Synlett

Issue eFirst

Liao, Lihao; Zhao, Xiaodan: Modern Organoselenium Catalysis: Opportunities and Challenges

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Battisti, Umberto M.; Müller, Marius; García-Vázquez, Rocío; Herth, Matthias Manfred: Labeling of Highly Reactive Tetrazines using [¹⁸F]SuFEx

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Zeng, Zhiwei; Zhao, Zichang; Yin, Zhaoyang; Tang, Mingjie; Liu, Yuji; Huang, Wei; Tang, Yongxing: Assembling Nitroamino and Amino Groups on a Pyrazolyl-1,3,4-Oxadiazole Framework for the Construction of High-Performance and Insensitive Energetic Materials

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Ran, You; Xia, Honglei; Song, Siwei; Wang, Kangcai; Zhang, Qinghua: Thermostable Insensitive Energetic Materials Based on a Triazolopyridine Fused Framework with Alternating Nitro and Amine Groups

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Roy, Tamal; Lee, Ji-Woong: Cyanide-Mediated Synthesis of Sulfones and Sulfonamides from Vinyl Sulfones

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Onuska, Nicholas P. R.; Schutzbach-Horton, Megan E.; Rosario Collazo, José L.; Nicewicz, David. A.: Anti-Markovnikov Hydroazidation of Activated Olefins via Organic Photoredox Catalysis

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Angelini, Lucrezia; Malet Sanz, Laia; Leonori, Daniele: Divergent Nickel-Catalysed Ring-Opening–Functionalisation of Cyclobutanone Oximes with Organozincs

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Ye, Fei; Xu, Li-Wen: A Glimpse and Perspective of Current Organosilicon Chemistry from the View of Hydrosilylation and Synthesis of Silicon-Stereogenic Silanes

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Reinhard, Dominik L.; Kutzinski, Dana; Hatta, Masahito; Engelage, Elric; Huber, Stefan M.: Evaluation of a Bidentate ‘Clamp-Like’ Halogen-Bond Donor Motif Based on Iodonium(III) Moieties

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Issue 04/2025

Dou, Chenguang; Yang, Ming: Synthetic Studies Toward Daphnezomines A and B

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Issue 19/2024

van Gemmeren, Manuel; Beller, Matthias: Late-Stage C–H Deuteration of Organic Compounds via Ligand-Enabled Palladium-Catalyzed Hydrogen Isotope Exchange

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Issue 17/2024

Huang, Haifeng; Yang, Jun: Cluster Preface: Synthesis of Energetic Molecules

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Issue 11/2024

Fukase, Koichi: Cluster Preface: Japan/Netherlands Gratama Workshop

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Rutjes, Floris P. J. T.; Bonger, Kimberly M.; Neumann, Kevin: Bioorthogonal Chemistry at Radboud University: Past, Present and Future

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de Paus, Laura V.; Janssen, Antonius P.A.; Halimi, Asad; van den Berg, Richard J. B. H. N.; Heitman, Laura H.; van der Stelt, Mario: Discovery of a Cannabinoid CB₂ Receptor Fluorescent Probe Based on a Pyridin-2-yl-benzyl-imidazolidine-2,4-dione Scaffold

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Aartsma-Rus, Annemieke: Applying Lessons Learned from Developing Exon Skipping for Duchenne to Developing Individualized Exon Skipping Therapy for Patients with Neurodegenerative Diseases

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Yano, Kumpei; Yoshimoto, Takuya; Tsutsui, Masato; Manabe, Yoshiyuki; Fukase, Koichi: Validation and Application of an Innovative Protective Group Concept: Enhancing Substrate Reactivity in Glycosylations by Disrupting Intermolecular Interactions

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Muta, Kensuke; Okamoto, Kazuhiro; Nagaki, Aiichiro: Reaction of Highly Volatile Organic Compounds with Organolithium Species in Flow Microreactor

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Kitano, Junya; Nishii, Yuji; Hirano, Koji; Miura, Masahiro: Rhodium-Catalyzed Direct Vinylene Annulation of 2-Aryloxazolines and Cascade Ring-Opening Using a Vinyl Selenone

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Umegawa, Yuichi; Fukunaga, Shiho; Yasuda, Tomokazu; Murata, Michio: A Fluorescent Probe for C₂₄ Fatty Acids to Report the Deep Interior of Lipid Bilayers

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Manabe, Yoshiyuki; Hizume, Koki; Takakura, Yohei; Takamatsu, Shinji; Miyoshi, Eiji; Kamada, Yoshihiro; Hurtado-Guerrero, Ramón; Fukase, Koichi: Systematic Strategy for the Development of Glycosyltransferase Inhibitors: Diversity-Oriented Synthesis of FUT8 Inhibitors

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Komine, Keita; Yamazaki, Yuta; Iwanaga, Taiga; Sakaguchi, Hikaru; Fukuda, Hayato; Ishihara, Jun: Visible-Light-Induced Three-Component Radical Coupling of Selenocarbamates, Enones, and Allylstannanes with Diphenyl (2,4,6-trimethylbenzoyl)phosphine Oxide

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Mikame, Yu; Maekawa, Nagisa; Kimura, Soichiro; Nakao, Juki; Yamayoshi, Asako: Modular Synthesis of Methyl-Substituted Novel Psoralen N-Hydroxysuccinimide Esters and Evaluation of DNA Photocrosslinking Properties of the Corresponding Triplex-Forming Oligonucleotide Conjugates

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Reintjens, Niels R. M.; Bartels, Imke M. A.; Marinus, Nittert; Massmann, Sarina C.; Bunt, Daan V.; Walvoort, Marthe T. C.; Witte, Martin D.; Minnaard, Adriaan J.: Practical Site-Selective Oxidation of Glycosides with Palladium(II) Acetate/Neocuproine

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Xu, Hang; Yamaguchi, Sho; Mitsudome, Takato; Mizugaki, Tomoo: Efficient Protosilylation of Unsaturated Compounds with Silylboronates over a Heterogeneous Cu₃N Nanocube Catalyst

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Omae, Tomoki; Nakahata, Masaki; Kamon, Yuri; Hashidzume, Akihito: Synthesis of an Alternating Polycation with the Dense 1,2,3-Triazole Backbone

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Tanaka, Yuya; Yashiro, Atsushi; Akita, Munetaka: Thermally Stable Monoruthenium Acetylide Radical Species

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Issue 10/2024

Zeng, Wei-Long; Jiang, Xu; Li, Wei: Chromium-Promoted Dearomative (Deutero)Hydrocyanoalkylation of (Hetero)Arenes Using Simple Alkylnitriles

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Rummler, Lénaic; Sater, Mariam Abd El; Blanchard, Nicolas; Bizet, Vincent: Copper-Catalyzed Regiodivergent Borylation of Fluorinated Alkynes and Palladium-Catalyzed Regiospecific Suzuki–Miyaura Cross-Coupling

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Ramakrishna, Isai; Hattori, Tomohiro; Ishiguro, Tomomi; Yamamoto, Hisashi: Triisobutylaluminium-Mediated Regioselective Protection of Sterically Hindered Amide NH of Cyclo-(AA-Gly): Key Building Block for Next-Generation Peptide Synthesis

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Zhang, Lanlan; Zhao, Lei; Zhu, Yuqin; Wang, Chao: Quinolinamide-Enabled Nickel-Catalyzed Regio- and Diastereoselective γ,δ-Arylalkylation of Nonactivated Alkenes

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Su, Gillian A.; Reiter, Paul; Schulz, Michael D.: Evaluating Catalyst Performance in Synthesizing Hydroxyl-Terminated Polybutadiene by Ring-Opening-Metathesis Polymerization

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Tang, Xinxin; Noda, Hidetoshi; Shibasaki, Masakatsu: anti-Selective Synthesis of Substituted β-Homoprolines by Rhodium Alkyl Nitrene C–H Insertion

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Herrera, Christian L.; Oliveira, Rafael L.; Silva, Rodrigo C.; Correia, Carlos R. D.; Pastre, Julio C.: Enantioselective Heterogeneous Heck–Matsuda Reaction with Polymer-Supported PyOx Ligands

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Banerjee, Somsuvra; Matsushita, Naoki; Nakamura, Eiichi; Patil, Nitin T.; Asako, Sobi; Ilies, Laurean: Molybdenum-Catalyzed Directed Activation of Aryl Chlorides and Fluorides

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Chiang, Hsin-Lun; Zhao, Wei-Ting; Chen, Yi-An; Lin, Yi-Ching; Chen, Pei-Lin; Wu, Yen-Ku: Palladium-Catalyzed α-Arylation of Meyers’s Chiral Bicyclic Lactams and a Deprotonative Ring-Opening Sideline

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Sanosa, Nil; Montiel-Cervantes, César; Rubio-Muñoz, Miguel; Sampedro, Diego; Funes-Ardoiz, Ignacio: Rationalizing the Regioselectivity of Azolation of Benzylic C–H Bonds under Photoredox Catalysis

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Ye, Xingchen; Wang, Zhaofeng: Synthesis of 2,4-Disubstituted Oxazoles by a Copper-Catalyzed [3+2] Annulation/Olefination Cascade between Amides and I^III/P^V Hybrid Ylides

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Yao, Bo-Ying; Xiao, Wei-Guo; Xiao, Li-Jun; Zhou, Qi-Lin: Nickel-Catalyzed Hydroalkynylation of 1,3-Dienes with Simple Alkynes

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Li, Wenjuan; Shen, Chaoren; Zhu, Yanping; Dong, Kaiwu: Practical Fischer Indolization Using Bench-Stable Arylhydrazine Sulfonate as the Surrogate of Arylhydrazine

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Zhang, Tianyu; Zhu, Can: Enzymatic Kinetic Resolution (EKR) of α-Allenols Enabled by a Commercially Available Immobilized Lipase

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Zhang, Guoxiang; Xue, Ting; Wang, Liting; Wang, Sichang; Ke, Congyu; Zeng, Rong: FeCl₃-Catalyzed Aerobic Oxidative Degradation of Polystyrene to Benzoic Acid: Scope and Mechanism

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Ngamnithiporn, Aurapat; Chuentragool, Padon; Songthammawat, Poramate; Punnita, Supakarn; Photong, Kittithuch; Ploypradith, Poonsakdi; Ruchirawat, Somsak: Sultines as o-Quinodimethane Precursors in an Oxa-Diels–Alder Reaction: Synthesis of Functionalized Isochromans

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Peng, Xiaolin; Wang, Yulin; Huang, Yixian; Zhang, Sheng; Jin, Zhichao; Ren, Shi-Chao: N-Heterocyclic Carbene Catalysis for Facile Access to Pentasubstituted 4H-Pyran Derivatives

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Nowak, Jan; Tryniszewski, Michał; Barbasiewicz, Michał: Are β-Lactones Involved in Carbon-Based Olefination Reactions?

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Issue 09/2024

Foja, Richard; Walter, Alexandra; Storch, Golo: Chemoselective Reduction of Barbiturates by Photochemically Excited Flavin Catalysts

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Geik, Dennis; Büker, Alina; Fornfeist, Felix; Schmidtmann, Marc; Doye, Sven: Catalytic C–H Functionalization of Trimethylamine

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Oliver, Gwyndaf A.; Kolb, Simon; Werz, Daniel B.: Electrocatalytic Synthesis of 1,2-Dioxolanes from Tetrasubstituted Donor–Acceptor Cyclopropanes

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Nandi, Shiny; Paffen, Alina; Patureau, Frederic W.: Aromatic Amine Catalysts for the O₂-Mediated Cross-Dehydrogenative Phenothiazination Reaction?

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Oelze, Silke; Bräuer, Nico; Michel, Tycho; Schaumann, Ernst; Kirschning, Andreas: [4+1] Cyclizations to Enantiopure Multifunctional Cyclopentanes from d-Glucose Using Formyl Dianion Synthons

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Fliegel, Lukas; Krauß, Julian; Christoffers, Jens: Ring Transformation of Annulated Benzofuran Derivatives to Medium-Sized Lactones

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Ahmed, Hussayn; Pöthig, Alexander; Truong, Khai-Nghi; Bach, Thorsten: Remote Enantioselective Epoxidation Reactions Catalyzed by Chiral Iron Porphyrin Complexes with a Hydrogen-Bonding Site

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Gorai, Mahadeb; Teichert, Johannes F.: Chiral Bifunctional NHC–Guanidine Ligands for Asymmetric Hydrogenation

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M. Bopape, Karabo; Shah, Aryan; Koenigs, Rene M.: Photocatalytic [2,3]-Sigmatropic Rearrangement Reactions of Ethyl Diazoacetate

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Friedmann, Till; Mireles-Chávez, Daniel A.; Walter, Frederik L.; Schneider, Christoph: Enantioselective (3+2)-Annulation of β-Keto Esters with Azoalkenes towards Bicyclic Dihydropyrroles via Cooperative Palladium and Brønsted Acid Catalysis

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Arnold, Andreas M.; Binder, Julia; Kretzschmar, Martin; Gulder, Tanja: Alkene versus Aryl Chlorination in Asymmetric Hypervalent Iodine Catalysis: A Case Study

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Heckmann, Felix; Ibrahim, Mohammad M.; Hampel, Frank; Tsogoeva, Svetlana B.: Synthesis of New Highly Functionalized Quinolines via a Novel Fe^III-Catalyzed Domino aza-Michael/Aldol/Aromatization Reaction

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Kail, Sascha; Hilt, Gerhard: The FeBr₃-Catalyzed Transfer Hydrogenation of Styrene Derivatives under Mild Reaction Conditions

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Spinnato, Davide; Leutzsch, Markus; Wang, Feng; Cornella, Josep: Internal Atom Exchange in Oxazole Rings: A Blueprint for Azole Scaffold Evaluation

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Große, Michel; Wegner, Hermann A.: Bidentate Lewis Acid-Catalyzed Inverse Electron-Demand Diels–Alder Reaction of Phthalazines and Cyclooctynes

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Langer, Lukas S.; Stahlberger, Mareen; Bär, Robin M.; Bräse, Stefan: A Novel Route towards Bicyclo[1.1.1]pentane Sulfoxides from a Bench-Stable Starting Material

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Hamad, Aboubakr; Mrozowicz, Michał; Xie, Yuanhao; Ritter, Tobias: Regioselective Double C–H Functionalization of Arenes via Aryl Thianthrenium Salt Analogues

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Stahlberger, Mareen; Mergel, Milada; dos Santos, John Marques; Matulaitis, Tomas; Nieger, Martin; Zysman-Colman, Eli; Bräse, Stefan: Design of Imidazo[1,2-a]pyridine-Based Donor–Acceptor Chromophores through a Multicomponent Approach

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Langhans, Alexander; Krummhaar, Michael; Roth, Christian; Koksch, Beate: Catalytically Competent Fluorinated Barnase Variants

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Rohlfs, Tabea; Gerken, Leon; Nova-Fernández, Jose L.; Malagón, Sara; Uygur, Mustafa; Cabrera, Silvia; Alemán, José; Mancheño, Olga García: Visible-Light-Mediated Selective Allylic C–H Oxygenation of Cycloalkenes

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Dressler, Friedemann; Öhler, Victoria; Topp, Christopher; Schreiner, Peter R.: Organocatalytic, Chemoselective, and Stereospecific House–Meinwald Rearrangement of Trisubstituted Epoxides

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Stahl, Jessica; Reiter, Thilo; König, Burkhard: Chemoselective Vicinal Dichlorination of Alkenes by Iron Ligand-to-Metal Charge-Transfer Catalysis

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Baumert, Benjamin; Terholsen, Henrik; Cziegler, Clemens; Thier, Isabel; Badenhorst, Christoffel P. S.; Siems, Karsten; Bornscheuer, Uwe T.: Enzymatic Synthesis of Hydroxycinnamic Acid Amides in Water Using the Promiscuous Hydrolase/Acyltransferase PestE from Pyrobaculum calidifontis VA1

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Issue 08/2024

Campeau, Louis-Charles: A Personal Account from Inside Keith Fagnou’s Research Laboratory

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Gallagher, Rory T.; Jha, Soocheta; Metze, Bryan E.; Stuart, David R.: Synthesis of Alkyl Aryl Ethers by O-Arylation of Alcohols with Diaryliodonium Salts: Scope, Limitations, and Mechanism

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Palermo, Anthony F.; Imbriaco, Bianca; Chan, Samantha C.; Doan, Brian A.; Rousseaux, Sophie A. L.: Asymmetric Cu(I)-Catalyzed Conjugate Borylation of α,β-Unsaturated Acyl Silanes

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Trofimova, Alina; Brien, Chelsey; Tan, Joanne; Trudel, Vincent; Yudin, Andrei K.: An Exploration of Regioselectivity During Formation of Aminoboronates from Epoxides

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Struwe, Julia; Oyama, Tsuyoshi; Gallou, Fabrice; Ackermann, Lutz: Manganese(I)-Catalyzed C–H Allylation of Tryptophans and Their Oligopeptides On Water

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Zheng, Yan-Long; Daneshfar, Omid; Li, Jia-Yi; Masson-Makdissi, Jeanne; Pinault-Masson, Émile; Newman, Stephen G.: Nickel-Catalyzed Transesterification of Methyl Esters

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Yatzoglou, Giorgos; Zambri, Matthew T.; Desai, Shrey P.; Taylor, Mark S.: Synergistic Organoboron/Palladium Catalysis for Regioselective N-Allylation of 2-Pyridones, 4-Pyridones, and Related Ambident Heterocycles

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Atsumi, Wataru; Kawabata, Keiichi; Yamane, Mina; Oi, Miku; Mitsunuma, Harunobu; Sohma, Youhei; Hori, Yukiko; Tomita, Taisuke; Kanai, Motomu: Rose Bengal Promoted Catalytic Amyloid-β Oxygenation by Sonoactivation

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Takishima, Ryo; Ghosh, Koushik; Nishii, Yuji; Miura, Masahiro: Synthesis of Axially Chiral Bibenzo[g]coumarin Derivatives by Rhodium-Catalyzed Oxidative Annulation of Thiocarbamates

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Rodríguez-Flórez, Lesly V.; Retamosa, María de Gracia; Martínez-Sánchez, Beatriz; Cazorla-Amorós, Diego; Nájera, Carmen; Yus, Miguel; Sansano, José M.: Microwave-Assisted Functionalization of Single-Walled Carbon Nanotubes as a Platform for a Supported Iridium Catalyst

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Choi, Eun Seo; Rousseaux, Sophie A. L.; Huestis, Malcolm P.: Nickel-Catalyzed Synthesis of Benzylamines from (Hetero)aryl Halides and Glycine-Derived N-Hydroxyphthalimide Esters

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Issue 06/2024

Kumpina, Ilze; Baskevics, Vladislavs; Walby, Grant D.; Tessier, Brandon R.; Saei, Sara Farshineh; Ryan, Christopher A.; MacKay, James A.; Katkevics, Martins; Rozners, Eriks: Synthesis of 2-Aminopyridine-Modified Peptide Nucleic Acids

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Shet, Harshita; Sahu, Rajesh; Sanghvi, Yogesh S.; Kapdi, Anant R.: Palladium-Catalyzed Cyanation of Nucleobases: Total Synthesis of Toyocamycin, Sangivamycin, and a Mycalisine A Precursor

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Benckendorff, Caecilie M. M.; Hawes, Chris S.; Smith, Mark; Miller, Gavin J.: Chemical Diversification of Carbocyclic Fluorinated Pyrimidine Nucleosides: Introducing 2′-Arabino Analogues and Ring Unsaturation

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El Mansouri, Az-eddine; Lachhab, Saida; Mehdi, Ahmad; Ait-Ali, Mustapha; Sanghvi, Yogesh S.; Zahouily, M.; Lazrek, Hassan B.: BF₃@K10: An Efficient Heterogeneous Montmorillonite Catalyst for the Halogenation of N-Heterocycles

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Li, Quanjian; Sanghvi, Yogesh S.; Yan, Hongbin: Solvent Selection in the Detritylation Reaction for the Solid-Phase Synthesis of Oligonucleotides

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Niogret, Germain; Röthlisberger, Pascal; Levi-Acobas, Fabienne; Bonhomme, Frédéric; Gasser, Gilles; Hollenstein, Marcel: Facilitated Synthetic Access to Boronic Acid-Modified Nucleoside Triphosphates and Compatibility with Enzymatic DNA Synthesis

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Maverick, Mary Anne; Noël, Mathieu; Vasseur, Jean-Jacques; Baraguey, Carine; Debart, Françoise; Smietana, Michael: Serendipitous Synthesis of 5-Hydroxyuridine from 2′,3′-O-Isopropylidene N4-Acetylcytidine by Hypervalent Iodine(III)-Mediated Reaction

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Meher, Sagarika; Gade, Chandrasekhar Reddy; Sharma, Nagendra K.: Fluorescent 2′-Deoxyuridine (dU) Analogue: Tropolonyl triazolyl-dU (tt-dU) Exhibits Solvatochromism/HeLa Cell Internalization and Its Triphosphate (tt-dUTP) Is Incorporated into DNA Enzymatically

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Prakash, Thazha P.; Yu, Jinghua; Vasquez, Guillermo; Allerson, Charels R.; Swayze, Eric E.: A Facile Synthesis of 3′-Fluoro Hexitol Adenosine and Guanosine Phosphoramidites

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Hou, Jiao; Wang, Jian-Hua; Yu, Wenquan; Chang, Junbiao: Synthesis of 2′-Deoxy-2′-β-fluoro-4′-azido-5-fluorouridine as a Potential Anti-HIV Agent

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Sarma, Daisy; Majumdar, Biju; Chaput, John C.: Alternative Synthesis of α-l-Threofuranosyl Guanosine 3′-triphosphate

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Oku, Yurino; Kai, Misaki; Kobayashi, Saika; Katoh, Ryuzi; Saito, Yoshio: Acyclic 2-Ethynylnaphthalene-Modified 8-Aza-3,7-dideaza-2′-deoxyadenosine Allows Thymine Discrimination by Probing the DNA Minor Groove Environment

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Fuchi, Yasufumi; Kawaguchi, Miho; Ito, Yuta; Hari, Yoshiyuki: Synthesis and Properties of 2′-Deoxyadenosine Mimics Bearing a Thieno[3,2-d]pyrimidine Ring

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Navarro, Natalia; Serantes, Sergio; Aviñó, Anna; Fàbrega, Carme; Eritja, Ramon: Synthesis and Evaluation of 3′-Oleyl–Oligonucleotide Conjugates as Potential Cellular Uptake Enhancers

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Kumamoto, Hiroki; Imoto, Shuhei; Kuwata-Higashi, Nobuyo; Mitsuya, Hiroaki; Haraguchi, Kazuhiro: Regio- and Stereoselective Synthesis of 2′-Deoxy-4′-thioguanine Nucleosides: Evaluation of Anti-Hepatitis B Virus Activity and ­Cytotoxicity Leading to Improved Selectivity Index by 4′-C-Cyanation

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Issue 05/2024

Sakamoto, Jukiya; Hiruma, Daiki; Kitajima, Mariko; Ishikawa, Hayato: Collective Total Synthesis of β-Carboline-Type Monoterpenoid Indole Alkaloid Glycosides

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Kuang, Yang; Chang, Le; Wang, Bingjian; Kang, Jingyi; Chong, Chuanke; Lu, Zhaoyong: Practical and Scalable Total Syntheses of (+)-Dysidavarones A–C

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Han, Shoule; Lou, Mingliang; Qi, Xiangbing: Bioinspired Formal Synthesis of Pancracine via Selective Hydro­genation of an Indole Derivative

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Park, Sangbin; Kim, Doyoung; Yang, Wooil; Han, Sunkyu: Total Synthesis of 4α-Hydroxyallosecurinine and Securingine F, Securinega Alkaloids with a C4-Hydroxy Handle for Biofunctional Derivatizations

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Deng, Jun; Tang, Yefeng: Cluster Preface: Biomimetic Synthesis

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Issue 04/2024

Sato, Tomohiko; Karad, Somnath N.; Shimokawa, Jun; Yorimitsu, Hideki: Regioselective anti-Silyllithiation of Propargylic Amines

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Yagita, Ryotaro; Irie, Kazuhiro; Tsukano, Chihiro: Toward the Total Synthesis of Schinortriterpenoids: Construction of the All-cis-Substituted Cyclopropane Unit

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Kage, Ayaha; Okuyama, Yuya; Kato, Erina; Matagawa, Tomoe; Kawano, Sayaka; Simizu, Siro; Chida, Noritaka; Okamura, Toshitaka; Sato, Takaaki: Synthesis and Evaluation of Saponins with All-Nitrogenated Sugars

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Hosoya, Masahiro; Mori, Atsunori; Okano, Kentaro: Regiodivergent Synthesis of Brominated Pyridylthiophenes by Overriding the Inherent Substrate Bias

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Inaba, Ryoto; Kikuchi, Takashi; Imoto, Hiroaki; Naka, Kensuke: Synthesis and Coordination Behavior of 9,10-Diarsatriptycene

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Ando, Yoshio; Ogawa, Daichi; Wakita, Fumihiro; Suzuki, Keisuke; Ohmori, Ken: Photochemical Reaction of 1,2-Naphthoquinone toward Enantioselective Synthesis of γ-Rubromycin: Viability Dependence on Chromophore

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Lezius, Lena; Reimler, Jannik; Döben, Nadine; Hamm, Michael; Daniliuc, Constantin G.; Studer, Armido: Aminoacylation of Alkenes by Cooperative NHC and Photoredox Catalysis

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Aida, Kazuhiro; Ota, Eisuke; Yamaguchi, Junichiro: Regioselective Ring Opening of Oxetanes Enabled by Zirconocene and Photoredox Catalysis

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Fujii, Ikuya; Higo, Ryota; Semba, Kazuhiko; Nakao, Yoshiaki: Magnesiation of Alkyl Fluorides Catalyzed by Rhodium–Aluminum Bimetallic Complexes

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De, Pinaki Bhusan; Ilies, Laurean; Takai, Kazuhiko; Asako, Sobi: Synthesis of 2,2′-Bipyridines via Dehydrogenative Dimerization of Pyridines Using Sodium Dispersion

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Yuan, Xiaobin; Qu, Yanjie; Li, Yajun; Bao, Hongli: Synthesis of Carbamoyl Azides from Redox-Active Esters and TMSN₃

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Ikeda, Kotaro; Harada, Shingo; Hashimoto, Yoshinori; Homma, Haruka; Kono, Masato; Zumbrägel, Nadine; Gröger, Harald; Nemoto, Tetsuhiro: Enantioselective Formal Synthesis of (–)-Catharanthine through Enzyme-Catalyzed Desymmetrization of a meso-Azabicyclo [2.2.2]octane

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Hayashi, Shunya; Takasu, Kiyosei; Takikawa, Hiroshi: Sequential Bromination/Dearomatization Reactions of 2-Methoxyphenols en route to Bromo-Substituted ortho-Quinonemonoacetals

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Mori, Taiki; Sumida, Sao; Furuya, Yasuaki; Shirakawa, Seiji: Chiral Bifunctional Sulfide-Catalyzed Enantioselective Synthesis of α-Substituted γ-Lactones Bearing a γ-Quaternary Stereocenter

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Issue 03/2024

Priya, V R Padma; Mercy, A Antony Haritha; Natarajan, K; Nandi, Ganesh Chandra: Sulfoximines as S-Aryl Surrogates: A Photocatalytic Rapid, Metal-Free, Mild Protocol to Access 3-Arylsulfenyl Indoles

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Smyth, Megan; Moody, Thomas S.; Wharry, Scott; Baumann, Marcus: Continuous-Flow Synthesis of Cyclobutenes Using LED Technology

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Sardar, Santosh Sing; De, Aramita; Pal, Satyajit; Sarkar, Subhankar; Santra, Sougata; Zyryanov, Grigory V.; Majee, Adinath: Visible-Light-Driven Denitrogenative C–C Bond Formation and Oxidative Difunctionalization of Vinyl Azides

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Cervantes-González, Javier; Mora-Rodríguez, Salma E.; Benitez-Puebla, Luis J.; López-Caamal, Fernando; García-Revilla, Marco A.; Vázquez, Miguel A.; Lagunas-Rivera, Selene: A Computational and Experimental Analysis of Aldehyde Photooxidation Driven by Visible Light in a Homemade Reactor

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Okumura, Shintaro; Takahashi, Teruki; Torii, Kaoru; Uozumi, Yasuhiro: Photocatalytic 1,4-Addition of Aromatic Aldehydes or Ketones via Umpoled Carbinol Anions

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Nowack, Marko H.; Moutet, Jules; Laursen, Bo W.; Gianetti, Thomas L.: Triangulenium Ions: Versatile Organic Photoredox Catalysts for Green-Light-Mediated Reactions

