jacobs, Wiebke C.; Christmann, Mathias: Enantioselective Rauhut–Currier-Type Cyclizations via Dienamine Activation: Scope and Mechanism

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Issue 07/2013

Hoshikawa, Tamaki; Yoshioka, Shun; Kamijo, Shin; Inoue, Masayuki: Photoinduced Direct Cyanation of C(sp³)–H Bonds

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Issue 06/2013

Perreault, Stéphane; Rovis, Tomislav: Enantioselective Synthesis of the Tricyclic Core of FR901483 Featuring a Rhodium-Catalyzed [2+2+2] Cycloaddition

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Issue 04/2013

Tian, Wei-Sheng; Ding, Kai; Sun, Yun-Shan; Chen, Ling; Lei, Zhen: Total Synthesis and Establishment of the Stereochemistry of Spiniferin-1, a Rare Planar Chiral Marine Natural Product with a 1,6-Methano[10]annulene Skeleton

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Issue 03/2013

Hintermann, Lukas; Schmitz, Marco; Maltsev, Oleg V.; Naumov, Panče: Organocatalytic Stereoisomerization versus Alkene Isomerization: Catalytic Asymmetric Synthesis of 1-Hydroxy-trans-2,5-diphenylphospholane 1-Oxide

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Issue 02/2013

Nugent, Thomas C.; Marinova, Sofiya M.: Step-Efficient Access to Chiral Primary Amines

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Issue 01/2013

Schüler, Peter; Fischer, Sebastian N.; Marsch, Michael; Oberthür, Markus: Efficient α-Mannosylation of Phenols: The Role of Carbamates as Scavengers for Activated Glycosyl Donors

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Issue 24/2012

Kovács, Szabolcs; Zih-Perényi, Katalin; Révész, Ádám; Novák, Zoltán: Copper on Iron: Catalyst and Scavenger for Azide–Alkyne Cycloaddition

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Issue 23/2012

Ghosh, Arun K.; Kass, Jorden; Nicponski, Daniel R.; Keyes, Chad: Diastereoselective Synthesis of Substituted Tetrahydropyrans by Copper(II)–Bisphosphine-Catalyzed Olefin Migration and Prins Cyclization

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Issue 22/2012

Mi, Xianwei; Wang, Yan; Zhu, Lili; Wang, Renxiao; Hong, Ran: Enantioselective Synthesis of (–)-Stemoamide

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Issue 21/2012

Shibata, Takanori; Fujimoto, Masako; Hirashima, Hiroyuki; Chiba, Tatsuya; Endo, Kohei: Facile Synthesis of Cyclic Polyphenylenes by Consecutive Inter- and Intramolecular Cycloadditions of ortho-, meta-, and para-Phenylene-Tethered Triynes

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Issue 20/2012

Zhu, Feng; Zhou, Feng; Cao, Zhong-Yan; Wang, Chao; Zhang, Yong-Xue; Wang, Cui-Hong; Zhou, Jian: A Facile Method for the Synthesis of 3-Substituted 3-(Alkylthio)oxindoles or 3-Alkoxyoxindoles

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Issue 19/2012

Kraft, Philip; Ahlin, Joachim S. E.; Büchel, Michelle; Sutter, Pascal: On the Crossroad of Dienone Musks and Cassyrane: Synthesis and Olfactory Properties of New High-Impact Orris Odorants

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Issue 18/2012

Maciejko, Magdalena; Stecko, Sebastian; Staszewska-Krajewska, Olga; Jurczak, Margarita; Furman, Bartłomiej; Chmielewski, Marek: An Entry to the Carbapenem Antibiotic Scaffold via the Asymmetric Kinugasa Reaction

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Issue 17/2012

Wakchaure, Satish; Einsiedel, Jürgen; Waibel, Reiner; Gmeiner, Peter: Conformationally Restricted Peptide Mimetics by Ring-Closing Olefin Metathesis

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Issue 15/2012

Samanta, Rajarshi; Kulikov, Katharina; Strohmann, Carsten; Antonchick, Andrey P.: Metal-Free Electrocyclization at Ambient Temperature: Synthesis of 1-Arylcarbazoles

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Issue 13/2012

Kirkham, James D.; Leach, Andrew G.; Row, Eleanor C.; Harrity, Joseph P. A.: Investigation of the Origins of Regiochemical Control in [4+2] Cycloadditions of 2-Pyrones and Alkynylboronates

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Issue 11/2012

Schmidt, Bernd; Krehl, Stefan; Sotelo-Meza, Veronica: Synthesis of Chromanes through RCM–Transfer Hydrogenation

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Issue 10/2012

Kim, Ju Hyun; Lee, Sang-gi: Tandem One-Pot Construction of Indoles via Palladium and Copper-Catalyzed Coupling Reactions of the Blaise Reaction Intermediate

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Issue 09/2012

Kuttner, Julian R.; Warratz, Svenja; Hilt, Gerhard: Straightforward Synthesis of Nonconjugated Cyclohex-3-enone and Conjugated 4-Methylenecyclohex-2-enone Derivatives

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Issue 07/2012

Yaren, Oezlem; Röthlisberger, Pascal; Leumann, Christian J.: Synthesis and Incorporation into Oligodeoxynucleotides of Carbocyclic exo-Amino Nucleosides

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Issue 06/2012

Aplander, Karolina; Lindström, U. Marcus; Wennerberg, Johan: Entropy-Controlled and Enantiodivergent Lewis Acid Catalysis in Water

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Issue 04/2012

Schotes, Christoph; Bigler, Raphael; Mezzetti, Antonio: Bicyclo[3.2.0]heptane-Based Enamides by Ru/PNNP-Catalyzed Enantioselective Ficini Reactions: Scope and Application in Ligand Design

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Issue 03/2012

Grove, Charles I.; Fettinger, James C.; Shaw, Jared T.: Second-Generation Synthesis of (-)-Viriditoxin

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Issue 02/2012

Rudzki, Martin; Alcalde-Aragonés, Ana; Dzik, Wojciech I.; Rodríguez, Nuria; Gooßen, Lukas J.: Selective Copper- or Silver-Catalyzed Decarboxylative Deuteration of Aromatic Carboxylic Acids

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Issue 01/2012

Marti, Alex; Peruncheralathan, Saravanan; Schneider, Christoph: Cationic Late-Transition-Metal Complexes Catalyze the Ring Opening of Aziridines with Amines

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Issue 24/2011

Schläger, Torsten; Schepmann, Dirk; Wünsch, Bernhard: Novel σ₁ Receptor Ligands by Oxa-Pictet-Spengler Reaction of Pyrazolylethanol

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Issue 23/2011

Knappke, Christiane E. I.; Arduengo, III, Anthony J.; Jiao, Haijun; Neudörfl, Jörg-Martin; Jacobi von Wangelin, Axel: On the Dual Role of N-Heterocyclic Carbenes as Bases and Nucleophiles in Reactions with Organic Halides

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Issue 22/2011

Kirsch, Stefan F.; Klahn, Philipp; Menz, Helge: The Use of COP-OAc in the Catalyst-Controlled Syntheses of 1,3-Polyols

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Issue 21/2011

Shibuya, Masatoshi; Sasano, Yusuke; Tomizawa, Masaki; Hamada, Toshimasa; Kozawa, Masami; Nagahama, Noriaki; Iwabuchi, Yoshiharu: Practical Preparation Methods for Highly Active Azaadamantane-Nitroxyl-Radical-Type Oxidation Catalysts

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Issue 17/2011

Wilkening, Ina; del Signore, Giuseppe; Ahlbrecht, Wiebke; Hackenberger, Christian P. R.: Lewis Acid or Alkyl Halide Promoted Rearrangements of Phosphor- and Phosphinimidates to N,N-Disubstituted Phosphor- and Phosphinamidates

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Issue 16/2011

Kakugawa, Kazumi; Nemoto, Tetsuhiro; Kohno, Yuta; Hamada, Yasumasa: Asymmetric Synthesis of 2-Substituted Hexahydroquinolin-4-ones Using a Pd-Catalyzed Asymmetric Allylic Amination and Intramolecular Mannich Reaction: Catalytic Asymmetric Synthesis of 2-epi-cis-195A

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Issue 15/2011

Ries, Oliver; Ochmann, Anne; Ducho, Christian: Synthesis of N-Alkyl-N-hydroxyguanidines: A Comparative Study Using Different Protecting Group Strategies