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Shanthi, Markabandhu; Perumal, Karuppaiah; Sivalingam, Soumya; Puhazhendhi, Arulmozhi; Kumar Mandali, Pavan; Ramesh, Subburethinam: Transition-Metal-Free and Photocatalyst-Free Sulfenylation of Halopyrazolamines under Visible-Light Irradiation via Electron Donor–Acceptor Complexes

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Singh, Shweta; Gremaud, Ludovic; Sen, Subhabrata; Maiti, Debajit: A Combination of Computational and Experimental Studies to Correlate Electronic Structure and Reactivity of Donor–Acceptor Singlet Carbenes

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Austin, Brooke E.; Palner, Ryan P.; Tobias, Elissa M.; Madiu, Rufai; Doran, Erin L.; Doran, Jenna M.; Howard, Amari M.; Stroud, James L.; Rossi, Morgan E.; Moskovitz, Dylan A.; Rivera, Dominic A.; Mullen, Michael D.; Zinsky, Amy H.; Rosario, Rose A.; Moura-Letts, Gustavo: Visible-Light-Promoted Synthesis of Vinyloxaziridines from Conjugated Carbonyls

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Gkizis, Petros L.; Serviou, Stamatis K.; Balaskas, Angelos; Constantinou, Constantinos T.; Triandafillidi, Ierasia; Kokotos, Christoforos G.: Anthraquinone-Catalyzed Photooxidation of Boronic Acids in a Bio-Based Solvent (2-Me-THF)

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Jung, Jaehyun; Kinoshita, Takumi; Makihara, Yuta; Sakakibara, Yota; Amaike, Kazuma; Murakami, Kei; Itami, Kenichiro: Nickel/Photoredox-Catalyzed Decarboxylative Coupling of Aryl Bromides with N-Protected Glycine as an Aminomethyl Source

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Kurtay, Gülbin; Lusseau, Jonathan; Robert, Frédéric; Landais, Yannick: Iron-Catalyzed Oxidative Decarboxylation of Oxamic Acids: A Safe and Efficient Photochemical Route to Urethanes

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Zhang, Yi; Nie, Guihua; Jin, Zhichao; Ren, Shichao: Photoredox Defluorinative Silylation of α-Trifluoromethyl Arylalkenes Using Silacarboxylic Acids as Silyl Radical Precursors

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Miyajima, Ryo; Okamura, Manon; Oomori, Kazuki; Iwamoto, Hajime; Wakamatsu, Kan; Hasegawa, Eietsu: Desulfonylative Radical Truce–Smiles Rearrangement Utilizing the Benzimidazoline and Benzimidazolium Redox Couple

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Hashimoto, Ryoga; Furutani, Toshiki; Suzuki, Hirotsugu; Yoshimi, Yasuharu: Effects of Electron-Donor and Counter-Cation in Photoinduced Deboronative and Decarboxylative Aryl Radical Generation Using Two-Molecule Photoredox Catalysts

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Morizumi, Haruka; Nakayama, Kaii; Kitano, Yoshikazu; Okada, Yohei: Redox-Tag-Guided Radical Cation Diels–Alder Reactions: Use of Enol Ethers as Dienophiles

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Issue 01/2024

Yang, Youjun; Fan, Jiangli: Cluster Preface: Functional Dyes

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Koli, Mrunesh; Mula, Soumyaditya: Synthesis of Heavy-Atom-Free Triplet Photosensitizers Based on Organoboron Complexes

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Zhou, Meizhu; Hu, Xinhu; Zhang, Dongxiang; Cui, Tianfang; Jiang, Xin-Dong: Synthesis of a Heavy-Atom-Free BODIPY and its Photooxygenation of 1-Naphthol to 1,4-Naphthoquinone

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Wu, Ruixin; Li, Zipeng; Xia, Tianping; Cai, Wenlin; Du, Jianjun; Fan, Jiangli; Peng, Xiaojun: Synthesis of an Azo-Cyanine Dye as an RNA Probe for Distinguishing Gram-Positive Bacteria from Gram-Negative Bacteria

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Li, Jin; Wei, Ruwei; Zhang, Xiaodong; Luo, Xiao; Qian, Xuhong; Yang, Youjun: A Practical Synthesis of Near-Infrared Benzannulated Xanthenoid Dyes

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Dong, Yunhong; Cheng, Lin; Duan, Yanjuan; Xu, Huiru; Dong, Ruonan; Guo, Baolin; Cao, Liping: Dual Responses of Fluorescence and Circular Dichroism for Antibiotics by a Cationic Cage in Water

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Shan, Shiquan; Pang, Songhao; Qu, Yunwei; Lu, Yongna; Cheng, Xiamin; Li, Lin: Photooxidative Coupling of Thiols Promoted by Bromo(trichloro)methane in a Basic Aqueous Medium

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Wang, Wanying; Yao, Qichao; Xu, Runfeng; Wang, Ankang; Chen, Pengzhong; Peng, Xiaojun: Novel Zinc(II) Phthalocyanine Dyes for Color Photoresists

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Roy, Tirupati; Debnath, Indraneel; Mahata, Kingsuk: Tunable Optical Properties and Self-Assemblies of a Water-Soluble Perimidinium Imide Dye

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Zeng, Zhi-Yong; Zhao, Xiaoli; Huang, Junhai; Zhu, Jing; Jin, Tongxia; Hu, Lianrui; Dou, Wei-Tao; Xu, Lin: Anthracene-Functionalized Metallacage with Fluorescence Response Behavior to Anions

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Shi, Lei; Yu, Ai-Wen; Meng, Wei-Han; Xie, Kun-Peng; Li, Kun: Purine-Based AIEgens with Different Morpholine Substitution Sites and Their Application in Lipophagy Imaging

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Wu, Shuyao; Zhang, Xinfu; Li, Xiaoxi; Sun, Shulan; Wang, Ze Hui; Li, Dingxuan; Xiao, Yi: A Novel Heterocyclic Xanthene-Analogous pH Probe for ­Quantitative Monitoring of Cell Surface pH by Fluorescence ­Lifetime Imaging

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Issue 20/2023

Yu, Shengyu; Liu, Jiahao; Wang, Zhe; Kato, Terumasa; Liu, Yan; Maruoka, Keiji: Design of Y-Shaped Trimers of Chiral Phase-Transfer Catalysts for the Asymmetric Alkylation of Amino Acid Derivatives

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Han, Jung Tae; Zhou, Hui; List, Benjamin: Brønsted Acid Catalyzed Asymmetric Silylation of Biaryl Diols

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Sun, Haoyi; Guo, Yongcheng; Li, Huajie; Wang, Meiling; Ding, Tiandi; Zhi, Ying; Zhao, Kun; Yao, Qingqiang: Synthesis of (2-Nitro-1-AfAlemphenylethyl)malononitriles by Michael Addition of Masked Acyl Cyanides to Nitroalkenes

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Yamaoka, Seiha; Fukuoka, Hiroyuki; Noda, Naoki; Okano, Kentaro; Horie, Masaki; Mori, Atsunori: Nickel(II) Thiocyanate Complex as a Catalyst for Cross-Coupling Reactions

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Li, Zegong; Zeng, Zi; Tang, Qi; Zhong, Ziwei; Liu, Xiaohua; Feng, Xiaoming: Asymmetric Synthesis of 3-Lactone-Substituted 2-Oxindoles with Vicinal Quaternary Carbon Centers through Vinylogous Conjugate Addition

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Wei, Jia-Hui; Jin, You-Xiang; Wang, Pu-Sheng; Gong, Liu-Zhu: Access to Fluorinated Quaternary Stereogenic Centers via Palladium-Catalyzed Asymmetric Allylic C–H Alkylation

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Ding, Nan; Li, Zhi: Acid-Catalyzed [4+1]-Dearomatization Spiroannulation of Hydroquinones and Naphthols

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Hayashi, Yujiro; Han, Xiaolei; Mori, Naoki: Bis(2-ethylhexyl)amine as an Effective Organocatalyst for the Racemic Reactions of α,β-Unsaturated Aldehydes Involving an Iminium Ion

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Zeng, Yiqun; Fei, Chao; Zhou, Xiao; Luo, Jisheng; Deng, Li: Chiral Betaine-Mediated Efficient Organocatalytic Asymmetric Isomerization of β,γ-Unsaturated Butenolides

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Thorve, Pradip Ramdas; Maji, Biplab: Synthesis of Furo- and Thienoquinolines by Using an Amine Oxidase-Inspired Catalyst

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Naruse, Yuji; Takamori, Atsushi; Oda, Kenji; Kosugi, Takuya: Lone Pair Participation in a Decarboxylation Reaction: A New Design of a Boradecarboxylation Reaction

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Uwaso, Yuki; Yokoyama, Naoki; Kano, Taichi: Short Synthesis of a Biphenyl-Based Amino Triflamide Catalyst and Its Application in Enamine Catalysis

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Liu, Guo; Li, Pingfan: Enantioselective Bromination of Silyl Enol Ethers with Chiral Pentacarboxycyclopentadienyl Bromide

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Mizoguchi, Haruki; Yoshida, Ryuji; Ikeda, Haruka; Sakakura, Akira: Visible-Light-Photoexcited Palladium-Catalyzed Silylmethylation of Benzyl Alcohol Derivatives

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Hori, Tatsuaki; Kakinuma, Shuya; Ohtsuka, Naoya; Fujinami, Takeshi; Suzuki, Toshiyasu; Momiyama, Norie: Synthesis of Halogen-Bond-Donor-Site-Introduced Functional Monomers through Wittig Reaction of Perfluorohalogenated Benzaldehydes: Toward Digitalization as Reliable Strategy in Small-Molecule Synthesis

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Xu, Changgong; Nader, Phillip; Xavier, Jonathan; Takenaka, Norito: Asymmetric Allenylation of N-Acylhydrazones with Propargyltrichlorosilane Catalyzed by Helical Chiral 2,2′-Bipyridine N-Monoxide

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Mondal, Swati Lekha; Patra, Koushik; Yadav, Rahul; Baidya, Mahiuddin: Organocatalyzed Regioselective α,γ-Difunctionalization of Deconjugated Butenolides: Synthesis of Butyrolactone–Butyrolactam Hybrid Molecules

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Yao, Hongqing; Wang, Chuan: Yttrium-Catalyzed Regioselective Aminolysis of 2,3-Epoxy Esters and Amides

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Nakahara, Yuki; Hirokawa, Ryo; Uchida, Shotaro; Yamashita, Kenji; Hamashima, Yoshitaka: Switching Regioselectivity in the Asymmetric Bromocyclization of Difluoroalkenes Catalyzed by a Chiral Bisphosphine Oxide

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Rahaman, Ajijur; Bhadra, Sukalyan: Copper-Catalyzed Construction of Amide Linkages via Coupling between Unactivated Acids and Amines

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Ano, Yusuke; Takahashi, Daichi; Yo, Kazumune; Nagamune, Ryosuke; Chatani, Naoto: Palladium-Catalyzed Ring Opening of Cyclobutanones with Carbon- and Heteroatom-Centered Nucleophiles

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Sawano, Takahiro; Yasumura, Yuki; Kuwabara, Kyohei; Sugiura, Hikaru; Takahashi, Kana; Ishikawa, Eri; Takeuchi, Ryo: Iridium-Catalyzed Asymmetric Allylation of Indoles via Kinetic Resolution of 1-Alken-4-yn-3-ols

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Pawar, Tushar Janardan; Valtierra-Galvan, Marco F.; Rodríguez-Hernández, Alfredo; Reyes-Luna, Alfonso; Bonilla-Landa, Israel; García-Barradas, Oscar; Barrera-Méndez, Felipe; Olivares-Romero, José L.: Synthesis of Novel C₂ Bishydroxamic Acid Ligands and their Application in Asymmetric Epoxidation Reactions

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Chen, Minghao; Watanabe, Takumi; Habaue, Shigeki: Smart Hydrogel Reactor of Poly(N-isopropylacrylamide)/Polyethylene Glycol Interpenetrating Polymer Networks for Oxidative Coupling of 2-Naphthol

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Hatano, Manabu; Nishioka, Chiaki; Mimura, Ayaka; Kimura, Risa; Okuda, Yuki; Yamada, Takeshi; Sakata, Ken: 2,2′-Biphenol-Derived Phosphoric Acid Catalyst for the Dehydrative Esterification of Carboxylic Acids with Alcohols

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Yanagisawa, Akira; Hinata, Yuki; Midorikawa, Koji; Watanabe, Takamichi: Asymmetric α-Cyanation of β-Keto Esters Catalyzed by Chiral Tin Alkoxides

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Sakai, Kazuho; Yagi, Yusuke; Nomura, Nobuyoshi: Stereoselective Ring-Opening Deacetonation Polymerization of Racemic 2,2,5-Trimethyl-1,3-dioxolan-4-one by Using Homosalen–Aluminum Complexes: A Novel Approach to Isotactic ­Poly(rac-lactic acid)

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Nohara, Shoya; Iwai, Suguru; Yamaguchi, Naoya; Asada, Yosuke; Kamiyama, Yusuke; Tanaka, Yuta; Tanaka, Kenta; Hoshino, Yujiro: Visible-Light-Induced Oxidative Generation of o-Quinone Methides for Inverse-Electron-Demand [4+2] Cycloaddition Reactions

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Issue 18/2023

Morken, James P.; Aggarwal, Varinder: Cluster Preface: Modern Boron Chemistry: 60 Years of the ­Matteson Reaction

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Bastick, Kane A. C.; Watson, Allan J. B.: Pd-Catalyzed Homologation of Arylboronic Acids as a Platform for the Diversity-Oriented Synthesis of Benzylic C–X Bonds

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Priester, Ronja; Kazmaier, Uli: A Straightforward Synthesis of Emericellamide A Using Matteson’s Homologation Approach

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Jung, Yongsuk; Cho, Seung Hwan: Chemo-, Regio-, and Stereoselective Access to (E)-Boryl-Substituted Allyl Fluorides via Electrophilic Fluorodesilylation

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Lee, Hyelee; Alvarado, Marisol; Ingram, Sarah; Li, Bo; Liu, Shih-Yuan: N-Functionalization of 1,2-Azaborines

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Rourke, Michael J.; McGill, Matthew J.; Yang, Daniel; Farnam, Emelia J.; Zhu, Joshua L.; Scheidt, Karl A.: Photoredox-Catalyzed Radical–Radical Coupling of Potassium Trifluoroborates with Acyl Azoliums

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Kuznetsov, Dmitry M.; Ready, Joseph M.: Asymmetric Catalytic Hydroboration of Enol Carbamates Enables an Enantioselective Matteson Homologation

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Sakuraba, Mahiro; Morishita, Taichi; Hashimoto, Taiki; Ogoshi, Sensuke; Hoshimoto, Yoichi: Remote Back Strain: A Strategy for Modulating the Reactivity of Triarylboranes

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Akram, Manjur O.; Vogels, Christopher M.; Santos, Webster L.; Westcott, Stephen A.; Martin, Caleb D.: Addition of a Phosphinoboronate Ester to Borole and Borafluorene

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Trammel, Grace L.; Kerlin, Abby C.; Zachau, Christian; Brown, M. Kevin: Synthesis of (±)-Phyltetralin by Cu/Pd-Catalyzed Arylboration

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Cao, Yang; Blakemore, Paul R.: Enantiocontrolled Connective Synthesis of Allenes by Carbenoid Eliminative Cross-Coupling between α-(Methylthio)vinylcuprate Species and α-(Carbamoyloxy)alkylboronates

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Nishino, Soshi; Nishii, Yuji; Hirano, Koji: Preparation and Use of (γ,γ-Dioxyallyl)boronates

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Sun, Kai; Huang, Chung-Yang Dennis; Sawamura, Masaya; Shimizu, Yohei: Direct α-Trifluoromethylthiolation of Carboxylic Acids Enabled by Boron Catalysis

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Rygus, Jason P. G.; Boateng, Daniel B.; Hall, Dennis G.: Hemiboronic Acid-Catalyzed Reduction of α,β-Unsaturated Ketones with Reagent-Controlled Chemoselectivity

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Jiang, Wang; Bai, Jingyi; Lv, Jiahang; Zhao, Yue; Yan, Chaoguo; Shi, Zhuangzhi: Metal-Free Directed C–H Borylation of Indoles at the Sterically Congested C2 Position

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Semba, Kazuhiko; Nagase, Kotaro; Nakao, Yoshiaki: Conjugate Addition of Organoboron Compounds to α,β-Unsaturated Ketones Catalyzed by Nickelacycles

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Vedani, Luca; Gnägi-Lux, Manuel; Dénès, Fabrice; Renaud, Philippe: Intramolecular Asymmetric Cyclopropanation Using Air-Stable Alkylboronic Esters

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Trofimova, Alina; Brien, Chelsey; Trinchera, Piera; Tien, Chieh-Hung; Yudin, Andrei K.: Boryl Acrylaldehyde: An Elusive Member of the α-Boryl Aldehyde Class of Reagent

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Xu, Jianeng; Qin, Yucheng; Liu, Chao: Direct Amination of Benzylic Pinacol Boronates by an Aminoazanium

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Issue 13/2023

Zhang, Dong-Yang; Gong, Liu-Zhu: Enantioselective Oxidative Dearomatization of 2-Naphthols ­Enabled by Chiral Organoiodine Catalysis

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Dentmon, Zackery W.; Butch, Christopher J.; Gold, Hannah B.; Liotta, Dennis C.: Synthesis and Antiviral Evaluation of 2′,3′-β-C-Disubstituted Nucleoside Analogue ProTides to Test a Conformational Model of Potency Against Hepatitis C

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Issue 12/2023

Martin, Ruben: Cluster Preface: Special Issue Honoring Masahiro Murakami’s Contributions to Science

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Shigeno, Masanori; Tohara, Itsuki; Nozawa-Kumada, Kanako; Kondo, Yoshinori: 1,5-Double-Carboxylation of 2-Alkylheteroarenes Mediated by a Combined Brønsted Base System

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Zhumagazy, Serik; Zhu, Chen; Yue, Huifeng; Rueping, Magnus: Nickel-Сatalyzed Carbon–Selenium Bond Formations under Mild Conditions

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Qu, Quan; Chen, Lin; Deng, Yu; Gui, Yong-Yuan; Yu, Da-Gang: Visible-Light Photocatalytic Barbier-Type Reaction of Aziridines and Azetidines with Nonactivated Aldehydes

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Yamanomoto, Ken; Matsudaira, Tadachika; Akiyama, Takahiko: Metal- and Additive-Free Synthesis of α-Hydroxyamino Ketones Enabled by Organophotocatalyst

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Zhang, Quan; Ma, Dawei: Ligand-Promoted Rosenmund–von Braun Reaction

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Yu, Xuewen; Wan, Saihong; Zhou, Wang: 1,4-Reduction of α,β-Unsaturated Ketones through Rhodium(III)-Catalyzed Transfer Hydrogenation

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Han, Feng; Xie, Yuanhao; Xie, Xiulan; Ivlev, Sergei I.; Meggers, Eric: Chiral-at-Ru Catalyst with Cyclometalated Imidazo[1,5-a]pyridin­ylidene for Enantioselective Intramolecular Cyclopropanations

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González, Sara; Fernández, Elena: Alkenylboronic Ester Activation to Nucleophilic Addition and Electrophilic Trapping with Carbonyl Groups

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Lotuzas, Aleksandras; El Khoury, Anton; Li, Liubo; Harran, Patrick G.: Synthesis and Reactivity of a Stable Prototropic Isomer of 2-Acetyl-3-methylpyrrole

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Isshiki, Ryota; Kubota, Koji; Ito, Hajime: Solid-State Silver-Catalyzed Ring-Opening Fluorination of Cyclobutanols by Using Mechanochemistry

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Morita, Nobuyoshi; Chiaki, Hitomi; Tanaka, Kosaku; Hashimoto, Yoshimitsu; Tamura, Osamu; Krause, Norbert: Sustainable Chemical Synthesis of 2,3-Dihydrobenzofurans/1,2,3-Trisubstituted Indanes in Water by Using a Permethylated β-Cyclodextrin-Tagged N-Heterocyclic Carbene–Gold Catalyst

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Kai, Nobushige; Kono, Hideya; Yagi, Akiko; Itami, Kenichiro: Synthesis and Properties of Methylene-Bridged [6]Cyclo-2,6-naphthylene

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Kim, Minseok; Lee, Kangjae; Kim, Seonyul; Hong, Sungwoo: Photoinduced Carboarylation of Alkenes by Using Bifunctional Reagents

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Zhou, Qiansujia; Yin, Si-Yong; Zheng, Dong-Song; Zhang, Wen-Wen; Zhang, Su-Zhen; Gu, Qing; You, Shu-Li: Enantioselective Synthesis of Axially Chiral 1-Arylisoquinolines by Iridium(I)-Catalyzed Hydroarylation of Alkynes

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Um, Hyun-Suk; Shin, Woong Sik; Son, Kyu Jin; Lee, Chulbom: Synthesis of 2-Sulfonylthiazoles via Heteroaryl C–H Sulfonylation of Thiazole N-Oxides

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Corneliussen, Nicklas P.; Grove, Ebbe K.; Schøler, Anne-Sofie O.; Andersen, Anton H.; Donslund, Aske S.; Neumann, Karoline T.; Skrydstrup, Troels: Nickel-Catalyzed Carbonylative Coupling of Alkylzinc Reagents and α-Bromo-α,α-difluoroacetamides

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Han, Shuxiong; He, Shuo; Huang, Zhibin; Zhao, Yingsheng; Chen, Gong: Facile Synthesis of Isoindolinones via Radical-Mediated Intramolecular Coupling of Two C–H Bonds

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Papucci, Costanza; Ventura, Francesco; Franchi, Daniele; Dessi, Alessio; Pucci, Andrea; Reginato, Gianna; Mordini, Alessandro; Calamante, Massimo; Zani, Lorenzo: A Direct Arylation Approach for the Preparation of Benzothiadiazole-Based Fluorophores for Application in Luminescent Solar ­Concentrators

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Wiethoff, Maxim-Aleksa; Abdellaoui, Mehdi; Deis, Thomas; Corcé, Vincent; Lemière, Gilles; Ollivier, Cyril; Fensterbank, Louis: Martin Silicates as Versatile Radical Precursors in Photoredox/ Nickel Dual Catalysis

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Viudes, Olivier; Guarnieri-Ibáñez, Alejandro; Besnard, Céline; Lacour, Jérôme: Regiodivergent Synthesis of Oxadiazocines via Dirhodium-Catalyzed Reactivity of Oxazolidines and α-Imino Carbenes

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Nguyen, Jennifer A.; Cabanero, David C.; Rovis, Tomislav: Electrochemically Controlled Ruthenium-Catalyzed Olefin ­Metathesis

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Kashihara, Myuto; Kosaka, Kohei; Matsushita, Naoki; Notsu, Shunta; Osawa, Ayumi; Nakao, Yoshiaki: Catalytic Generation of Radicals from Nitroalkanes

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Su, Siyuan; Lee, Daesung: Synthesis of N-Acyl Pyrroles and Isoindoles from Oxime Ester Precursors via Transition-Metal-Catalyzed Iminocarboxylation

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Hayashi, Minoru; Fujimoto, Shion; Ohta, Hidetoshi: Fused λ⁵-Phosphinines: Design, Syntheses, and Properties

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Sun, Minghe; Wei, Linsheng; Li, Changkun: Rhodium-Catalyzed N-Reverse Prenylation of Nonactivated Indoles

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Ono, Shunya; Sugiyama, Aya; Sakamoto, Nao; Kuwabara, Kazuma; Minoura, Mao; Murai, Toshiaki: Two-Step Substitution Reaction of Phosphonates Carrying a Binaphthyl Group with Grignard Reagents Leading to the Formation of P-Chirogenic Phosphine Oxides

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Ouyang, Wenbai; Huo, Jingfeng; Wang, Jianbo: Rh(II)-Catalyzed Ring Expansion of Cyclopropyl N-Tosylhydrazones to 1-Substituted Cyclobutenes

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Heikinheimo, Annakaisa; Nieger, Martin; Koskinen, Ari M. P.: Diastereoselective Synthesis of Substituted Chromenopyrrolidinones from Amino Acid Derived Nitriles

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Peters, Bram B. C.; Birke, Norman; Massaro, Luca; Andersson, Pher G.: Enantioselective Synthesis of α-Chiral Amides by Catalytic Hydrogenation with Iridium N,P-Complexes

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Gunawan, Nina; Nutt, Michael J.; Bissember, Alex C.; Smith, Jason A.; Stewart, Scott G.: N-Tosyl-1,2,3-triazoles as Scaffolds for Morpholines: The Total Synthesis of (–)-Chelonin A

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Chen, Yuhao; Lan, Ping; White, Lorenzo V.; Yang, Weiguang; Banwell, Martin G.: Total Syntheses of Dysidealactams E and F and Dysidealactone B, Drimane-Type Sesquiterpenes Derived from a Dysidea sp. of Marine Sponge

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Zhang, Cheng; Liu, Jianzhong; Cheng, Zengrui; Li, Junhua; Song, Song; Jiao, Ning: Aminotetrazole Synthesis from Secondary Amides by C–C Bond Nitrogenation

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Issue 10/2023

Kondage, Savini Suduweli; Roemmele, Tracey L.; Boeré, René T.: Dispersion in Crystal Structures of 1-Chloro-3-aryl-5-trihalomethyl-1λ⁴,2,4,6-thiatriazines: Towards an Understanding of the Supramolecular Organization of Covalent Thiazyl Chlorides

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Holtrop, Flip; Helling, Christoph; Lutz, Martin; van Leest, Nicolaas P.; de Bruin, Bas; Slootweg, J. Chris: Enhancement of London Dispersion in Frustrated Lewis Pairs: Towards a Crystalline Encounter Complex

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Rummel, Lars; Hanke, Kai; Becker, Jonathan; Schreiner, Peter R.: London Dispersion Stabilizes Chloro-Substituted cis-Double Bonds

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Gorges, Johannes; Bädorf, Benedikt; Grimme, Stefan; Hansen, Andreas: Efficient Computation of the Interaction Energies of Very Large Non-covalently Bound Complexes

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Shimajiri, Takuya; Kawakami, Yuta; Kawaguchi, Soki; Hayashi, Yuki; Hada, Kazuto; Suzuki, Takanori; Ishigaki, Yusuke: Ultralong C(sp³)–C(sp³) Single Bonds Shortened and Stabilized by London Dispersion

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Schatz, Dominic; Kunz, Anne; Raab, Aileen R.; Wegner, Hermann A.: Investigation of Alkyl–Aryl Interactions Using the Azobenzene Switch – The Influence of the Electronic Nature of Aromatic London Dispersion Donors

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Verevkin, Sergey P.; Samarov, Artemiy A.; Zherikova, Kseniya V.: Noncovalent Interactions in Crowded Benzene Systems: How Much Strain Is Too Much? Attractions Overcome Repulsions!

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Loir-Mongazon, Lucas; Antuña-Hörlein, Carmen; Deraedt, Christophe; Cornaton, Yann; Djukic, Jean-Pierre: Activation Barriers for Cobalt(IV)-Centered Reductive Elimination Correlate with Quantified Interatomic Noncovalent Interactions

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Zhai, Jianyu; Reid, Jolene P.: Reaction Mechanisms for Chiral-Phosphate-Catalyzed Transformations Involving Cationic Intermediates and Protic Nucleophiles

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Issue 09/2023

Cao, Lujing; Wu, Yejian; Zhuang, Yixin; Xiong, Linan; Zhan, Zhajun; Ma, Liefeng; Duan, Hongliang: A Novel Application of a Generation Model in Foreseeing ‘Future’ Reactions

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Issue 07/2023

Pavithra, Thangavel; Karthiyayini, Gnanaoli; Nagarajan, Subbiah; Sridharan, Vellaisamy; Maheswari, C. Uma: Metal- and Solvent-Free Synthesis of m-Terphenyls by an Iodine-Catalyzed Tandem Formal [3+3]-Cycloaddition/Oxidation

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Kalita, Gitumoni; Khatua, Snehadrinarayan; Chatterjee, Paresh Nath: A Brønsted Acid Catalyzed Easy Access to Conjugated Diene-­Diones from Tertiary Propargyl Alcohols and 1,3-Dicarbonyl ­Compounds

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Ahmad, Sarwat Asma Ziya; Khan, Faiz Ahmed: Boron Trifluoride Etherate-Controlled Reactions of Methyl Enol Ethers: Selective Synthesis of Dihydrofuro[3,2-c]chromenone and Furo[3,2-c]chromenone Derivatives

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Mouli, M. S. S. Vinod; Katyal, Sahil; Mishra, Ashutosh Kumar: Design and Synthesis of a Flavin–Samarium Complex as an Efficient Photocatalyst for Sulfoxidation Reactions

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Ghosh, Sayan; Dutta, Jhilik; Halder, Atreyee; De Sarkar, Suman: Easy Access to N-(Pyridin-2-yl)benzamides through Electro-oxidative Ring Opening of 2-Arylimidazo[1,2-a]pyridines

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Kotha, Sambasivarao; Agrawal, Arpit: Synthesis of Linear Tetraquinanes by [3+2] Cycloaddition, Chemoselective Allylation of 7-Ketonorbornene, and Ring-Rearrangement Metathesis as Key Steps

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Kotha, Sambasivarao; Mehta, Gulazarahind: Strain-Induced Regioselective Ring-Opening Cross-Metathesis of Hybrid Cage Propellane Containing both Bicyclo[2.2.1]heptene and Bicyclo[2.2.2]octene Units

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Kotha, Sambasivarao; Jena, Kunkumita: Ring-Rearrangement Metathetic Approach to Fused 6/5/6/5/6-Oxacyclic Ring System and Bipentalene Derivatives

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Dinesh, Votarikari; Nagarajan, Rajagopal: Photochemical Decarboxylative Formylation of Indoles with Aqueous Glyoxylic Acid

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Yadav, Abhinay; Majumder, Satyajit; Das, Mrinal Kanti; Mondal, Ayan; Bisai, Alakesh: Asymmetric Total Syntheses of (–)-Dihydromaritidine and (–)-Oxomaritidine

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Ray, Sayan; Mukherjee, Santanu: Catalytic Enantioselective Desymmetrization of meso-Cyclopropane-Fused Cyclohexene-1,4-diones by a Formal C(sp²)–H Alkylation

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Ramachandran, Kuppan; Anbarasan, Pazhamalai: Chelation-Assisted Rhodium-Catalyzed Alkylation of a 1-Arylpyrazole C–H Bond with Cyclopropanols

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Issue 06/2023

Maiti, Debabrata; Mukherjee, Santanu: Cluster Preface: Chemical Synthesis and Catalysis in India

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Biswas, Nandita; Sharma, Rahul; Sardar, Bitan; Srimani, Dipankar: Acridine-Based SNS–Ruthenium Pincer Complex-Catalyzed Borrowing Hydrogen-Mediated C–C Alkylation Reaction: Application to the Guerbet Reaction

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Mahato, Rina; Khan, Jabir; Tyagi, Aparna; Hazra, Chinmoy Kumar: Lewis Acid Promoted Homodimerization of Styrene Diols: An Efficient Approach toward 2-Phenylnaphthalenes

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Chakraborty, Gargi; Pal, Subhasree; Chakraborty, Subhajit; Paul, Nanda D.: Nickel-Catalyzed Sustainable and Selective Alkylation of Alcohols to α-Alkylated Ketones via Borrowing Hydrogen Approach

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Akhtar, Sk Md Samim; Hajra, Saumen: Catalytic Enantioselective Synthesis of 4-Amino-5-aryltetrahydro-1H-benzo[c]azepines by an Aminoarylation Reaction

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Bhattacharyya, Dipanjan; Senapati, Siddhartha Kumar; Das, Animesh: Concise Synthesis of N-Aryl Tetrahydroquinolines via a One-Pot Sequential Reduction of Quinoline/Chan–Evans–Lam Coupling ­Reaction

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Mukherji, Ananya; Kancharla, Pavan K.: Cl^–···H–N Interaction Assisted Addition of Sulfonamides to Enol Ethers: Synthesis of 2-Deoxy and 2,6-Dideoxy Sulfonamido Glycosides

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Bania, Nimisha; Barman, Dipankar; Pan, Subhas Chandra: Organocatalytic Asymmetric Oxa-Michael–Michael Reaction of 3-Aryl-2-Nitroprop-2-Enols with Unsaturated Pyrazolones: Synthesis of Spirotetrahydropyranopyrazolones

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Saha, Suman K.; Jain, Anshul; Kumari, Akanksha; Bhutia, Tshering Sangmo; Agrawat, Chanchal; Rana, Nirmal K.: Use of Polymer-Supported 4-(N,N-Dimethylamino)pyridine in a Formal Conjugate Addition/Elimination Mediated by an N-Ylide Generated In Situ for the Construction of Highly Functionalized Itaconimides/Alkenes

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Mandal, Gour Hari; Saha, Dhiman; Auddy, Sourya Shankar; Goswami, Rajib Kumar: Synthesis of the Key Skeleton of Phosphoeleganin

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Padma Priya, V. R.; Irfana Jesin, C. P.; Nandi, Ganesh Chandra: Transition-Metal-Free N-(o-Halo)arylation of Sulfoximines/Sulfonimidamides

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Issue 05/2023

Gong, Guanfei; Xie, Fei; Wang, Lu; Wang, Jike; Chen, Shigui: Construction and Characterization of a Diphase Two-Dimensional Halogen-Bonded Organic Framework Based on a Pyrene Derivative

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Xu, Zeyu; Su, Shuaisong; Li, Xue; Jia, Tiezheng: A Facile and Mild Alkylation Protocol of NH-Diphenyl Sulfondiimines

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Murphy, Grace K.; Richards, Corey A.; Applegate, Seth A.; Neely, Jamie M.: Two-Step, One-Pot Pyrrole Synthesis by Iron-Catalyzed ­Carboamination/Copper-Mediated Cyclization

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Meyrelles, Ricardo; Fetisleam, Yener; Maryasin, Boris: Computational Investigation of the Aza-Cope Rearrangement Leading to Angularly Substituted 1-Azabicyclic Rings

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Akkarasamiyo, Sunisa; Sakonnakhon, Hatairat Promsaka Na; Kuntiyong, Punlop; Ploypradith, Poonsakdi; Samec, Joseph S. M.: Concise Synthesis of 1,4-Dideoxy-1,4-imino-l-arabinitol (LAB) from d-Xylose by Intramolecular Stereospecific Substitution of a Hydroxy Group

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Stubbs, James M.; Nanuwa, Amrit S.; Hoffman, Matthew D.; Blacquiere, Johanna M.: Catalyst Comparison for Additive-Free Acceptorless Dehydro­genation of Indoline Derivatives

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Miao, Han-Zhe; Liu, Yang; Chen, Ye-Wei; Lu, Han-Yu; Li, Jian; Lin, Guo-Qiang; He, Zhi-Tao: Stereoselective Pd-Catalyzed Remote Hydroamination of Skipped Dienes with Azoles

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Shi, Anzai; Xiang, Panjie; Wu, Yanxuan; Ge, Chang; Liu, Yan; Sun, Kai; Yu, Bing: Visible-Light-Promoted Metal-Free 3-Arylation of 2-Aryl-2H-­indazoles with Triarylsulfonium Salts

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Singh, Bandana; Bera, Tishyasoumya; Singh, Vinod P.; Priyasha, Priyasha; Das, Dinabandhu; Saha, Jaideep: Construction of Spiropyrroloindolines by Dearomative [3+2]-Cycloaddition of Indoles with Oxindole-Embedded Azaoxyallyl ­Cations

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Wang, Peng; Li, Shao-Jie; Zhang, Honghai; Yang, Na; Liao, Saihu: Photo-organocatalytic Synthesis of β-Keto Sulfonyl Fluorides via Radical Fluorosulfonylation of Vinyl Acetates

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Full, Felix; Wildervanck, Martijn J.; Volland, Daniel; Nowak-Król, Agnieszka: Synthesis of Enantioenriched Azaborole Helicenes by Chirality Transfer from Axially Chiral Biaryls

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Li, XinXin; Yang, Qingxing; Zhang, Yuna; Xu, Tao: Rhodium(III) Iodide Catalyzed Carboamination of Alkynes through C–N Bond Activation

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Issue 02/2023

Xu, Shitang; Yi, Rongnan; Zeng, Chunling; Cui, Yue; Wang, Xue-Qiang; Xu, Xinhua; Li, Ningbo: CsOH-Promoted Regiospecific Sulfenylation, Selenylation, and Telluration of Indoles in H₂O

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Issue 20/2022

Lange, Manuel; Sennert, Elisabeth; Suhm, Martin A.: London Dispersion-Assisted Low-Temperature Gas Phase Synthesis of Hydrogen Bond-Inserted Complexes

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Issue 18/2022

Zhang, Zhipeng; Zhao, Baoguo: Cluster Preface: Development and Applications of Novel Ligands/Catalysts and Mechanistic Studies on Catalysis

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Takeshima, Aika; Kano, Taichi: The Design and Synthesis of Phenylcyclopropane-Based Secondary Amine Catalysts and Their Applications in Asymmetric Reactions

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Yan, Yao-Hong; Li, Long; Ye, Long-Wu: Claisen Rearrangement Triggered by Brønsted Acid Catalyzed Alkyne Alkoxylation

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Dong, Jia-Wei; Cao, Ren-Fei; Chen, Zhi-Min: Catalytic Enantioselective Dihalogenation of Alkenes

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Pan, Shulei; Zhu, Qiongqiong; Zhang, Yanghui: Palladium-Catalyzed Coupling of Biphenyl-2-yl Trifluoromethanesulfonates with Dibromomethane to Access Fluorenes

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Hayashi, Yujiro; Hatano, Yutaro; Mori, Naoki: Asymmetric Michael Reaction of Malononitrile and α,β-Unsaturated Aldehydes Catalyzed by Diarylprolinol Silyl Ether

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Dong, Zhan; Zhong, Dayou; Li, Zi-Meng; Liu, Wei-Min; Zhao, Jing; Liu, Wen-Bo: Palladium-Catalyzed Stereospecific Coupling of BINOL-bistriflates and Zinc Cyanide and Applications in the Synthesis of 1,1′-Binaphthyl-2,2′-bisoxazolines (BOXAX)

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Brennan, Therese B.; Müller-Bunz, Helge; Guiry, Patrick J.: The Synthesis of Novel P,N-Ferrocenylpyrrolidine-Containing Ligands and Their Application in Pd-Catalyzed Allylic Alkylation – A Synthetic and Mechanistic Investigation

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Luan, Baixue; Tang, Zaiquan; Wu, Xianqing; Chen, Yifeng: 8-Quinolinyl Oxazoline: Ligand Exploration in Enantioselective Ni-Catalyzed Reductive Carbamoyl-Alkylation of Alkene to Access the Chiral Oxindoles

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Kondoh, Azusa; Yamaguchi, Sho; Watanabe, Yushi; Terada, Masahiro: Brønsted Base Catalyzed Conjugate Addition of β-Acylvinyl Anion Equivalents to α,β-Unsaturated Ketones

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Wang, Chengyi; Deng, Shaomin; Chen, Rui; Liu, Guohua; Cheng, Tanyu; Liu, Rui: Mechanochemical Asymmetric Transfer Hydrogenation of Diketones to Access Chiral 1,3-Diols under Solvent-Free Conditions

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Li, Bing; Li, Changkun: Rhodium-Catalyzed Regio- and Enantioselective Direct Allylation of Methyl Ketones

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Tang, Jingjing; Li, Jian; Yang, Xueyan; Zhang, Zhipeng: Synthesis of Novel Chiral Phenanthroline Ligands and a Copper Complex

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Issue 14/2022

Wacharasindhu, Sumrit: Cluster Preface: Organic Chemistry in Thailand

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Songthammawat, Poramate; Phumjan, Tanawat; Ruchirawat, Somsak; Ploypradith, Poonsakdi: 4b-Aryltetrahydroindeno[1,2-a]indenes by Acid-Catalyzed Trans­annular Cyclization of Benzannulated Cyclooctene Alcohols

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Meesin, Jatuporn; Chotsaeng, Nawasit; Kuhakarn, Chutima: Dimerization of 3-Chlorooxindoles Mediated by Potassium Ethyl­xanthate: Synthesis of Isoindigos

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Phae-nok, Supasorn; Kuhakarn, Chutima; Leowanawat, Pawaret; Reutrakul, Vichai; Soorukram, Darunee: Decarboxylation of Paraconic Acids by a Silver(I) Nitrate/Persulfate Combination: An Entry to β-Nitro- and β-Hydroxy γ-Butyrolactones

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Ruengsangtongkul, Sureeporn; Kuribara, Takahito; Chaisan, Nattawadee; Tummatorn, Jumreang; Thongsornkleeb, Charnsak; Ruchirawat, Somsak: Ceric Ammonium Nitrate Promoted Oxidative Coupling of Terminal Alkynes and 1,3-Keto Esters: A Synthesis of Unsymmetrical 1,1,2-Triacylalkenes

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Pham, Quynh Nguyen Nhu; Silpcharu, Komthep; Vchirawongkwin, Viwat; Sukwattanasinitt, Mongkol; Rashatasakhon, Paitoon: 2,3-Diaryl-1,1,4,4-tetracyanobutadienes as Colorimetric Sensors for Sulfide Ion in Aqueous Media

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Thiraporn, Aticha; Iawsipo, Panata; Tadpetch, Kwanruthai: Total Synthesis and Cytotoxic Activity of 7-O-Methylnigrosporolide and Pestalotioprolide D

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Soonthonhut, Siraporn; Acharasatian, Peera: Ionic Liquid Driven Nucleophilic Substitution of Squaric Acid to Squaramides

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Akkarasamiyo, Sunisa; Chitsomkhuan, Saranya; Buakaew, Supawadee; Samec, Joseph S. M.; Chuawong, Pitak; Kuntiyong, Punlop: Synthesis of (Z)-Cinnamate Esters by Nickel-Catalyzed Stereoinvertive Deoxygenation of trans-3-Arylglycidates

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Khanthong, Adisorn; Khamphaijun, Korawit; Ruengsuk, Araya; Docker, Andrew; Limpanuparb, Taweetham; Tantirungrotechai, Jonggol; Bunchuay, Thanthapatra: Pillar[4]arene[1]thioarenes: Synthesis and Host–Guest Binding Properties

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Yimyaem, Jirapat; Chantana, Chayamon; Boonmee, Suthimon; Jaratjaroonphong, Jaray: Expedient Access to Indolyl-Substituted Tri- and Diarylmethanes and (±)-Colletotryptin E by Silica Sulfuric Acid Catalyzed Transindolylation

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Saebang, Yotsakorn; Kaeobamrung, Juthanat; Rukachaisirikul, Vatcharin: Synthesis of Eleven-Membered Cyclic Urea Fused Quinazolinones

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Kuntiyong, Punlop; Inprung, Nantachai; Attanonchai, Sineenart; Kheakwanwong, Wichita; Bunrod, Pijitra; Akkarasamiyo, Sunisa: Diastereoselective Synthesis of Tetrahydrofurano[2,3-g]indolizidines and 8-Aminoindolizidines from l-Asparagine

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Rinkam, Suttida; Senapak, Warapong; Watchasit, Sarayut; Saeeng, Rungnapha; Sirion, Uthaiwan: Brønsted Acidic Ionic Liquid Catalyzed Three-Component Friedel–Crafts Reaction for the Synthesis of Unsymmetrical Triarylmethanes

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Chooppawa, Tianchai; Janprasert, Penpicha; Padungros, Panuwat: One-Pot Synthesis of Glycosyl Chlorides from Thioglycosides Mediated by a Bromodiethylsulfonium Salt as a Mild Oxidant

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Saejong, Peerawat; Somprasong, Siriphong; Rujirasereesakul, Chaiwat; Luanphaisarnnont, Torsak: Direct Synthesis of Coumarin Derivatives from Alkynoic Esters via Dual Organocatalysis

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Mansawat, Woraluk; Yukhet, Phanomsak; Bhanthumnavin, Worawan; Reiser, Oliver; Vilaivan, Tirayut: Kinetic Resolution of dl-Hydrobenzoins Catalyzed by Copper(II) Complexes of C₂-Symmetric Thiophene-Derived Ligands

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La-ongthong, Kannika; Sawekteeratana, Natthapat; Klaysuk, Jasarin; Soorukram, Darunee; Leowanawat, Pawaret; Reutrakul, Vichai; Krobthong, Sucheewin; Wongtrakoongate, Patompon; Kuhakarn, Chutima: Cyclization of o-Alkynylisocyanobenzenes with 1,3-Dicarbonyl Compounds

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Chatsirisupachai, Jirat; Sudyoadsuk, Taweesak; Namuangrak, Supawadee; Promarak, Vinich: Chrysene-Cored Fluorescent Dendrimers as Nondoped Deep-Blue Emitters for Solution-Processable Electroluminescent Devices

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Chaisan, Nattawadee; Ruengsangtongkul, Sureeporn; Thongsornkleeb, Charnsak; Tummatorn, Jumreang; Ruchirawat, Somsak: Dihalooxygenation of Alkynes and Alkynols: Preparation of 2,2-Dihaloketones and gem-Dihalolactols

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Worayuthakarn, Rattana; Suddee, Nattanit; Nealmongkol, Prattya; Ruchirawat, Somsak; Thasana, Nopporn: Copper-Mediated C–O/C–N Bond Formation: A Facile Synthesis of 3-Amidocoumarin, 3-Amidoazacoumarin, and N-Aroylindole ­Derivatives

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Dolsophon, Kulvadee; Soponpong, Jakapun; Kornsakulkarn, Jittra; Thongpanchang, Chawanee; Thongpanchang, Tienthong: Methods for Determination of Absolute Configurations of Chiral Diols by THENA Ester and NMR Shift Difference

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Kraikruan, Panitan; Rakchaya, Intouch; Sang-aroon, Pattarapon; Chuanopparat, Nutthawat; Ngernmeesri, Paiboon: One-Pot Synthesis of 2-Arylindole Derivatives under Transition-Metal-Free Conditions

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Chumkaeo, Peerapong; Poonsawat, Thinnaphat; Yunita, Isti; Temnuch, Natcha; Meechai, Titiya; Kumpan, Nuttapong; Khamthip, Achjana; Chuaitammakit, Laksamee Chaicharoenwimolkul; Chairam, Sanoe; Somsook, Ekasith: Accelerated Decomposition of Potassium Permanganate in Ferrocenium Ion as Ferrocenium-Doped Manganese(IV) Oxide for Selective Oxidation of Alcohols

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Ajavakom, Vachiraporn; Pandokrak, Potchanee; Salim, Sofia S.; Moustafa, Gamal A. I.; Bellingham, Richard K.; Hill-Cousins, Joseph T.; Ajavakom, Anawat; Brown, Richard C. D.: Formation of Seven-Membered Rings by Ring-Closing Metathesis of Vinyl Bromides

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Yamano, Dolnapa; Wiriya, Nittaya; Phakhodee, Wong; Wet-osot, Sirawit; Pattarawarapan, Mookda: Mechanochemical Synthesis of 2,5-Disubstituted 1,3,4-Oxadiazoles Mediated by PPh₃-TCCA

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Lamor, Anphisa; Uipanit, Suwanan; Yakhampom, Sujitra; Ngernmeesri, Paiboon; Kongkathip, Ngampong; Kongkathip, Boonsong; Chuanopparat, Nutthawat: Asymmetric Formal Synthesis of (–)-Swainsonine from Chiral-Pool Precursors d-Mannose and d-Arabinose

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Wiriya, Nittaya; Yamano, Dolnapa; Hongsibsong, Surat; Pattarawarapan, Mookda; Phakhodee, Wong: Direct Synthesis of N-Monosubstituted Benzimidazol-2-ones via Ph₃P–I₂-Mediated Reaction of Hydroxamic Acids

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Issue 13/2022

Tyagarajan, Sriram; Guiadeen, Deodial; Streckfuss, Eric; Gao, Xiaolei; Buevich, Alexei V.; Doss, George; Liu, Jian; Vachal, Petr; Krska, Shane W.: Late-Stage Functionalization for the Optimization of Reversible BTK Inhibitors

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Issue 12/2022

Nicewicz, David: Cluster Preface: Organic Photoredox Catalysis in Synthesis – Honoring Professor Shunichi Fukuzumi’s 70th Birthday

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Kamada, Kenji; Okuwa, Hiroko; Wakabayashi, Taku; Sekizawa, Keita; Sato, Shunsuke; Morikawa, Takeshi; Jung, Jieun; Saito, Susumu: A Highly Durable, Self-Photosensitized Mononuclear Ruthenium Catalyst for CO₂ Reduction

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Jeong, Dong Yeun; You, Youngmin: Organic Photoredox Catalysts Exhibiting Long Excited-State Lifetimes

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Wu, Yanyu; Kim, Dooyoung; Teets, Thomas S.: Photophysical Properties and Redox Potentials of Photosensitizers for Organic Photoredox Transformations

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Hutskalova, Valeriia; Sparr, Christof: The Versatility of the Aryne–Imine–Aryne Coupling for the ­Synthesis of Acridinium Photocatalysts

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Hyodo, Yuki; Takahashi, Keigo; Chitose, Youhei; Abe, Manabu; Yoshizawa, Michito; Koike, Takashi; Akita, Munetaka: Assemblies of 1,4-Bis(diarylamino)naphthalenes and Aromatic Amphiphiles: Highly Reducing Photoredox Catalysis in Water

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He, Min; Yang, Shilei; Yu, Xiaoqiang; Bao, Ming: 7,10-Dibromo-2,3-dicyanopyrazinophenanthrene Aggregates as a Photosensitizer for Nickel-Catalyzed Aryl Esterification

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Stull, Savannah M.; Mei, Liangyong; Gianetti, Thomas L.: Red-Light-Induced N,N′-Dipropyl-1,13-dimethoxyquinacridinium-Catalyzed [3+2] Cycloaddition of Cyclopropylamines with Alkenes or Alkynes

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Weick, Fabian; Steuernagel, Desirée; Belov, Arina; Wagenknecht, Hans-Achim: Complementary Photocatalytic Toolbox: Control of Intramolecular endo- versus exo-trig Cyclizations of α-Phenyl Olefins to Oxaheterocyclic Products

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Nicholls, Bryce T.; Qiao, Tianzhang; Hyster, Todd K.: A Photoenzyme for Challenging Lactam Radical Cyclizations

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Issue 09/2022

Jung, Sangmin; Yoon, Hyo Jae: Heterocyclic Mechanophores in Polymer Mechanochemistry

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Baumann, Christoph; Göstl, Robert: Triazole-Extended Anthracenes as Optical Force Probes

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Li, Qing; Wang, Qi; Yuan, Yuan; Chen, Yulan: Mechanochemiluminescent Hydrogels for Real-Time Visualization of Chemical Bond Scission

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Wang, Zi; Kouznetsova, Tatiana B.; Craig, Stephen L.: Pulling Outward but Reacting Inward: Mechanically Induced Symmetry-Allowed Reactions of cis- and trans-Diester-Substituted Dichlorocyclopropanes

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Wu, Lik Chun; De Bo, Guillaume: Stereoelectronic Effects in Force-Accelerated Retro-Diels–Alder Reactions

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van Bonn, Pit; Bolm, Carsten: Mechanochemical Synthesis of Diarylethynes from Aryl Iodides and CaC₂

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Kubota, Koji; Kondo, Keisuke; Seo, Tamae; Ito, Hajime: Insight into the Reactivity Profile of Solid-State Aryl Bromides in Suzuki–Miyaura Cross-Coupling Reactions Using Ball Milling

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Issue 05/2022

Fischer, Christian; Vepřek, Nynke A.; Peitsinis, Zisis; Rühmann, Klaus-Peter; Yang, Chao; Spradlin, Jessica N.; Dovala, Dustin; Nomura, Daniel K.; Zhang, Yingkai; Trauner, Dirk: De novo Design of SARS-CoV-2 Main Protease Inhibitors

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Hung, Kevin; Liu, Yugang; Simon, Oliver; Zhang, Lei; Lu, Peichao; Yeung, Bryan K. S.; Sarko, Christopher; Yokokawa, Fumiaki: Synthesis of a Potent Pan-Serotype Dengue Virus Inhibitor Having a Tetrahydrothienopyridine Core

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Issue 04/2022

Kang, Qi-Kai; Shi, Hang: Catalytic Hydrogen Isotope Exchange Reactions in Late-Stage Functionalization

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Rogge, Torben; Müller, Thomas; Simon, Hendrik; Hou, Xiaoyan; Wagschal, Simon; Broggini, Diego; Ackermann, Lutz: Triazole-Enabled Ruthenium(II) Carboxylate-Catalyzed C–H Arylation with Electron-Deficient Aryl Halides

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Luo, Huanhuan; Wang, Dawei; Wang, Minyan; Shi, Zhuangzhi: Rhodium-Catalyzed, Phosphorus(III)-Directed Hydroarylation of Internal Alkynes: Facile and Efficient Access to New Phosphine Ligands

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Santiago, Carlos; Chen, Hao; Mondal, Arup; van Gemmeren, Manuel: Dual Ligand-Enabled Late-Stage Fujiwara–Moritani Reactions

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Issue 01/2022

Padilla, Robin; Vollhardt, K. Peter C.; Houk, Kendall N.; Wong, Jonathan J.: Bis(η⁵-cyclopentadienyl)[μ-(4b,5,5a-η³:9b,10,10a-η³)-2,3,7,8-tetrakis(trimethylsilyl)benzo[3,4]cyclobuta[1,2-b]biphenylene]-syn-dicobalt (Co–Co), a Dinuclear π-Complex of the Linear [3]Phenylene Framework

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Höfler, Denis; List, Benjamin: A Chiral, Dendralenic C–H Acid

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Suzuka, Toshimasa; Niimi, Ryoko; Uozumi, Yasuhiro: Cyanide-Free Cyanation of Aryl Iodides with Nitromethane by Using an Amphiphilic Polymer-Supported Palladium Catalyst

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Höfler, Denis; Kaupmees, Karl; Leito, Ivo; List, Benjamin: A Chiral Sulfoxide-Based C–H Acid

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Roth, Hudson G.; Nicewicz, David A.: Diastereoselective Synthesis of the ABCD Ring System of Rubriflordilactone B

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Sau, Miriam; Pericàs, Miquel A.; Martin, Ruben: Pd-Catalyzed Arylation of 1,2-Amino Alcohol Derivatives via β-Carbon Elimination

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Issue 18/2021

Zankov, D.; Polishchuk, P.; Madzhidov, T.; Varnek, A.: Multi-Instance Learning Approach to Predictive Modeling of Catalysts Enantioselectivity

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Xu, Li-Cheng; Li, Xin; Tang, Miao-Jiong; Yuan, Luo-Tian; Zheng, Jia-Yu; Zhang, Shuo-Qing; Hong, Xin: A Molecular Stereostructure Descriptor Based On Spherical Projection

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Yada, Akira; Matsumura, Tarojiro; Ando, Yasunobu; Nagata, Kenji; Ichinoseki, Sakina; Sato, Kazuhiko: Ensemble Learning Approach with LASSO for Predicting Catalytic Reaction Rates

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Issue 16/2021

Ishida, Naoki; Kamino, Yuka; Murakami, Masahiro: Nickel-Catalyzed α-1,3-Dienylation of 1,3-Dicarbonyl Compounds with Propargylic Carbonates

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Ye, Yang; Ma, Guobin; Yao, Ken; Gong, Hegui: Zn-Mediated Hydrodeoxygenation of Tertiary Alkyl Oxalates

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Kathe, Prasad M.; Berkefeld, Andreas; Fleischer, Ivana: Nickel Hydride Catalyzed Cleavage of Allyl Ethers Induced by Isomerization

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Higginson, Bradley; Sanjosé-Orduna, Jesus; Gu, Yiting; Martin, Ruben: Nickel-Catalyzed Photodehalogenation of Aryl Bromides

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Shuai, Bin; Fang, Ping; Mei, Tian-Sheng: Nickel-Catalyzed Favorskii-Type Rearrangement of Cyclobutanone Oxime Esters to Cyclopropanecarbonitriles

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Liu, Shengzhang; Yang, Lingyun; Tao, Jiasi; Yu, Weijie; Wang, Tao; Fu, Junkai: Nickel-Catalyzed Oxidative Transamidation of Tertiary Aromatic Amines with N-Acylsaccharins

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Xue, Yuhang; Chen, Jian; Song, Peihong; He, Yuli; Zhu, Shaolin: Nickel-Catalyzed Regiodivergent Reductive Hydroarylation of Styrenes

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Zhang, Pengpeng; Cantrell, Rachel L.; Newhouse, Timothy R.: Role of Benzylic Deprotonation in Nickel-Catalyzed Benzylic Dehydrogenation

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Li, Yuqiang; Yin, Guoyin: Bathocuproine-Enabled Nickel-Catalyzed Selective Ullmann Cross-Coupling of Two sp²-Hybridized Organohalides

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Xiao, Jian; Wang, Ya-Wen; Qiu, Zhong-Ping; Peng, Yu: Ni-Catalyzed Intramolecular Reductive 1,2-Dicarbofunctionalization of Alkene: Facile Access to Podophyllum Lignans Core