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Issue 14/2011

Nedolya, Nina A.; Tarasova, Ol’ga A.; Volostnykh, Ol’ga G.; Albanov, Alexander I.; Klyba, Ludmila V.; Trofimov, Boris A.: Reactions of Lithiated Alkynes and Allenes with Isothiocyanates: A Simple and Efficient Synthesis of New Aryl- or Hetaryl-Substituted 3H-Azepines and 4,5-Dihydro-3H-azepines

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Issue 13/2011

Barjau, Joaquin; Schnakenburg, Gregor; Waldvogel, Siegfried R.: Short Domino Sequence to Dioxa[4.3.3]propellanes

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Issue 12/2011

Wu, Ming-Yu; Li, Kun; Wang, Na; He, Ting; Yu, Xiao-Qi: A Novel Catalyst-Free Tandem Reaction for the Synthesis of 5-Hydroxy-1,5-dihydro-2H-pyrrol-2-ones in Water Medium

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Issue 11/2011

Schäfer, Ines; Opatz, Till: Pyrroles and Indolizidines from Deprotonated α-(Alkylideneamino)nitriles

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Issue 10/2011

Prechter, Agnes; Heinrich, Markus R.: Hydrogen Peroxide and Arenediazonium Salts as Reagents for a Radical Beckmann-Type Rearrangement

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Issue 09/2011

Chemla, Fabrice; Dulong, Florian; Ferreira, Franck; Nüllen, Max P.; Pérez-Luna, Alejandro: Radical Zinc-Atom Transfer Based Multicomponent Approaches to 3-Alkylidene-Substituted Tetrahydrofurans

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Issue 08/2011

Blecking, C. J.; Hu, W.; Zadmard, R.; Dasgupta, A.; Schrader, T.: A Modular Synthetic Route to Dimeric Calixarenes: A New Family of DNA Major Groove Binders

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Issue 07/2011

Cao, Hua; Jiang, Huanfeng; Huang, Huawen: Transition-Metal-Catalyzed Domino Reactions: Efficient One-Pot Regiospecific Synthesis of Highly Functionalized Polysubstituted Furans from Electron-Deficient Alkynes and 2-Yn-1-ols

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Issue 04/2011

Jennum, Karsten; Vestergaard, Mikkel; Pedersen, Anders Holmen; Fock, Jeppe; Jensen, Jonas; Santella, Marco; Led, Jens Jørgen; Kilså, Kristine; Bjørnholm, Thomas; Nielsen, Mogens Brøndsted: Synthesis of Oligo(phenyleneethynylene)s with Vertically Disposed Tetrathiafulvalene Units

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Issue 02/2011

Rose, Christopher A.; Gundala, Sivaji; Connon, Stephen J.; Zeitler, Kirsten: Chemoselective Crossed Acyloin Condensations: Catalyst and Substrate Control

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Issue 24/2010

Peng, Cheng; Yan, Guobin; Wang, Yan; Jiang, Yubo; Zhang, Yan; Wang, Jianbo: Palladium-Catalyzed Coupling Reaction of α-Diazocarbonyl Compounds with Aromatic Boronic Acids or Halides

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Issue 23/2010

El Sous, Mariana; Ganame, Danny; Tregloan, Peter; Rizzacasa, Mark A.: Total Synthesis of (-)-Reveromycin A via a Hetero-Diels-Alder Approach

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Issue 22/2010

Hatano, Manabu; Ishihara, Kazuaki: Highly Practical BINOL-Derived Acid-Base Combined Salt Catalysts for the Asymmetric Direct Mannich-Type Reaction

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Issue 18/2010

Upadhyay, Puspesh K.; Kumar, Pradeep: A Concise Synthesis of (2S,3S,4S)-2-(Hydroxymethyl)pyrrolidine-3,4-diol (LAB1)

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Issue 16/2010

Campbell, Matthew J.; Johnson, Jeffrey S.: Enantioselective Synthesis of (+)-Polyanthellin A via Cyclopropane-Aldehyde (3+2)-Annulation

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Issue 15/2010

Adachi, Shinya; Tanaka, Fumi; Watanabe, Kazuya; Watada, Atsushi; Harada, Toshiro: Enantioselective Friedel-Crafts Alkylation of Furans and Indoles with Simple α,β-Unsaturated Ketones Catalyzed by Oxazaborolidinone

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Issue 14/2010

Kamijo, Shin; Amaoka, Yuuki; Inoue, Masayuki: Unified Oxidation Protocol for the Synthesis of Carbonyl Compounds Using a Manganese Catalyst

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Issue 09/2010

Chassaing, Stefan; Alix, Aurélien; Boningari, Thirupathi; Sani Souna Sido, Karim; Keller, Murielle; Kuhn, Philippe; Louis, Benoit; Sommer, Jean; Pale, Patrick: Copper(I)-Zeolites as New Heterogeneous and Green Catalysts for Organic Synthesis

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Issue 08/2010

Kraus, George A.; Guo, Haitao; Kumar, Ganesh; Pollock III, Gerald; Carruthers, Heather; Chaudhary, Divya; Beasley, Jonathan: A Flexible Synthesis of Indoles from ortho-Substituted Anilines: A Direct Synthesis of Isocryptolepine

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Issue 07/2010

Sabitha, Gowravaram; Reddy, S. Siva Sankara; Bhaskar, Vangala; Yadav, Jhillu S.: A Concise Synthesis of (-)-(3S,6R)-3,6-Dihydroxy-10-methylundecanoic Acid Using a Cross-Metathesis Approach

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Issue 05/2010

Ambrosini, Lisa M.; Cernak, Tim A.; Lambert, Tristan H.: Development of Oxidative Formylation and Ketonylation Reactions

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Issue 04/2010

Uria, Uxue; Vicario, Jose L.; Badía, Dolores; Carrillo, Luisa; Reyes, Efraim; Pesquera, Amaia: ‘On Water’ Iminium/Enamine Catalysis: Organocatalytic Enantioselective Cyclopropanation of α,β-Unsaturated Aldehydes

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Issue 03/2010

Bischop, Martina; Doum, Verena; Nordschild née Rieche, Anja C. M.; Pietruszka, Jörg; Sandkuhl, Diana: Total Synthesis of Halicholactone and Neohalicholactone

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Issue 02/2010

McConville, Matthew; Blacker, John; Xiao, Jianliang: Heck Reaction in Diols and Cascade Formation of Cyclic Ketals

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Issue 01/2010

Gioia, Claudio; Bernardi, Luca; Ricci, Alfredo: Asymmetric Diels-Alder Reactions of Vinylindoles Using Organocatalysis

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Issue 24/2009

Rück-Braun, Karola; Kempa, Stefan; Priewisch, Beate; Richter, Anja; Seedorff, Sabine; Wallach, Lukas: Azobenzene-Based ω-Amino Acids and Related Building Blocks: Synthesis, Properties, and Application in Peptide Chemistry

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Issue 23/2009

Shu, Wan-Ting; Zhou, Shuangliu; Gau, Han-Mou: Palladium-Catalyzed Cross-Coupling Reaction of AlArEt₂(THF) with Aryl Bromides

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Issue 22/2009

Su, Xianbin; Thomas, Gemma L.; Galloway, Warren R. J. D.; Surry, David S.; Spandl, Richard J.; Spring, David R.: Synthesis of Biaryl-Containing Medium-Ring Systems by Organocuprate Oxidation: Applications in the Total Synthesis of Ellagitannin Natural Products

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Issue 21/2009

Inoue, Masahiro; Nakada, Masahisa: Structure Elucidation and Enantioselective Total Synthesis of the HMG-CoA Reductase Inhibitors FR901512 and FR901516

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Issue 19/2009

García Ruano, José Luis; Marcos, Vanesa; Alemán, José: Synthesis of Enantiomerically Pure Allenes with Central and Axial Chirality Mediated by a Remote Sulfinyl Group

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Issue 18/2009

Feldman, Ken S.; Fodor, Matthew D.; Skoumbourdis, Amanda P.: Synthesis of Dibromophakellin, Dibromophakellstatin, and Dibromo­agelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives

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Issue 16/2009

Judd, Katie E.; Mahon, Mary F.; Caggiano, Lorenzo: Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates

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Issue 15/2009

Concellón, José M.; Rodríguez-Solla, Humberto; del Amo, Vicente; Díaz, Pamela: Stereoselective Olefination Reactions Promoted by Rieke Manganese

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Issue 14/2009

Yoshida, Masahiro; Al-Amin, Mohammad; Shishido, Kozo: Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media

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Issue 11/2009

Hodgson, David M.; Kloesges, Johannes; Evans, Brian: Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine

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Issue 10/2009

Wang, Jiang; Shi, Jianmei; Zhang, Xiaodong; Lin, Daizong; Jiang, Hualiang; Liu, Hong: Highly Diastereoselective Conjugate Addition-Elimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives

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Issue 20/2008

Gnamm, Christian; Franck, Géraldine; Miller, Nicole; Stork, Timon; Brödner, Kerstin; Helmchen, Günter: Enantioselective Iridium-Catalyzed Allylic Aminations of Allylic Carbonates with Functionalized Side Chains. Asymmetric Total Synthesis of (S)-Vigabatrin

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Issue 18/2008

Ferjancic, Zorana; Quiclet-Sire, Béatrice; Zard, Samir Z.: Generation and Intermolecular Additions of Pyridylmethyl Radicals

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Issue 15/2008

Gehring, Timo; Podlech, Joachim; Rothenberger, Alexander: Intramolecular Michael-Type Additions to Vinyl Bissulfoxides: Enantioselective Synthesis of Chiral Aldehydes

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Issue 10/2008

Yamada, Tohru: Enantioselective Borohydride Reduction Catalyzed by Cobalt Complexes: Discovery, Analysis, and Design for a Halogen-Free System

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Issue 09/2008

Ito, Nobuhiro; Watahiki, Tsutomu; Maesawa, Tsuneaki; Maegawa, Tomohiro; Sajiki, Hironao: H-D Exchange Reaction Taking Advantage of the Synergistic Effect of Heterogeneous Palladium and Platinum Mixed Catalyst

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Issue 08/2008

Maki, Brooks E.; Chan, Audrey; Scheidt, Karl A.: Protonation of Homoenolate Equivalents Generated by N-Heterocyclic Carbenes

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Issue 04/2008

Perez, Lark J.; Micalizio, Glenn C.: Titanium-Mediated Fragment Union Processes in Complex Molecule Synthesis: Development of a Branched Reaction Pathway of High Step Economy for the Synthesis of Complex and Diverse Polyketides

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Issue 02/2008

García Ruano, José Luis; Parra, Alejandro; Yuste, Francisco; Mastranzo, Virginia M.: Mild and General Method for the Synthesis of Sulfonamides

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Issue 01/2008

Broggi, Julie; Díez-González, Silvia; Petersen, Jeffrey L.; Berteina-Raboin, Sabine; Nolan, Steven P.; Agrofoglio, Luigi A.: Study of Copper(I) Catalysts for the Synthesis of Carbanucleosides via Azide-Alkyne 1,3-Dipolar Cycloaddition

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Issue 24/2007

Böge, Nicolas; Krüger, Sarah; Schröder, Marcus; Meier, Chris: A New Short and Efficient Synthetic Route to C8-N-Acetylarylamine 2′-Deoxyguanosine Phosphoramidites

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Issue 23/2007

Erdsack, Jörg; Krause, Norbert: Synthesis of Furanomycin Derivatives by Gold-Catalyzed Cycloisomerization of α-Hydroxyallenes

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Issue 21/2007

Tang, Feili; Chen, Ceng; Moeller, Kevin D.: Electrochemistry and Umpolung Reactions: New Tools for Solving Synthetic Challenges of Structure and Location

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Issue 19/2007

Lohr, Andreas; Gress, Tobias; Deppisch, Manuela; Knoll, Marina; Würthner, Frank: Synthesis of Merocyanine Dye Nanorods: The Importance of Solvent, Kinetic and Thermodynamic Control, and Steric Effects on Self-Assembly

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Issue 18/2007

Matsubara, Hiroshi; Maeda, Louis; Sugiyama, Hiroyuki; Ryu, Ilhyong: Chiral and Achiral Lithium Amides Having a Fluorous Ponytail: Preparation and Evaluation as a Recycling Reagent for Lithium Enolate Generation

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Issue 17/2007

Guo, Hao; Ma, Shengming: Highly Regio- and Stereoselective Palladium(0)-Catalyzed Addition of Organoboronic Acids with 1,2-Allenic Sulfones, Sulfoxides, or Alkyl- or Aryl-Substituted Allenes in the Presence of Acetic Acid: An Efficient Synthesis of E-Alkenes

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Issue 14/2007

Fernandes, Carlos; Gauzy, Christine; Yang, Yi; Roy, Olivier; Pereira, Elisabeth; Faure, Sophie; Aitken, David J.: [2+2] Photocycloadditions with Chiral Uracil Derivatives: Access to All Four Stereoisomers of 2-Aminocyclobutanecarboxylic Acid

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Issue 10/2007

Restorp, Per; Dressel, Martina; Somfai, Peter: Synthesis of Functionalized Pyrrolidines by a Highly Stereoselective [3+2]-Annulation Reaction of N-Tosyl-α-Amino Aldehydes and 1,3-Bis(silyl)propenes

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Issue 09/2007

Margaretha, Paul; Schmidt, Kerstin; Kopf, Jürgen; Sinnwell, Volker: Photocycloaddition of 2,3-Dihydro-2,2-dimethyl-4H-thiopyran-4-one (a 4-Thiacyclohex-2-enone) to bona fide Triplet Quenchers. A Contradiction?

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Issue 07/2007

Bomkamp, Martin; Artiukhov, Aleksander; Kataeva, Olga; Waldvogel, Siegfried R.: Facile Synthesis of Enantiomerically Pure Architectures Based on Triphenylene Ketals

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Issue 06/2007

Ziessel, Raymond; Goze, Christine; Ulrich, Gilles: Design and Synthesis of Alkyne-Substituted Boron in Dipyrromethene Frameworks

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Issue 05/2007

Kotke, Mike; Schreiner, Peter R.: Generally Applicable Organocatalytic Tetrahydropyranylation of Hydroxy Functionalities with Very Low Catalyst Loading

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Issue 04/2007

Inoue, Munenori; Yokota, Wakako; Katoh, Tadashi: Enantioselective Total Synthesis of (+)-Scyphostatin, a Potent and Specific Inhibitor of Neutral Sphingomyelinase

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Issue 03/2007

Wessig, Pablo; Müller, Gunnar; Pick, Charlotte; Matthes, Annika: The Photo-Dehydro-Diels-Alder (PDDA) Reaction - A Powerful Method for the Preparation of Biaryls

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Issue 02/2007

Kashin, Dmitry; Meyer, Axel; Wittenberg, Rüdiger; Schöning, Kai-Uwe; Kamlage, Stefan; Kirschning, Andreas: A Practical Synthesis of the Ansa Chain of Benzenic Ansamycin Antibiotics: Total Synthesis of an Ansatrienol Derivative

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Issue 01/2007

Marcseková, Klaudia; Doye, Sven: HI-Catalyzed Hydroamination and Hydroarylation of Alkenes

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Issue 24/2006

Vogler, Thomas; Studer, Armido: The Effect of Additives on TEMPO-Mediated Alkoxyamine Isomerizations: Experiments and Simulations

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Issue 22/2006

Schobert, Rainer; Dietrich, Matthias; Mullen, Gillian; Urbina-Gonzalez, Juan-Manuel: Phosphorus Ylide Based Functionalizations of Tetronic and Tetramic Acids

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Issue 20/2006

Čapek, Petr; Vrábel, Milan; Hasník, Zbyněk; Pohl, Radek; Hocek, Michal: Aqueous-Phase Suzuki-Miyaura Cross-Coupling Reactions of Free Halopurine Bases

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Issue 17/2006

Abarbri, Mohamed; Parrain, Jean-Luc; Duchêne, Alain; Thibonnet, Jérôme: Stereoselective Synthesis of Trienoic Acids: Synthesis of Retinoic Acids and Analogues

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Issue 14/2006

Burstein, Christian; Tschan, Serena; Xie, Xiulan; Glorius, Frank: N-Heterocyclic Carbene-Catalyzed Conjugate Umpolung for the Synthesis of γ-Butyrolactones

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Issue 11/2006

Schmidt, Andreas; Beutler, Ariane; Habeck, Tobias; Mordhorst, Thorsten; Snovydovych, Bohdan: Pseudo-Cross-Conjugated Mesomeric Betaines and N-Heterocyclic Carbenes of Indazole

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Issue 09/2006

Granzhan, Anton; Bats, Jan W.; Ihmels, Heiko: Synthesis and Spectroscopic Properties of 4a,14a-Diazoniaanthra[1,2-a]anthracene and 13a,16a-Diazoniahexaphene Derived from 1,7-Dimethylnaphthalene

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Issue 08/2006

Vincze, Zoltán; Bíró, A. Beatrix; Csékei, Márton; Timári, Géza; Kotschy, András: The Palladium-Catalyzed Preparation of Condensed Tetracyclic Heterocycles and their Application to the Synthesis of rac-Mangochinine