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Lundrigan, Travis; Tassone, Joseph P.; Stradiotto, Mark: Nickel-Catalyzed N-Arylation of Amides with (Hetero)aryl Electrophiles by Using a DBU/NaTFA Dual-Base System

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Wei, Shichao; Mao, Yongjun; Shi, Shi-Liang: Nickel-Catalyzed Ligand-Free Hiyama Coupling of Aryl Bromides and Vinyltrimethoxysilane

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Issue 15/2021

Martin, Ruben; Molander, Gary A.: Cluster Preface: Modern Nickel-Catalyzed Reactions

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Diao, Haiyan; Shi, Zhangjie; Liu, Feng: Biaryl Construction Based on Nickel-Catalyzed C–O Bond Activation

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Abdellaoui, Mehdi; Millanvois, Alexandre; Levernier, Etienne; Ollivier, Cyril; Fensterbank, Louis: Visible-Light-Mediated Z-Stereoselective Monoalkylation of β,β-Dichlorostyrenes by Photoredox/Nickel Dual Catalysis

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Feng, Xiaoliang; Guo, Lei; Zhu, Shengqing; Chu, Lingling: Borates as a Traceless Activation Group for Intermolecular Alkylarylation of Ethylene through Photoredox/Nickel Dual Catalysis

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Lucas, Erika L.; McGinnis, Tristan M.; Castro, Anthony J.; Jarvo, Elizabeth R.: Nickel-Catalyzed Cross-Electrophile Coupling of the Difluoromethyl Group for Fluorinated Cyclopropane Synthesis

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Kerackian, Taline; Reina, Antonio; Krachko, Tetiana; Boddaert, Hugo; Bouyssi, Didier; Monteiro, Nuno; Amgoune, Abderrahmane: C(sp³)–H Bond Acylation with N-Acyl Imides under Photoredox/ Nickel Dual Catalysis

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Ashida, Keita; Hoshimoto, Yoichi; Ogoshi, Sensuke: Ni(0)-Catalyzed Synthesis of Polycyclic α,β-Unsaturated γ-Lactams via Intramolecular Carbonylative Cycloaddition of Yne-imines with CO

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Minami, Hiroko; Nogi, Keisuke; Yorimitsu, Hideki: Nickel-Catalyzed Negishi-Type Arylation of Trialkylsulfonium Salts

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Lin, Zhiyang; Lan, Yun; Wang, Chuan: Ligand-Free Nickel-Catalyzed Reductive Allylic Defluorinative Cross-Coupling of α-Trifluoromethyl Alkenes with Epoxides

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Luo, Ying; Chan, Bun; Fukuda, Tsutomu; Onodera, Gen; Kimura, Masanari: Nickel-Catalyzed Carboxylation of Conjugated Dienes with Carbon Dioxide and DIBAL-H for the Synthesis of β,γ-Unsaturated Carboxylic Acids

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Iizumi, Keiichiro; Kurosawa, Miki B.; Isshiki, Ryota; Muto, Kei; Yamaguchi, Junichiro: Decarbonylative Synthesis of Aryl Nitriles from Aromatic Esters and Organocyanides by a Nickel Catalyst

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Chen, Qiang; Fu, Liyan; You, Jingwen; Nishihara, Yasushi: Nickel-Catalyzed Decarbonylative Alkynylation of Acyl Fluorides with Terminal Alkynes under Copper-Free Conditions

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Zhao, Qing-Wei; Yang, Zhi-Fang; Fu, Xia-Ping; Zhang, Xingang: Access to α,α-Difluoro-γ-amino Acids by Nickel-Catalyzed Reductive Aryldifluoroacetylation of N-Vinylacetamide

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Kim, Nana; Tran, Van T.; Apolinar, Omar; Wisniewski, Steven R.; Eastgate, Martin D.; Engle, Keary M.: Ni(COD)(DMFU): A Heteroleptic 16-Electron Precatalyst for 1,2-Diarylation of Alkenes

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Issue 13/2021

Jiang, Xuefeng: Cluster Preface: Perspectives on Organoheteroatom and Organometallic Chemistry

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Wong, Jonathan; Yeung, Ying-Yeung: Recent Advances in C–Br Bond Formation

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Lou, Qin-Xin; Li, Jing-Yu; Yang, Shang-Dong: Iridium(III)-Catalyzed C−H Functionalization of Triarylphosphine Oxides with Diazo Dicarbonyl Compounds: Synthesis of α-Aryl 1,3-Dicarbonyl Derivatives

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Issue 05/2021

Lang, Yatao; Li, Chao-Jun; Zeng, Huiying: Dearomatization–Rearomatization Strategy for Palladium-Catalyzed C–N Cross-Coupling Reactions

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Brutiu, Bogdan R.; Klose, Immo; Maulide, Nuno: Facile C–S Bond Cleavage of Aryl Sulfoxides Promoted by Brønsted Acid

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Drießen, Daniel; Biesen, Lukas; Müller, Thomas J. J.: Sequentially Catalyzed Three-Component Masuda–Suzuki–Sonogashira Synthesis of Fluorescent 2-Alkynyl-4-(7-azaindol-3-yl)pyrimidines: Three Palladium-Catalyzed Processes in a One-Pot Fashion

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Li, Longbo; Schneider, Yanika; Hoeglund, Adrienne B.; Braslau, Rebecca: Advances in Internal Plasticization of PVC: Copper-Mediated Atom-Transfer Radical Polymerization from PVC Defect Sites To Form Acrylate Graft Copolymers

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Yasukawa, Tomohiro; Zhu, Zhiyuan; Yamashita, Yasuhiro; Kobayashi, Shu: Carbonylative Suzuki–Miyaura Coupling Reactions of Aryl Iodides with Readily Available Polymer-Immobilized Palladium Nanoparticles

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Xu-Xu, Qing-Feng; Yang, Pusu; Zhang, Xiao; You, Shu-Li: Enantioselective Synthesis of 4-Silyl-1,2,3,4-tetrahydroquinolines via Copper(I) Hydride Catalyzed Asymmetric Hydrosilylation of 1,2-Dihydroquinolines

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Gargaro, Samantha L.; Dunson, Bre'Shon; Sieber, Joshua D.: Identification of a Surprising Boronic Acid Homocoupling Process in Suzuki–Miyaura Cross-Coupling Reactions Utilizing a Hindered Fluorinated Arene

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Tosi, Eleonora; Spielmann, Kim; de Figueiredo, Renata Marcia; Campagne, Jean-Marc: Copper-Catalyzed Ring Expansion of Vinyl Aziridines under Mild Conditions

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Shin, Sang Ik; Nguyen, Nguyen H.; Im, Jangbin; Shin, Seunghoon: Zinc-Catalyzed Transacetalization of N,O-Acetals into N,N-Acetals with Benzotriazoles, Indazoles, and Azides

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Aubineau, Thomas; Dupas, Alexandre; Zeng, Tian; Cossy, Janine: Iron-Catalyzed Diastereoselective Synthesis of Disubstituted Morpholines via C–O or C–N Bond Formation

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Mino, Takashi; Yamaguchi, Daiki; Kumada, Manami; Youda, Junpei; Saito, Hironori; Tanaka, Junya; Yoshida, Yasushi; Sakamoto, Masami: Chiral P,Olefin Ligands with Rotamers for Palladium-Catalyzed Asymmetric Allylic Substitution Reactions

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Issue 04/2021

Zhu, Chen; Liu, Xin-Yuan: Cluster Preface: Radicals – by Young Chinese Organic Chemists

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Zhang, Zheng-Hua; Wei, He; Li, Zhong-Liang; Liu, Xin-Yuan: Recent Advances in Radical-Involved Alkynylation of Unactivated C(sp³)–H Bonds by Hydrogen Atom Abstraction

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Xu, Fan; Lai, Xiao-Li; Xu, Hai-Chao: C–H Alkylation of Heteroarenes with Alkyl Oxalates by Molecular Photoelectrocatalysis

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He, Bin-Qing; Gao, Yuan; Wang, Peng-Zi; Wu, Hong; Zhou, Hong-Bin; Liu, Xiao-Peng; Chen, Jia-Rong: Dual Photoredox/Palladium-Catalyzed C–H Acylation of 2-Arylpyridines with Oxime Esters

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Jiang, Yue-Ming; Liu, Jie; Fu, Qiang; Yu, Yu-Ming; Yu, Da-Gang: Visible-Light-Driven Phosphonoalkylation of Alkenes

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Zhuang, Bi-Yang; Jin, Ji-Kang; Zhang, Feng-Lian; Wang, Yi-Feng: Radical-Hydroboration-Involved One-Pot Synthesis of Boron-Handled Glycol Derivatives

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Li, Yantao; Xu, Wentao; Zhu, Chengjian; Xie, Jin: Direct Deoxygenative Intramolecular Acylation of Biarylcarboxylic Acids

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Zhao, Jia-Jia; Yu, Shouyun: Synthesis of Chiral Fluorides by Sequential Organocatalyzed Desymmetrization of Glutaric Anhydrides and Photoredox-Catalyzed Decarboxylic Fluorination

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Su, Min; Zhu, Nengbo; Chiou, Mong-Feng; Bao, Hongli: Synthesis of Amidine Derivatives by Intermolecular Radical ­Addition to Nitrile Groups of AIBN Derivatives

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Zhang, Huihui; Ji, Meishan; Wei, Youhao; Chen, Haodong; Wu, Xinxin; Zhu, Chen: Radical-Mediated Hetaryl Functionalization of Nonactivated Alkenes through Distal ipso-Migration of O- or S-Hetaryls

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Liu, Haiwang; Xue, Fei; Wang, Mu; Tang, Xinxin; Wu, Jie: Neutral-Eosin Y-Catalyzed Regioselective Hydroacylation of Aryl Alkenes under Visible-Light Irradiation

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Issue 02/2021

Liu, Saiwen; Deng, Guo-Jun; Huang, Huawen: Recent Advances in Sulfur-Containing Heterocycle Formation via Direct C–H Sulfuration with Elemental Sulfur

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Zhou, Fei-Yu; Jiao, Lei: Recent Developments in Transition-Metal-Free Functionalization and Derivatization Reactions of Pyridines

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Hadrys, Barbara W.; Phipps, Robert J.: Acid and Solvent Effects on the Regioselectivity of Minisci-Type Addition to Quinolines Using Amino Acid Derived Redox Active Esters

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Gallardo-Alfonzo, Salvador; Cortés-Garcia, Carlos Jesus; Mejía-Farfán, Itzel; López, Yliana; Mojica, Martha; Contreras-Celedón, Claudia; Chacón-García, Luis: A Two-Step Synthesis of a Novel 7,8-Dihydro-5,8-ethanoindolizine-6,9(5H)-dione

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Liu, Zhuqing; Hyde, Alan M.; Klapars, Artis; Chung, John Y. L.; Lam, Yu-hong; Yasuda, Nobuyoshi: Selective 1,4-Addition of Organolithiums to Maleate Monoesters with Application for a Short Efficient Route to Azaindanones

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Shevlin, Michael; Strotman, Neil A.; Anderson, Laura L.: Concise Synthesis of Furo[2,3-b]indolines via [3,3]-Sigmatropic Rearrangement of N-Alkenyloxyindoles

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Barber, Joyann S.; Kong, Dehuan; Li, Wei; McAlpine, Indrawan J.; Nair, Sajiv K.; Sakata, Sylvie K.; Sun, Nicole; Patman, Ryan L.: Rhodium(III)-Catalyzed C–H Activation: Annulation of Petrochemical Feedstocks for the Construction of Isoquinolone Scaffolds

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Qian, Hui; Sun, Jianwei: Synthesis of Coumarins via [4+2] Cyclization of Siloxy Alkynes and Salicylaldehydes

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Spurlin, Racheal M.; Harris, Amber L.; Pratt, Cameron J.; Jui, Nathan T.: Synthesis of Spirocyclic Piperidines by Radical Hydroarylation

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Boyle, Benjamin T.; Koniarczyk, J. Luke; McNally, Andrew: Facile Pyridine S_NAr Reactions via N-Phosphonium–Pyridinium Intermediates

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Issue 19/2020

Fuse, Shinichiro: Cluster Preface: Integrated Synthesis Using Continuous-Flow Technologies

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Harenberg, Johannes H.; Weidmann, Niels; Knochel, Paul: Continuous-Flow Reactions Mediated by Main Group Organometallics

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Monos, Timothy M.; Jaworski, Jonathan N.; Stephens, John C.; Jamison, Timothy F.: Continuous-Flow Synthesis of Tramadol from Cyclohexanone

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Amri, Nasser; Wirth, Thomas: Accelerating Electrochemical Synthesis through Automated Flow: Efficient Synthesis of Chalcogenophosphites

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Lee, Hyune-Jea; Torii, Daiki; Jeon, Yongju; Yoshida, Jun-ichi; Kim, Heejin: Integrated Synthesis Using Isothiocyanate-Substituted Aryllithiums by Flow Chemistry

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Iwata, Takayuki; Yoshinaga, Tatsuro; Shindo, Mitsuru: Flow Synthesis of Triptycene via Triple Cycloaddition of Ynolate to Benzyne

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Griffiths, Oliver M.; Ruggeri, Michele; Baxendale, Ian R.: Photochemical Flow Oximation of Alkanes

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Okano, Kentaro; Yamane, Yoshiki; Nagaki, Aiichiro; Mori, Atsunori: Trapping of Transient Thienyllithiums Generated by Deprotonation of 2,3- or 2,5-Dibromothiophene in a Flow Microreactor

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Iio, Takuya; Nagai, Kohei; Kozuka, Tomoki; Sammi, Akhtar Mst; Sato, Kohei; Narumi, Tetsuo; Mase, Nobuyuki: Fine-Bubble–Slug-Flow Hydrogenation of Multiple Bonds and Phenols

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Sagandira, Cloudius R.; Watts, Paul: Continuous-Flow Synthesis of (–)-Oseltamivir Phosphate (Tamiflu)

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Ota, Kazuki; Fukumoto, Shinya; Iwase, Taiki; Mizota, Isao; Shimizu, Makoto; Hachiya, Iwao: Umpolung Reactions of α-Tosyloximino Esters in a Flow System

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Jiang, Yiyuan; Ashikari, Yosuke; Guan, Kaiteng; Nagaki, Aiichiro: Accelerating Heat-Initiated Radical Reactions of Organic Halides with Tin Hydride Using Flow Microreactor Technologies

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Oltmanns, Mona; Kirschning, Andreas: Subsupercritical Water Generated by Inductive Heating Inside Flow Reactors Facilitates the Claisen Rearrangement

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Issue 06/2020

Burke, Anthony J.: Cluster Preface: Special Edition Dedicated to ISySyCat2019

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Elumalai, Vijayaragavan; Hansen, Jørn H.: A Green, Scalable, One-Minute Synthesis of Benzimidazoles

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Alves, Cláudia; Grosso, Carla; Barrulas, Pedro; Paixão, José A.; Cardoso, Ana L.; Burke, Anthony J.; Lemos, Américo; Pinho e Melo, Teresa M. V. D.: Asymmetric Neber Reaction in the Synthesis of Chiral 2-(Tetrazol-5-yl)-2H-Azirines

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Massé, Paul; Choppin, Sabine; Chiummiento, Lucia; Hanquet, Gilles; Colobert, Françoise: Unintended Formation of a 26-Membered Cycle in the Course of a Novel Approach to Myricanol, a Strained [7,0]-Metacyclophane

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Trofymchuk, Serhii A.; Kliukovskyi, Denys V.; Semenov, Sergey V.; Khairulin, Andrii R.; Shevchenko, Valerii O.; Bugera, Maksym Y.; Tarasenko, Karen V.; Volochnyuk, Dmitriy M.; Ryabukhin, Sergey V.: Semi-Industrial Fluorination of β-Keto Esters with SF₄: Safety vs Efficacy

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Zi, You; Lange, Markus; Schüler, Philipp; Krieck, Sven; Westerhausen, Matthias; Vilotijevic, Ivan: Synthesis of β-Lactams via Enantioselective Allylation of Anilines with Morita–Baylis–Hillman Carbonates

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Rahman, MD Taifur; Wharry, Scott; Smyth, Megan; Manyar, Haresh; Moody, Thomas S.: FAST Hydrogenations as a Continuous Platform for Green Aromatic Nitroreductions

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Qu, Bo; Samankumara, Lalith P.; Saha, Anjan; Schumer, Mac G.; Han, Zhengxu S.; Haddad, Nizar; Busacca, Carl A.; Yee, Nathan K.; Kozlowski, Marisa C.; Song, Jinghua J.; Senanayake, Chris H.: Rational Design of New Dihydrobenzooxophosphole-Based Lewis Base Organocatalysts

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Di Mauro, Giovanni; Drescher, Martina; Tkaczyk, Sara; Maulide, Nuno: Aminoxylation of Thioalkynes through Radical-Polar Crossover

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Xu, Di; Frank, Lena; Nguyen, Tina; Stumpf, Andreas; Russell, David; Angelaud, Remy; Gosselin, Francis: Magnesium-Catalyzed N2-Regioselective Alkylation of 3-Substituted Pyrazoles

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Salgado, Mateo M.; Manchado, Alejandro; Nieto, Carlos T.; Díez, David; Garrido, Narciso M.: Asymmetric Synthesis of 2,3,6-Trisubstituted Piperidines via Baylis–Hillman Adducts and Lithium Amide through Domino Reaction

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Sebest, Filip; Haselgrove, Samuel; White, Andrew J. P.; Díez-González, Silvia: Metal-Free 1,2,3-Triazole Synthesis in Deep Eutectic Solvents

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Roux, Amélie; Cisnetti, Federico: Click Variations on the Synthesis of 2-Nitrophenyl-4-aryl-1,2,3-triazoles without Isolation of 2-Nitrophenyl Azides

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Carreiro, Elisabete P.; Sena, Ana M.; Puerta, Adrián; Padrón, José M.; Burke, Anthony J.: Synthesis of Novel 1,2,3-Triazole-Dihydropyrimidinone Hybrids Using Multicomponent 1,3-Dipolar Cycloaddition (Click)–Biginelli Reactions: Anticancer Activity

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Capretz-Agy, André; Fernandes, Fábio S.; Rodrigues, Manoel T.; Conti, Caroline; Coelho, Fernando: Aza-Morita–Baylis–Hillman Reaction with Vinyl-oxadiazoles: An Expeditious Approach to Access New Heterocyclic Arrangements

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Reeves, Ryan D.; Kinkema, Caitlin N.; Landwehr, Eleanor M.; Vine, Logan E.; Schomaker, Jennifer M.: Stereodivergent Metal-Catalyzed Allene Cycloisomerizations

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Ferreira, Joana R. M.; Nunes da Silva, Raquel; Rocha, João; Silva, Artur M. S.; Guieu, Samuel: 1,2,4-Triphenylpyrroles: Synthesis, Structure and Luminescence Properties

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Issue 03/2020

Hyster, Todd K.: Cluster Preface: Biocatalysis

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Steck, Viktoria; Sreenilayam, Gopeekrishnan; Fasan, Rudi: Selective Functionalization of Aliphatic Amines via Myoglobin-Catalyzed Carbene N–H Insertion

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Doyon, Tyler J.; Narayan, Alison R. H.: Synthetic Utility of One-Pot Chemoenzymatic Reaction Sequences

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Kudalkar, Gaurav P.; Tiwari, Virendra K.; Lee, Joshua D.; Berkowitz, David B.: A Hammett Study of Clostridium acetobutylicum Alcohol Dehydrogenase (CaADH): An Enzyme with Remarkable Substrate Promiscuity and Utility for Organic Synthesis

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Issue 02/2020

Osako, Takao; Srisa, Jakkrit; Torii, Kaoru; Hamasaka, Go; Uozumi, Yasuhiro: Iterative Preparation of Platinum Nanoparticles in an Amphiphilic Polymer Matrix: Regulation of Catalytic Activity in Hydrogenation

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Yanagi, Tomoyuki; Nogi, Keisuke; Yorimitsu, Hideki: Sulfoxide-Directed Iterative Assembly into Oligoarenes

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Issue 17/2019

Cluster Cover Page

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Morandi, Bill: Cluster Preface: Metathesis Reactions beyond Olefins

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Lambert, Tristan H.: Development of a Hydrazine-Catalyzed Carbonyl-Olefin Metathesis Reaction

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Oss, Giulia; Nguyen, Thanh Vinh: Iodonium-Catalyzed Carbonyl–Olefin Metathesis Reactions

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Pemba, Alexander G.; Miller, Stephen A.: Acetal Metathesis: Mechanistic Insight

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Naraoka, Asuka; Naka, Hiroshi: Transfer Hydration of Dinitriles to Dicarboxamides

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Patrzałek, Michał; Piątkowski, Jakub; Kajetanowicz, Anna; Grela, Karol: Anion Metathesis in Facile Preparation of Olefin Metathesis Catalysts Bearing a Quaternary Ammonium Chloride Tag

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Bothe, Michael; Orrillo, A. Gastón; Furlan, Ricardo L. E.; von Delius, Max: Trithioorthoester Exchange and Metathesis: New Tools for Dynamic Covalent Chemistry

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Masuya, Yoshihiro; Kawashima, Yuki; Kodama, Takuya; Chatani, Naoto; Tobisu, Mamoru: Thiolate-Initiated Synthesis of Dibenzothiophenes from 2,2′-Bis(methylthio)-1,1′-Biaryl Derivatives through Cleavage of Two Carbon–Sulfur Bonds

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Issue 14/2019

Yeung, Ying-Yeung: Cluster Preface: Organosulfur and Organoselenium Compounds in Catalysis

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Cluster Cover Page

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Dinh, Andrew N.; Nguyen, Ashley D.; Aceves, Ernesto Millan; Albright, Samuel T.; Cedano, Mario R.; Smith, Diane K.; Gustafson, Jeffrey L.: Photocatalytic Oxidative C–H Thiolation: Synthesis of Benzothiazoles and Sulfenylated Indoles

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Robb, Kevin A.; Athavale, Soumitra V.; Denmark, Scott E.: Unusual Kinetic Profiles for Lewis Base-Catalyzed Sulfenocyclization of ortho-Geranylphenols in Hexafluoroisopropyl Alcohol

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Tsuchihashi, Ayano; Shirakawa, Seiji: Catalyst-Controlled Regio- and Stereoselective Bromolactonization with Chiral Bifunctional Sulfides

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Jana, Sadhan; Verma, Ajay; Rathore, Vandana; Kumar, Sangit: Synthesis of Novel C₂-Symmetric Sulfur-Based Catalysts: Asymmetric Formation of Halo- and Seleno-Functionalized Normal- and Medium-Sized Rings

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Wonner, P.; Steinke, T.; Huber, S. M.: Activation of Quinolines by Cationic Chalcogen Bond Donors

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Otsuka, Yuta; Shimazaki, Yuto; Nagaoka, Hitoshi; Maruoka, Keiji; Hashimoto, Takuya: Scalable Synthesis of a Chiral Selenium π-Acid Catalyst and Its Use in Enantioselective Iminolactonization of β,γ-Unsaturated Amides

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Cao, Hongen; Chen, Tian; Yang, Chenggen; Ye, Jianqing; Zhang, Xu: Diphenyl Diselenide Catalyzed Oxidative Degradation of Benzoin to Benzoic Acid

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Li, Huimin; Liao, Lihao; Zhao, Xiaodan: Organoselenium-Catalyzed Aza-Wacker Reactions: Efficient Access to Isoquinolinium Imides and an Isoquinoline N-Oxide

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Chen, Diao; Liu, Jian-Guo; Zhang, Xu; Xu, Ming-Hua: Rhodium-Catalyzed Asymmetric Addition of Arylboronic Acids to Glyoxylates: Access to Optically Active Substituted Mandelic Acid Esters

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Liu, Yonghong; Ling, Hai; Chen, Chao; Xu, Qing; Yu, Lei; Jiang, Xuefeng: Sodium Selenosulfate from Sodium Sulfite and Selenium Powder: An Odorless Selenylating Reagent for Alkyl Halides to Produce Dialkyl Diselenide Catalysts

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Gao, Ge; Han, Jie; Yu, Lei; Xu, Qing: Organoselenium-Catalyzed Polymerization of Aniline with Hydrogen Peroxide as Oxidant

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Issue 10/2019

Cluster Cover Page

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Kawamata, Yu; Baran, Phil S.: Cluster Preface: Electrochemical Synthesis and Catalysis

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Song, Chunlan; Liu, Kun; Dong, Xin; Chiang, Chien-Wei; Lei, Aiwen: Recent Advances in Electrochemical Oxidative Cross-Coupling for the Construction of C–S Bonds

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Qiu, Youai; Struwe, Julia; Ackermann, Lutz: Metallaelectro-Catalyzed C–H Activation by Weak Coordination

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Lips, Sebastian; Franke, Robert; Waldvogel, Siegfried R.: Electrochemical Synthesis of 2-Hydroxy-para-terphenyls by Dehydrogenative Anodic C–C Cross-Coupling Reaction

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Takahira, Yusuke; Chen, Miao; Kawamata, Yu; Mykhailiuk, Pavel; Nakamura, Hugh; Peters, Byron K.; Reisberg, Solomon H.; Li, Chao; Chen, Longrui; Hoshikawa, Tamaki; Shibuguchi, Tomoyuki; Baran, Phil S.: Electrochemical C(sp³)–H Fluorination

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Amri, Nasser; Skilton, Ryan A.; Guthrie, Duncan; Wirth, Thomas: Efficient Flow Electrochemical Alkoxylation of Pyrrolidine-1-carbaldehyde

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Klunder, Kevin J.; Cass, Ashley C.; Anderson, Scott L.; Minteer, Shelley D.: Phthalocyanines as a π–π Adsorption Strategy to Immobilize Catalyst on Carbon for Electrochemical Synthesis

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Tanaka, Kenta; Yoshizawa, Hirona; Atobe, Mahito: A Flow Microreactor Approach to a Highly Efficient Diels–Alder Reaction with an Electrogenerated o-Quinone

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Lu, Lingxiang; Fu, Niankai; Lin, Song: Three-Component Chlorophosphinoylation of Alkenes via Anodically Coupled Electrolysis

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Yamamoto, Kosuke; Ishimaru, Keiko; Mizuta, Satoshi; Minato, Daishirou; Kuriyama, Masami; Onomura, Osamu: Diastereodivergent Synthesis of Bromoiminolactones: Electrochemical and Chemical Bromoiminolactonization of α-Allylmalonamides

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Mitsudo, Koichi; Yoshioka, Kazuki; Hirata, Takayuki; Mandai, Hiroki; Midorikawa, Koji; Suga, Seiji: 1,10-Phenanthroline- or Electron-Promoted Cyanation of Aryl Iodides

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Pandolfi, Fabiana; Chiarotto, Isabella; Mattiello, Leonardo; Rocco, Daniele; Feroci, Marta: Cathodic Reduction of Caffeine: Synthesis of an Amino-Functionalized Imidazole from a Biobased Reagent

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Xu, P.; Xu, H.-C.: Electrochemical Deoxygenation of N-Heteroaromatic N-Oxides

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Issue 20/2018

Ayalew, Hailemichael; Wang, Tian-lin; Wang, Tsai-Hui; Hsu, Hsiu-Fu; Yu, Hsiao-hua: Direct C–H Arylation Polymerization to form Anionic Water-Soluble Poly(3,4-ethylenedioxythiophenes) with Higher Yields and Molecular Weights

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Issue 19/2018

Cluster Cover Page

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Swager, Timothy M.: Cluster Preface: Synthesis of Materials

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Messersmith, Reid E.; Siegler, Maxime A.; Tovar, John D.: A Heptacyclic Heptacycle: A Doubly Naphtho[b]thiophene Fused Borepin

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Torelli, M.; Domenichelli, I.; Pedrini, A.; Guagnini, F.; Pinalli, R.; Terenziani, F.; Artoni, F.; Brighenti, R.; Dalcanale, E.: pH-Driven Conformational Switching of Quinoxaline Cavitands in Polymer Matrices

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Yoshinaga, Kosuke; Swager, Timothy M.: Fluorofluorescent Perylene Bisimides

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Jones, Daniel R.; Vallee, Ryan; Levine, Mindy: Novel Fluorescent Fluorene-Containing Conjugated Polymers: Synthesis, Photophysical Properties, and Application for the Detection of Common Bisphenols

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Xu, Liguo; Yang, Kou; Hu, Rongrong; Tang, Ben Zhong: Multicomponent Polymerization of Alkynes, Sulfonyl Azide, and Iminophosphorane at Room Temperature for the Synthesis of Hyperbranched Poly(phosphorus amidine)s

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Stężycki, Rafał; Reger, David; Hoelzel, Helen; Jux, Norbert; Gryko, Daniel T.: Synthesis and Photophysical Properties of Hexaphenylbenzene–Pyrrolo[3,2-b]pyrroles