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Issue 07/2006

Gómez Arrayás, Ramón; Cabrera, Silvia; Carretero, Juan Carlos: Copper-Catalyzed Ring-Opening of Heterobicyclic Alkenes with Grignard Reagents: Remarkably High anti-Stereocontrol

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Issue 04/2006

Hanessian, Stephen; Talbot, Clément; Saravanan, Parthasarathy: Diastereoselective [3,2]-Stevens and Sommelet-Hauser Rearrangements in the Dihydromethanodibenzoazocine Series

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Issue 03/2006

Díez, Elena; Prieto, Auxiliadora; Simon, Monika; Vázquez, Juan; Álvarez, Eleuterio; Fernández, Rosario; Lassaletta, José María: Asymmetric Mannich-Type Addition of Ketene Silyl Acetals and Thioacetals to N,N-Dialkylhydrazones

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Issue 02/2006

Keller, Jan; Schlierf, Clemens; Nolte, Christoph; Mayer, Peter; Straub, Bernd F.: One-Pot Syntheses of Sterically Shielded Phosphorus Ligands by Selective Stepwise Nucleophilic Substitution at Triphenyl Phosphite

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Issue 01/2006

Commeiras, Laurent; Bourdron, Julien; Douillard, Soazig; Barbier, Pascale; Vanthuyne, Nicolas; Peyrot, Vincent; Parrain, Jean-Luc: Total Synthesis of Terpenoids Isolated from Caulerpale Algae and Their Inhibition­ of Tubulin Assembly

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Issue 20/2005

Nad, Sukanya; Breinbauer, Rolf: Electroorganic Synthesis of 2,5-Dialkoxydihydrofurans and Pyridazines on Solid Phase Using Polymer Beads as Supports

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Issue 18/2005

Luu, Thanh; Shi, Wei; Lowary, Todd L.; Tykwinski, Rik R.: A Divergent Synthesis of Triyne Natural Products and Glycosylated Analogues Using a Carbenoid Rearrangement

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Issue 17/2005

Pirc, Samo; Bevk, David; Jakše, Renata; Rečnik, Simon; Golič, Ljubo; Golobič, Amalija; Meden, Anton; Stanovnik, Branko; Svete, Jurij: Synthesis of N-Substituted 3-Aminomethylidenetetramic Acids

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Issue 16/2005

Kraft, Philip; Popaj, Kasim; Abate, Agnese: Design, Synthesis and Olfactory Properties of 2-Substituted 2-tert-Butyl-5-­methyl-2,5-dihydrofurans: seco-Derivatives of Theaspiranes

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Issue 14/2005

Bartoschek, Anna; El-Idreesy, Tamer T.; Griesbeck, Axel G.; Höinck, Lars-Oliver; Lex, Johann; Miara, Claus; Neudörfl, Jörg M.: A Family of New 1,2,4-Trioxanes by Photooxygenation of Allylic Alcohols in Sensitizer-Doped Polymers and Secondary Reactions

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Issue 13/2005

Harthong, Steven; Billard, Thierry; Langlois, Bernard R.: Towards the Syntheses of α-Trifluoromethylated Oxygenated Heterocycles and Their Precursors

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Issue 11/2005

Lesch, Bernhard; Toräng, Jakob; Nieger, Martin; Bräse, Stefan: The Diels-Alder Approach towards Cannabinoids

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Issue 08/2005

Kawabata, Takeo; Chen, Jianyong; Suzuki, Hideo; Fuji, Kaoru: Stereochemical Study on α-Alkylation of β-Branched α-Amino Acid Derivatives­ via Memory of Chirality

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Issue 07/2005

Hassfeld, Jorma; Eggert, Ulrike; Kalesse, Markus: Synthesis of the C1-C17 Macrolactone of Tedanolide

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Issue 06/2005

Lang, Martin; Steglich, Wolfgang: An Effective Method for the Synthesis of ¹³C-Labeled Polyprenylhydroxy­benzoic Acids

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Issue 05/2005

Takami, Kazuaki; Usugi, Shin-ichi; Yorimitsu, Hideki; Oshima, Koichiro: Radical Allylation, Vinylation, Alkynylation, and Phenylation Reactions of α-Halo Carbonyl Compounds with Organoboron, Organogallium, and Organoindium Reagents

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Issue 04/2005

Lopez, Roman; Poupon, Jean-Christophe; Prunet, Joëlle; Férézou, Jean-Pierre; Ricard, Louis: Diastereocontrolled Synthesis of Highly Functionalized Spiroketals: Application to the Synthesis of a Precursor of the C-12-C-25 Fragment of Bafilomycin A₁

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Issue 03/2005

Pena, Miguel A.; Pérez Sestelo, José; Sarandeses, Luis A.: New Synthetic Applications of Indium Organometallics in Cross-Coupling Reactions

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Issue 02/2005

Lomberget, Thierry; Bouyssi, Didier; Balme, Geneviève: New Method for the Synthesis of Functionalized 1,3-Bis-Exocyclic Dienes via a Palladium-Catalyzed Reaction. Scope and Synthetic Applications

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Issue 01/2005

Breit, Bernhard; Breuninger, Daniel: Enantioselective Copper-Mediated Allylic Substitution with Grignard Reagents Employing a Chiral Reagent-Directing Leaving Group

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Issue 17/2004

Kulkarni, Mukund G.; Davawala, Saryu I.; Doke, Aniruddha K.; Pendharkar, Dhananjay S.: An Expedient Protocol for Cyclopentenone Annulation

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Issue 15/2004

Luis, Ana Liza; Krische, Michael J.: Nucleophilic Catalysis via Phosphine Conjugate Addition: Vinyl Sulfones as Reacting Partners in Catalytic Cross-Michael Cycloisomerization

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Issue 14/2004

Braun, Roland U.; Müller, Thomas J. J.: Coupling-Isomerization-Stetter and Coupling-Isomerization-Stetter-Paal-Knorr Sequences - A Multicomponent Approach to Furans and Pyrroles

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Issue 12/2004

Gingras, Marc; Chabre, Yoann M.; Raimundo, Jean-Manuel: Fundamental Reactivity of Sulfur with Organotins: Underexploited Ar-S Bond Formation under Aqueous and Aerobic Conditions

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Issue 11/2004

Kilroy, Tim G.; Cozzi, Pier Giorgio; End, Nicole; Guiry, Patrick J.: The Application of HETPHOX Ligands to the Asymmetric Intermolecular Heck Reaction of 2,3-Dihydrofuran and 2,2-Disubstituted-2,3-Dihydrofurans

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Issue 10/2004

Karsch, Sandra; Freitag, Dirk; Schwab, Pia; Metz, Peter: Ring Closing Metathesis in the Synthesis of Sultones and Sultams

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Issue 08/2004

Gravel, Michel; Lachance, Hugo; Lu, Xiaosong; Hall, Dennis G.: Scope and Limitations of the Scandium-Catalyzed Enantioselective Addition of Chiral Allylboronates to Aldehydes

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Issue 07/2004

Kang, Sung Ho; Kang, Suk Youn; Choi, Hyeong-wook; Kim, Chul Min; Jun, Hyuk-Sang; Youn, Joo-Hack: Stereoselective Total Synthesis of the Natural (+)-Lasonolide A

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Issue 06/2004

Tsuji, Riichiro; Arai, Shigeru; Nishida, Atsushi: General Method for the Synthesis of Chiral 2,3-Bisarylmethoxy-1,4-Butanediols from l-(+)-Tartrate

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Issue 04/2004

Bunte, Jens O.; Rinne, Stefanie; Mattay, Jochen: Synthesis of Novel Steroid Backbones via Photoinduced Electron Transfer Initiated Domino Cyclizations of Silyl Enol Ethers

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Issue 03/2004

Radix-Large, Sylvie; Kucharski, Stéphanie; Langlois, Bernard R.: Trifluoromethylated Vinylic and Aromatic Compounds from α-(Trifluoro­methyl)allyl Alcohols

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Issue 02/2004

Salem, Bahaâ; Klotz, Philippe; Suffert, Jean: Cascade Cyclization via a 4-exo-dig-Cyclocarbopalladation for an Easy Access to New Polycyclic Structures

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Issue 01/2004

Rimkus, Audrius; Sewald, Norbert: Conjugate Addition of Organozinc Compounds to Nitroolefins

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Issue 17/2003

Oestreich, Martin; Schmid, Ulrike K.; Auer, Gertrud; Keller, Manfred: A Convergent Method for the Synthesis of Highly Enantiomerically Enriched Cyclic Silanes with Silicon-Centered Chirality

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Issue 16/2003

Haeuseler, Andreas; Henn, Wolfgang; Schmittel, Michael: Stereoselective Assembly of Three Different Carbonyl Components by Two Successive Aldol Reactions Using Group IVa and IVb Metals

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Issue 15/2003

Kitamura, Mitsuru; Yoshida, Masayuki; Kikuchi, Takashi; Narasaka, Koichi: Synthesis of Quinolines and 2H-Dihydropyrroles by Nucleophilic Substitution at the Nitrogen Atom of Oxime Derivatives

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Issue 13/2003

Ludek, Olaf R.; Meier, Chris: New Convergent Synthesis of Carbocyclic Nucleoside Analogues

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Issue 12/2003

Gomes, Paulo; Gosmini, Corinne; Périchon, Jacques: Allylation of Carbonyl Compounds by Allylic Acetates Using a Cobalt Halide as Catalyst

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Issue 10/2003

Kellogg, Richard M.; Nieuwenhuijzen, José W.; Pouwer, K.; Vries, Ton R.; Broxterman, Quirinus B.; Grimbergen, Reinier F. P.; Kaptein, Bernard; Crois, René M. La; de Wever, Ellen; Zwaagstra, Karen; van der Laan, Alexander C.: Dutch Resolution: Separation of Enantiomers with Families of Resolving Agents. A Status Report

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Issue 08/2003

Cravotto, Giancarlo; Nano, Gian Mario; Palmisano, Giovanni; Tagliapietra, Silvia: The Reactivity of 4-Hydroxycoumarin under Heterogeneous High-Intensity Sonochemical Conditions

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Issue 07/2003

Jørgensen, Karl Anker: Asymmetric Friedel-Crafts Reactions: Catalytic Enantioselective Addition of Aromatic and Heteroaromatic C-H Bonds to Activated Alkenes, Carbonyl Compounds, and Imines

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Issue 06/2003

Petri, Andreas F.; Kühnert, Sven M.; Scheufler, Frank; Maier, Martin E.: Applications of Size-Selective Macrolactonizations to the Synthesis of Benzolactone-Enamide Core Structures

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Issue 04/2003

Dias, Luiz C.; Diaz, Gaspar; Ferreira, Andrea A.; Meira, Paulo R. R.; Ferreira, Edílson: Allyltrichlorostannane Additions to α-Amino Aldehydes: Application to the Total Synthesis of the Aspartyl Protease Inhibitors l-682,679, l-684,414, l-685,434, and l-685,458

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Issue 03/2003

Mamane, Victor; Ledoux-Rak, Isabelle; Deveau, Sandrine; Zyss, Joseph; Riant, Olivier: Palladium-Catalyzed Cross-Coupling Reaction of a Chiral Ferrocenyl Zinc Reagent with Aromatic Bromides: Application to the Design of Chiral Octupoles­ for Second Harmonic Generation

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Issue 01/2003

Shionhara, Tomoichi; Suzuki, Keisuke: Facile One-Pot Procedure for Et₃Al-Promoted Asymmetric Pinacol-Type Rearrangement

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Issue 18/2002

Smitrovich, Jacqueline H.; Woerpel, K. A.: Reactions of Silylmethyl Allylic Silanes: Synthesis of Tetrahydrofurans

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Issue 16/2002

Lin, Wen-Li; Taduri, B. Pratap; Liu, Rai-Shung: Stereocontrolled Construction of Tricyclic Furan and Pyrrolyl Derivatives via Tungsten-Mediated [3+2] Cycloaddition and Intramolecular Diels-Alder Reaction

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Issue 15/2002

Ambroise, Lydia; Dumez, Estelle; Szeki, Andrea; Jackson, Richard F. W.: Stereocontrolled Synthesis of anti-α-Hydroxy-β-Amino and anti-α,β-Diamino Acid Derivatives by Epoxidation of 1-Arylthio-1-nitroalkenes

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Issue 13/2002

Ichikawa, Junji; Wada, Yukinori; Fujiwara, Masaki; Sakoda, Kotaro: The Nucleophilic 5-endo-trig Cyclization of 1,1-Difluoro-1-alkenes: Ring-Fluorinated Hetero- and Carbocycle Synthesis and Remarkable Effect of the Vinylic Fluorines on the Disfavored Process

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Issue 12/2002

Krause, Norbert; Hoffmann-Röder, Anja; Canisius, Johannes: From Amino Acids To Dihydrofurans: Functionalized Allenes in Modern
Organic Synthesis

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Issue 10/2002

Hodgson, David M.; Stent, Matthew A. H.; Wilson, Francis X.: Organolithium-Induced Synthesis of Unsaturated Diols from Epoxides of Dihydrofurans and Dihydropyrans

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Issue 08/2002

Gandon, Vincent; Bertus, Philippe; Szymoniak, Jan: Conversion of Imines into C,N-Dimagnesiated Compounds and Trapping with Electrophiles. One-Pot Access to 1-Azaspirocyclic Framework

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Issue 05/2002

Hilt, Gerhard; Smolko, Konstantin I.: Cobalt(I)-catalyzed Neutral Diels-Alder Reactions of 1,3-Diynes with Acyclic 1,3-Dienes

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Issue 04/2002

Knölker, Hans-Joachim; Fröhner, Wolfgang; Reddy, Kethiri R.: Indoloquinones, Part 7. Total Synthesis of the Potent Lipid Peroxidation Inhibitor Carbazoquinocin C by an Intramolecular Palladium-Catalyzed Oxidative Coupling of an Anilino-1,4-benzoquinone

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Issue 03/2002

Bargiggia, Frédéric; Dos Santos, Sylvia; Piva, Olivier: Asymmetric Photodeconjugation: Highly Stereoselective Synthesis of α-Fluorocarboxylic Derivatives

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Issue 02/2002

Ooi, Takashi; Miura, Tomoya; Itagaki, Yoshifumi; Ichikawa, Hayato; Maruoka, Keiji: Catalytic Meerwein-Ponndorf-Verley (MPV) and Oppenauer (OPP) Reactions: Remarkable Acceleration of the Hydride Transfer by Powerful Bidentate Aluminum Alkoxides

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Issue 01/2002

Arisawa, Mieko; Miyagawa, Chie; Yamaguchi, Masahiko: Equatorial Preference in the GaCl₃-Promoted Ethenylation of Cyclic Ketones

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Issue 16/2001

Gansäuer, Andreas; Pierobon, Marianna; Bluhm, Harald: Titanocene Catalysed 5-exo Cyclisations of Unsaturated Epoxides- Reagent Control in Radical Chemistry

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Issue 14/2001

Kim, Byeang Hyean; Jeong, Eun Jeong; Hwang, Gil Tae; Venkatesan, Natarajan: Multiple Cycloadditive Macrocyclization: An Efficient Method for Crown Ether-Type Cyclophanes, Bis-Calix[4]arenes and Silamacrocycles

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Issue 13/2001

Bernardinelli, Gérald; Gillet, Sandra; Kündig, E. Peter; Liu, Ronggang; Ripa, Alberto; Saudan, Lionel: Diastereoselective Transformation of Arenes into Highly Enantiomerically Enriched Substituted Cyclohexadienes

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Issue 12/2001

Carretero, Juan Carlos; Adrio, Javier: Asymmetric Pauson-Khand Cyclizations of 1-Sulfinylenynes

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Issue 10/2001

Ollivier, Cyril; Panchaud, Philippe; Renaud, Philippe: A One-Pot Conversion of Carboxylic Acids into Homoallylic Alcohols

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Issue 09/2001

Vossmann, Petra; Hornig, Knut; Fröhlich, Roland; Würthwein, Ernst-Ulrich: Asymmetric Addition of Aldehydes and Ketones to Chiral 2-Azapentadienyl Lithium Compounds: Diastereoselective Synthesis of 4-Vinyl-4,5-dihydro-oxazoles

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Issue 07/2001

Beller, Matthias; Mägerlein, Wolfgang; Indolese, Adriano F.; Fischer, Christine: Efficient Palladium-Catalyzed Alkoxycarbonylation of N-Heteroaryl Chlorides - A Practical Synthesis of Building Blocks for Pharmaceuticals and Herbicides

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Issue 05/2001

Charonnet, Emmanuelle; Filippini, Marie-Hélène; Rodriguez, Jean: Novel DBU-MeOH-Promoted One-Pot Stereoselective γ-Functionalization of 1,3-Dicarbonyls: An Easy Access to γ-Arylidene, γ-Alkylidene and γ-Allylidene α-Ketoesters and -amides

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Issue 04/2001

Mori, Miwako; Kitamura, Tsuyoshi; Sato, Yoshihiro: Synthesis of Medium-Sized Ring Compounds Using Enyne Metathesis