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Li, Kelvin; McNelles, Stuart A.; Adronov, Alex: Preparation and Properties of a Hydrolytically Stable Cyclooctyne-Containing Polymer

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Anderson, Trent E.; Culver, Evan W.; Almyahi, Furqan; Dastoor, Paul C.; Rasmussen, Seth C.: Poly(2,3-dihexylthieno[3,4-b]pyrazine-alt-2,3-dihexylquinoxaline): Processible, Low-Bandgap, Ambipolar-Acceptor Frameworks via Direct Arylation Polymerization

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Jin, Zexin; Teo, Yew Chin; Teat, Simon J.; Xia, Yan: Iterative Synthesis of Edge-Bent [3]Naphthylene

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Selmani, Serxho; Vanderzwet, Luke; Kukor, Andrew J.; Schipper, Derek J.: Synthesis of Poly(heteroarylenevinylene) Derivatives via Rhodium-Catalyzed Hydroarylation of Alkynes

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Sugiyasu, Kazunori; Inoue, Ryota; Shomura, Ryo; Matsushita, Yoshitaka; Takeuchi, Masayuki: Synthesis and Redox Behavior of a Sheathed Cross-Conjugated Polythiophene

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Frederickson, Conerd K.; Barker, Joshua E.; Dressler, Justin J.; Zhou, Zheng; Hanks, Evan R.; Bard, Jeremy P.; Zakharov, Lev N.; Petrukhina, Marina A.; Haley, Michael M.: Synthesis and Characterization of a Fluorescent Dianthraceno­indacene

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Bulumulla, Chandima; Gunawardhana, Ruwan; Gamage, Prabhath L.; Kularatne, Ruvanthi N.; Biewer, Michael C.; Stefan, Mihaela C.: π-Spacer-Linked Bisthienopyrroles with Tunable Optical Properties

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Kulkarni, Gajanan C.; Morales-Cruz, Jean L.; Hussain, Waseem A.; Garvey, Ian J.; Plunkett, Kyle N.: Electron Acceptors Based on Cyclopentannulated Tetracenes

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Nitti, Andrea; Osw, Peshawa; Abdullah, Media N.; Galbiati, Alessandro; Pasini, Dario: Scalable Synthesis of Naphthothiophene-based D-π-D Extended Oligomers through Cascade Direct Arylation Processes

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Harnoy, Assaf J.; Papo, Nitsan; Slor, Gadi; Amir, Roey J.: Mixing End Groups in Thiol-Ene/Yne Reactions as a Simple Approach toward Multienzyme-Responsive Polymeric Amphiphiles

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Issue 16/2018

Cluster Cover Page

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Siegel, Jay S.: Cluster Preface: Atropisomerism

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Siegel, Jay S.: Prologue: Atropisomerism

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Matsuoka, Mizuki; Iida, Asumi; Kitagawa, Osamu: α-Alkylation of N–C Axially Chiral Quinazolinone Derivatives Bearing Various ortho-Substituted Phenyl Groups: Relation between Diastereoselectivity and the ortho-Substituent

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Ni, Cailing; Wang, Meng; You, Lei: Dynamic Covalent Chemistry within Biphenyl Scaffolds: Effects from Endocyclic to Exocyclic Sulfonamides

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Toyota, Shinji; Saibara, Toyoaki; Fujise, Kei; Oki, Tomohiro; Iwanaga, Tetsuo: Synthesis and Conformational Analysis of 10-Mesitylanthracene-1,8-diyl Oligomers

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Tabata, Hidetsugu; Tsuji, Yuka; Yoneda, Tetsuya; Tasaka, Tomohiko; Oshitari, Tetsuta; Takahashi, Hideyo; Natsugari, Hideaki: Atropisomerism in the 2,3,4,5-Tetrahydro-1H-1,5-benzodiazepine Nucleus: Effects of Central Chirality at C3 on the N-Mesylation Reaction

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Ishigaki, Yusuke; Iwai, Tomohiro; Hayashi, Yuki; Nagaki, Aiichiro; Katoono, Ryo; Fujiwara, Kenshu; Yoshida, Jun-ichi; Suzuki, Takanori: Transmission of Point Chirality to Axial Chirality for Strong Circular Dichroism in Triarylmethylium-o,o-dimers

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Dinh, Andrew N.; Noorbehesht, Ryan R.; Toenjes, Sean T.; Jackson, Amy C.; Saputra, Mirza A.; Maddox, Sean M.; Gustafson, Jeffrey L.: Toward a Catalytic Atroposelective Synthesis of Diaryl Ethers Through C(sp²)–H Alkylation with Nitroalkanes

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Pagano, Angela; Marotta, Emanuela; Mazzanti, Andrea; Petrillo, Giovanni; Tavani, Cinzia; Mancinelli, Michele: Stereodynamic Analysis of New Atropisomeric 4,7-Di(naphthalen-1-yl)-5,6-dinitro-1H-indoles

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Nagata, Yuuya; Shimada, Yasuo; Nishikawa, Tsuyoshi; Takeda, Ryohei; Uno, Makoto; Ogoshi, Tomoki; Suginome, Michinori: A Planar-Chiral Pillar[5]arene-Based Monophosphine Ligand with Induced Chirality at the Biaryl Axis

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Mátravölgyi, Béla; Deák, Szilvia; Erdélyi, Zsuzsanna; Hergert, Tamás; Ábrányi-Balogh, Péter; Faigl, Ferenc: Effect of Regioisomerism on the Efficiency of 1-Phenylpyrrole-Type Atropisomeric Amino Alcohol Ligands in Enantioselective Organometallic Reactions

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Fischer, Christian; Sparr, Christof: Configurationally Stable Atropisomeric Acridinium Fluorophores

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Issue 06/2018

Cluster Cover Page

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Murakami, Masahiro: Cluster Preface: C–C Activation

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Kondo, Teruyuki; Taniguchi, Ryosuke; Kimura, Yu: Ruthenium- and Rhodium-Catalyzed Ring-Opening Coupling Reactions of Cyclopropenones with Alkenes or Alkynes

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Shima, Yusuke; Igarashi, Emiko; Yoshimura, Tomoyuki; Matsuo, Jun-ichi: Reactions of Nitrosobenzenes with Cyclobutanones by Activation with a Lewis Acid

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Kuwabara, Takuya; Takamori, Shuhei; Kishi, Satoshi; Watanabe, Takahiro; Ikeda, Yousuke; Kodama, Shintaro; Minami, Yasunori; Hiyama, Tamejiro; Ishii, Youichi: Activation of a Carbon–Carbon Bond in Internal Alkynes: Vinylidene Rearrangement of Disubstituted Alkynes at an Ir Complex

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Mao, Wenbin; Zhu, Chen: Rhodium-Catalyzed C–C Bond Olefination of Ring-Fused Benzocyclobutenols and Application in the Construction of Polycyclic Compounds

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Lee, Chang-Hee; Jun, Chul-Ho: Chelation-Assisted C–H and C–C Bond Activation of Allylic Alcohols by a Rh(I) Catalyst under Microwave Irradiation

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Mori, Yasuyuki; Shigeno, Chieko; Luo, Ying; Chan, Bun; Onodera, Gen; Kimura, Masanari: Ni-Catalyzed Formal Carbonyl-Ene Reaction of Terminal Alkenes via Carbon Dioxide Insertion

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Swartz, Brett D.; Brennessel, William W.; Jones, William D.: Lewis Acid Assisted C–CN Cleavage of Benzonitrile Using [(dippe)NiH]₂

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Matsuda, Takanori; Matsumoto, Takeshi; Murakami, Akira: Palladium-Catalyzed Ring-Opening Coupling of Cyclobutenols with Aryl Halides

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Feng, Shiyu; Chan, Kin Shing: Regioselective and Room-Temperature Carbon–Carbon Bond Activation of Cyclopropanes by Rhodium(II) Porphyrin

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Liu, Cheng-Hang; Yu, Zhi-Xiang: Rh(I)-Catalyzed Intramolecular [3+2] Cycloaddition of trans-2-Allene-Vinylcyclopropanes

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Issue 04/2018

Cluster Cover Page

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Johnston, Jeffrey N.; Rovis, Tomislav: Cluster Preface: Alkene Halofunctionalization

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Ortiz, Gerardo X.; Chansaenpak, Kantapat; Wang, Mengzhe; Ma, Xiaofen; Wang, Hui; Li, Zibo; Wang, Qiu: A Novel ¹⁸F-Labeling Method for the Synthesis of [¹⁸F]-Piperidine-Containing Ligands as Potential PET Radiotracers for σ Receptors

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Hokamp, Tobias; Storm, Alena Therese; Yusubov, Mekhman; Wirth, Thomas: Iodine Monoacetate for Efficient Oxyiodinations of Alkenes and Alkynes

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Ng, Wing Hin; Shing, Tony K. M.; Yeung, Ying-Yeung: Mild and Efficient Vicinal Dibromination of Olefins Mediated by Aqueous Ammonium Fluoride

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Suzuki, Satoru; Kamo, Tomohiro; Fukushi, Kazunobu; Tokunaga, Etsuko; Sumii, Yuji; Shibata, Norio: Intramolecular Aminotrifluoromethanesulfinyloxylation of ω-Aminoalkenes by CF₃SO₂Na/Pd(OAc)₂/PhI(OAc)₂/^tBuOCl/PivOH System

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Klosowski, Daniel W.; Martin, Stephen F.: Enantioselective Synthesis of F-Ring Fragments of Kibdelone C via Desymmetrizing Bromolactonization of 1,4-Dihydrobenzoic Acid

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Böse, Dietrich; Denmark, Scott E.: Investigating the Enantiodetermining Step of a Chiral Lewis Base Catalyzed Bromocycloetherification of Privileged Alkenes

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Issue 19/2017

Cluster Cover Page

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Tobisu, Mamoru; Chatani, Naoto; Snieckus, Victor: Cluster Preface: C–O And Related Bond Activation

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Yoshida, Yuto; Nogi, Keisuke; Yorimitsu, Hideki: C–S Bond Alkynylation of Diaryl Sulfoxides with Terminal Alkynes by Means of a Palladium–NHC Catalyst

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Yang, Ze-Kun; Wang, Chao; Uchiyama, Masanobu: DFT Studies Provide Mechanistic Insight into Nickel-Catalyzed Cross-Coupling Involving Organoaluminum-Mediated C–O Bond Cleavage

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Yasui, Kosuke; Higashino, Masaya; Chatani, Naoto; Tobisu, Mamoru: Rhodium-Catalyzed Reductive Cleavage of Aryl Carbamates Using Isopropanol as a Reductant

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Makida, Yusuke; Matsumoto, Yasutaka; Kuwano, Ryoichi: Palladium-Catalyzed Decarboxylation of Benzyl Fluorobenzoates

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Tang, Jinghua; Luo, Meiming; Zeng, Xiaoming: Chromium-Catalyzed, Regioselective Cross-Coupling of C–O Bonds by Using Organic Bromides as Reactants

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Gui, Yong-Yuan; Chen, Xiao-Wang; Zhou, Wen-Jun; Yu, Da-Gang: Arylation of Amide and Urea C(sp³)–H Bonds with Aryl Tosylates Generated In Situ from Phenols

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da Frota, Livia C. R. M.; Schneider, Cédric; de Amorim, Mauro B.; da Silva, Alcides J. M.; Snieckus, Victor: Chemoselective Ruthenium-Catalyzed C–O Bond Activation: Orthogonality of Nickel- and Palladium-Catalyzed Reactions for the Synthesis of Polyaryl Fluorenones

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Lee, Shao-Chi; Guo, Lin; Yue, Huifeng; Liao, Hsuan-Hung; Rueping, Magnus: Nickel-Catalyzed Decarbonylative Silylation, Borylation, and Amination of Arylamides via a Deamidative Reaction Pathway

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Isshiki, Ryota; Takise, Ryosuke; Itami, Kenichiro; Muto, Kei; Yamaguchi, Junichiro: Catalytic α-Arylation of Ketones with Heteroaromatic Esters

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Martin-Montero, R.; Krolikowski, T.; Zarate, C.; Manzano, R.; Martin, R.: Stereospecific Nickel-Catalyzed Borylation of Secondary Benzyl Pivalates

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Izumoto, Akiko; Kondo, Hikaru; Kochi, Takuya; Kakiuchi, Fumitoshi: Synthesis of Fluorine-Containing Tetraarylanthracenes via Ruthenium-Catalyzed C–O or C–F Arylation and their Crystal Structures

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Issue 18/2017

Cluster Cover Page

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Oestreich, Martin: Cluster Preface: Silicon in Synthesis and Catalysis

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Gandhamsetty, Narasimhulu; Park, Sehoon; Chang, Sukbok: Boron-Catalyzed Hydrogenative Reduction of Substituted Quinolines to Tetrahydroquinolines with Hydrosilanes

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Das, Manas; Manvar, Atul; Fox, Ian; Roberts, Dilwyn J.; O’Shea, Donal F.: Bu₄N⁺-Controlled Addition and Olefination with Ethyl 2-(Trimethylsilyl)acetate via Silicon Activation

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Minami, Yasunori; Komiyama, Takeshi; Shimizu, Kenta; Uno, Shu-ichi; Hiyama, Tamejiro; Goto, Osamu; Ikehira, Hideyuki: Nickel-Catalyzed N-Arylation Using N-Trimethylsilyl-carbazole

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Wübbolt, Simon; Oestreich, Martin: Exhaustive Chemoselective Reduction of Nitriles by Catalytic Hydrosilylation Involving Cooperative Si–H Bond Activation

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Denmark, Scott E.; Ambrosi, Andrea: Understanding Site Selectivity in the Palladium-Catalyzed Cross-Coupling of Allenylsilanolates

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Ren, Xiaoyu; Han, Caifang; Feng, Xiangqing; Du, Haifeng: A Borane-Catalyzed Metal-Free Hydrosilylation of Chromones and Flavones

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Lee, Yong Ho; Morandi, Bill: Ether Synthesis through Reductive Cross-Coupling of Ketones with Alcohols Using Me₂SiHCl as both Reductant and Lewis Acid

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Moyer, Brandon S.; Gagné, Michel R.: Taming Silylium Ions for Synthesis: N-Heterocycle Synthesis via Stereoselective C–C Bond Formation

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De, Chandra Kanta; Mitra, Raja; List, Benjamin: Design and Synthesis of Enantiopure Tetrakis(pentafluorophenyl) Borate Analogues for Asymmetric Counteranion Directed Catalysis

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Flinker, Mathias; Lopez, Sara; Nielsen, Dennis U.; Daasbjerg, Kim; Jensen, Frank; Skrydstrup, Troels: Experimental and Theoretical Studies on the Reduction of CO₂ to CO with Chloro(methyl)disilane Components from the Direct Process

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Igawa, Kazunobu; Kuroo, Akihiro; Yoshihiro, Daisuke; Yamanaka, Yuki; Tomooka, Katsuhiko: Synthesis of Stereoselectively Functionalized Silacyclopentanes

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Bo, Yingjian; Sieburth, Scott McN.: A Quantitative NMR Method for Silyllithium Analysis

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Xie, Hengmu; Lu, Ji; Gui, Yingying; Gao, Lu; Song, Zhenlei: (HMe₂SiCH₂)₂: A Useful Reagent for B(C₆F₅)₃-Catalyzed Reduction–Lactonization of Keto Acids: Concise Syntheses of (–)-cis-Whisky and (–)-cis-Cognac Lactones

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Yamamoto, Eiji; Ukigai, Satoshi; Ito, Hajime: Formal Nucleophilic Silyl Substitution of Aryl Halides with Silyllithium Reagents via Halogenophilic Attack of Silyl Nucleophiles

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Cornelissen, Loïc; Nagy, Audric; Leyssens, Tom; Riant, Olivier: Tetrabutylammonium Bifluoride as an Efficient Activating Agent for Copper-Catalyzed Vinylsilane Cross-Coupling Reactions

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Fang, Huaquan; He, Qiaoxing; Liu, Guixia; Huang, Zheng: Pincer Ruthenium Catalyzed Intramolecular Silylation of C(sp²)–H Bonds

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Godou, Timothé; Chauvier, Clément; Thuéry, Pierre; Cantat, Thibault: Iron-Catalyzed Silylation of Alcohols by Transfer Hydrosilylation with Silyl Formates

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Sanzone, Jillian R.; Woerpel, K. A.: Reactivity of Seven-Membered-Ring trans-Alkenes with Electrophiles

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Issue 15/2017

Cluster Cover Page

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Liu, Lei: Cluster Preface: Recent Advances in Protein and Peptide Synthesis

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Jiang, Yan-Hong; Zhao, Hui; Tian, Yuan; Li, Zi-Gang: Lipid–Cell-Penetrating-Peptide Conjugates as Effective Delivery Systems

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Tornøe, Christian W.; Johansson, Eva; Wahlund, Per-Olof: Divergent Protein Synthesis of Bowman–Birk Protease Inhibitors, their Hydrodynamic Behavior and Co-crystallization with α-Chymotrypsin

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Qi, Yun-Kun; He, Qiao-Qiao; Ai, Hua-Song; Li, Jia-Bin; Zheng, Ji-Shen: Convergent Total Synthesis of Histone H2B Protein with Site-Specific Ubiquitination at Lys120

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Li, Kaicheng; Gao, Jianmin: Iminoboronate-Mediated Peptide Cyclization with Lysine Homologues

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Guan, Xiaoyang; Chaffey, Patrick K.; Ruan, Yuan; Hurd, Connor K.; Taatjes, Dylan J.; Tan, Zhongping: Chemical Synthesis of the Multiply Phosphorylated and Biotinylated N-Terminal Transactivation Domain of Human p53 (p53TAD)

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Castillo-Pazos, Durbis J.; Macmillan, Derek: Investigation of Cysteine as an Activator of Side-Chain N→S Acyl Transfer and Tail-to-Side-Chain Cyclization

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Rohrbacher, Florian; Baldauf, Simon; Wucherpfennig, Thomas G.; Bode, Jeffrey W.: Product Selectivity in KAHA Ligations: Ester vs. Amide Formation with Cyclic Hydroxylamines

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Wang, Jian; Zhang, Ru-Yan; Wang, Ya-Cong; Chen, Xiang-Zhao; Yin, Xu-Guang; Du, Jing-Jing; Lei, Ze; Xin, Ling-Ming; Gao, Xiao-Fei; Liu, Zheng; Guo, Jun: Polyfluorophenyl Ester-Terminated Homobifunctional Cross-Linkers for Protein Conjugation

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He, Qiaoqiao; Qi, Yunkun; Liu, Chao; Li, Jiabin; Hu, Honggang: Synthesis of a Ubiquitinated Histone Mimic Bearing a New Thioether Linkage

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Aihara, Keisuke; Inokuma, Tsubasa; Jichu, Takahisa; Lin, Zhenjian; Fu, Feixue; Yamaoka, Kosuke; Shigenaga, Akira; Hutchins, David A.; Schmidt, Eric W.; Otaka, Akira: Cysteine-Free Intramolecular Ligation of N-Sulfanylethylanilide Peptide Using 4-Mercaptobenzylphosphonic Acid: Synthesis of Cyclic Peptide Trichamide

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Matveenko, Maria; Becker, Christian F. W.: Synthetic Approach to Argpyrimidine as a Tool for Investigating Nonenzymatic Posttranslational Modification of Proteins

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Tsuda, Shugo; Uemura, Tsuyoshi; Mochizuki, Masayoshi; Nishio, Hideki; Yoshiya, Taku: Preparation of Peptide o-Aminoanilides Using a Modified Dawson's Linker for Microwave-Assisted Peptide Synthesis

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Chen, Pu-Guang; Huang, Zhi-Hua; Sun, Zhan-Yi; Li, Qian-Qian; Chen, Yong-Xiang; Zhao, Yu-Fen; Li, Yan-Mei: Synthesis of an MUC1 Glycopeptide Dendrimer Based on β-Cyclodextrin by Click Chemistry

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Tian, Xiaobo; Yu, Pengqiu; Tang, Yubo; Le, Zhiping; Huang, Wei: Aspartic Acid Side-Chain Benzyl Ester as a Multifunctionalization Precursor for Synthesis of Branched and Cyclic Arginylglycylaspartic Acid Peptides

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Issue 14/2017

Reiser, Oliver: Heterocyclic Chemistry – Old Science or the Forefront of Chemistry?

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Hossain, Asik; Pagire, Santosh K.; Reiser, Oliver: Visible-Light-Mediated Synthesis of Pyrazines from Vinyl Azides Utilizing a Photocascade Process

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Mei, Ruhuai; Zhang, Shou-Kun; Ackermann, Lutz: Concise Synthesis of Lamellarin Alkaloids by C–H/N–H Activation: Evaluation of Metal Catalysts in Oxidative Alkyne Annulation

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Sato, Shogo; Kawada, Takuma; Takikawa, Hiroshi; Suzuki, Keisuke: Preparation of 2-Substituted 3-Methoxycarbonyl-4-methoxyfurans that Allow Access to Highly Functionalized Naphthalenes via Regioselective Cycloaddition with Alkoxybenzyne

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Jarrige, Lucie; Merad, Jeremy; Zaied, Siwar; Blanchard, Florent; Masson, Géraldine: Easy Access to Quinolin-2(1H)-ones via a One-Pot Tandem Oxa-Michael–Aldol Sequence

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Patil, Pravin C.; Luzzio, Frederick A.: Unnatural Amino Acid Derivatives through Click Chemistry: Synthesis of Triazolylalanine Analogues

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Kippo, Takashi; Kimura, Yuki; Ueda, Mitsuhiro; Fukuyama, Takahide; Ryu, Ilhyong: Bromine-Radical-Mediated Synthesis of β-Functionalized β,γ- and δ,ε-Unsaturated Ketones via C–H Functionalization of Aldehydes

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Aitken, R. Alan; Harper, Andrew D; Slawin, Alexandra M. Z.: Base-Induced Cyclisation of ortho-Substituted 2-Phenyloxazolines to Give 3-Aminobenzofurans and Related Heterocycles

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Lessing, Timo; Müller, Thomas J. J.: One-Pot Coupling–Cyclization–Alkylation Synthesis of 1,2,5-Trisubstituted 7-Azaindoles in a Consecutive Three-component Fashion

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Talero, Alexánder G.; Burtoloso, Antonio C. B.: Sharpless Asymmetric Dihydroxylation on α,β-Unsaturated Diazoketones: A New Entry for the Synthesis of Disubstituted Furanones

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Parra, Claudio; Solís, Pablo; Bonjoch, Josep; Bradshaw, Ben: A One-Pot Methodology for the Synthesis of the Yohimban Skeleton

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Mai, Duy N.; Uchenik, Dmitriy; Vanderwal, Christopher D.: Efforts Toward a Synthesis of Crotogoudin and Crotobarin

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Issue 13/2017

Cluster Cover Page

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Stahl, Shannon S.; Rovis, Tomislav: Cluster Preface: Catalytic Aerobic Oxidations

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Kwon, Ohhyeon; Esguerra, Kenneth Virgel N.; Glazerman, Michael; Petitjean, Laurène; Xu, Yalun; Ottenwaelder, Xavier; Lumb, Jean-Philip: Development of 3,5-Di-tert-butylphenol as a Model Substrate for Biomimetic Aerobic Copper Catalysis

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Shibuya, Masatoshi; Furukawa, Keisuke; Yamamoto, Yoshihiko: Selective Aerobic Oxidation of Primary Alcohols to Aldehydes

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Singh, Atul K.; Yi, Hong; Zhang, Guoting; Bian, Changliang; Pei, Pengkun; Lei, Aiwen: Photoinduced Oxidative Cross-Coupling for O–S Bond Formation: A Facile Synthesis of Alkyl Benzenesulfonates

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Sterckx, Hans; Sambiagio, Carlo; Lemière, Filip; Tehrani, Kourosch Abbaspour; Maes, Bert U. W.: Iron-Catalyzed Aerobic Oxidation of (Alkyl)(aryl)azinylmethanes

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Lo, Kai-Yip; Ye, Liu; Yang, Dan: Palladium-Catalyzed Aerobic Oxidative Cyclization of Aliphatic Alkenyl Amides for the Construction of Pyrrolizidine and Indolizidine Derivatives

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Tanaka, Hirotaka; Oisaki, Kounosuke; Kanai, Motomu: Ligand-Free, Copper-Catalyzed Aerobic Benzylic sp³ C–H Oxygenation

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Li, Ziyuan; Wang, Xiaoyang; Ma, Lifang; Jiao, Ning: Copper-Catalyzed Aerobic Oxidation and Oxygenation of Anilines and Acetaldehydes with Dioxygen for the Concise Synthesis of 2-Aroylquinolines

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Issue 11/2017

Cluster Cover Page

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Tan, Choon-Hong; List, Benjamin: Cluster Preface: Asymmetric Brønsted Base Catalysis

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Teng, Bo; Lim, Wei Chun; Tan, Choon-Hong: Recent Advances in Enantioselective Brønsted Base Organocatalytic Reactions

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Eröksüz, Serap; Neudörfl, Jörg M.; Berkessel, Albrecht: Kinetic Resolution of 5-Substituted Oxazinones with Bifunctional Chiral Base/Squaramide Organocatalysts

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Schnitzer, Tobias; Wennemers, Helma: Thieme Chemistry Journals Awardees – Where Are They Now?
A Stereoselective Tripeptide Catalyst for Conjugate Addition Reactions of Acetophenones to Dicyanoolefins

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Yamashita, Yasuhiro; Igarashi, Ryo; Suzuki, Hirotsugu; Kobayashi, Shū: Catalytic Asymmetric Direct-Type 1,4-Addition Reactions of Alkanesulfonamides

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Ohmatsu, Kohsuke; Ando, Yuichiro; Ooi, Takashi: In Situ Electrophilic Activation of Hydrogen Peroxide for Catalytic Asymmetric α-Hydroxylation of 3-Substituted Oxindoles

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March, Taryn; Murata, Akihiro; Kobayashi, Yusuke; Takemoto, Yoshiji: Enantioselective Synthesis of anti-β-Hydroxy-α-amino Esters via an Organocatalyzed Decarboxylative Aldol Reaction

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Wang, Fei; Chen, Jiean; Huang, Yong: Synthesis of Optically Active Oxazolines by an Organocatalytic Isocyanoacetate Aldol Reaction with α-Keto Esters

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Odagi, Minami; Hosoya, Keisuke; Yamamoto, Yoshiharu; Nagasawa, Kazuo: Oxidative Kinetic Resolution of cis-Fused Tricyclic 1-Tetralone Derivatives by Guanidine–Bisurea Bifunctional Organocatalyst

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Zhang, Gao; Yin, Yanli; Zhao, Xiaowei; Jiang, Zhiyong: Organocatalytic Asymmetric Tandem Conjugate Addition–Protonation of Azlactones to N-Itaconimides

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Issue 01/2017

Cluster Cover Page

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Krishnamurthy, Ramanarayanan; Snieckus, Victor: Prebiotic Organic Chemistry and Chemical pre-Biology: Speaking to the Synthetic Organic Chemists

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Ritson, Dougal J.; Xu, Jiangfeng; Sutherland, John D.: Thiophosphate – A Versatile Prebiotic Reagent?

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Leman, Luke J.; Ghadiri, M. Reza: Potentially Prebiotic Synthesis of α-Amino Thioacids in Water

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Liu, Ziwei; Hanson, Cassandra; Ajram, Ghinwa; Boiteau, Laurent; Rossi, Jean-Christophe; Danger, Grégoire; Pascal, Robert: 5(4H)-Oxazolones as Effective Aminoacylation Reagents for the 3′-Terminus of RNA

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Fernández-García, Christian; Powner, Matthew W.: Selective Acylation of Nucleosides, Nucleotides, and Glycerol-3-phosphocholine in Water

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Biondi, Elisa; Howell, Layne; Benner, Steven A.: Opal Adsorbs and Stabilizes RNA – A Hierarchy of Prebiotic Silica Minerals

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Gherase, Dragos; Hazen, Robert M.; Krishnamurthy, Ramanarayanan; Blackmond, Donna G.: Mineral-Induced Enantioenrichment of Tartaric Acid

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Mohammed, Fiaz S.; Chen, Ke; Mojica, Mike; Conley, Mark; Napoline, Jonathan W.; Butch, Christopher; Pollet, Pamela; Krishnamurthy, Ramanarayanan; Liotta, Charles L.: A Plausible Prebiotic Origin of Glyoxylate: Nonenzymatic Transamination Reactions of Glycine with Formaldehyde

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Rice, Gavin B.; Yerabolu, Jayasudhan R.; Krishnamurthy, Ramanarayanan; Springsteen, Greg: The Abiotic Oxidation of Organic Acids to Malonate

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Mattia, Elio; Pal, Asish; Leonetti, Giulia; Otto, Sijbren: Mechanism of Building Block Exchange in Stacks of Self-Replicating Macrocycles

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Brea, Roberto J.; Bhattacharya, Ahanjit; Devaraj, Neal K.: Spontaneous Phospholipid Membrane Formation by Histidine Ligation

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Issue 14/2016

Cluster Cover Page

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Kuck, Dietmar: Cluster Preface: Nonplanar Polyaromatic Compounds

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Yano, Yuuta; Ito, Hideto; Segawa, Yasutomo; Itami, Kenichiro: Helically Twisted Tetracene: Synthesis, Crystal Structure, and Photophysical Properties of Hexabenzo[a,c,fg,j,l,op]tetracene

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Yamada, Kenta; Shibamoto, Hiroshi; Tanigawa, Yusuke; Ishikawa, Hiroyuki; Nishida, Jun-ichi; Kitamura, Chitoshi; Kurata, Hiroyuki; Kawase, Takeshi: Fulvalene Derivatives Containing a Tetrabenzofluorene Unit: New Nonplanar Fulvalenes with High Electron Affinity

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Yang, Xuejin; Miao, Qian: Studies toward the Synthesis of Hepta-peri-heptabenzo-[7]circulene

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Deng, Chun-Lin; Hau, Sam C. K.; Peng, Xiao-Shui; Wong, Henry N. C.: Synthesis of Unexpected trans-meso Macrocycle from Novel Unsymmetrical Tetraphenylene

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Rajeshkumar, Venkatachalam; Marc, Courte; Fichou, Denis; Stuparu, Mihaiela C.: Synthesis and Properties of a Buckybowl/Buckyball Dyad

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Cocq, Kévin; Saffon-Merceron, Nathalie; Poater, Albert; Maraval, Valérie; Chauvin, Remi: Aromatic Rings and Aromatic Rods: Nonplanar Character of an Indeno-dehydro[14]annulene

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Zhang, Baozhong; Zhao, Yuming; Bodwell, Graham J.: Kinetic Stabilization of a Highly Bent Pyrene System

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Maag, Roman; Siegel, Jay S.: Synthesis of a Five-Fold-Differentiated 1,3,5,7,9-Pentasubstituted Corannulene: A Maximal Labeling Problem in the Context of Corannulene

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Yu, Yuming; Xu, Liang; Huang, Xinchen; Liang, Sisi; Gan, Liangbing: Synthesis of C₅₈ Open-Cage Fullerene Derivatives

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Amaya, Toru; Katoh, Shun; Hirao, Toshikazu: Bowl-to-Bowl Inversion Accelerated by the Introduction of Bulky 1,1,4,4-Tetramethylbutane-1,4-diyl Groups on Sumanene

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Kurata, Hiroyuki; Inoue, Taihei; Suzuki, Takeshi; Hirao, Yasukazu; Matsumoto, Kouzou; Kubo, Takashi: Synthesis, Structure, and Properties of Quinone Methides Incorporating Thiophene and Bithiophene Derivatives: New Overcrowded Extended Quinonoid π-Systems

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Nobusue, Shunpei; Tobe, Yoshito: Twisted Polycyclic Aromatic Hydrocarbon with a Cyclooctatetraene Core via Formal [4+4] Dimerization of Indenofluorene

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Sharafi, Mona; Weinert, Zackariah J.; Cohen, Ian M.; Liao, Chenyi; Ivancic, Monika; Li, Jianing; Schneebeli, Severin T.: Controlled Self-Assembly inside C-Shaped Polyaromatic Strips

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Lehne, Verena; Ernst, Ludger; Hopf, Henning: Exploring the Chemistry of [2.2.2]Paracyclophane

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Issue 08/2016

Cluster Cover Page

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Hierso, Jean-Cyrille; Uozumi, Yasuhiro: Cluster Preface: Heterogeneous Catalysis

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Murakami, Ryo; Iwai, Tomohiro; Sawamura, Masaya: Site-Selective and Stereoselective C(sp³)–H Borylation of Alkyl Side Chains of 1,3-Azoles with a Silica-Supported Monophosphine-Iridium Catalyst

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Gholinejad, Mohammad; Hamed, Fatemeh; Nájera, Carmen: Gold Nanoparticles Supported on Polyacrylamide Containing a Phosphorus Ligand as an Efficient Heterogeneous Catalyst for Three-Component Synthesis of Propargylamines in Water

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Ohtaka, Atsushi; Kotera, Takamasa; Sakon, Akira; Ueda, Kouhei; Hamasaka, Go; Uozumi, Yasuhiro; Shinagawa, Tsutomu; Shimomura, Osamu; Nomura, Ryôki: Fluoride-Free Hiyama Coupling Reaction Catalyzed by Linear Polystyrene-Stabilized PdO Nanoparticles in Water: Specific Reactivity of PdO Nanoparticles over Pd Nanoparticles

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Ma, Shuang; Toy, Patrick H.: Chromatography-Free Esterification Reactions Using a Bifunctional Polymer

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Reay, Alan J.; Neumann, Lydia K.; Fairlamb, Ian J. S.: Catalyst Efficacy of Homogeneous and Heterogeneous Palladium Catalysts in the Direct Arylation of Common Heterocycles

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Akagawa, Kengo; Hirata, Tomoaki; Kudo, Kazuaki: Asymmetric Epoxidation of Enones by Peptide-Based Catalyst: A Strategy Inverting Juliá–Colonna Stereoselectivity

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Okumura, Kazu: Formation and Catalysis of Gold Nanoparticles Generated through the Physical Mixing of AuCl(PPh₃) and Oxides

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Bizouard, Pierre; Testa, Christelle; Zinovyeva, Veronika A.; Roger, Julien; Hierso, Jean-Cyrille: Palladium–Polypyrrole Nanocomposites Pd@PPy for Direct C–H Functionalization of Pyrroles and Imidazoles with Bromoarenes

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Issue 07/2016

Cluster Cover Page

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Phipps, Robert J.: Cluster Preface: Non-Covalent Interactions in Asymmetric Catalysis

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Akamatsu, Masaaki; Matile, Stefan: Expanded Chiral Surfaces for Asymmetric Anion–π Catalysis

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Ohmatsu, Kohsuke; Hara, Yoshiyuki; Kusano, Yuya; Ooi, Takashi: Anion-Stoichiometry-Dependent Selectivity Enhancement in Ion-Paired Chiral Ligand–Palladium Complex Catalyzed Enantioselective Allylic Alkylation

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Molnár, István Gábor; Holland, Mareike C.; Daniliuc, Constantin; Houk, K. N.; Gilmour, Ryan: Organocatalysis Intermediates as Platforms to Study Noncovalent Interactions: Integrating Fluorine Gauche Effects in Iminium Systems to Facilitate Acyclic Conformational Control

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Böhm, Alexander; Bach, Thorsten: Synthesis of Supramolecular Iridium Catalysts and Their Use in Enantioselective Visible-Light-Induced Reactions

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Hatano, Manabu; Hayashi, Kazushi; Sakamoto, Tatsuhiro; Makino, Yuma; Ishihara, Kazuaki: Enantioselective Diels–Alder Reaction Induced by Chiral Supramolecular Lewis Acid Catalysts Based on CN···B and PO···B Coordination Bonds

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Yuan, Pengfei; Meng, Sixuan; Chen, Jiean; Huang, Yong: Asymmetric Sulfa-Michael Addition of α,β-Unsaturated Esters/Amides Using a Chiral N-Heterocyclic Carbene as a Noncovalent Organocatalyst

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Issue 05/2016

Cluster Cover Page

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Shenvi, Ryan A.: Cluster Preface: Reinventing Radical Reactions

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Hartmann, Marcel; Gerleve, Carolin; Studer, Armido: Intramolecular Radical Carboaminoxylation of Aryl Amines

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Chenneberg, Ludwig; Lévêque, Christophe; Corcé, Vincent; Baralle, Alexandre; Goddard, Jean-Philippe; Ollivier, Cyril; Fensterbank, Louis: Single-Electron-Transfer Oxidation of Trifluoroborates and Silicates with Organic Reagents: A Comparative Study

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Li, Yanjie; Koike, Takashi; Akita, Munetaka: Radical Pentafluorosulfanylphenylation of Styrenes by Photoredox Catalysis

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Ueno, Ryota; Shimizu, Takashi; Shirakawa, Eiji: Reduction of Aryl Halides into Arenes with 2-Propanol Promoted by a Substoichiometric Amount of a tert-Butoxy Radical Source

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Meyer, Daniel; Vin, Estelle; Wyler, Benjamin; Lapointe, Guillaume; Renaud, Philippe: Facile Preparation of Functionalized 1-Substituted Cycloalkenes via an Iodine Atom Transfer Radical Addition–Elimination Process

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Huo, Haohua; Huang, Xiaoqiang; Shen, Xiaodong; Harms, Klaus; Meggers, Eric: Visible-Light-Activated Enantioselective Perfluoroalkylation with a Chiral Iridium Photoredox Catalyst

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Swift, Elizabeth C.; Williams, Theresa M.; Stephenson, Corey R. J.: Intermolecular Photocatalytic C–H Functionalization of Electron-Rich Heterocycles with Tertiary Alkyl Halides

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Pascual, Laura M. M.; Dunford, Damian G.; Goetz, Adam E.; Ogawa, Kelli A.; Boydston, Andrew J.: Comparison of Pyrylium and Thiopyrylium Photooxidants in Metal-Free Ring-Opening Metathesis Polymerization

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Issue 04/2016

Cluster Cover Page

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Akiyama, Takahiko: Cluster Preface: BINOL Phosphates for Chemistry

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Mao, Zhenjun; Mo, Fan; Lin, Xufeng: Diastereo- and Enantioselective Assembly of Spirooxindole Tetrahydroquinoline Skeletons through Asymmetric Binary Acid Catalyzed Hydride Transfer–Cyclization

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Tay, Jia-Hui; Nagorny, Pavel: ³¹P NMR Based Method for Determining Enantiopurity of Chiral Phosphoric Acids and Its Application to the BINOL- and H8-BINOL-Based Chiral Phosphoric Acid Thermal Racemization Studies

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Lai, Zengwei; Sun, Jianwei: Enantioselective Addition of Thiols to ortho-Quinone Methides Catalyzed by Chiral Phosphoric Acids

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Lebée, Clément; Blanchard, Florent; Masson, Géraldine: Highly Enantioselective Intermolecular Iodo- and Chloroamination of Enecarbamates Catalyzed by Chiral Phosphoric Acids or Calcium Phosphate Salts

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Hatano, Manabu; Ishihara, Hideyuki; Goto, Yuta; Ishihara, Kazuaki: Remote Tris(pentafluorophenyl)borane-Assisted Chiral Phosphoric Acid Catalysts for the Enantioselective Diels–Alder Reaction

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Qin, Long; Wang, Pei; Zhang, Yixin; Ren, Zhengxiang; Zhang, Xin; Da, Chao-Shan: Direct Asymmetric Friedel–Crafts Reaction of Naphthols with Acetals Catalyzed by Chiral Brønsted Acids

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Jiang, Fei; Zhang, Yu-Chen; Yang, Xue; Zhu, Qiu-Ning; Shi, Feng: Catalytic Asymmetric Cascade Dearomatization of Tryptamines with Indol-3-ylmethanols: Diastereo- and Enantioselective Synthesis of Structurally Complex Indole Derivatives

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Kanomata, Kyohei; Terada, Masahiro: Study of Stereocontrolling Elements in Chiral Phosphoric Acid Catalyzed Addition Reaction of Vinylindoles with Azlactones

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Zhou, Yong; Liu, Xiao-Wei; Gu, Qing; You, Shu-Li: Enantioselective Synthesis of Tetrahydroindolizines via Ruthenium–Chiral Phosphoric Acid Sequential Catalysis

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Monaco, Mattia R.; Properzi, Roberta; List, Benjamin: An Approach to Highly Hindered BINOL Phosphates

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Issue 20/2015

Cluster Cover Page

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Snieckus, Victor; Knochel, Paul: Cluster Preface: Resurgence of Synthetic Aromatic Chemistry

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Zhang, Zhan; Xu, Lijun; Chen, Zhengkai; Liu, Zhubo; Miao, Maozhong; Song, Jinyu; Ren, Hongjun: Nickel-Catalyzed Regioselective Reductive Cross-Coupling of Aryl Halides with Polysubstituted Allyl Halides in the Presence of Imidazolium Salts

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Martina, Katia; Rinaldi, Laura; Baricco, Francesca; Boffa, Luisa; Cravotto, Giancarlo: Highly Efficient Mechanochemical N-Arylation of Amino Alcohols and Diamines with Cu⁰ Powder

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dos Santos, Fernanda M.; Batista, João H. C.; Vessecchi, Ricardo; Clososki, Giuliano C.: Directed Functionalization of Cyano-Substituted Furans and Thiophenes with TMPMgCl·LiCl

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Koga, Rintaro; Oishi, Tohru; Torikai, Kohei: Tuned Classical Thermal Aromatization Furnishing an Estrogenic Benzoacridine

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Rasheed, Omer K.; Raftery, James; Quayle, Peter: A New Benzannulation Reaction of Azoaromatics

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Marquise, Nada; Nguyen, Tan Tai; Chevallier, Floris; Picot, Laurent; Thiéry, Valérie; Lozach, Olivier; Bach, Stéphane; Ruchaud, Sandrine; Mongin, Florence: Azine and Diazine Functionalization Using 2,2,6,6-Tetramethylpiperidino-Based Lithium–Metal Combinations: Application to the Synthesis of 5,9-Disubstituted Pyrido[3′,2′:4,5]pyrrolo[1,2-c]pyrimidines

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Wu, Hao; Sheng, Wei-Jian; Chen, Bin; Liu, Ren-Rong; Gao, Jian-Rong; Jia, Yi-Xia: Nickel-Catalyzed Enantioselective Friedel–Crafts Alkylation of Indoles with β,β-Disubstituted Nitroalkenes

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Zhang, Xiao-Yan; Hu, Li-Li; Shen, Ze; Chen, Zhong-Zhu; Xu, Zhi-Gang; Li, Shi-Qiang; Xie, Jian-Wu; Cui, Hai-Lei: Copper-Catalyzed Synthesis of Furo[3,2-c]coumarins and Dihydrofuro[3,2-c]coumarins through a Propargylation/Alkyne Oxacyclization/Isomerization Cascade under Microwave Irradiation

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Yang, De-Suo; Ke, Sen; Fan, Ming-Jin; Zhu, Hai-Tao; Wang, Xiao-Ling; Guan, Zheng-Hui: A Facile and Efficient Synthesis of Six-Membered Enol Carbocyclic Compounds

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Chen, Jie; Xiong, Xiaoyu; Chen, Zenghua; Huang, Jianhui: Imidazolium Salt Catalyzed para-Selective Halogenation of Electron-Rich Arenes

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Issue 17/2015

Mordini, Alessandro; Snieckus, Victor: Cluster Preface: In Memory of Professor Manfred Schlosser

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Stead, Darren; O’Brien, Peter; Sanderson, Adam: Investigation of the Lithiation-Trapping of an N-Boc Bispidine-Ketal: Reactivity and Diastereoselectivity

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Maddaluno, Jacques; Durandetti, Muriel: Dimerization of Aryl Sulfonates by in situ Generated Nickel(0)

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Franchi, Daniele; Calamante, Massimo; Reginato, Gianna; Zani, Lorenzo; Peruzzini, Maurizio; Taddei, Maurizio; Fabrizi de Biani, Fabrizia; Basosi, Riccardo; Sinicropi, Adalgisa; Colonna, Daniele; Di Carlo, Aldo; Mordini, Alessandro: Two New Dyes with Carboxypyridinium Regioisomers as Anchoring Groups for Dye-Sensitized Solar Cells

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Shimada, Yukako; Haraguchi, Ryosuke; Matsubara, Seijiro: Preparation of an Arenylmethylzinc Reagent with Functional Groups by Chemoselective Cross-Coupling Reaction of Bis(iodo­zincio)methane with Iodoarenes

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Behloul, Cherif; Bouchelouche, Kenza; Guijarro, David; Foubelo, Francisco; Nájera, Carmen; Yus, Miguel: Indium-Mediated Cleavage of the Trityl Group from Protected 1H-Tetrazoles

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Kitazawa, Yu; Otsuka, Mai; Kanazawa, Junichiro; Takita, Ryo; Uchiyama, Masanobu: Palladium-Catalyzed Cross-Coupling Reaction of Lithiated Monocarba-closo-dodecaborate at the Carbon Vertex

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Mehdi, Mariam A.; Djurdjevic, Sinisa; Green, James R.: Lewis Acid Catalyzed Synthesis of Allocolchicinoids

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Ryu, Ilhyong; Yamamura, Go-hei; Minakata, Satoshi; Komatsu, Mitsuo; Kubo, Haruka; Ueda, Mitsuhiro: Intramolecular Carbolithiation of 3-Lithioxy-5-alkenyllithiums as a Platform for Cyclopentanols and Cyclopentanones

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Milen, Mátyás; Földesi, Tamás; Dancsó, András; Simig, Gyula; Volk, Balázs: Synthesis of Three New Tricyclic Ring Systems: Pyrrolotriazepines Condensed with an Imidazole, a Triazole, or a Tetrazole Ring

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Issue 03/2015

Cluster Cover Page

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Gaunt, Matthew J.; Chow, Hak-Fun; Rovis, Tomislav: Cluster Preface: Catalysis Using Sustainable Metals – Part II

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Zhong, Yao; Spahn, Nathan A.; Stolley, Ryan M.; Nguyen, Minh H.; Louie, Janis: 3,5-Disubstituted 2-Aminopyridines via Nickel-Catalyzed Cycloaddition of Terminal Alkynes and Cyanamides

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Westerhaus, Felix A.; Sorribes, Iván; Wienhöfer, Gerrit; Junge, Kathrin; Beller, Matthias: Reduction of Nitroarenes Using CO and H₂O in the Presence of a Nanostructured Cobalt Oxide/Nitrogen-Doped Graphene (NGr) Catalyst

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Semba, Kazuhiko; Kameyama, Ryohei; Nakao, Yoshiaki: Copper-Catalyzed Semihydrogenation of Alkynes to Z-Alkenes

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Caputo, Jill A.; Naodovic, Marina; Weix, Daniel J.: Nickel-Catalyzed Allylation of α-Amido Sulfones To Form Protected Homoallylic Amines

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Baralle, Alexandre; Otsuka, Shinya; Guérin, Vincent; Murakami, Kei; Yorimitsu, Hideki; Osuka, Atsuhiro: Nickel–NHC-Catalyzed Cross-Coupling of 2-Methylsulfanylbenzofurans with Alkyl Grignard Reagents

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Jefferies, Latisha R.; Weber, Savannah R.; Cook, Silas P.: Iron-Catalyzed C–N Bond Formation via the Beckmann Rearrangement

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Liwosz, Timothy W.; Chemler, Sherry R.: Copper-Catalyzed Synthesis of N-Aryl and N-Sulfonyl Indoles from 2-Vinyl­anilines with O₂ as Terminal Oxidant and TEMPO as Cocatalyst

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Yamakawa, Takeshi; Seto, Yuan Wah; Yoshikai, Naohiko: Cobalt-Catalyzed Directed Alkylation of Olefinic C–H Bond with Primary and Secondary Alkyl Chlorides

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Zhu, Cheng-Liang; Zhang, Yong-Qiang; Yuan, Yong-An; Xu, Hao: Copper-Catalyzed Aerobic C–H Trifluoromethylation of Phenanthrolines

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Choi, Bonnie; Saxena, Aakarsh; Smith, Joshua J.; Churchill, Gwydion H.; Lam, Hon Wai: Enantioselective Copper-Catalyzed Reductive Coupling of Vinylazaarenes with N-Boc Aldimines

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Issue 01/2015

Cluster Cover Page

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Browne, Duncan L.: Cluster Preface: Progress in Organo-Fluorine Chemistry

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Xu, Peng; Guo, Shuo; Wang, Liyan; Tang, Pingping: Recent Advances in the Synthesis of Difluoromethylated Arenes

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Dai, Xiaoyang; Cahard, Dominique: Regio- and Stereocontrolled Nucleophilic Trifluoromethylthiolation of Morita–Baylis–Hillman Carbonates

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Lishchynskyi, Anton; Mazloomi, Zahra; Grushin, Vladimir V.: Trifluoromethylation and Pentafluoroethylation of Vinylic Halides with Low-Cost R_fH-Derived CuR_f (R_f = CF₃, C₂F₅)

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Breen, Jessica R.; Sandford, Graham; Patel, Bhairavi; Fray, Jonathan: Synthesis of 4,4-Difluoro-1H-pyrazole Derivatives

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Tarui, Atsushi; Miyata, Erina; Tanaka, Ayumi; Sato, Kazuyuki; Omote, Masaaki; Ando, Akira: Stereoselective Suzuki Coupling Reaction of an α-Bromo-α-fluoro-β-lactam

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Zhang, Zhikun; Feng, Jiajie; Xu, Yan; Zhang, Songnan; Ye, Yuxuan; Li, Tianjiao; Wang, Xi; Chen, Jun; Zhang, Yan; Wang, Jianbo: Synthesis of Trifluoromethylated Cycloheptatrienes from N-Tosylhydrazones: Transition-Metal-Free Büchner Ring Expansion

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Kageshima, Yoshiya; Suzuki, Chiharu; Oshiro, Kojun; Amii, Hideki: Highly Controlled Ring-Opening of Siloxydifluorocyclopropanes: A Versatile Route to Cyclic Fluoroketones

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Liu, Yingle; Yang, Yi; Huang, Yangen; Xu, Xiu-Hua; Qing, Feng-Ling: Regio- and Diastereoselective Vinylogous Mannich Addition of 3-Alkenyl-2-oxindoles to α-Fluoroalkyl Aldimines

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Hendriks, Christine M. M.; Reball, Jens; Bolm, Carsten: Methyl 4-Pentafluorosulfanylphenyl Sulfoximines

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Alazet, Sébastien; Billard, Thierry: Electrophilic Aromatic Trifluoromethylthiolation with the Second Generation of Trifluoromethanesulfenamide

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Issue 19/2014

Cluster Cover Page

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Gaunt, Matthew; Rovis, Tomislav; Chow, Hak-Fun: Catalysis Using Sustainable Metals – Part I

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Feng, Peng; Song, Song; Zhang, Li-He; Jiao, Ning: CAN-Catalyzed Rapid C–O Bond Formation towards α-Aminoxylation of Ketones

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Chen, Junjie; Chen, Chao; Chen, Jing; Gao, Hongpeng; Qu, Hongmei: An Unprecedented Tandem Annulation of ω-Azido-1-alkynes with Diaryl­iodonium Salts: A Facile Synthesis of Polycyclic Quinolines

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Mao, Liu-Liang; Zhou, An-Xi; Liu, Na; Yang, Shang-Dong: Copper-Catalyzed Oxidative Cross-Coupling of H-Phosphine Oxides with Alkenes in the Synthesis of Alkenylphosphine Oxides

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Xue, Zhi-Yong; Xiong, Yong; Wang, Chun-Jiang: Catalytic Asymmetric Construction of Azabicyclo[2.2.1]heptanes Bearing Two Quaternary Stereogenic Centers via Silver(I)-Catalyzed 1,3-Dipolar Cyclo­addition of Cyclic Azomethine Ylides

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He, Lisi; Ho, Chun-Yu: Nitrate-Enhanced NHC-NiH Catalyzed Tail-to-Tail Vinyl Ether Dimerization

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Lee, Hang Wai; Yung, Ka Fu; Kwong, Fuk Yee: Iron-Catalyzed S-Arylation of Benzothiazole with Aryl Iodides under Aqueous Medium: Facile Synthesis of Aryl(2-aminoaryl) Sulfides

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Fu, Ming-Chen; Shang, Rui; Huang, Zheng; Fu, Yao: Conversion of Levulinate Ester and Formic Acid into γ-Valerolactone Using a Homogeneous Iron Catalyst

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Issue 16/2014

Cluster Cover Page

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Green, James R.; Snieckus, Victor: Activated Cyclopropanes: A Remarkable Breadth of Recent Chemistry

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Ren, Jun; Bao, Jilai; Ma, Weiwei; Wang, Zhongwen: Tandem Diels–Alder [4+2] Cycloadditions and Intramolecular [3+2] Cross-Cycloadditions of Dienylcyclopropane 1,1-Diesters

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Reich, Dorian; Müller, Dennis S.; Schefzig, Luise; Zimmer, Reinhold; Reissig, Hans-Ulrich: One-Pot Generation of C≡X Bonds from Methyl 2-Siloxycyclopropane­carboxylates: Simple Syntheses of Functionalized Nitriles and Alkynes

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Li, Ling; Wei, Enxiang; Lin, Shaoxia; Liu, Bing; Liang, Fushun: 1,4-Diazabicyclo[2.2.2]octane-Mediated Ring Opening of 1-Acetylcyclopropanecarboxamides and Its Application to the Construction of 3-Alkylated γ-Lactams

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Mikhaylov, Andrey A.; Novikov, Roman A.; Khomutova, Yulia A.; Arkhipov, Dmitry E.; Korlyukov, Alexander A.; Tabolin, Andrey A.; Tomilov, Yury V.; Ioffe, Sema L.: Novel Formal [3+3] Cycloaddition of Silyl Nitronates with Activated Cyclo­propanes and Its Application in the Synthesis of Pyrroline-N-oxides

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Tombe, Rihoko; Iwamoto, Takahiro; Kurahashi, Takuya; Matsubara, Seijiro: Regio- and Diastereoselective Nickel-Catalyzed Cycloaddition of Activated Cyclopropanes with Allenes

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Serrano, Eloisa; de Nanteuil, Florian; Waser, Jerome: Diester-Substituted Aminocyclopropanes: Synthesis and Use in [3+2]-Annulation Reactions

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Ivanova, Olga A.; Budynina, Ekaterina M.; Skvortsov, Dmitriy A.; Trushkov, Igor V.; Melnikov, Mikhail Ya.: Shortcut Approach to Cyclopenta[b]indoles by [3+2] Cyclodimerization of Indole-Derived Cyclopropanes

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Sun, Run; Zhang, Di-Han; Shi, Min: Lewis Acid Catalyzed Intramolecular Ring-Opening of Triazole-Substituted Methylenecyclopropanes: An Approach to 4H-[1,2,3]Triazolopyrazines and 4H-[1,2,3]Triazolo[1,4]diazepines

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Flisar, Michelle E.; Emmett, Michael R.; Kerr, Michael A.: Catalyst-Free Tandem Ring-Opening/Click Reaction of Acetylene-Bearing Donor–Acceptor Cyclopropanes

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Nikolaev, Andrei; Nithiy, Nisha; Orellana, Arturo: One-Step Synthesis of Quinolines via Palladium-Catalyzed Cross-Coupling of Cyclopropanols with Unprotected ortho-Bromoanilines

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Hirata, Goki; Onodera, Gen; Kimura, Masanari: Synthesis of Lactones and Lactams from Vinylcyclopropane by Palladium- Catalyzed Nucleophilic Allylation

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Chen, Gen-Qiang; Tang, Xiang-Ying; Shi, Min: Rhodium-Catalyzed Carbonylative Skeleton Rearrangement of 1,4-Enynes Tethered by a Cyclopropane Group

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Pursley, Dominik; Plietker, Bernd: Insertion of Imines into Vinylcyclopropanes Catalyzed by Nucleophilic Iron Complexes: A Formal [3+2]-Cycloaddition Strategy for the Synthesis of Substituted Pyrrolidine Derivatives

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Issue 11/2014

Cluster Cover Page

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Alcarazo, Manuel: Frustrated Lewis Pairs: An Elegant Concept for Catalysis

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Dornan, Peter K.; Longobardi, Lauren E.; Stephan, Douglas W.: Reversible Frustrated Lewis Pair Addition of N-Heterocycles to Unsaturated C–C Bonds

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Dorkó, Éva; Varga, Eszter; Gáti, Tamás; Holczbauer, Tamás; Pápai, Imre; Mehdi, Hasan; Soós, Tibor: Steric Control of Geminal Lewis Pair Behavior: Frustration Induced Dyotropic Rearrangement

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Feldhaus, Philipp; Wibbeling, Birgit; Fröhlich, Roland; Daniliuc, Constantin G.; Kehr, Gerald; Erker, Gerhard: Formation of Allenes by 1,4-Addition of Intermolecular Phosphane/Borane Frustrated Lewis Pairs to a Conjugated Enyne

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He, Jianghua; Zhang, Yuetao; Chen, Eugene Y.-X.: Synthesis of Pyridine- and 2-Oxazoline-Functionalized Vinyl Polymers by Alane-Based Frustrated Lewis Pairs