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Issue 03/2001

Mues, Heike; Kazmaier, Uli: The Asymmetric Chelate-Claisen Rearrangement as a Key Step in the Syntheses of Non-Proteinogenic Amino Acids

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Issue 02/2001

Andreassen, Vinni; Svensson, Birte; Bols, Mikael: Synthesis of an 1′-Azasugar Analogue of Maltose

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Issue 01/2001

Bringmann, Gerhard; Hinrichs, Jürgen; Pabst, Thomas; Henschel, Petra; Peters, Karl; Peters, Eva-Maria: From Dynamic to Non-Dynamic Kinetic Resolution of Lactone-Bridged Biaryls: Synthesis of Mastigophorene B

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Issue 14/2000

Ziessel, Raymond; El-ghayoury, Abdelkrim: Facile and Multistep Synthesis of Functionalized Nitroxide Radicals Containing a Bipyridine Frame

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Issue 12/2000

Bentz, Dagmar; Laschat, Sabine: Synthesis of Perhydroindenes and Perhydroisoindoles via One-Pot Enyne Metathesis/Diels-Alder Reaction; Remarkable Stability of Grubbs Catalyst under Lewis Acidic Conditions

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Issue 11/2000

Kim, Sunggak; Yoon, Joo-Yong: Carbene Reactions of α-Oxacyclo- and α-Azacyclo-N-aziridinylimines: Effect of Heteroatom and Ring Size in the Ring Expansion Reaction

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Issue 10/2000

Meyer, Oliver G. J.; Fröhlich, Roland; Haufe, Günter: Asymmetric Cyclopropanation of Vinyl Fluorides: Access to Enantiopure Monofluorinated Cyclopropane Carboxylates

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Issue 09/2000

von Zezschwitz, Paultheo; Voigt, Katharina; Noltemeyer, Matthias; de Meijere, Armin: A New Methodology for Ring Enlargements by the Oxy-Cope Rearrangement: Ready Access to Highly Functionalized Medium-Size Rings

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Issue 08/2000

Roussi, Fanny; Chauveau, Ariane; Bonin, Martine; Micouin, Laurent; Husson, Henri-Philippe: Diastereoselective Cycloadditions of Chiral Non-racemic Azomethine Imines

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Issue 05/2000

Steif, Frank; Wibbeling, Birgit; Meyer, Oliver; Hoppe, Dieter: Enantio- and Diastereoselective Synthesis of (Protected) 2-Formyl- and 2-(Hydroxymethyl)-1-phenylalkane-1,3-diols from Chiral 2-Methoxy-3-tosyl-1,3-oxazolidines by Subsequent Asymmetric Formylation and Aldolization

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Issue 04/2000

Gebauer, Olaf; Brückner, Reinhard: β-Alkoxycarbonyl Enol Triflates as Precursors of Stereopure 3-Ene-1,5-diyne Building Blocks for the Chromophores of Neocarzinostatin, C-1027, Kedarcidin, Maduropeptin, and N1999A2

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Issue 03/2000

Huang, Wenwei; Tidwell, Thomas T.: Allenylketenes: Versatile Substrates in Nucleophilic, Electrophilic, and Cycloaddition Reactions

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Issue 02/2000

Bach, Thorsten; Krüger, Christa; Harms, Klaus: The Stereoselective Synthesis of 2-Substituted 3-Azabicyclo[3.2.0]heptanes by Intramolecular [2+2]-Photocycloaddition Reactions

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Issue 01/2000

Reddy, Katamreddy Subba; Solà, Lluís; Moyano, Albert; Pericàs, Miquel A.; Riera, Antoni: Synthesis of a 9-Fluorenone Derived β-Amino Alcohol Ligand Depicting High Catalytic Activity and Pronounced Non-linear Stereochemical Effects

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Issue 12/1999

Thum, Oliver; Hertweck, Christian; Simon, Helmut; Boland, Wilhelm: (6R,7R)-[4,5,6,7-²H₄]-Palmitoate and (8S,9R)-[8,9-²H₂]-l-erythro-Sphinganine: Probes for the Analysis of the Stereochemical Course of Δ⁶-Desaturases from Plants and Insects

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Issue 10/1999

Albrecht, Markus; Blau, Oliver; Witt, Karen; Wegelius, Elina; Nissinen, Maija; Rissanen, Kari; Fröhlich, Roland: Di(8-hydroxyquinoline) Derivatives for Supramolecular Chemistry: Syntheses and Solid State Superstructures

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Issue 09/1999

Menzel, Andreas; Öhrlein, Reinhold; Griesser, Helmut; Wehner, Volkmar; Jäger, Volker: A Short Synthesis of l-Acosamine Based on Nitroaldol Addition (Henry Reaction). Analysis of the Key Step Concerning Solvent and Temperature Effects

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Issue 08/1999

Shimizu, Takeshi; Ohzeki, Tomoya; Hiramoto, Katsuya; Hori, Nobuyuki; Nakata, Tadashi: Chloromethanesulfonate as an Efficient Leaving Group: Rearrangement of the Carbon-Carbon Bond and Conversion of Alcohols into Azides and Nitriles

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Issue 07/1999

Bolm, Carsten; Muñiz, Kilian; Aguilar, Núria; Kesselgruber, Martin; Raabe, Gerhard: The Search for Benchrotrenes and Ferrocenes Containing a Chiral Sulfoximido Group: Preparation and Structural Properties

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Issue 06/1999

Cossy, Janine; Blanchard, Nicolas; Meyer, Christophe: Stereoselective Synthesis of Cyclopropanes Bearing Adjacent Stereocenters

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Issue 05/1999

Kita, Yasuyuki; Egi, Masahiro; Takada, Takeshi; Tohma, Hirofumi: Development of Novel Reactions Using Hypervalent Iodine(III) Reagents: Total Synthesis of Sulfur-Containing Pyrroloiminoquinone Marine Product, (±)-Makaluvamine F

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Issue 04/1999

Chinchilla, Rafael; Galindo, Nuria; Nájera, Carmen: Chiral 3,6-Dihydro-2H-1,4-oxazin-2-ones as Alanine Equivalents for the Asymmetric Synthesis of α-Methyl α-Amino Acids (AMAAs) under Mild Reaction Conditions

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Issue 03/1999

Foubelo, Francisco; Gutiérrez, Ana; Yus, Miguel: Functionalized Organolithium Compounds by DTBB-Catalyzed Sulfur-Lithium Exchange

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Issue 02/1999

Takeuchi, Miwako; Taniguchi, Takahiko; Ogasawara, Kunio: Back to the Sugars: A New Enantio and Diastereocontrolled Route to Hexoses from Furfural

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Issue 12/1998

Aggarwal, Varinder K.; Vennall, Graham P.: Sc(OTf)₃, an Efficient Catalyst for Addition of Allyltrimethylsilane to Aldehydes; Chemoselective Addition to Aldehydes in Presence of Ketones and in situ Acylation (3 Component Coupling)

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Issue 11/1998

Kraft, Philip; Cadalbert, Riccardo: 4-Substituted 1,7-Dioxacycloalkan-8-ones: Preparation and Olfactory Properties

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Issue 10/1998

Shirakawa, Eiji; Yamasaki, Kenji; Hiyama, Tamejiro: Cross-Coupling Reaction of Organostannanes with Aryl Halides Catalyzed by Nickel-Triphenylphosphine or Nickel-Lithium Halide Complex

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Issue 09/1998

Effenberger, Franz; Grube, Gunther: Synthesis of Oligothienylfullerenes

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Issue 08/1998

Cahiez, Gérard; Avedissian, Hovsep: Highly Stereo- and Chemoselective Iron-Catalyzed Alkenylation of Organomagnesium Compounds

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Issue 07/1998

Ullmann, Astrid; Schnaubelt, Jürgen; Reissig, Hans-Ulrich: Synthesis of Highly Functionalized Cyclodecenone Derivatives from Siloxycyclopropanes: Scope and Limitations

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Issue 06/1998

Boßhammer, Stephan; Gais, Hans-Joachim: Synthesis and Alkylation of Cyclic α-Sulfonimidoyl Carbanions: Non-transferable Chiral Carbanionic Ligands in Copper-Mediated Enantioselective Conjugate Addition

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Issue 05/1998

Taylor, Richard J. K.; Alcaraz, Lilian; Kapfer-Eyer, Isabelle; Macdonald, Gregor; Wei, Xudong; Lewis, Norman: The Synthesis of Alisamycin, Nisamycin, LL-C10037α and Novel Epoxyquinol and Epoxyquinone Analogues of Manumycin A

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Issue 04/1998

Phansavath, Phannarath; Stammler, Robert; Aubert, Corinne; Malacria, Max: Synthesis of Variously Substituted Spirobenzocyclobutenes

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Issue 03/1998

Dünnwald, Thomas; Parham, Amir Hossain; Vögtle, Fritz: Non-ionic Template Synthesis of Amide-linked Rotaxanes: Axles with Benzophenone and Cinnamic Acid Units

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Issue 02/1998

Seela, Frank; Becher, Georg: Synthesis of 7-Halogenated 8-Aza-7-deaza-2′-deoxyguanosines and Related Pyrazolo[3,4-d]pyrimidine 2′-Deoxyribonucleosides

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Issue 01/1998

Lindström, Ulf M.; Somfai, Peter: Aminolysis of Vinyl Epoxides as an Efficient Entry to N-H Vinylaziridines

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Issue 12/1997

Gewehr, Markus; Kunz, Horst: Comparative Lipase-Catalyzed Hydrolysis of Ethylene Glycol Derived Esters. The 2-Methoxyethyl Ester as a Protective Group in Peptide and Glycopeptide Synthesis

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Issue 11/1997

Loiseleur, Olivier; Hayashi, Masahiko; Schmees, Norbert; Pfaltz, Andreas: Enantioselective Heck Reactions Catalyzed by Chiral Phosphinooxazoline-Palladium Complexes

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Issue 10/1997

Prévôté, Delphine; Le Roy-Gourvennec, Sylvie; Caminade, Anne-Marie; Masson, Serge; Majoral, Jean-Pierre: Application of the Horner-Wadsworth-Emmons Reaction to the Functionalization of Dendrimers: Synthesis of Amino Acid Terminated Dendrimers

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Issue 09/1997

Sebastian, Dagmar; Heuser, Axel; Schulze, Sonja; Waldmann, Herbert: Selective Enzymatic Removal of Protecting Groups from Phosphopeptides: Chemoenzymatic Synthesis of a Characteristic Phosphopeptide Fragment of the Raf-1 Kinase

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Issue 08/1997

Barluenga, José; Tomás, Miguel; López, Luis A.; Suárez-Sobrino, Angel: Efficient Approaches to the Stereoselective Synthesis of Chiral 2-Alkoxydienes and Heterodienes

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Issue 07/1997

Fürstner, Alois; Langemann, Klaus: Macrocycles by Ring-Closing Metathesis

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Issue 06/1997

Gompper, Rudolf; Mair, Hans-Jürgen; Polborn, Kurt: Synthesis of Oligo(diazaphenyls). Tailor-Made Fluorescent Heteroaromatics and Pathways to Nanostructures

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Issue 05/1997

Jahn, Ullrich; Andersch, Jens; Schroth, Werner: 3,3-Dichloroprop-2-ene Iminium Salts (Vinylogous Viehe Salts): A Study of Their Reactivity Towards Nucleophiles

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Issue 04/1997

Ashton, Peter R.; Horn, Thomas; Menzer, Stephan; Preece, Jon A.; Spencer, Neil; Stoddard, J. Fraser; Williams, David J.: Towards a Molecular Anchor Chain. Synthesis and Catenations of Spiro Crown Ethers

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Issue 03/1997

Mikoajczyk, Marian; urawiski, Remigiusz; Kiebasiski, Piotr; Wieczorek, Micha W.; Baszczyk, Jarosaw; Majzner, Wiesaw R.: Total Synthesis of Racemic and Optically Active Sarkomycin

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Issue 02/1997

Wirschun, Wolfgang; Jochims, Johannes C.: 1,3-Diaza-2-azoniaallene Salts, Novel N₃-Building Blocks: Preparation and Cycloadditions to Olefins

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Issue 01/1997

Kotora, Matin; Negishi, Ei-ichi: Highly Efficient and Selective Procedures for the Synthesis of γ-Alkylidenebutenolides via Palladium-Catalyzed Ene-Yne Coupling and Palladium- or Silver Catalyzed Lactonization of (Z)-2-En-4-ynoic Acids. Synthesis of Rubrolides A, C, D, and E

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Issue 12/1996

Creton, Isabelle; Marek, Ilane; Normant, Jean F.: Synthesis of Polysubstituted Stereodefined Olefins via the Reactivity of sp² Organo-gem-bismetallics

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Issue 11/1996

Yamago, Shigeru; Takeichi, Atsuo; Nakamura, Eiichi: Synthesis of Dimethyleneketene Acetals and Their [2+2] Cycloaddition to Olefins and [60]Fullerene as Cyclopropanecarboxylate Synthons

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Issue 10/1996

Eisenbrand, G.; Lauck-Birkel, S.; Tang, W. C.: An Approach Towards More Selective Anticancer Agents

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Issue 09/1996

Geyer, M.; Plenzig, F.; Rauschnabel, J.; Hanack, M.; del Rey, B.; Sastre, A.; Torres, T.: Subphthalocyanines: Preparation, Reactivity and Physical Properties

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Issue 08/1996

Slany, Michael; Stang, Peter J.: The Synthesis and Characterisation of Chiral Atropisomeric 4,4’-Biquinolines

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Issue 07/1996

Hudlicky, Tomas; Abboud, Khalil A.; Entwistle, David A.; Fan, Rulin; Maurya, Rakesh; Thorpe, Andrew J.; Bolonick, Joel; Myers, Brian: Toluene-Dioxygenase-Mediated cis-Dihydroxylation of Aromatics in Enantioselective Synthesis. Iterative Glycoconjugate CouplingStrategy and Combinatorial Design for the Synthesis of Oligomers of nor-Saccharides,Inositols and Pseudosugars with Interesting Molecular Properties

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Issue 06/1996

Hsung, Richard P.; Wulff, William D.; Challener, Cynthia A.: Stereoselective Benzannulations and Cyclohexadienone Annulations of Fischer Carbene Complexes in the Synthesis of Decala-2,4-dien-1-ones and in the Synthesis of Tetralin Chromium Tricarbonyl Complexes

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Issue 05/1996

Smith, Nicholas D.; Kocienski, Philip J.; Street, Stephen D. A.: A Synthesis of (+)-Herboxidiene A

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Issue 04/1996

Lange, Tim; Loon, Jan-Dirk van; Tykwinski, Rik R.; Schreiber, Martin; Diederich, François: Towards the Synthesis of Tetraethynylallene

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Issue 03/1996

Simonsen, Klaus B.; Svenstrup, Niels; Lau, Jesper; Simonsen, Ole; Mørk, Pernille; Kristensen, Gitte J.; Becher, Jan: Sequential Functionalisation of Bis-Protected Tetrathiafulvalene-dithiolates

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Issue 02/1996

Markó, István E.; Bayston, Daniel J.: Towards the Total Synthesis of Ambruticin: Preparation of the Fully Functionalised Right-Hand Portion Using the Intramolecular Silyl-Modified Sakurai (ISMS) Annulation

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Issue 01/1996

Lattmann, E.; Coombs, J.; Hoffmann, H. M. R.: Pyranofuranones via Lewis Acid Mediated Hetero-Diels-Alder Reactions of 4-Furan-2(5H)-ones: A Convergent Route to the Manoalide Substructure

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Issue 12/1995

Wipf, Peter; Kim, Yuntae; Jahn, Heike: Synthesis of (-)-LL-C10037α and Related Manumycin-Type Epoxyquinols

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Issue 11/1995

Matzeit, Agnes; Schäfer, Hans J.; Amatore, Christian: Radical Tandem Cyclizations by Anodic Decarboxylation of Carboxylic Acids

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Issue 10/1995

Katritzky, Alan R.; Wu, Hong; Xie, Linghong; Rachwal, Stanislaw; Rachwal, Bogumila; Jiang, Jinlong; Zhang, Guifen; Lang, Hengyuan: The Origins of the Benzotriazole Project, Its Versatility Illustrated by a New ^-C=CHCH⁺OEt Synthon, and Novel Syntheses of α,β-Unsaturated Aldehydes and Ketones, Furans, Pyrroles and Allyl Ethers

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Issue 09/1995

Kobayashi, Sh.; Ishitani, Haruro; Nagayama, Satoshi: Lanthanide Triflate Catalyzed Imino Diels-Alder Reactions; Convenient Syntheses of Pyridine and Quinoline Derivatives

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Issue 08/1995

Alexakis, Alex; Lensen, Nathalie; Tranchier, Jean-Philippe; Mangeney, Pierre; Feneau-Dupont, J.; Declercq, J. P.: Chiral Aminal Templates: Diastereoselective Addition to Hydrazones; An Asymmetric Synthesis of α-Amino Aldehydes