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Inés, Blanca; Holle, Sigrid; Bock, Dominique A.; Alcarazo, Manuel: Polyfluorinated Cyclopentadienones as Lewis Acids

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Issue 19/2013

Cluster Cover Page

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Ishikawa, Tsutomu; Harwood, Laurence M.: Organic Superbases: The Concept at a Glance

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Suzuki, Noriyuki; Kishimoto, Kaito; Yamazaki, Kohei; Kumamoto, Takuya; Ishikawa, Tsutomu; Margetić, Davor: Immobilized 1,2-Bis(guanidinoalkyl)benzenes: Potentially Useful for the Purification of Arsenic-Polluted Water

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Filatova, Ekaterina A.; Pozharskii, Alexander F.; Gulevskaya, Anna V.; Vistorobskii, Nikolay V.; Ozeryanskii, Valery A.: Synthesis of 2-Alkynyl-, 4-Alkynyl-, and 2,7-Dialkynyl-1,8-bis(dimethyl­amino)naphthalenes and the Unexpected Influence of ortho-Alkynyl Groups on Their Basicity

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Biswas, Abul Kalam; Lo, Rabindranath; Ganguly, Bishwajit: Is the Isodesmic Reaction Approach a Better Model for Accurate Calculation of pK_a of Organic Superbases? A Computational Study

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Carrera, Gonçalo V. S. M.; Costa, Alexandra; da Ponte, Manuel Nunes; Branco, Luis C.: Use of Organic Superbases and Temperature Effects for the Development of Reversible Protic Amino Acid Salts

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Terada, Masahiro; Goto, Kengo; Oishi, Masafumi; Takeda, Tadahiro; Kwon, Eunsang; Kondoh, Azusa: Design and Synthesis of Helically Chiral Spirocyclic P3 Phosphazenes and Characterization of Their Onium Salts

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Selig, Philipp; Turočkin, Aleksej; Raven, William: Guanidine-Catalyzed γ-Selective Morita–Baylis–Hillman Reactions on α,γ-Dialkyl-Allenoates: Access to Densely Substituted Heterocycles

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Glasovac, Zoran; Trošelj, Pavle; Jušinski, Iva; Margetić, Davor; Eckert-Maksić, Mirjana: Synthesis of Highly Basic Hexasubstituted Biguanides by Environmentally Friendly Methods

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Issue 10/2013

Cluster Cover Page

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Rovis, Tomislav; Nolan, Steven P.: Stable Carbenes: From ‘Laboratory Curiosities’ to Catalysis Mainstays

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Chen, Ming-Tsz; Navarro, Oscar: N-Heterocyclic Carbene (NHC)–Copper(I) Complexes as Catalysts for A³ Reactions

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Abbas, Muddasar; Leitgeb, Anita; Slugovc, Christian: Low Catalyst Loading in the Cross Metathesis of Olefins with Methyl Vinyl Ketone

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Hao, Lin; Chuen, Chan Wei; Ganguly, Rakesh; Chi, Yonggui Robin: NHC-Catalyzed Ester Activation: Access to Sterically Congested Spirocyclic Oxindoles via Reaction of α-Aryl Esters and Unsaturated Imines

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Jia, Min-Qiang; You, Shu-Li: Desymmetrization of Cyclohexadienones via Intramolecular Stetter Reaction to Construct Tricyclic Carbocycles

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Gondo, Chenaimwoyo A.; Bode, Jeffrey W.: Catalytic Redox Amidations of Aldehydes with a Polymer-Supported Peptide–N-Heterocyclic Carbene Multifunctional Catalyst

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Ondrusek, Brian A.; Opalka, Suzanne M.; Hietsoi, Oleksandr; Shatruk, Michael; McQuade, D. Tyler: Structure and Reactivity of a Copper(I)-Fused N-Heterocyclic Carbene ­Complex: Reactivity toward Styrenic and Strained Alkenes

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Wu, Linglin; Salvador, Alvaro; Ou, Arnold; Shi, Ming Wen; Skelton, Brian W.; Dorta, Reto: Monodentate Chiral N-Heterocyclic Carbene–Palladium-Catalyzed Asymmetric Suzuki–Miyaura and Kumada Coupling

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Dong, Xiuqin; Zhao, Yu-Ming; Sun, Jianwei: N-Heterocyclic Carbene (NHC) Catalyzed Synthesis of α,α-Difluoro Esters

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Gundala, Sivaji; Fagan, Claire-Louise; Delany, Eoghan G.; Connon, Stephen J.: Organocatalytic Aerobic Oxidative Cleavage of Cyclic 1,2-Diketones

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Zhao, Xiaodan; Glover, Garrett S.; Oberg, Kevin M.; Dalton, Derek M.; Rovis, Tomislav: S_NAr-Derived Decomposition By-products Involving Pentafluorophenyl Triazolium Carbenes

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Hepperle, Johannes A. M.; Samanta, Ramesh C.; Studer, Armido: N-Heterocyclic Carbene Catalyzed Transesterification of Polytrifluoroethyl Acrylates

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Gung, Benjamin W.; Conyers, Ryan C.; Wonser, Josh: Gold(I)-Catalyzed Intramolecular [4+3]-Cycloaddition Reactions with Furan Propargyl Esters as the Substrates: Carbenoid vs. Stabilized Allyl Cation

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Leckie, Stuart M.; Fallan, Charlene; Taylor, James E.; Brown, T. Bruce; Pryde, David; Lébl, Tomáš; Slawin, Alexandra M. Z.; Smith, Andrew D.: Enantioselective NHC-Catalysed Formal [4+2] Cycloaddition of Alkylaryl­ketenes with β,γ-Unsaturated α-Ketophosphonates

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Gawin, Rafał; Pieczykolan, Michał; Malińska, Maura; Woźniak, Krzysztof; Grela, Karol: Testing New Ruthenium Complexes bearing Chiral 1,2,4-Triazol-5-ylidene ­Ligands as Catalysts for Asymmetric Olefin Metathesis

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Gu, Peng; Xu, Qin; Shi, Min: Synthesis of Novel N-Heterocyclic Carbene-Oxazoline Palladium Complexes and Their Applications in Suzuki–Miyaura Cross-Coupling Reaction

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Brahmi, Malika Makhlouf; Malacria, Max; Curran, Dennis P.; Fensterbank, Louis; Lacôte, Emmanuel: Substituent Effects in NHC–Boranes: Reactivity Switch in the Nucleophilic Fluorination of NHC–Boranes

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Issue 03/2013

Cluster Cover Page

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Yasuda, Nobuyoshi: Cluster Preface: Process Chemistry

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Chen, Ying; Crockett, Richard D.; Wang, Xin; Larsen, Robert D.; Cui, Sheng; Faul, Margaret M.: Development of a Scalable Synthesis of a VEGFR Inhibitor

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Mudryk, Boguslaw; Joshi, Amit; Ortiz, Adrian; Young, Ian S.; Sawyer, James R.; Zheng, Bin; Sugiyama, Masano; Shi, Zhongping; Müslehiddinoğlu, Jale; Corbett, R. Michael; Kronenthal, David R.; Conlon, David A.: Evolution of the Process for the Preparation of a Selective ErbB VEGF Receptor Inhibitor

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Houpis, Ioannis N.; Lemaire, Sebastien; Farina, Vittorio; Xiao, Tingting; Liu, Renmao; Nettekoven, Ulrike; Wang, Youchu: New Synthesis of 2′,4′-Functionalized Nucleotides via Stereospecific Hydrogenation and Azidation Reactions

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Lu, Bruce Z.; Li, Guisheng; Rodriguez, Sonia; Liu, Jianxu; Eriksson, Magnus C.; Tan, Zhulin; Song, Jinhua J.; Yee, Nathan K.; Farina, Vittorio; Senanayake, Chris H.: Development of a Practical Synthesis of 4-[6-(Morpholinomethyl)-pyridin-3-yl]naphthalen-1-amine, a Key Intermediate for the Synthesis of BIRB 1017, a Potent p38 MAP Kinase Inhibitor

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Chase, Charles E.; Fang, Francis G.; Lewis, Bryan M.; Wilkie, Gordon D.; Schnaderbeck, Matthew J.; Zhu, Xiaojie: Process Development of Halaven^®: Synthesis of the C1–C13 Fragment from d-(–)-Gulono-1,4-lactone

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Austad, Brian C.; Benayoud, Farid; Calkins, Trevor L.; Campagna, Silvio; Chase, Charles E.; Choi, Hyeong-wook; Christ, William; Costanzo, Robert; Cutter, James; Endo, Atsushi; Fang, Francis G.; Hu, Yongbo; Lewis, Bryan M.; Lewis, Michael D.; McKenna, Shawn; Noland, Thomas A.; Orr, John D.; Pesant, Marc; Schnaderbeck, Matthew J.; Wilkie, Gordon D.; Abe, Taichi; Asai, Naoki; Asai, Yumi; Kayano, Akio; Kimoto, Yuichi; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Mizuno, Masanori; Nakamura, Taiju; Omae, Takao; Ozeki, Naoki; Suzuki, Taeko; Takigawa, Teiji; Watanabe, Tomohiro; Yoshizawa, Kazuhiro: Process Development of Halaven^®: Synthesis of the C14–C35 Fragment via Iterative Nozaki–Hiyama–Kishi Reaction–Williamson Ether Cyclization

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Austad, Brian C.; Calkins, Trevor L.; Chase, Charles E.; Fang, Francis G.; Horstmann, Thomas E.; Hu, Yongbo; Lewis, Bryan M.; Niu, Xiang; Noland, Thomas A.; Orr, John D.; Schnaderbeck, Matthew J.; Zhang, Huiming; Asakawa, Naoki; Asai, Naoki; Chiba, Hiroyuki; Hasebe, Takashi; Hoshino, Yorihisa; Ishizuka, Hiroyuki; Kajima, Takashi; Kayano, Akio; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Miyazawa, Mamoru; Tagami, Katsuya; Watanabe, Tomohiro: Commercial Manufacture of Halaven^®: Chemoselective Transformations En Route to Structurally Complex Macrocyclic Ketones

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Issue 19/2012

Cluster Cover Page

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White, M. Christina: C–H Bond Functionalization & Synthesis in the 21^st Century: A Brief History and Prospectus

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Zhang, Hao; Chen, Pinhong; Liu, Guosheng: Palladium-Catalyzed Oxidative Arylalkylation of Unactivated Alkenes: Dual C–H Bond Cleavage of Anilines and Acetonitrile

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Lo, Vanessa Kar-Yan; Thu, Hung-Yat; Chan, Yu-Man; Lam, Tsz-Lung; Yu, Wing-Yiu; Che, Chi-Ming: Stereoselective Intramolecular Carbene C–H Insertion Catalyzed by Rhodium(III) Porphyrin Complexes

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Jia, Zhenhua; Li, Xingshu; Chan, Albert S. C.; Li, Chao-Jun: Silver-Catalyzed Direct Addition of Terminal Alkynes to Simple Cyclic Ketones in Water

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Ano, Yusuke; Tobisu, Mamoru; Chatani, Naoto: Ruthenium-Catalyzed Direct ortho-Alkynylation of Arenes with Chelation Assistance

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Bigi, Marinus A.; Liu, Peng; Zou, Lufeng; Houk, K. N.; White, M. Christina: Cafestol to Tricalysiolide B and Oxidized Analogues: Biosynthetic and Derivatization Studies Using Non-heme Iron Catalyst Fe(PDP)

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Issue 01/2012

Toste, F. Dean: Cluster Preface: Gold Catalysis for Organic Synthesis: Opportunities Abound

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Huguet, Núria; Echavarren, Antonio M.: Gold-Catalyzed Cyclization of Oxo-1,5-enynes

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Sun, Sheng; Kroll, Julien; Luo, Yingdong; Zhang, Liming: Gold-Catalyzed Regioselective Dimerization of Aliphatic Terminal Alkynes

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Kojima, Masafumi; Mikami, Koichi: Enantioselective Intramolecular Hydroamination of N-Alkenyl Ureas Catalyzed by tropos BIPHEP-Gold(I) Complexes with Au-Au Interaction

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Martín-Rodríguez, María; Nájera, Carmen; Sansano, José M.: Enantioselective 1,3-Dipolar Cycloadditions of Azlactones and Electrophilic Alkenes Catalyzed by Dimeric BinapAuTFA Complexes

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Asao, Naoki; Menggenbateer; Seya, Yohei; Yamamoto, Yoshinori; Chen, Mingwei; Zhang, Wei; Inoue, Akihisa: Nanoporous Gold-Catalyzed [4+2] Benzannulation between ortho-Alkynylbenzaldehydes and Alkynes

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Davies, Paul W.; Albrecht, Sebastien J.-C.: A Reactivity Switch in the Gold-Catalysed Coupling of Allyl Sulfides with Propargylic Carboxylates

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Pradal, Alexandre; Chen, Qian; Faudot dit Bel, Pierre; Toullec, Patrick Yves; Michelet, Véronique: Gold-Catalyzed Cycloisomerization of Functionalized 1,5-Enynes - An Entry to Polycyclic Framework

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Issue 09/2011

Wilcke, David; Herdtweck, Eberhardt; Bach, Thorsten: Enantioselective Brønsted Acid Catalysis in the Friedel-Crafts Reaction of Indoles with Secondary ortho-Hydroxybenzylic Alcohols

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Zhang, Jun-Wei; Cai, Quan; Shi, Xiao-Xin; Zhang, Wei; You, Shu-Li: Enantioselective Synthesis of Tetrahydropyrano[3,4-b]indoles Catalyzed by Chiral N-Triflyl Phosphoramide via Intramolecular Friedel-Crafts Alkylation Reaction

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Rueping, Magnus; Hubener, Lukas: Enantioselective Synthesis of Quinolizidines and Indolizidines via a Catalytic Asymmetric Hydrogenation Cascade

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Hatano, Manabu; Sugiura, Yoshihiro; Akakura, Matsujiro; Ishihara, Kazuaki: Enantioselective Friedel-Crafts Aminoalkylation Catalyzed by Chiral Ammonium 1,1′-Binaphthyl-2,2′-disulfonates

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Zhu, Chen; Akiyama, Takahiko: Brønsted Acid Catalyzed Reductive Amination with Benzothiazoline as a Highly Efficient Hydrogen Donor

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Terada, Masahiro; Kanomata, Kyohei: Metal-Free Chiral Phosphoric Acid or Chiral Metal Phosphate as Active Catalyst in the Activation of N-Acyl Aldimines

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Aguado, Andreina; Takenaka, Norito: Intramolecular Nitroalkene Diels-Alder Reaction Catalyzed by Brønsted Acids

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Zhang, Zhiguo; Jakab, Gergely; Schreiner, Peter R.: Enantioselective Synthesis of 2-Aryl-3-nitro-2H-chromenes Catalyzed by a Bifunctional Thiourea

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Uraguchi, Daisuke; Kinoshita, Natsuko; Kizu, Tomohito; Ooi, Takashi: Enantioselective Aza-Michael Addition to Conjugated Nitroenynes Catalyzed by Chiral Arylaminophosphonium Barfates

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Issue 04/2011

List, Benjamin: Cluster Preface: Challenges of Proline-Based Aminocatalysis

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Alza, Esther; Sayalero, Sonia; Cambeiro, Xacobe C.; Martín-Rapún, Rafael; Miranda, Pedro O.; Pericàs, Miquel A.: Catalytic Batch and Continuous Flow Production of Highly Enantioenriched Cyclohexane Derivatives with Polymer-Supported Diarylprolinol Silyl Ethers

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Enders, Dieter; Wang, Chuan; Yang, Xuena; Raabe, Gerhard: One-Pot Organocatalytic Asymmetric Synthesis of 1H-Pyrrolo[1,2a]indol-3(2H)-ones via a Michael-Hemiaminalization-Oxidation Sequence

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Wang, Jian; Zhang, Man-Man; Zhang, Shieli; Xu, Zi-An; Li, Hao; Yu, Xin-Hong; Wang, Wei: Chiral Pyrrolidine Sulfonamide Catalyzed Enantioselective Michael Addition of Cyclohexanones to Maleimides

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Lu, Min; Lu, Yunpeng; Tan, Puay Kah Amy; Lau, Qiu Ying; Zhong, Guofu: Highly Enantioselective Synthesis of Fluorinated β-Amino Ketones via Asymmetric Organocatalytic Mannich Reactions: A Case Study of Unusual Reversal of Regioselectivity

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Bisai, Vishnumaya; Singh, Vinod K.: Organocatalytic Enantioselective Direct Aldol Reaction in Aqueous Media Catalyzed by a Bifunctional Diamine Catalyst

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Hayashi, Yujiro; Yasui, Yusuke; Kawamura, Tsuyoshi; Kojima, Masahiro; Ishikawa, Hayato: Diarylprolinol in the Direct Asymmetric Aldol Reaction of Trifluoromethylacetaldehyde Ethyl Hemiacetal with Aldehyde

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Vera, Silvia; Liu, Yankai; Marigo, Mauro; Escudero-Adán, Eduardo C.; Melchiorre, Paolo: Asymmetric Michael Addition of Nitrobenzyl Pyridines to Enals via Iminium Catalysis

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Qiao, Yupu; Zhang, Long; Luo, Sanzhong; Cheng, Jin-Pei: Chiral Zwitterions from Vicinal Diamines: Effective and Recoverable Asymmetric Enamine Catalysts

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Messerer, Matthias; Wennemers, Helma: Reversing the Enantioselectivity of a Peptidic Catalyst by Changing the Solvent

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Freund, Matthias H.; Tsogoeva, Svetlana B.: l-Proline-Catalyzed Asymmetric Michael Addition of 2-Oxindoles to Enones: A Convenient Access to Oxindoles with a Quaternary Stereocenter

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Ward, Dale E.; Jheengut, Vishal; Beye, Garrison E.; Gillis, H. Martin; Karagiannis, Athanasios; Becerril-Jimenez, Fabiola: Enantioselective Direct Aldol Reactions of Achiral Ketones with Racemic Enolizable α-Substituted Aldehydes: Scope and Limitations

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Issue 13/2010

Uozumi, Yasuhiro: Green Chemistry - A New Paradigm of Organic Synthesis

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Hagiwara, Hisahiro; Sasaki, Hirokazu; Tsubokawa, Norio; Hoshi, Takashi; Suzuki, Toshio; Tsuda, Tetsuya; Kuwabata, Susumu: Immobilization of Pd on Nanosilica Dendrimer as SILC: Highly Active and Sustainable Cluster Catalyst for Suzuki-Miyaura Reaction

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Leung, Peter Shu-Wai; Teng, Yan; Toy, Patrick H.: Rasta Resin-PPh₃ and its Use in Chromatography-Free Wittig Reactions

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Zeng, Tieqiang; Song, Gonghua; Moores, Audrey; Li, Chao-Jun: Magnetically Recoverable Iron Nanoparticle Catalyzed Cross-Dehydrogena­tive Coupling (CDC) between Two Csp^³-H Bonds Using Molecular Oxygen

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Ceylan, Sascha; Klande, Tobias; Vogt, Carla; Friese, Carsten; Kirschning, Andreas: Chemical Synthesis with Inductively Heated Copper Flow Reactors

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Matsubara, Hiroshi; Tsukida, Masaaki; Ishihara, Daisuke; Kuniyoshi, Kenji; Ryu, Ilhyong: A Photoirradiative Phase-Vanishing Method: Efficient Generation of HBr from Alkanes and Molecular Bromine and Its Use for Subsequent Radical Addition to Terminal Alkenes

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Karimi, Babak; Behzadnia, Hesam: Novel Periodic Mesoporous Silica Chlorides (PMSCl) with 2D P₆mm Hexagonal Structures: Efficient Catalysts for the Beckmann Rearrangement

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Hatano, Manabu; Mizuno, Tomokazu; Ishihara, Kazuaki: A Concise Synthesis of (S)-(+)-Ginnol Based on Catalytic Enantioselective Addition of Commercially Unavailable Di(n-alkyl)zinc to Aldehydes and Ketones

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Xiao, Jian; Liu, Yan-Ling; Loh, Teck-Peng: The Organocatalytic Enantioselective Michael Addition of Aldehydes to Vinyl Sulfones in Water

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Kobayashi, Shu; Kitanosono, Taku; Ueno, Masaharu: Copper(II) and Bismuth(III) Hydroxide Catalyzed Addition Reactions of Hydrazonoester with Allenylboronate in Aqueous Media

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Ulbrich, Kathrin; Kreitmeier, Peter; Reiser, Oliver: Microwave- or Microreactor-Assisted Conversion of Furfuryl Alcohols into 4-Hydroxy-2-cyclopentenones

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Huang, Shenlin; Voigtritter, Karl R.; Unger, John B.; Lipshutz, Bruce H.: Asymmetric CuH-Catalyzed 1,4-Reductions in Water at Room Temperature

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Issue 11/2010

Overman, Larry E.: Cluster Preface: Stereoselective Synthesis of Stereogenic Quaternary Carbons: A Formidable Challenge and Remarkable Recent Progress

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Müller, Daniel; Hawner, Christine; Tissot, Matthieu; Palais, Laëtitia; Alexakis, Alexandre: Creation of Quaternary Stereogenic Centers via Copper-Catalyzed Asymmetric Conjugate Addition of Alkenyl Alanes to α,β-Unsaturated Cyclic Ketones

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Seiser, Tobias; Cathomen, Gino; Cramer, Nicolai: Enantioselective Construction of Indanones from Cyclobutanols Using a Rhodium-Catalyzed C-C/C-H/C-C Bond Activation Process

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Pesciaioli, Fabio; Tian, Xu; Bencivenni, Giorgio; Bartoli, Giuseppe; Melchiorre, Paolo: Organocatalytic Asymmetric Conjugate Additions of Oxindoles and Benzofuranones to Cyclic Enones

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Hsieh, Jen-Chieh; Ebata, Shiro; Nakao, Yoshiaki; Hiyama, Tamejiro: Asymmetric Synthesis of Indolines Bearing a Benzylic Quaternary Stereocenter through Intramolecular Arylcyanation of Alkenes

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McDougal, Nolan T.; Virgil, Scott C.; Stoltz, Brian M.: High-Throughput Screening of the Asymmetric Decarboxylative Alkylation Reaction of Enolate-Stabilized Enol Carbonates

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Gu, Zhenhua; Herrmann, Aaron T.; Stivala, Craig E.; Zakarian, Armen: Stereoselective Construction of Adjacent Quaternary Chiral Centers by the Ireland-Claisen Rearrangement: Stereoselection with Esters of Cyclic Alcohols

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Denmark, Scott E.; Wilson, Tyler W.: Construction of Quaternary Stereogenic Carbon Centers by the Lewis Base Catalyzed Conjugate Addition of Silyl Ketene Imines to α,β-Unsaturated Aldehydes and Ketones

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Issue 02/2010

He, Guangke; Xue, Can; Fu, Chunling; Ma, Shengming: An Efficient Synthesis of Allenyl Perfluoroalkyl Ketones from Mono-1,2-Addition-Elimination Reaction of Allenoates with R_fMgX

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Satoh, Tsuyoshi; Kasuya, Takashi; Miyagawa, Toshifumi; Nakaya, Nobuhito: Cyclobutylmagnesium Carbenoids: Generation from 1-Chlorocyclobutyl p-Tolyl Sulfoxides with Ethylmagnesium Chloride, Properties, and Some Synthetic Uses

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Tuulmets, Ants; Ploom, Anu; Panov, Dmitri; Järv, Jaak: Selectivity in the Grignard Reaction with Silanes

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Ackermann, Lutz; Wechsler, Cindy; Kapdi, Anant R.; Althammer, Andreas: Air-Stable Diaminophosphine Sulfides as Preligands for Nickel-Catalyzed Cross-Couplings of Unactivated Fluoro(hetero)arenes

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Cahiez, Gérard; Gager, Olivier; Buendia, Julien: New Insights into the Copper-Catalyzed Alkylation of Grignard and Organolithium Reagents

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Monzon, Gabriel; Knochel, Paul: Directed ortho- and meta-Magnesiation or Zincation of Polyfunctional Aryl Nonaflates

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Mitamura, Yukihiro; Someya, Hidenori; Yorimitsu, Hideki; Oshima, Koichiro: Silver-Catalyzed Diallylation and Dibenzylation of gem-Dibromoalkanes with Grignard Reagents

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Yoshikai, Naohiko; Matsumoto, Arimasa; Norinder, Jakob; Nakamura, Eiichi: Iron-Catalyzed Direct Arylation of Aryl Pyridines and Imines Using Oxygen as an Oxidant

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Ladjel, Chehla; Fuchs, Nicolas; Gremaud, Ludovic; Alexakis, Alexandre: Copper-Catalysed Kinetic Resolution of Cyclic Alkenyl Cyclopropane Malonates with Organoaluminium and Grignard Reagents

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Hatano, Manabu; Suzuki, Shinji; Ishihara, Kazuaki: Highly Chemoselective Stoichiometric Alkylation of Ketones with Grignard Reagent Derived Zinc(II) Ate Complexes

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Kobayashi, Yuichi; Tani, Yukio; Nakata, Kenya; Kaneko, Yuki: Allylic Substitution of 4-Cyclopentene-1,3-diol Monoacetate with Copper Reagents Derived from Functionalized Aryl Grignard Reagents

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Levin, Anat; Basheer, Ahmad; Marek, Ilan: Regiodivergent Carbometalation Reactions of Ynol Ether Derivatives

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Issue 10/2009

Ito, Masato; Shibata, Yuji; Watanabe, Akira; Ikariya, Takao: (η⁶-Arene)Ru^II/Chiral SN Ligand: A Novel Bifunctional Catalyst System for Asymmetric Transfer Hydrogenation of Aromatic Ketones

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Inokuma, Tsubasa; Sakamoto, Shota; Takemoto, Yoshiji: Enantioselective Nitrocyclopropanation of α,β-Unsaturated α-Cyanoimides Catalyzed by Bifunctional Thiourea

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Hamashima, Yoshitaka; Tamura, Toshihiro; Suzuki, Shoko; Sodeoka, Mikiko: Enantioselective Protonation in the Aza-Michael Reaction Using a Combination of Chiral Pd-µ-Hydroxo Complex with an Amine Salt

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Kato, Yuko; Chen, Zhihua; Matsunaga, Shigeki; Shibasaki, Masakatsu: Catalytic Asymmetric Synthesis of Nitrogen-Containing gem-Bisphosphonates Using a Dinuclear Ni₂-Schiff Base Complex

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Nakamura, Shuichi; Sakurai, Yuki; Nakashima, Hiroki; Shibata, Norio; Toru, Takeshi: Organocatalytic Enantioselective Aza-Friedel-Crafts Alkylation of Pyrroles with N-(Heteroarenesulfonyl)imines

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Takada, Keisuke; Tanaka, Shinji; Nagasawa, Kazuo: Asymmetric Mannich-Type Reaction of Aromatic α-Amido Sulfone with Malonate Using Guanidine-Thiourea Bifunctional Organocatalyst

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Sakakura, Akira; Umemura, Shuhei; Ishihara, Kazuaki: 3-Pyrroline-1-carbonyl (Pyroc) Group: A Removable Protecting Group for the Kinetic Resolution of Racemic Carboxylic Acids and Alcohols through Catalytic Asymmetric Acylation

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Abraham, Ciby J.; Paull, Daniel H.; Dogo-Isonagie, Cajetan; Lectka, Thomas: Diastereoselective Synthesis of trans-β-Lactams Using a Simple Multifunctional Catalyst

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Wang, Wentao; Shen, Ke; Hu, Xiaolei; Wang, Jun; Liu, Xiaohua; Feng, Xiaoming: Highly Enantioselective Synthesis of α-Diazo-β-hydroxy Esters Using a Bifunctional Titanium Complex

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Iwasaki, Takanori; Maegawa, Yusuke; Hayashi, Yukiko; Ohshima, Takashi; Mashima, Kazushi: A Simple, General, and Highly Chemoselective Acetylation of Alcohols Using Ethyl Acetate as the Acetyl Donor Catalyzed by a Tetranuclear Zinc Cluster

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Akiyama, Takahiko; Katoh, Takuya; Mori, Keiji; Kanno, Kazuaki: Enantioselective Mannich-Type Reaction Catalyzed by a Chiral Phosphoric Acid Bearing an (S)-Biphenol Backbone

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Takizawa, Shinobu; Rajesh, Doss; Katayama, Tomomi; Sasai, Hiroaki: One-Pot Preparation of Chiral Dinuclear Vanadium(V) Complex

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Nakano, Megumi; Terada, Masahiro: Acid-Base Dual-Functional Catalysis by Axially Chiral Guanidine in Enantioselective [3+2] Cycloaddition of Maleate to Schiff Bases as a Precursor of Azomethine Ylides