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Issue 07/1995

Schmidt, Richard R.; Bär, Thomas; Wild, Robert: Sphingosines - an Oxa-Cope Rearrangement Route for Their Synthesis

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Issue 06/1995

Trauner, Hans; Le Floch, Pascal; Lefour, Jean-Michel; Ricard, Louis; Mathey, François: Insertion of Palladium(0) and Nickel(0) Complexes into the α-Carbon-Bromine Bonds of 2-Bromo- or 2,6-Dibromophosphinines: A Versatile Route to α-Functionalised Phosphinines

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Issue 05/1995

Blechert, Siegfried; Knier, Ruth; Schroers, Harald; Wirth, Thomas: Domino Reactions - New Concepts in the Synthesis of Indole Alkaloids and Other Polycyclic Indole Derivatives

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Issue 04/1995

Pirrung, Frank O. H.; Hiemstra, Henk; Speckamp, W. Nico; Kaptein, Bernard; Schoemaker, Hans E.: Synthesis of Enantiomerically Pure Eight- and Nine-Membered Lactones by Copper(I) Chloride/2,2’-Bipyridine-Catalyzed Cyclization

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Issue 03/1995

Bruns, Wilfried; Horns, Stefan; Redlich, Hartmut: Botrylactone Synthesis and Structure Revision: A Convergent Approach from D-Glucose

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Issue 02/1995

Kauffmann, Thomas; Nienaber, Hubert: Alkyl Cyanoferrates, Cyanocobaltates, and Cyanonickelates as New Reagents for Cross-Coupling with Organic Halides

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Issue 01/1995

Mulzer, Johann; Funk, Günther: Synthesis of Optically Active β,γ-Unsaturated α-Amino Acids and of α,β-Unsaturated

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Issue 12/1994

Boese, Roland; Van Sickle, Andrew P.; Vollhardt, K. Peter C.: The Cobalt-Mediated [2+2+2] Cycloaddition of α,ω-Diynes to the 2,3-Double Bond of Indole

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Lipshutz, Bruce H.; Hayakawa, Hiroyuki; Kato, Kaneyoshi; Lowe, Richard F.; Stevens, Kirk L.: A Novel Route to Pyrimidine Nucleosides via Intramolecular Couplings of Bases with 2′-Deoxyribosides: Quick and Stereospecific...but with a 'Twist'

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Issue 11/1994

Tietze, Lutz F.; Bachmann, Jürgen; Wichmann, Jürgen; Burkhardt, Olaf: Inter- and Intramolecular Hetero-Diels-Alder Reactions; Part 50: Domino Reactions in Organic Chemistry: The Knoevenagel-hetero-Diels-Alder-Hydrogenation Sequence for the Biomimetic Synthesis of Indole Alkaloids via Strictosidine Analogues

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Issue 10/1994

Endo, Yasuyuki; Uchida, Takuya; Hizatate, Shoji; Shudo, Koichi: Anionic Hetero[3,3] and [3,5] Rearrangements of Hydroxylamine Derivatives Accompanied with N-O Bond Cleavage

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Issue 09/1994

Padwa, Albert; Harring, Scott R.; Hertzog, Donald L.; Nadler, William R.: Cycloaddition Chemistry of Anhydro-4-hydroxy-1,3-thiazolium Hydroxides (Thioisomünchnones) for the Synthesis of Heterocycles

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Issue 08/1994

De Brabander, Jef; Vandewalle, Maurits: Bryostatins: The Asymmetric Synthesis of the C₁-C₉ and C₁₇-C₂₇ Fragments

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Issue 07/1994

Reetz, Manfred T.; Hübel, Marcus; Jaeger, Ralf; Schwickardi, Renate; Goddard, Richard: Stereoselective Synthesis of α,β-Diamino Nitriles from Amino Acids

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Issue 06/1994

Hoffmann, Reinhard W.; Dahmann, Georg; Andersen, Marc W.: Stereoselective Synthesis of Alcohols, XLV: Recent Developments in the Generation of the Stereotriad "D"

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Issue 05/1994

Hayashi, Tamio; Iwamura, Hiroshi; Uozumi, Yasuhiro; Matsumoto, Yonetatsu; Ozawa, Fumiyuki: A New Optically Active Monodentate Phosphine Ligand, (R)-(+)-3-Diphenylphosphino-3′-methoxy-4,4′-biphenanthryl (MOP-phen): Preparation and Use for Palladium-Catalyzed Asymmetric Reduction of Allylic Esters with Formic Acid

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Issue 04/1994

Cabezas, Jorge A.; Oehlschlager, Allan C.: Regioselective Addition of Stannylcyanocuprates to Acetylenic Ethers: A Chemical and Spectroscopic Study

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Issue 03/1994

Mcneill, Alan H.; Thomas, Eric J.: Effective 1,5-Asymmetric Induction in Tin(IV) Chloride Promoted Reactions Between Aldehydes and (4-Alkoxy-2-alkenyl)tributylstannanes

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Issue 02/1994

Erker, Gerhard; Berlekamp, Martin; Lopez, Luis; Grehl, Matthias; Schönecker, Bruno; Krieg, Reimar: Syntheses of Substituted 6-Hydroxyhexenoic Acids and Related Tetrahydrofuran Systems by Metallocene-Template Directed 1,4-Selective Coupling of 1,3-Butadiene with Carbonyl Compounds

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Issue 01/1994

Adam, Waldemar; Peters, Karl; Sauter, Markus: Dimethyldioxirane Epoxidation of 3-Phenyl-Substituted Benzofurans: A Reversible Valence Isomerization between Benzofuran Epoxides and Quinone Methides

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Issue 12/1993

Juaristi, Eusebio; Beck, Albert K.; Hansen, Jesper; Matt, Thomas; Mukhopadhyay, Triptikumar; Simson, Malgorzata; Seebach, Dieter: Enantioselective Aldol and Michael Additions of Achiral Enolates in the Presence of Chiral Lithium Amides and Amines

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Issue 11/1993

Dondoni, Alessandro; Perrone, Daniela: 2-Thiazolyl α-Amino Ketones: A New Class of Reactive Intermediates for the Stereocontrolled Synthesis of Unusual Amino Acids

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Issue 10/1993

Rück, Karola; Kunz, Horst: Stereoselective Conjugate Addition of Organoaluminum Chlorides to α,β-Unsaturated Carboxylic Acid Derivatives

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Issue 09/1993

Kondo, Kazuhiro; Sodeoka, Mikiko; Mori, Miwako; Shibasaki, Masakatsu: Asymmetric Heck Reaction: Catalytic Asymmetric Syntheses of Bicyclic Enones, Dienones and the Key Intermediate for Vernolepin

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Issue 08/1993

Trost, Barry M.; Chang, Virginia K.: An Approach to Botrydianes: On the Steric Demands of a Metal Catalyzed Enyne Metathesis

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Issue 07/1993

Gonda, Josef; Helland, Anne-Charlotte; Ernst, Beat; Belluš, Daniel: Diastereoselective Synthesis of 1,2-Diamines by Palladium Catalyzed Aza-Claisen Rearrangement

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Issue 06/1993

Hanack, Michael; Schmid, Ulrich; Echinger, Stefan; Teichert, Frank; Hieber, Jürgen: Synthesis of Precursor Molecules for Low Band Gap Polymers

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Issue 05/1993

Tucker, Charles E.; Knochel, Paul: Preparation of Functionalized Z-Olefins Using 1,1-Dimetalloalkanes

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Issue 04/1993

Murahashi, Shun-Ichi; Naota, Takeshi: Ruthenium-Catalyzed Oxidations for Selective Syntheses of Ketones and Acyl Cyanides. Selective Acylation of Amino Compounds with Acyl Cyanides

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Issue 03/1993

Bäckvall, Jan-E.; Gatti, Roberto; Schink, Hans E.: Enzyme and Palladium Catalysis as a Powerful Combination in Asymmetric Transformations of meso-2-Alkene-1,4-diol Derivatives. Application to Enantiodivergent Synthesis of (R)- and (S)-(2,4-Cycloalkadienyl)acetic Acids

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Issue 02/1993

Meyers, A. I.; Schmidt, Wolfgang; Mckennon, Marc J.: Asymmetric Addition to Chiral Aromatic and Unsaturated Oxazolines Using a Novel Chiral Auxiliary

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Issue 01/1993

Balkenhohl, F.; Brüning, I.; Winterfeldt, E.: Stereoselective Synthesis of Acceptor Stabilized Prostacyclins

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