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Chidara, Sridhar; Lin, Yun-Ming: Reaction Rate Acceleration Enabled by Tethered Lewis Acid-Lewis Base Bifunctional Catalysis: A Catalytic, Enantioselective [2+2] Ketene Aldehyde Cycloaddition Reaction

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Mita, Tsuyoshi; Jacobsen, Eric N.: Bifunctional Asymmetric Catalysis with Hydrogen Chloride: Enantioselective Ring Opening of Aziridines Catalyzed by a Phosphinothiourea

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Liu, Xiaofeng; Sun, Bingfeng; Deng, Li: Catalytic Enantioselective Electrophilic Aminations of Acyclic α-Alkyl β-Carbonyl Nucleophiles

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Issue 04/2009

Christiansen, Michael A.; Butler, Aaron W.; Hill, Amanda R.; Andrus, Merritt B.: Synthesis of Kurasoin B Using Phase-Transfer-Catalyzed Acylimidazole Alkylation

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Uraguchi, Daisuke; Asai, Yoshihiro; Seto, Yuki; Ooi, Takashi: Asymmetric Synthesis of α,α-Disubstituted α-Amino Acids via Enantioselective Alkylation of Azlactones under Biphasic Conditions Using P-Spiro Chiral Tetraaminophosphonium Salts as a Phase-Transfer Catalyst

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Hashimoto, Takuya; Sasaki, Keigo; Fukumoto, Kazuhiro; Murase, Yuichi; Ooi, Takashi; Maruoka, Keiji: Phase-Transfer-Catalyzed Enantioselective Alkylation of α-Benzoyloxy-β-Keto Ester

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Ding, Changhua; Maruoka, Keiji: Enantioselective Alkylation of α-Fluoro-β-Keto Esters by Asymmetric Phase-Transfer Catalysis

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Tanaka, Shinji; Nagasawa, Kazuo: Guanidine-Urea Bifunctional Organocatalyst for Asymmetric Epoxidation of 1,3-Diarylenones with Hydrogen Peroxide

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Kim, Taek-Soo; Lee, Yeon-Ju; Lee, Kyoungyim; Jeong, Byeong-Seon; Park, Hyeung-geun; Jew, Sang-sup: Enantioselective Synthesis of (R)-α-Alkylhomoserines and (R)-α-Alkylhomocysteines via Phase-Transfer Catalytic Alkylation

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Lygo, Barry; Allbutt, Bryan; Beaumont, Douglas J.; Butt, Umar; Gilks, James A. R.: Synthesis and Evaluation of Chiral Dibenzazepinium Halide Phase-Transfer Catalysts

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Issue 01/2009

Lovely, Carl J.; Flores, Jaime A.; Meng, Xiaofeng; Dias, H. V. Rasika: Silver-Catalyzed C-H Insertion Reactions with Donor-Acceptor Diazoacetates

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Pillekamp, Marcus; Aniol, Alexandra; Heppekausen, Johannes; Neukirchen, Saskia; Seel, Stephanie; Oppel, Iris M.; Dyker, Gerald: Palladium-Catalyzed Four-Membered Ring Annelation Reactions at Dibenzobarrelene

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Yoo, Woo-Jin; Correia, Camille A.; Zhang, Yuhua; Li, Chao-Jun: Oxidative Alkylation of Cyclic Benzyl Ethers with Malonates and Ketones Using Oxygen as the Terminal Oxidant

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Zalatan, David N.; Du Bois, J.: Oxidative Cyclization of Sulfamate Esters Using NaOCl - A Metal-Mediated Hoffman-Löffler-Freytag Reaction

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Harrisson, Peter; Morris, James; Steel, Patrick G.; Marder, Todd B.: A One-Pot, Single-Solvent Process for Tandem, Catalyzed C-H Borylation-Suzuki-Miyaura Cross-Coupling Sequences

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Nadeau, Etienne; Li, Zhanjie; Morton, Daniel; Davies, Huw M. L.: Rhodium Carbenoid Induced Intermolecular C-H Functionalization at Tertiary C-H Bonds

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Issue 10/2008

Shirakawa, Seiji; Shimizu, Shoichi: Dehydrative Amination of Alcohols in Water Using a Water-Soluble Calix[4]resorcinarene Sulfonic Acid

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Egami, Hiromichi; Katsuki, Tsutomu: Optimization of Asymmetric Oxidation of Sulfides with the Fe(salan) Complex in Water and the Expanded Scope of its Application

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Beletskaya, Irina P.; Kashin, Alexander N.; Khotina, Irina A.; Khokhlov, Alexey R.: Efficient and Recyclable Catalyst of Palladium Nanoparticles Stabilized by Polymer Micelles Soluble in Water for Suzuki-Miyaura Reaction, Ostwald Ripening Process with Palladium Nanoparticles

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Lee, Hang Wai; Kwong, Fuk Yee; Chan, Albert S. C.: Rh-Catalyzed Aqueous Pauson-Khand-Type Cycloaddition in Microwave-Irradiated Medium

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Uozumi, Yasuhiro; Takenaka, Hiroe; Suzuka, Toshimasa: Allylic Substitution of meso-1,4-Diacetoxycycloalkenes in Water with an Amphiphilic Resin-Supported Chiral Palladium Complex

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Kokubo, Masaya; Kobayashi, Shu: Scandium(III) Fluoride as a Novel Catalyst for Hydroxymethylation of Dimethylsilyl Enolates in Aqueous Media

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Hayashi, Yujiro; Itoh, Takahiko; Nagae, Norio; Ohkubo, Masahiro; Ishikawa, Hayato: The Effectiveness of Proteinogenic Amino Acids in the Asymmetric Aldol Reaction in DMSO and Aqueous DMSO

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Deng, Guo-Jun; Li, Chao-Jun: Efficient Direct Alkynylation of Trifluoromethyl Ketones Catalyzed by AgF in Water and Organic Solvents

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Bonollo, Simona; Fringuelli, Francesco; Pizzo, Ferdinando; Vaccaro, Luigi: Zn(II)-Catalyzed Desymmetrization of meso-Epoxides by Aromatic Amines in Water

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Issue 05/2008

McLaughlin, Martin; Shimp, Heidi L.; Navarro, Raul; Micalizio, Glenn C.: Regio- and Stereoselective Direct Cross-Coupling of Aromatic Imines with Allenic Alcohols

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Antoline, Jennifer E.; Hsung, Richard P.: An Unexpected Reversal of Diastereoselectivity in the [4+3]-Cycloaddition Reaction of Nitrogen-Stabilized Oxyallyl Cations with Methyl 2-Furoate

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Abu Sohel, Shariar Md; Lin, Sheng-Hsun; Liu, Rai-Shung: Platinum-Catalyzed Tandem Cyclization-Nazarov Cylization Reactions: An Easy Access to Complex Carbocyclic Molecules from 2-Alkenyl-(1′-hydroxyl-4-en-2-ynyl)benzenes

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Buisine, Olivier; Gandon, Vincent; Fensterbank, Louis; Aubert, Corinne; Malacria, Max: Thermal Intramolecular Alder-Ene Cycloisomerization of 1,6-Allenynes

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Onodera, Gen; Matsuzawa, Masayoshi; Aizawa, Takahiro; Kitahara, Takeshi; Shimizu, Yoshihisa; Kezuka, Satoko; Takeuchi, Ryo: [Ir(cod)Cl]₂/FDPPE-Catalyzed Chemo- and Regioselective Cyclotrimerization of Two Different Terminal Alkynes To Give 1,3,5-Trisubstituted Benzenes

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Brummond, Kay M.; Chen, Daitao; Painter, Thomas O.; Mao, Shuli; Seifried, Darla D.: A Rh(I)-Catalyzed Cycloisomerization Reaction Affording Cyclic Trienones

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Shibata, Takanori; Nishizawa, Go; Endo, Kohei: Iridium-Catalyzed Enantioselective Formal [4+2] Cycloaddition of Biphenylene and Alkynes for the Construction of Axial Chirality

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Dugovič, Branislav; Reissig, Hans-Ulrich: A New Alkoxyallene-Based [3+2] Approach to the Synthesis of Highly Substituted Cyclopentenones

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Nakao, Yoshiaki; Takeda, Masahide; Chen, Jinshui; Hiyama, Tamejiro: Rhodium-Catalyzed Hydroarylation and Hydroalkenylation of Alkynes Using Organo[2-(hydroxymethyl)phenyl]dimethylsilanes

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Oh, Chang Ho; Kim, Ahyun: Gold-Catalyzed [2+2] Cyclization of Alkyne-propargylic Pivaloates to Fused Bicyclic Compounds

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Issue 11/2007

Hashmi, A. Stephen K.; Wölfle, Michael; Teles, J. Henrique; Frey, Wolfgang: Bisphenols from Furfurals by Organocatalysis and Gold Catalysis

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Cabello, Noemí; Rodríguez, Cristina; Echavarren, Antonio M.: Gold-Catalyzed Cyclizations of 1,7-Enynes

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Skouta, Rachid; Li, Chao-Jun: Au(I)-Catalyzed Annulation of 2-Tosylaminobenzaldehyde and Alkynes

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Hashmi, A. Stephen K.; Salathé, Ralph; Frey, Wolfgang: Gold-Catalyzed Cyclization of N-Alkynyl Carbamates

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Nishina, Naoko; Yamamoto, Yoshinori: Gold-Catalyzed Intermolecular Hydroamination of Allenes: First Example of the Use of an Aliphatic Amine in Hydroamination

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Corma, Avelino; González-Arellano, Camino; Iglesias, Marta; Pérez-Ferreras, Susana; Sánchez, Félix: Heterogenized Gold(I), Gold(III), and Palladium(II) Complexes for C-C Bond Reactions

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Ambrogio, Ilaria; Arcadi, Antonio; Cacchi, Sandro; Fabrizi, Giancarlo; Marinelli, Fabio: Gold-Catalyzed Synthesis of 2-Substituted, 2,3-Disubstituted and 1,2,3-Trisubstituted Indoles in [bmim]BF₄

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Genin, Emilie; Leseurre, Lucie; Toullec, Patrick Yves; Genêt, Jean-Pierre; Michelet, Véronique: Gold-Catalyzed Hydroxy- and Alkoxycyclization of Functionalized Enynes

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Brouwer, Chad; Rahaman, Ronald; He, Chuan: Gold(I)-Mediated Hydrothiolation of Conjugated Olefins

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Deutsch, Carl; Gockel, Birgit; Hoffmann-Röder, Anja; Krause, Norbert: Golden Opportunities in Stereoselective Catalysis: Optimization of Chirality Transfer and Catalyst Efficiency in the Gold-Catalyzed Cycloisomerization of α-Hydroxyallenes to 2,5-Dihydrofurans

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Issue 07/2007

Kang, Young Ku; Cho, Min Je; Kim, Sun Mi; Kim, Dae Young: Asymmetric Electrophilic Fluorination of α-Cyanoalkylphosphonates ­Catalyzed by Chiral Palladium Complexes

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Moriya, Ken-ichi; Hamashima, Yoshitaka; Sodeoka, Mikiko: Pd(II)-Catalyzed Asymmetric Fluorination of α-Aryl-α-cyanophosphonates with the Aid of 2,6-Lutidine

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Ramírez, Jesús; Huber, Dominique P.; Togni, Antonio: Asymmetric Electrophilic Fluorination of α-Nitro Esters

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Hidaka, Asami; Zagipa, Bakenova; Nagura, Hirokatsu; Fuchigami, Toshio: Regioselective Anodic Fluorination of α-(Arylthio)benzylphosphonate Esters, α-(Arylthio)methylphosphonate Esters and Their Analogues

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Shibata, Norio; Yasui, Hiroyuki; Nakamura, Shuichi; Toru, Takeshi: DNA-Mediated Enantioselective Carbon-Fluorine Bond Formation

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Prakash, G. K. Surya; Linares-Palomino, Pablo J.; Glinton, Kevin; Chacko, Sujith; Rasul, Golam; Mathew, Thomas; Olah, George A.: Friedel-Crafts Alkylations of Arenes with Mono- and Bis(trifluoro­methyl)oxiranes in Superacid Medium: Facile Synthesis of α-(Trifluoro­methyl)- and α,α-Bis(Trifluoromethyl)-β-Arylethanols

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Shimizu, Masaki; Higashi, Masahiro; Takeda, Youhei; Jiang, Guofang; Murai, Masahito; Hiyama, Tamejiro: Novel Generation of 3,3,3-Trifluoropropynyllithium and Transformation of the Carbonyl Adducts to Trifluoromethyl-Substituted Allenes

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Purser, Sophie; Wilson, Christopher; Moore, Peter R.; Gouverneur, Véronique: Highly Diastereoselective Electrophilic Fluorination of Cyclic syn-β-
Hydroxysilanes

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Mori, Takashi; Ichikawa, Junji: Radical 6-endo-trig Cyclization of β,β-Difluoro-o-isocyanostyrenes: A Facile Synthesis of 3-Fluoroquinolines and Their Application to the ­Synthesis of 11-Alkylated Cryptolepines

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Issue 20/2006

Colladon, Marco; Scarso, Alessandro; Strukul, Giorgio: Tailoring Pt(II) Chiral Catalyst Design for Asymmetric Baeyer-Villiger ­Oxidation of Cyclic Ketones with Hydrogen Peroxide

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Zhao, Gui-Ling; Dziedzic, Pawel; Ibrahem, Ismail; Córdova, Armando: Organocatalytic Asymmetric Synthesis of 1,2,3-prim,sec,sec-Triols

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Bourhani, Zaïnaba; Malkov, Andrei V.: Vanadium-Catalyzed Asymmetric Epoxidation: Proline-Derived Hydroxamic Acids Revisited

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Chen, Zhihua; Morimoto, Hiroyuki; Matsunaga, Shigeki; Shibasaki, Masakatsu: Catalytic Asymmetric Epoxidation of α-Methyl α,β-Unsaturated Anilides as Ester Surrogates

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Ebner, David C.; Novák, Zoltán; Stoltz, Brian M.: Oxidative Kinetic Resolution-Claisen Rearrangement Sequence to ­Enantioenriched Arylcycloalkenes

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Mohammadpoor-Baltork, Iraj; Hill, Mathias; Caggiano, Lorenzo; Jackson, Richard F. W.: Oxidative Kinetic Resolution of Alkyl Aryl Sulfoxides

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Matsumoto, Kazuhiro; Sawada, Yuji; Katsuki, Tsutomu: Catalytic Enantioselective Epoxidation of Unfunctionalized Olefins: Utility of a Ti(Oi-Pr)₄-Salan-H₂O₂ System

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Issue 14/2006

Miller, Aubry K.; Trauner, Dirk: Mapping the Chemistry of Highly Unsaturated Pyrone Polyketides

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Zhang, Hongjun; Padwa, Albert: Utilization of Some Novel Cascade Reactions for the Synthesis of Various Hydroxylated Phenanthridones

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Sinclair, Alex; Arini, Louise G.; Rejzek, Martin; Szeto, Peter; Stockman, Robert A.: Combining Two-Directional Synthesis and Tandem Reactions, Part 8: A Novel Condensation/Michael Addition/Cycloaddition/Fragmentation/Lactamisation Cascade

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Sromek, Anna W.; Rheingold, Arnold L.; Wink, Donald J.; Gevorgyan, Vladimir: Chemodivergent Transformations of Alkynyl Imines

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Heffron, Timothy P.; Jamison, Timothy F.: Concerning Lewis Acid Promoted, Directing-Group-Free Epoxide-Ring-Opening Cascades

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Werner, Stefan; Turner, David M.; Lyon, Michael A.; Huryn, Donna M.; Wipf, Peter: A Focused Library of Tetrahydropyrimidinone Amides via a Tandem Biginelli-Ugi Multi-Component Process

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Tanguy, Chloé; Bertus, Philippe; Szymoniak, Jan; Larionov, Oleg V.; de Meijere, Armin: Convenient Access to 2-Arylpyrroles from 2-Lithio-N,N-dibenzylcyclopropylamine and Nitriles

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Uenoyama, Yoshitaka; Fukuyama, Takahide; Ryu, Ilhyong: Cascade Radical Carbonylations Leading to 3-Substituted Cyclohexanones

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Issue 01/2006

Katayama, Mayumi; Nagase, Ryohei; Mitarai, Kumi; Misaki, Tomonori; Tanabe, Yoo: Isolation of Intermediary anti-Aldol Adducts of the Horner-Wadsworth-­Emmons Reaction Utilizing Direct Titanium-Aldol Addition and Successive Brønsted Acid Promoted Stereoselective Elimination Leading to (Z)-α,β-Unsaturated Esters

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Terada, Masahiro; Sorimachi, Keiichi; Uraguchi, Daisuke: Phosphorodiamidic Acid as a Novel Structural Motif of Brønsted Acid Catalysts for Direct Mannich Reaction of N-Acyl Imines with 1,3-Dicarbonyl Compounds

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Xu, Xuenong; Yabuta, Takaya; Yuan, Pei; Takemoto, Yoshiji: Organocatalytic Enantioselective Hydrazination of 1,3-Dicarbonyl ­Compounds: Asymmetric Synthesis of α,α-Disubstituted α-Amino Acids

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Akiyama, Takahiko; Tamura, Yukio; Itoh, Junji; Morita, Hisashi; Fuchibe, Kohei: Enantioselective Aza-Diels-Alder Reaction Catalyzed by a Chiral Brønsted Acid: Effect of the Additive on the Enantioselectivity

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Sohtome, Yoshihiro; Takemura, Nobuko; Iguchi, Toshitsugu; Hashimoto, Yuichi; Nagasawa, Kazuo: Diastereoselective Henry Reaction Catalyzed by Guanidine-Thiourea Bifunctional Organocatalyst

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Hess, Abram S.; Yoder, Ryan A.; Johnston, Jeffrey N.: Chiral Proton Catalysis: pK_a Determination for a BAM-HX Brønsted Acid

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Nakashima, Daisuke; Yamamoto, Hisashi: Titanium Tetrachloride and Chiral Aliphatic Alcohol as a New Lewis Acid Assisted Chiral Brønsted Acid for the Enantioselective Protonation of Silyl Enol Ether

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Issue 11/2005

Molander, Gary A.; Petrillo, Daniel E.; Landzberg, Nicole R.; Rohanna, John C.; Biolatto, Betina: Palladium-Catalyzed Suzuki-Miyaura Reactions of Potassium Aryl- and Heteroaryltrifluoroborates with Aryl- and Heteroaryl Triflates

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Ma, Dawei; Cai, Qian; Xie, Xiaoan: CuI/N,N-Dimethylglycine-Catalyzed Cross-Coupling Reaction of Vinyl Halides with Phenols and its Application to the Assembly of Substituted Benzofurans

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Saeki, Tomoyuki; Takashima, Yohei; Tamao, Kohei: Nickel- and Palladium-Catalyzed Cross-Coupling Reaction of Polyfluorinated Arenes and Alkenes with Grignard Reagents

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Uozumi, Yasuhiro; Kikuchi, Makoto: Controlled Monoarylation of Dibromoarenes in Water with a Polymeric Palladium Catalyst

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Charette, André B.; Mathieu, Simon; Fournier, Jean-François: Diastereoselective Synthesis of 1,2,3-Substituted Potassium Cyclopropyl Trifluoroborates via an Unusual Zinc-Boron Exchange

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Terao, Jun; Begum, Shameem Ara; Oda, Akihiro; Kambe, Nobuaki: Zr-Catalyzed Coupling Reaction of Alkyl Halides, Tosylates, and Sulfates with β-Phenethyl Grignard Reagents via Styrene-Zirconate Intermediates

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Hirano, Koji; Fujita, Kazuya; Yorimitsu, Hideki; Oshima, Koichiro: Nickel-Catalyzed Cross-Coupling Reaction of Aryl Halides with Allylic Zirconium Reagents Generated in situ from Zirconocene(alkene) Complexes

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Qian, Mingxing; Negishi, Ei-ichi: Palladium-Catalyzed Cross-Coupling of Alkynylzincs with Allylic Electrophiles: An Efficient and Selective Synthesis of Stereo- and Regio-Defined 1,4-Enynes

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Nakamura, Masaharu; Ito, Shingo; Matsuo, Keiko; Nakamura, Eiichi: Iron-Catalyzed Chemoselective Cross-Coupling of Primary and Secondary Alkyl Halides with Arylzinc Reagents

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Berman, Ashley M.; Johnson, Jeffrey S.: Nickel-Catalyzed Electrophilic Amination of Organozinc Halides

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Tonogaki, Keisuke; Soga, Kazuya; Itami, Kenichiro; Yoshida, Jun-ichi: Versatile Synthesis of 1,1-Diaryl-1-alkenes Using Vinylboronate Ester as a Platform

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Issue 04/2005

Kozuch, Sebastian; Leifels, Tycho; Meyer, Dominik; Sbaragli, Laura; Shaik, Sason; Woggon, Wolf-D.: New Synthetic Models of Cytochrome P450: How Different Are They from the Natural Species?

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Mulzer, Johann; Sieg, Andreas; Brücher, Christoph; Müller, Dieter; Martin, Harry J.: Horner-Wadsworth-Emmons Reactions as a Facile Entry to Biogenetic Key Substructures

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Dastlik, Kim A.; Sundermeier, Uta; Johns, Deidre M.; Chen, Yuyin; Williams, Robert M.: An Improved Synthesis of Optically Pure 4-Boc-5,6-Diphenylmorpholin-2-one and 4-Cbz-5,6-Diphenylmorpholin-2-one

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Clark, J. Stephen; Myatt, James; Roberts, Lee; Walshe, Nigel: Investigation of the Biomimetic Synthesis of Emindole SB Using a Fluorinated Polyene Cyclisation Precursor

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Olson, Brooke S.; Trauner, Dirk: Concise Synthesis of (±)-Smenochromene D (= Likonide B)

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Imagawa, Hiroshi; Iyenaga, Tomoaki; Nishizawa, Mugio: Biomimetic Tandem Cyclization Catalyzed by Hg(OTf)₂ Affording ­Polycarbocycles

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Krattiger, Philipp; Wennemers, Helma: Water-Soluble Diketopiperazine Receptors - Selective Recognition of Arginine-Rich Peptides

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Issue 13/2004

Denmark, Scott E.; Heemstra, John R.: Lewis Base Activation of Lewis Acids: Vinylogous Aldol Additions of Silyl Dienol Ethers to Aldehydes

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Anaya de Parrodi, Cecilia; Walsh, Patrick J.: trans-1,2-Diaminocyclopentane-Based Catalyst for the Asymmetric Addition of Alkyl-, Aryl-, and Vinyl Groups to Ketones

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Sibi, Mukund P.; Prabagaran, Narayanasamy: Chiral Relay in Enantioselective Conjugate Radical Additions Using ­Pyrazolidinone Templates. How Does Metal Geometry Impact Selectivity?

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Valenzuela, Marcela; Doyle, Michael P.; Hedberg, Christine; Hu, Wenhao; Holmstrom, Alexandra: Influence of the Diene in the Hetero-Diels-Alder Reaction Catalyzed by Dirhodium(II) Carboxamidates

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Morrison, Darryl J.; Piers, Warren E.; Parvez, Masood: (R)-1,1′-Binaphthyl-2-bis(pentafluorophenyl)borane Lewis Acids

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Abiko, Yumi; Yamagiwa, Noriyuki; Sugita, Mari; Tian, Jun; Matsunaga, Shigeki; Shibasaki, Masakatsu: Catalytic Asymmetric Cyano-Phosphorylation of Aldehydes Promoted by Heterobimetallic YLi₃tris(binaphthoxide) (YLB) Complex

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Xia, Guoyao; Shibatomi, Kazutaka; Yamamoto, Hisashi: Novel Lewis Acid-Assisted Chiral Lewis Acid (LLA) System: Development of Boroxin-Ti-BINOL-Catalyzed Asymmetric Allylation of Aldehydes

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McGilvra, Jeff D.; Rawal, Viresh H.: Carbon-Substituted Co(III) Salens as Effective Catalysts for Enantioselective Diels-Alder Reactions

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Sasaki, Mikio; Yudin, Andrei K.: One-Pot Reduction-Aldol Reaction of Esters

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Issue 01/2004

Lee, Dongwhan; Swager, Timothy M.: Defining Space Around Conjugated Polymers: New Vistas in Self-Amplifying Sensory Materials

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Dyke, Christopher A.; Stewart, Michael P.; Maya, Francisco; Tour, James M.: Diazonium-Based Functionalization of Carbon Nanotubes: XPS and GC-MS Analysis and Mechanistic Implications

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Scott, John L.; Parkin, Sean R.; Anthony, John E.: Radical-Induced Cycloaromatization: Routes to Fluoranthenes and Acephenanthrylenes

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Miller, Jeremie J.; Marsden, Jeremiah A.; Haley, Michael M.: Synthesis and Optical Properties of Donor-Acceptor Tetrakis(phenyl­ethynyl)benzenes

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Bangcuyo, Carlito G.; Smith, Mark D.; Bunz, Uwe H. F.: Tetraethynylbenzo[2,1,3]thiadiazole

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Bancu, Mihail; Rai, Amarjit K.; Cheng, Peichao; Gilardi, Richard D.; Scott, Lawrence T.: Corannulene Polysulfides: Molecular Bowls with Multiple Arms and Flaps

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Miyasaka, Makoto; Rajca, Andrzej: Synthesis of Functionalized Carbon-Sulfur [5]Helicene: Pd-Catalyzed Negishi Cross-Coupling Between the β-Positions of Thiophenes

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Campbell, Katie; Tiemstra, Natasha M.; Prepas-Strobeck, Natasha S.; McDonald, Robert; Ferguson, Michael J.; Tykwinski, Rik R.: Synthesis of a Pyridinophane with endo-Annular Donor Sites

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Jones, Carissa S.; Elliott, Eric; Siegel, Jay S.: Synthesis and Properties of Monosubstituted Ethynylcorannulenes

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Marsella, Michael J.; Estassi, Samia; Wang, Li-Sheng; Yoon, Kunsang: Revisiting Cyclobutadienemetal Complexes: High-Content Dewar Benzene Polymers and a One-Pot Synthesis of Permethylated Ladderanes

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Issue 12/2003

Martin, Harry J.; List, Benjamin: Mining Sequence Space for Asymmetric Aminocatalysis: N-Terminal Prolyl-Peptides Efficiently Catalyze Enantioselective Aldol and Michael Reactions

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Pojarliev, Peter; Biller, William T.; Martin, Harry J.; List, Benjamin: Highly Enantioselective Synthesis of 1,2-Amino Alcohol Derivatives via Proline-Catalyzed Mannich Reaction

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Chowdari, Naidu S.; Ramachary, D. B.; Barbas III, Carlos F.: Organocatalysis in Ionic Liquids: Highly Efficient l-Proline-Catalyzed Direct Asymmetric Mannich Reactions Involving Ketone and Aldehyde Nucleophiles

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Ramachary, D. B.; Chowdari, Naidu S.; Barbas III, Carlos F.: The First Organocatalytic Hetero-Domino Knoevenagel-Diels-Alder-Epimerization Reactions: Diastereoselective Synthesis of Highly Substituted Spiro[cyclohexane-1,2′-indan]-1′,3′,4-triones

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Bøgevig, Anders; Poulsen, Thomas B.; Zhuang, Wei; Jørgensen, Karl Anker: Formation of Optically Active Functionalized β-Hydroxy Nitrones Using a Proline Catalyzed Aldol Reaction of Aldehydes with Carbonyl Compounds and Hydroxylamines

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Wenzel, Anna G.; Lalonde, Mathieu P.; Jacobsen, Eric N.: Divergent Stereoinduction Mechanisms in Urea-Catalyzed Additions to Imines

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Griswold, Keith S.; Horstmann, Thomas E.; Miller, Scott J.: Acyl Sulfonamide Catalysts for Glycosylation Reactions with Trichloroacetimidate Donors

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Hang, Jianfeng; Deng, Li: Dynamic Kinetic Resolution for Asymmetric Synthesis of α-Alkyl Amino Acids via Dual-Function Catalysis of Modified Cinchona Alkaloids

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Ooi, Takashi; Kubota, Yasushi; Maruoka, Keiji: A New N-Spiro C₂-Symmetric Chiral Quaternary Ammonium Bromide Consisting of 4,6-Disubstituted Biphenyl Subunit as an Efficient Chiral Phase-Transfer Catalyst

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Kerr, Mark S.; Rovis, Tomislav: Effect of the Michael Acceptor in the Asymmetric Intramolecular Stetter Reaction

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Shah, Meha H.; France, Stefan; Lectka, Thomas: Bicarbonate Salts as Cost-Effective Bases for the Synthesis of Ketenes and Their Synthetic Equivalents Applied to the Asymmetric Synthesis of β-Lactams

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